Compounds and compositions for prevention of overdose of oxycodone
Patent 7169752 Issued on January 30, 2007. Estimated Expiration Date: September 30, 2024. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.
514/2, Peptide containing (e.g., protein, peptones, fibrinogen, etc.) DOAI514/14, 12 to 15 peptide repeating units in known peptide chain514/15, 9 to 11 peptide repeating units in known peptide chain514/16, 7 or 8 peptide repeating units in known peptide chain514/17, 5 or 6 peptide repeating units in known peptide chain514/18, 3 or 4 peptide repeating units in known peptide chain514/19, 2 peptide repeating units in known peptide chain514/563, RC(=O)N containing (i.e., carboxamide) (R is C or H)530/300, PEPTIDES OF 3 TO 100 AMINO ACID RESIDUES530/327, 11 to 14 amino acid residues in defined sequence530/328, 8 to 10 amino acid residues in defined sequence530/329, 6 to 7 amino acid residues in defined sequence530/330, 4 to 5 amino acid residues in defined sequence530/331Tripeptides, e.g., tripeptide thyroliberin (TRH), melanostatin (MIF), etc.
The invention relates to pharmaceutical compounds and compositions comprised of a chemical moiety attached to an opioid such as oxycodone in a manner that substantially decreases the potential of the opioid to cause overdose. When delivered at the proper dosage the pharmaceutical composition provides therapeutic activity similar to that of the parent active agent. Further the compounds and compositions of the invention are useful in preventing addiction and susceptibility to addiction.
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September 30, 2024. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.
