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Inhibitors of proteasomal activity for stimulating hair growth

Patent 6838252 Issued on January 4, 2005. Estimated Expiration Date: Icon_subject January 15, 2022. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.

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Inventors

Application

No. 10052832 filed on 01/15/2002

US Classes:

435/23, Involving proteinase435/6, Involving nucleic acid514/880, HAIR TREATMENT (THERAPEUTIC-SCALP)530/350, PROTEINS, I.E., MORE THAN 100 AMINO ACID RESIDUES514/457, Coumarins (including hydrogenated)514/263.35, Nitrogen attached indirectly to the purine ring system by acyclic nonionic bonding514/18, 3 or 4 peptide repeating units in known peptide chain548/472, Chalcogen bonded directly to ring carbon of the five-membered hetero ring (e.g., phthalimidines, etc.)514/526, Acyclic514/64, Boron containing DOAI514/12, 25 or more peptide repeating units in known peptide chain structure548/453, Plural ring hetero atoms in the bicyclo ring system, or ring nitrogen is shared by the two cyclos of the bicyclo ring system514/100Polycyclo ring system having the hetero ring as one of the cyclos

Examiners

Primary: Gitomer, Ralph

Attorney, Agent or Firm

Foreign Patent References

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  • 0 931 544 EP 07/01/1999
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International Class

C12Q 137

Abstract

The present invention relates to compounds that inhibit the activity of the proteasome or the production of proteasomal proteins and promote the production of hair follicles and are thus useful in stimulating hair growth, including hair density, in subject where this is desirable.

Other References

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