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US Patent 6734186 - Compounds for the treatment of female sexual dysfunction

US Patent Issued on May 11, 2004
Estimated Patent Expiration Date: Icon_subject November 8, 2020Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.
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Abstract

A method of treating a female suffering from FSD, in particular FSAD, is described. The method comprises delivering to the female an agent that is capable of potentiating cAMP in the sexual genitalia; wherein the agent is in an amount to cause potentiation of cAMP in the sexual genitalia of the female. The agent may be admixed with a pharmaceutically acceptable carrier, diluent or excipient.

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Inventors

Assignee

Application

No. 09708392 filed on 11/08/2000

US Classes:

514/263.1, Purine (including hydrogenated)544/224, The six-membered hetero ring consists of two nitrogens and four carbons (e.g., 1,2-diazines, etc.)544/2421,3-diazines

Field of Search

514/263.1, Purine (including hydrogenated)544/262, The other cyclo in the bicyclo ring system is five-membered544/224, The six-membered hetero ring consists of two nitrogens and four carbons (e.g., 1,2-diazines, etc.)544/2421,3-diazines

Examiners

Primary: Padmanabhan, Sreeni
Assistant: Wells, Lauren Q.

Attorney, Agent or Firm

US Patent References

4666908, 5-Substituted pyrazolo[4,3-d]pyrimidine-7-ones and methods of use
Issued on: 05/19/1987
Inventor: Hamilton
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Issued on: 11/12/1996
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Issued on: 03/18/1997
Inventor: Stamler, et al.
5861396, 5981527, Cyclic GMP-specific phosphodiesterase inhibitors
Issued on: 11/09/1999
Inventor: Daugan, et al.
6043252, Carboline derivatives
Issued on: 03/28/2000
Inventor: Bombrun
6235742, 5-substituted pyrazolo[4,3-D]pyrimidin-7-ones
Issued on: 05/22/2001
Inventor: Bell, et al.
6294550, Treatment of female sexual dysfunction
Issued on: 09/25/2001
Inventor: Place, et al.
6306841, Treatment of female sexual dysfunction
Issued on: 10/23/2001
Inventor: Place, et al.
6316457Nitrosated and nitrosylated phosphodiesterase inhibitor compounds, compositions and their uses
Issued on: 11/13/2001
Inventor: Garvey, et al.

Foreign Patent References

  • 0274434 EP 07/01/1988
  • 0771799 EP 07/01/1997
  • 0911333 EP 04/01/1999
  • WO9104042 WO 04/01/1991
  • WO9720821 WO 06/01/1997
  • WO9735989 WO 10/01/1997
  • WO9739760 WO 10/01/1997
  • WO9803492 WO 01/01/1998
  • WO9920266 WO 04/01/1999
  • WO9921562 WO 05/01/1999
  • WO9922731 WO 05/01/1999
  • WO0015228 WO 03/01/2000
  • WO0015639 WO 03/01/2000

International Classes

A01N 4390
A61K 3152
C07D23700
C07D23702
C07D23900

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