Patent References 3717634 Buspirone anti-anxiety method 2-[4-[(4,4 -Dialkyl-2,6-piperidinedion-1-yl)butyl]-1-piperazinyl]pyrimidines Quinoline derivatives which are 5-hydroxytryptamine antagonists Succinimide derivatives, compositions and method of use Quinoline derivatives Quinoline derivatives which are 5-hydroxytryptamine antagonists Acetaminophen/hydroxyzine analgesic combinations Formulation of 5-HT agonist and NSAID for treatment of migraine Patent #: 5872145 InventorsAssigneeApplicationNo. 860181 filed on 05/17/2001US Classes:514/252.14, The additional hetero ring is a 1,3 diazine ring514/252.15, Spiro ring system containing514/252.16, Polycyclo ring system having the additional 1,3-diazine ring as one of the cyclos514/252.17, The polycyclo ring system is quinazoline (including hydrogenated)514/252.18, Additional six-membered hetero ring consisting of five ring carbons and one ring nitrogen attached directly or indirectly to the 1,3-diazine by nonionic bonding514/252.19, Five-membered nitrogen hetero ring attached directly or indirectly to the 1,3-diazine ring by nonionic bonding514/922SIDE EFFECT REDUCTION BY INCORPORATION OF A SECOND DESIGNATED INGREDIENTExaminersPrimary: Krass, FrederickAttorney, Agent or FirmForeign Patent References
International ClassA61K 031/497Foreign Application Priority Data1999-06-30 FRAbstractA method of treating pain with acetaminophen comprises the concurrent administration of an azapirone such as buspirone. This combination of agents surprisingly results in a strengthened analgesic response characterized by rapid onset, greater pain relief, and a longer duration of action.Other References
Field of SearchThe additional hetero ring is a 1,3 diazine ringSpiro ring system containing Polycyclo ring system having the additional 1,3-diazine ring as one of the cyclos The polycyclo ring system is quinazoline (including hydrogenated) Additional six-membered hetero ring consisting of five ring carbons and one ring nitrogen attached directly or indirectly to the 1,3-diazine by nonionic bonding Five-membered nitrogen hetero ring attached directly or indirectly to the 1,3-diazine ring by nonionic bonding SIDE EFFECT REDUCTION BY INCORPORATION OF A SECOND DESIGNATED INGREDIENT | |