Patent 6124282 Issued on September 26, 2000. Estimated Expiration Date: May 22, 2018. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.
514/227.5, 1,4-Thiazines514/284, Tetracyclo ring system having the six-membered hetero ring as one of the cyclos514/357Nitrogen attached indirectly to the six-membered hetero ring by nonionic bonding
Various compounds that can inhibit the enzyme CYP2D6 are disclosed. The compounds are useful in increasing the effectiveness and reducing the abuse potential of drugs that are metabolised by CYP2D6.
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