U.S. patents available from 1976 to present.
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Methods for prevention and treatment of attention deficit disorder

Patent 5885998 Issued on March 23, 1999. Estimated Expiration Date: Icon_subject February 12, 2018. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.

Patent References

3870794

Devices and methods for treating memory impairment
Patent #: 4680172
Issued on: 07/14/1987
Inventor: Leeson

Method for treatment of neurodegenerative diseases
Patent #: 5212188
Issued on: 05/18/1993
Inventor: Caldwell, et al.

Compounds of 1,2,5,6-tetrahydropyridin-3-carboxaldehyde oxime which are useful as cholinergic agents
Patent #: 5219872
Issued on: 06/15/1993
Inventor: Galliani, et al.

Compounds of 1,2,5,6-tetrahydropyridine which are useful as cholinergic agents
Patent #: 5219873
Issued on: 06/15/1993
Inventor: Galliani, et al.

Heterocyclic acetylenic amines having central nervous system activity Patent #: 5225567
Issued on: 07/06/1993
Inventor: Moon, et al.

Inventors

Application

No. 023040 filed on 02/12/1998

US Classes:

514/256, 1,3-diazines (e.g., pyrimidines, etc.)514/277, Hetero ring is six-membered consisting of one nitrogen and five carbon atoms514/344, Cyano bonded directly to the six-membered hetero ring514/357Nitrogen attached indirectly to the six-membered hetero ring by nonionic bonding

Examiners

Primary: Jarvis, William R. A.

Attorney, Agent or Firm

International Classes

A61K 031/505
A61K 031/44
A61K 031/435

Abstract

Patients susceptible to or suffering from attention deficit disorder are treated by administering an effective amount of an aryl subsistituted aliphatic compound, an aryl substituted olefinic amine compound or an aryl substituted acetylenic compound. Exemplary compounds are (E)-4-(5-pyrimidinyl)-3-butene-1-amine, (E)-4-›3-(5-methoxypyridin)yl!-3-butene-1-amine, (E)-N-methyl-4-(5-pyrimidinyl)-3-butene-1-amine, (E)-N-methyl-4-›3-(5-methoxypyrindin)yl!-3-butene-1-amine, (Z)-metanicotine, (E)-metanicotine, N-methyl-(3-pyridinyl)-butane-1-amine, N-methyl-4-(3-pyridinyl)-3-butyne-1-amine and (E)-N-methyl-4-›3-(6-methylpyrindin)yl!-3-butene-1-amine.

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