3-arylcarbonyl-1(C-attached-N-heteryl)-1H-indoles

Patent 5607933 Issued on March 4, 1997. Estimated Expiration Date:

March 16, 2014. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.

Abstract Claims Description Full Text

Patent References

3489770

Indole derivatives
Patent #: 3946029
Issued on: 03/23/1976
Inventor: Descamps , et al.

3-arylcarbonyl-and 3-cycloalkylcarbonyl-1-aminoalkyl-1H-indoles Patent #: 4634776
Issued on: 01/06/1987
Inventor: Bell

Inventors

Assignee

Sterling Winthrop Inc.

Application

No. 213777 filed on 03/16/1994

US Classes:

514/254.09, Indole ring system (including hydrogenated) attached directly or indirectly to the piperazine ring by nonionic bonding544/373The five-membered hetero ring is one of the cyclos in a bicyclo ring system

Examiners

Primary: Springer, David B.

Attorney, Agent or Firm

Alexander; Michael D., Dupont; Paul E., Davis; William J.

International Classes

C07D 403/06
A61K 031/495

Abstract

2--R2 --R4 -substituted-3--R3 --CO--1--[(C-attached-N-heteryl)-(Alk)n ]--1H-indoles useful as analgesic, anti-rheumatic, anti-inflammatory or anti-glaucoma agents.

Other References

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