Azacycloalkane derivatives, absorption promoters containing the derivatives as the effective ingredient and external preparations containing the absorption promoters
Patent 4882359 Issued on November 21, 1989. Estimated Expiration Date: 
November 18, 2007. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.
November 18, 2007. Estimated Expiration Date is calculated based on simple USPTO term provisions. It does not account for terminal disclaimers, term adjustments, failure to pay maintenance fees, or other factors which might affect the term of a patent.Patent References 3188317 3228955 3232952 N-(substituted-thiomethyl)-2-pyrrolidinones Vehicle composition containing 1-substituted azacyclopentan-2-ones Vehicle composition containing 1-substituted azacyclononan-2-ones Vehicle composition containing 1-substituted azacyclohexan-2-ones Vehicle composition containing 1-substituted azacycloalkan-2-ones Vehicle composition containing 1-substituted azacyclopentan-2-ones Patent #: 4444762 InventorsAssigneeApplicationNo. 131193 filed on 11/18/1987US Classes:514/2, Peptide containing (e.g., protein, peptones, fibrinogen, etc.) DOAI424/94.1, ENZYME OR COENZYME CONTAINING424/443, Web, sheet or filament bases; compositions of bandages; or dressings with incorporated medicaments514/171, With additional active ingredient514/183, Heterocyclic carbon compounds containing a hetero ring having chalcogen (i.e., O,S,Se or Te) or nitrogen as the only ring hetero atoms DOAI514/212.03, Chalcogen double bonded directly to a ring carbon of the seven-membered hetero ring which is adjacent to the ring nitrogen514/424, Chalcogen bonded directly to the five-membered hetero ring by nonionic bonding514/946, PENETRANT OR ABSORBENT (ENHANCES PENETRATION INTO SUBJECT TREATED)540/451, Chalcogen double bonded directly to a ring carbon of the hetero ring which is adjacent to the ring nitrogen (e.g., laurolactam, etc.)548/551Chalcogen attached indirectly to the five-membered hetero ring by acyclic nonionic bondingExaminersPrimary: Springer, David B.Attorney, Agent or FirmForeign Patent References
International ClassesA61K 031/40A61K 031/395 A61K 047/00 Foreign Application Priority Data1986-04-08 JPAbstractAn azacycloalkane derivative useful for promoting the absorption of a medicine, an absorption promoting agent comprising at least one of the azacycloalkane derivatives as the effective ingredient for promoting the absorption and an external preparation containing the absorption promoting agent, the derivative being represented by the following formula ##STR1## wherein A is --CH2 -- or --S-- for example, B is sulfur or oxygen, R is --SR" in which R" is an alkyl group or alkylthioalkyl group for example, or --OR" in which R" is as defined above, an alkyl group or substituted amino group, R' is a hydrogen atom, alkyl group or alkyloxy group for example, m is an integer of 0-5 and n is an integer of 1-15.Field of SearchChalcogen attached indirectly to the five-membered hetero ring by acyclic nonionic bondingChalcogen double bonded directly to a ring carbon of the hetero ring which is adjacent to the ring nitrogen (e.g., laurolactam, etc.) Topical application Chalcogen bonded directly to the five-membered hetero ring by nonionic bonding Heterocyclic carbon compounds containing a hetero ring having chalcogen (i.e., O,S,Se or Te) or nitrogen as the only ring hetero atoms DOAI |
| ||||||||||||||
