|8618327||Antibacterial agents and methods of use thereof|
The present invention relates generally to compounds providing antibacterial therapeutic agents and preparations, and related methods of using and making antibacterial compounds. Antibacterial compounds of the present invention include chalcone, alkylpyrimidine, ami...
|8461390||Method for producing substituted biphenyls|
A process for preparing substituted biphenyls of the formula I where R1=nitro or amino, R2=cyano, halogen, C1-C4-haloalkyl, C1-C4-haloalkoxy ...
|8269045||Substituted pyrazinecarboxylic acid anilide derivatives or salts thereof, intermediates of the same, pesticides for agricultural and horticultural use, and usage thereof|
Substituted pyrazinecarboxylic acid anilide derivatives represented by the general formula (I) or salts thereof; intermediates of them; pesticides (such as insecticides and acaricides) for agricultural and horticultural use, containing the compounds as the active in...
|8115032||Process for the synthesis of a propargylic alcohol|
A process for the preparation of the compound of formula ...
|8088952||Ionic bronsted acid|
A new ionic compound is provided that is derived from N,N-dimethylaniline and pentafluorophenol in amounts such that there are at least 2 equivalents of pentafluorophenol per equivalent of the N,N-dimethylaniline. ...
|7825280||Fluorine-containing polymerizable monomer and polymer compound using same|
The present invention relates to a fluorine-containing polymerizable monomer represented by the formula , [Chem. 31] wherein “a” represents an integer of 1-4. This monomer has a plurality of polymerizable amin...
|7439400||Amino alcohol ligand and its use in preparation of chiral proparglic tertiary alcohols and tertiary amines via enantioselective addition reaction|
The invention disclosed a new process of asymmetric alkynylation of ketone or ketimine, involving the chiral ligand-mediated asymmetric addition of zinc or copper acetylide to a trifluoromethyl ketone or ketimine intermediate to give a chiral tertiary proparglic alc...
|7365085||Compounds and methods|
Disclosed is a compound having the formula: pharmaceutically acceptable salts or solvates thereof and pharmaceutical compositions containing the same, wherein the structural variables are as defined...
|7227036||Production process of aminomethyl group-containing benzamide compound|
There is provided a process for producing an aminomethyl group-containing benzamide compound represented by the general formula (II): wherein —CONH2 and —X represent a substituent on the benzene ring and —CONH2 exists at the meta- or para-position of —CH2NH2...
|7176334||Process for the preparation of substituted halogenated aniline|
A process for the preparation of substituted halogenated anilines from substituted halogenated 1-chlorobenzenes which comprises a) reacting a substituted halogenated 1-chlorobenzene selectively with an imine in the presence of a transition metal catalyst complex and...
This invention relates to novel phthalamide derivatives of formula (I) wherein R1, R2, R3, R4, and R5 have the meanings given in the...
|7087778||Process for producing benzoxazine derivative and production intermediate thereof|
Processes for producing antibacterial agents and intermediates useful in producing antibacterial agents are provided and include producing compound (VI-a) in accordance with the following reaction schema, as well as production intermediates thereof
|7084138||Active ingredient combinations with insecticidal and acaricidal properties|
The invention relates to novel active compound combinations having very good insecticidal and acaricidal properties and containing (a) cyclic ketoenols having the formula in which the gro...
A selectively herbicidal composition which comprises, besides customary inert formulation auxiliaries, as active ingredient a mixture of: a) a herbicidally active amount of a herbicide selected from the group consisting of the compounds of formula (Ia), and/or (Ib),...
|7060850||Fluorous tagging and scavenging reactants and methods of synthesis and use thereof|
The present invention includes methods and compositions for increasing the fluorous nature of an organic compound by reacting it with at least one fluorous compound to produce a fluorous tagged organic compound. The increased fluorous nature of the fluorous tagged o...
|7053123||Substituted (e)-styryl benzylsulfones for treating proliferative disorders|
(E)-Styryl benzylsulfones useful as antiproliferative agents, including, for example, anticancer agents, are provided according to formula I: wherein: R1 is selected from the group consisting of halogen, C1–C6 alkoxy, nitro, phosphonato, amino, sulfamyl...
|7045660||Compounds as PDE IV and TNF-inhibitors|
This invention is directed to a [di(ether or thioether)heteroaryl or fluoro substituted aryl] compound or an N-oxide thereof or a pharmaceutically acceptable salt thereof, which is useful for inhibiting the production or physiological effects of TNF in the treatment...
The present invention relates to a process for preparing perfluoroalkylanilines and to their use for preparing active ingredients, in particular for agrochemicals. ...
|6974837||Compositions comprising sibutramine metabolites in combination with phosphodiesterase inhibitors|
Pharmaceutical compositions and dosage forms are disclosed that comprise a racemic or optically pure sibutramine metabolite and a phosphodiesterase inhibitor. ...
Described herein are compounds of formula I wherein M1, M2 and M3 have the meanings recited in the disclosure, liquid crystalline mixtures and polymers containing them, and the use of t...
|6900245||Pharmaceutical composition comprising crystalline sibutramine methanesulfonate hemihydrate|
The present invention relates to a pharmaceutical composition for treating or preventing obesity, comprising novel crystalline sibutramine methanesulfonate hemihydrate of formula (I). The crystalline sibutramine methanesulfonate hemihydrate according to the present ...
Aminomethyl-phenyl-cyclohexanone derivatives of formula I or Ia, their diastereomers, enantiomers and salts formed with a physiologically tolerated acid. Also disclosed are processes for preparing the same, pharmaceuti...
|6849766||1,4-diamino-2-alkenylbenzene derivatives, and dyes containing these compounds|
1,4-Diamino-2-alkenylbenzene derivatives of general formula (I) or physiologically tolerated water-soluble salts thereof as well as agents for oxidative dyeing of fibers, containing these compounds. ...
|6828466||Process for the synthesis of phenols from arenes|
A process to synthesize substituted phenols such as those of the general formula RR′R″Ar(OH) wherein R, R′, and R″ are each independently hydrogen or any group which does not interfere in the process for synthesizing the substituted phenol including, but not...
|6803388||(R)-Chiral halogenated substituted n,n-bis-phenyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity|
The invention relates to substituted aryl and heteroaryl (R)-Chiral Halogenated 1-Substitutedamino-(n+1)-Alkanol compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for ...
|6784318||Vinyl polymer and organic electroluminescent device|
An organic electroluminescent device has an organic layer between a pair of electrodes. The organic layer (in particular, a hole-transporting layer) has a polymer of a vinyl compound represented by the following formula (1):
|6784311||Method of producing 3-aminoalkanoic acid esters|
Process for the preparation of 3-aminoalkanoic acid esters of the general formula: in which R is C1-6-alkyl and R1 is hydrogen, C1-6-alkyl or phenyl, or their salts, by catalytic hydrogen...
|6765023||Use of substituted N, N-disubstituted reverse aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity|
The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for treating atheroscle...
|6747175||Chlorination of an aniline in a hydrofluoric medium|
The invention concerns a method for the synthesis of chlorinated aniline on the ring and comprising at least a sp3 hybridization carbon atom both perhalogenated and bearing a fluorine atom. Said method is characterized in that it comprises a step which consists in c...
|6747149||Glucamine salts for treating hepatitis virus infections|
N-Substituted glucamine compounds of formula I are effective in treatment of hepatitis infections, including hepatitis B and hepatitis C. In treating hepatitis infections the compounds of formular I may be used alone, or in combinatioin with another antiviral agent ...
|6717013||Perfluoroalkylated aniline compound and process for producing the same|
The present invention provides an aniline derivative represented by the formula (I) wherein R1 and R2 are each H, (C1-12)alkyl, (C3-8)cycloalkyl, hydroxy(C1-12)alkyl...
|6683099||Substituted N,N-disubstituted cycloalkyl aminoalcohol compounds useful for inhibiting cholesteryl ester transfer protein activity|
The invention relates to substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamine compounds useful as inhibitors of cholesteryl ester transfer protein (CETP; plasma lipid transfer protein-I) and compounds, compositions and methods for treating...
|6673794||Substituted aminomethyl-phenyl-cyclohexane derivatives|
A substituted aminomethyl-phenyl-cyclohexane derivative of formula I or Ia, ##STR1## and their a diastereomer, enantiomer, or of a salt formed with a physiologically tolerated acid. Also disclosed are method for preparing the substituted aminomethyl-pheny...
|6600074||Perfluoroalkylated aniline compound and process for producing the same|
The present invention provides an aniline derivative represented by the formula (I) ##STR1## wherein R1 and R2 are each H, (C1-12)alkyl, (C3-8)cycloalkyl, hydroxy(C1-12)alkyl, hydroxycarbonyl (C
|6559341||Phthalic acid diamide derivatives, fluorine-containing aniline compounds as starting material, agricultural and horticultural insecticides, and a method for application of the insecticides|
The present invention provides a phthalic acid diamide derivative represented by the general formula (I) ##STR1## (wherein R1, R2 and R3 are each H, C3 -C6 cycloalkyl group, group of the formula --A
|6555959||Material for light emitting device, light emitting device using thereof, and amine compound|
A material for a light emitting device which is a compound represented by the following formula (I): ##STR1## wherein Ar1 and Ar6, which are the same or different, each represents a divalent aryl group or a divalent heterocyclic grou...
A compound comprises a blocked halogenated hydroxydiphenyl ether of the formula: ##STR1## where X1 is a halogen, X2 is chlorine or bromine, X3 is hydrogen, chlorine or bromine, X4 is chlorine, bromine, alkyl hav...
|6552161||Polarizable amines and polymides for optical alignment of liquid crystals|
The present invention relates to amine compositions and the preparation of polyimides. The polyimides can be used for inducing alignment of a liquid crystal medium with polarized light in liquid crystal display elements....
|6521793||Catalyst ligands, catalytic metal complexes and processes using same|
New ligands having a backbone comprised of NCCX can be combined with a metal or metal precursor compound or formed into a metal-ligand complex to catalyze a number of different chemical transformations, including polymerization....
|6521794||Method for production of aromatic compounds|
For the production of an aromatic compound by hydrolyzing and decarboxylating a corresponding aromatic cyano compound in the presence of an acidic substance, this invention provides a method for the production of the aromaic compound, characterized by car...