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| Number | Title | Issue Date |
| 7632972 | Compounds and methods for treatment of cancer and modulation of programmed cell death for melanoma and other cancer cells Compounds and related methods for synthesis, and the use of compounds and combination therapies for the treatment of cancer and modulation of apoptosis in cells are disclosed. The generation of synthetic combinatorial libraries and the evaluation of library member c... | 12/15/2009 |
| 7435849 | Process for the production of acid chlorides A process for the preparation of acid halides of formula I which are useful as intermediates in the preparation of i.a. pharmaceutically active compounds. ... | 10/14/2008 |
| 7038085 | Stereoisomers of p-hydroxy-milnacipran, and methods of use thereof The present invention relates generally to the enantiomers of para-hydroxy-milnacipran or congeners thereof. Biological assays revealed that racemic para-hydroxy-milnacipran is approximately equipotent in inhibiting serotonin and norepinephrine uptake (IC50 | 05/02/2006 |
| 7015349 | Reduction of hair growth Compositions including a conjugate of α-difluoromethylornithine can be applied topically to reduce hair growth. ... | 03/21/2006 |
| 6992220 | Process and intermediates for the preparation of 3-(amino)-3-cyclobutylmethyl-2-hydroxy-propionamide or salts thereof In one embodiment, the present application relates to a process of making a compound of formula I: and to certain intermediate compounds that are made within the process of making the compound of formula I. ... | 01/31/2006 |
| 6960687 | Derivatives and pharmaceutical compositions of n-hydroxyalkyl tetramethylcyclopropane-carboxamide, having anti-epiletic, neurological, and CNS activity, and method for their preparation New derivatives of N-Hydroxyalkyl-tetramethylcyclopropane carboxamide, pharmaceutical compositions thereof, methods for their preparation, and use thereof for the treatment of epilepsy, neurological, affective and psychotic disorders and for the treatment of pain an... | 11/01/2005 |
| 6703379 | Benzene derivatives and pharmaceutical use thereof The present invention provides an AP-1 activation inhibitor, NF-kappa B activation inhibitor, inflammatory cytokine production inhibitor, matrix metalloprotease production inhibitor, inflammatory cell adhesion molecule expression inhibitor, anti-inflammat... | 03/09/2004 |
| 6683212 | Fungicidally active carboxylic acid amides ##STR1## Compounds of Formula (I) are disclosed which are useful as fungicides wherein R1 is hydrogen; halogen; C1 -C2 alkoxy; C1 -C2 haloalkoxy, cyano; or C1 -C2 alkyl optionally ... | 01/27/2004 |
| 6596898 | Process for preparing halogenated cyclopropane derivatives A process for preparing compounds represented by the following general formula (I) wherein X represents chlorine atom, bromine atom, or iodine atom, and R includes alkoxy group and amino group which comprises the step of allowing a compound represented by... | 07/22/2003 |
| 6576792 | 2-halo-1-cycloalkenecarboxamides and their preparation The invention relates to a 2-halo-1-cycloalkenecarboxamides represented by Formula I: ##STR1## wherein n is 1 or 2; R is hydrogen or an alkyl group; and X is a halogen.... | 06/10/2003 |
| 6552217 | Process for the preparation of alkyl 1-methylcyclopropanecarboxylate Disclosed is a 4-step process for the preparation of alkyl esters of 1-methylcyclopropanecarboxylic acid which comprises the steps of (1) converting γ-butyrolactone to -methyl-γ-butyrolactone; (2) converting the -methyl-γ-butyrolactone fr... | 04/22/2003 |
| 6441044 | Cycloalkyl carboxylic acid amides, their production and their use as fungicides in agriculture The present invention relates to cycloalkylcarboxamides of formula I ##STR1## where: A is optionally substituted C3 -C6 -cycloalkyl; Alk is straight-chain or branched C1 -C6 -alkylene; R1 is optionally substitu... | 08/27/2002 |
| 6426365 | CETP activity inhibitors The present invention provides a CETP activity inhibitor comprising as an active ingredient a compound represented by the formula (I): ##STR1## wherein R represents a straight chain or branched alkyl group; a straight chain or branched alkenyl group; a lo... | 07/30/2002 |
| 6423748 | Amido polybiguanides and the use thereof as antimicrobial agents Amido polybiguanides and their use as antimicrobial agents in pharmaceutical compositions are disclosed. A method of synthesis of amido polybiguanides is also disclosed. The amido polybiguanides are useful in the preservation of pharmaceutical composition... | 07/23/2002 |
| 6362183 | Aromatic sulfonyl alpha-hydroxy hydroxamic acid compounds An aromatic sulfonyl alpha-hydroxy hydroxamic acid compound that, inter alia, inhibits matrix metalloprotease activity is disclosed, as is a treatment process that comprises administering a contemplated aromatic sulfonyl alpha-hydroxy hydroxamic acid comp... | 03/26/2002 |
| 6316669 | Bis-amido polybiguanides and the use thereof to disinfect contact lenses and preserve pharmaceutical compositions Bis-amido polybiguanides and their use as antimicrobial agents in pharmaceutical compositions are disclosed. A method of synthesis of bis-amido polybiguanides is also disclosed. The bis-amido polybiguanides are useful in the preservation of pharmaceutical... | 11/13/2001 |
| 6251947 | Fungicidal carboxamides ##STR1## Compounds of Formula (I) are disclosed which are useful as fungicides, wherein Q is: (Q-1) or (Q-2), Z is (Z-1); (Z-2); (Z-3) or (Z-4); X is --O--, --CH(R11)-- or .dbd.C(R11)--; R1 is H or C1 -C | 06/26/2001 |
| 6242609 | Method for manufacturing a color coupler used in a silver halide photographic light-sensitive material A method for manufacturing a color coupler used in a silver halide photographic light-sensitive material using an ammonium trihalide. Said method for manufacturing the color coupler comprising the following step: a step for halogenating a coupling position of ... | 06/05/2001 |
| 6172262 | Amphiphilic agents for membrane protein solubilization Disclosed are amphiphilic compounds comprising Formula I: ##STR1## wherein R1, R2, and R3 are C2 -C12 straight or branched alkyl; unsubstituted phenyl, biphenyl, C3 -C8 cycloalky... | 01/09/2001 |
| 6143789 | Naphthalene compounds Compound of formula (I): ##STR1## wherein: T represents alkylene, A and B together form a naphthalene, dihydronaphthalene, or tetrahydronaphthalene group, R represents hydrogen, hydroxy, R' or OR', R' being as defined in the description, G1 | 11/07/2000 |
| 6136887 | Vinylcyclopropane-(meth)acrylates and their use The invention relates to vinylcyclopropane derivatives according to the formula ##STR1## in which A is --[--Y--CO--C(.dbd.CH2)R4 ]m or --C(.dbd.CH2)CO--O--C1-4 -alkyl, U and X, independently of e... | 10/24/2000 |
| 6028112 | Spirocyclopropyl fluorenes as melatonergic agents There is provided novel spirocyclopropyl fluorene derivatives having the general Formula I ##STR1## wherein R, R1 and X are as defined herein which are useful as melatonergic agents.... | 02/22/2000 |
| 5939554 | Diarylaminopropanediol and diarylmethyl-oxazolidinone compounds A method for preparing a diarylalanine compound is provided. The method includes reacting a diarylaminopropanediol with a reducing agent to form a diarylaminopropanol compound and/or contacting a serine ester derivative with an aryl metal reagent to form ... | 08/17/1999 |
| 5925674 | Cycloalkylcarboxanilides This invention relates to cycloalkylcarboxanilides of the formula ##STR1## which are used to combat pests.... | 07/20/1999 |
| 5922771 | Benzocycloalkene compounds, their production and use A compound of the formula ##STR1## wherein R1 and R2 independently represent H or an optionally substituted hydrocarbon group; R3 represents an optionally substituted hydrocarbon group; R4 represents H or a... | 07/13/1999 |
| 5889031 | N-acyl-2-aryl cyclopropylmethylamine derivatives as melatonergics Certain N-acyl 2-aryl cyclopropylmethylamine derivatives are useful as melatonergic agents.... | 03/30/1999 |
| 5886223 | Process for the preparation of substituted ଲ-ketoanilide compounds There is provided a process for the preparation of substituted ଲ-ketoanilide compounds having the structural formula I ##STR1## The substituted ଲ-ketoanilide compounds are useful for the control of insect pests.... | 03/23/1999 |
| 5880157 | Derivatives of tetramethylcyclopropane The present invention relates to derivatives of 2,2,3,3-tetramethylcyclopropane carboxylic acid (TMCA) of general formula (I), ##STR1## wherein R is lower alkyl group (C1 -C6), an aryl group, an aralkyl group or an amide of... | 03/09/1999 |
| 5808134 | Cyclopropane derivatives and method of preparing the same An intermediate for the production of (3-oxo-2-oxobicyclo3,1,0!hexan-1-yl) methanol represented by formula (II): ##STR1## selected from the group of compounds (9)-(11) as shown below, wherein R1 represents a lower alkyl group, R3 | 09/15/1998 |
| 5808151 | Biphenylamido derivatives as melatonergic agents There is provided novel biphenylamido derivatives of the formula ##STR1## wherein Z is ##STR2## and Y is H or Z is H and Y is ##STR3## n is 0 or 1; R is C1-6 alkyl; R1 is C1-3 alkyl, C3-6 cycloal... | 09/15/1998 |
| 5780512 | Alkylated (hetero) cyclic compounds The invention relates to a compounds selected from these of formula (I): ##STR1## in which: R1, R2, R3 and A are as defined in the description, and a medicinal product containing the same useful for treating a melaton... | 07/14/1998 |
| 5760087 | Glycylanilide derivatives, their preparation and their application in therapy The invention relates to new derivatives of glycylanilides having general formula (I), wherein, particularly, R1, R3, R4, R8, R9 represent CH3 ; R2, R5, R6, R | 06/02/1998 |
| 5753652 | Antiretroviral hydrazine derivatives The invention relates to compounds of formula ##STR1## and salts, pharmaceutical compositions, intermediates and processes of preparation thereof.... | 05/19/1998 |
| 5753709 | N-acyl-2 aryl cyclopropylmethylamine derivatives as melatonergics Certain N-acyl 2-aryl cyclopropylmethylamine derivatives are useful as melatonergic agents.... | 05/19/1998 |
| 5739399 | Process for the preparation of cyclopropanecarboxylic acid amides Cyclopropanecarboxylic acid amides ##STR1## wherein R represents hydrogen, straight-chain or branched C1 -C4 -Alkyl, optionally substituted aryl or optionally substituted aralkyl, can be prepared directly from the corresponding cyclo... | 04/14/1998 |
| 5736578 | Ethylamido fluorenes and improved method of making same Novel substituted fluorene compunds of Formula I are active as melatonergic agents: ##STR1## wherein: X=H, halogen, OH or OZ; Z=C1-6 alkyl; --(CH2)m --CF3 (m=0-2); CD3 ; or ##STR2## n=1 or 2... | 04/07/1998 |
| 5710331 | Preparation of N-alkenyl carboxamides Preparation of N-alkenyl carboxamides of the general formula I ##STR1## in which the radicals R1 to R4 independently stand for hydrogen or for aliphatic, cycloaliphatic, or aromatic radicals, which optionally carry inert substit... | 01/20/1998 |
| 5693630 | Phenylethyl and phenylpropylamines Compounds of the general formula ##STR1## or pharmaceutically acceptable salts thereof, wherein Z is a saturated or unsaturated 3 to 6 carbon chain, m is 2 or 3, R1 is a hydrogen atom, or a straight or branched C1-4 alkyl group,... | 12/02/1997 |
| 5684198 | Method of preparing therapeutic amides Amides having formula I: ##STR1## wherein E, X, R2 and R3 have the meanings given in the specification, and pharmaceutically acceptable salts and pharmaceutically acceptable in vivo hydrolysable esters thereof, which are useful ... | 11/04/1997 |
| 5663418 | Processes for the preparation of cyclopropanecarboxylic acid and derivatives thereof Disclosed is a process for the preparation of cyclopropanecarboxylic acid by the non-catalytic, oxidation of cyclopropanecarboxaldehyde using molecular oxygen as the oxidant. Also disclosed are processes for the preparation of amides, esters and acid chlo... | 09/02/1997 |
