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Patent No. 5996127

Wearable Device For Feeding and Observing Birds and Other Flying Animals

A device for feeding and observing flying animals comprising a hat, a support mounted on the hat and extending outward from the hat, and a feeder mounted on the support.

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Class 562/458 - Carboxyl, or salt thereof, bonded directly to a ring


Subclass of Class 562 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the acid contains a carboxyl group bonded
No. of patents: 104
Last issue date: 05/24/2011


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NumberTitleIssue Date
79478511,1′-(1,2-ethynediyl)bis-benzene derivatives as PTP 1-B inhibitors
The present invention is related to carboxylic acids of Formula (I) and use thereof for the treatment and/or prevention of obesity and/or metabolic disorders mediated by insulin resistance or hyperglycemia, comprising diabetes type I and/or II, inadequate glucose to...
05/24/2011
7408078Anthranilic acid derivatives useful in treating infection with hepatitis C virus
The present invention provides pharmaceutical compositions useful in treating hepatitis C infection. The present invention also provides methods of treating hepatitis C infection by administering to a mammal the pharmaceutical compositions of the present invention.
08/05/2008
74080762-Bromoanaline and 2-chloroaniline compounds
Disclosed are 2-bromoaniline or 2-chloroaniline compounds of formula (I): wherein R, R1 and X are as defined. The compounds are useful as intermediates for preparing indole compounds. ...
08/05/2008
7371896Tetrafluorobenzyl derivatives and pharmaceutical composition for preventing and treating acute and chronic neurodegenerative diseases in central nervous system containing the same
The present invention relates to a tetrafluorobenzyl derivative and a pharmaceutical composition for prevention and treatment of acute and chronic neurodegenerative disease in central nervous system and ophthalmic diseases containing the same. The tetrafluorobenzyl ...
05/13/2008
7279597Phenyl amine carboxylic acid compounds and compositions for delivering active agents
Phenyl amine carboxylic acid compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well. ...
10/09/2007
72682483-Cyano-2,4,5-trifluorobenoxyl fluoride and intermediate products for the production thereof
The present invention relates to 3-cyano-2,4,5-trifluorobenzoyl fluoride and to intermediates for its preparation and to the process for the preparation of 3-cyano-2,4,5-trifluoro-benzoyl fluoride, which starts from 5-fluoro-1,3-xylene (VIII); which is bichlorinated...
09/11/2007
RE39682Farnesyl derivatives and pharmaceutical compositions containing them
Novel farnesyl derivatives which are inhibitors of the prenylated protein methyltransferase enzyme, and useful as anti-cancer drugs, have the following formula: wherein R1represents f...
06/05/2007
6936597Prodrugs of anticancer agents employing substituted aromatic acids
Polymeric prodrugs of the formula: wherein B is selected from the group consisting of OH, leaving groups, residues of amine-containing moieties and a residues of hydroxyl-containing m...
08/30/2005
6747170Thermosensitive recording material and color developer compound therefor
A thermosensitive recording material has a support and a thermosensitive coloring layer formed thereon containing a leuco dye and a color developer capable of inducing color formation in the leuco dye upon application of heat thereto, with the color developer includ...
06/08/2004
6727098Biaryl-type compounds, CD color fixing agent and method for determination of absolute configuration
A novel achiral biaryl-type compound and a circular dichroism (CD) color fixing agent are provided. Furthermore, a method for determining an absolute configuration of a chiral compound is carried out by introducing the above achiral biaryl-type compound into the chi...
04/27/2004
6710205Benzoic acid derivatives, processes for producing the same and drugs containing the same as the active ingredient
An agent comprising the benzoic acid of formula (I) wherein A, B, R6, R7 are carbocyclic ring, heterocyclic ring, etc.; R1 is hydroxy etc.; R2, R3, R4 are...
03/23/2004
6699909Aminoindanes
The present invention relates to therapeutically active novel aminoindanes of formula (I). Also provided is a method of preparing compounds of formula (I), and pharmaceutical compositions comprising the compounds. The novel compounds act as modulators of ...
03/02/2004
6603041Bicyclic enamide derivatives
Enamide derivatives of formula (1) are described: ##STR1## wherein R1 is a group Ar1 L2 Ar2 Alk- in which Ar1 is an optionally substituted aromatic or heteroaromatic group, L2 is a covalent...
08/05/2003
6504052Excitatory amino acid receptor modulators
Compounds of the formula (I) in which R1 is C1-10 allyl; C2-10 alkenyl; C2-10 alkynyl; phenyl-C2-10 alkyl or phenyl-C2-10 alkenyl; and salts and esters thereof, modulate metabotropic glutam...
01/07/2003
6172239Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin receptors, their preparation and pharamaceutical compositions containing them
The invention relates to compounds of the formula ##STR1## The compounds have agreat affinity for the neurotensin receptors....
01/09/2001
6172058Compounds with pharmaceutical properties
A pharmaceutical compound of the formula ##STR1## in which R1 is C1-10 alkyl, C2-10 alkenyl, C2-10 alkynyl, C3-10 cycloalkyl, C3-10 cycloalkyl-C1-10 alkyl, C3-10 cyclo...
01/09/2001
6150412Catechol derivatives
The invention relates to compounds of formula (I) ##STR1## wherein R1 is an electronegative substituent, preferably nitro, cyano, formyl or carboxy, R2 is --A--R4, wherein A is a branched or straight chain C1-9
11/21/2000
6127392Anthranilic acid analogs
Compounds of the formula: wherein: R1, R2, R3, R4,R5, R6, R7 and R8 are, independently, hydrogen, COOR15, halogen, nitro, cyano, C1-10 alkoxy, C1...
10/03/2000
6114386Inhibitors of bacterial sialidase
A sialidase inhibitor of the shown formula I: ##STR1## where dashed lines d1 and d2, X1, R1, R2, R6, R3, R4 and R5 are as described in the specificatio...
09/05/2000
5965592Acyl compounds
Compounds of the formula ##STR1## and their salts, in which R1, is a C1 -C7 aliphatic hydrocarbon radical; X1 is --CO; X2 is a divalent aliphatic hydrocarbon radical which comprises an ethyl grou...
10/12/1999
5935585Biaromatic amido compounds and pharmaceutical/cosmetic compositions comprised thereof
Novel pharmaceutically/cosmetically-active biaromatic amido compounds have the structural formula (I): ##STR1## in which Ar is a radical selected from among those of the following formulae (a)-(e): ##STR2## and are useful for the treatment ...
08/10/1999
5936119Chemical process
The invention provides a process for the preparation of 3-(N,N-dimethylamino)benzoic acid which comprises subjecting an aqueous solution of an alkali metal salt or ammonium salt of 3-aminobenzoic acid to reductive methylation in the presence of a supporte...
08/10/1999
5872282Allosteric modifiers of hemoglobin
A family of compounds has been found to be useful for right-shifting hemoglobin towards a low oxygen affinity state. The compounds are capable of acting on hemoglobin in whole blood. In addition, the compounds can maintain the oxygen affinity in blood dur...
02/16/1999
5744638Process for the preparation of haloanthranilic acids
The present invention relates to a process for the preparation of compounds of the general formula I ##STR1## in which X and Y, independently of each other, represent hydrogen, fluorine, chlorine or bromine, but cannot simultaneously represent h...
04/28/1998
5741926Aniline derivatives having antihyperglycemic activity
Aniline derivatives useful as antihyperglycemic agents, pharmaceutical compositions comprising the aniline derivatives and methods for their use are described. The aniline derivatives are useful for the treatment of insulin-dependent diabetes mellitus (ID...
04/21/1998
5717109Excitatory amino acid receptor antagonists
The present invention provides compounds of formula ##STR1## in which R represents an organic group, or a pharmaceutically acceptable metabolically labile ester or amide thereof, or a pharmaceutically acceptable salt thereof, which are useful as anta...
02/10/1998
5705528Farnesyl derivatives and pharmaceutical compositions containing them
Novel farnesyl derivatives which are inhibitors of the prenylated protein thyltransferase enzyme, and useful as anti-cancer drugs, have the following formula: ##STR1## wherein R1 represents farnesyl, geranyl or geranyl-geranyl; Z represent...
01/06/1998
5599814Pyridazinedione compounds useful in treating neurological disorders
The present invention relates to pyridazino[4,5-b]quinolines, and pharmaceutically useful salts thereof, which are excitatory amino acid antagonists and which are useful when such antagonism is desired such as in the treatment of neurological disorders. T...
02/04/1997
5543550Process for the preparation of 5-fluoroanthranilic alkyl esters and/or 5-fluoroanthranilic acid
The present invention relates to a process for the preparation of 5-fluoroanthranilic alkyl esters and/or 5-fluoroanthranilic acid, which comprises dissolving a 3-fluorobenzoic alkyl ester in sulfuric acid and reacting the solution with a nitrating acid a...
08/06/1996
5536878Method for preparing aromatic secondary amino compound
Disclosed are (1) a method for preparing an aromatic secondary amino compound which comprises reacting an N-cyclohexylideneamino compound in the presence of a hydrogen moving catalyst and a hydrogen acceptor by the use of a sulfur-free polar solvent and/o...
07/16/1996
5523472Process for the preparation of 5-fluoroanthranilic acid
The present invention relates to a process for the preparation of 5-fluoroanthranilic acid, which comprises reacting 5-fluoro-2-bromotoluene in the presence of a catalyst and of an acidic solvent, with oxygen or an oxygen-containing gas at from 80° to 22...
06/04/1996
5482942(3,4-dioxocyclobuten-1-yl)chromene, indene, and dihydronaphthalenone derivatives as smooth muscle relaxants
This invention relates to novel 4-(3,4-dioxocyclobuten-1-yl)chromenes and dihydronaphthalenones and 3-(3,4-dioxocyclobuten-1-yl)indenes and salts thereof having smooth muscle relaxing activity, to their use in the treatment of hypertension as well as for ...
01/09/1996
5436368Intermediates in the preparation of 4,5-difluoroanthranillic acid
Compounds of the formula ##STR1## which are intermediates in the preparation of 4,5-difluoroanthranilic acid, an intermediate itself in the synthesis of quinolone antibacterials, and methods of preparing these intermediates....
07/25/1995
5410082Process for preparing amines
Process for preparing amines by reacting amides in aqueous-alkaline solutions and/or suspensions with halogens or hypohalites in the presence of alcohols, and converting the reaction products into the amines by hydrolysis, hydrogenation or reductive metho...
04/25/1995
5403853Substituted N-aryl-1,2-diaminocyclobutene-3,4-diones
The compounds of the formula: ##STR1## wherein R1 and R2 are, independently, hydrogen, straight or branched chain alkyl or mono- or bi-cyclic alkyl; A is a substituted phenyl group containing one or two substituents selected fro...
04/04/1995
5393902Process for the preparation of bis(amidocarboxylic acids)
A process is reported for the preparation of bis(amidocarboxylic acid) involving reacting an ester with an aminocarboxylate compound, the latter being formed from lactams or aminocarboxylic acids and salts thereof. The ester and aminocarboxylate compound ...
02/28/1995
5387594Di(aromatic) compounds and their use in human and veterinary medicine and in cosmetics
Di(aromatic) compounds corresponding to the following formula: ##STR1## in which: Ar represents either ##STR2## n=1 or 2 or: ##STR3## X represents a divalent radical, Z represents O, S or a divalent radical, and R1, R2...
02/07/1995
5359120Improvements relating to the production of prodrugs
The invention provides compounds of the formula XX: M-Ar-CONH-R, where Ar represents an aromatic ring system, R-NH is the residue of an ଱-amino acid R-NH2 or oligopeptide R-NH2 and contains at least one carboxylic acid group in...
10/25/1994
5344959Tetrahydronaphthyl and cyclopropyl substituted 1,3-butadienes having retinoid-like activity
Compounds of the formula ##STR1## wherein m is 1-4; R1 -R4 independently are hydrogen, lower alkyl of 1 to 6 carbons, Cl, Br, or I; R5 is hydrogen, lower alkyl of 1 to 6 carbons, Cl, Br, I, lower alkoxy or lower thioa...
09/06/1994
5310682Fluorogenic reagents for detection of glycoconjugates, ଱-ketoacids and diketones
Compounds containing ଱-discarbonyl groups are rendered capable of fluorescent emission by conjugation with carboxylic acid-terminated ortho-diaminoaryl reagents. The carboxylic acid groups serve as ionizable moieties which facilitate the conjugation...
05/10/1994
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