Class 560/251 - Plural nitrogens in alcohol moiety

Subclass of Class 560 - Organic compounds -- part of the class 532-570 series
No. of patents: 210
Last issue date: 01/22/2008

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Number	Title	Issue Date
7320998	Carbohydrate analog inhibitors of alpha-amylase The present invention provides carbohydrate analogs of the formula: wherein X is CH2, O, or NH, and R1-8 are independently H, a short hydrocarbon, a substituted amine, an alcohol, a substitu...	01/22/2008
7253210	Methylene-bridged selective androgen receptor modulators and methods of use thereof This invention provides a class of androgen receptor targeting agents (ARTA). The agents define a new subclass of compounds, which are selective androgen receptor modulators (SARM). Several of the SARM compounds have been found to have an unexpected androgenic and a...	08/07/2007
7220781	Meta-benzamidine derivatives as serine protease inhibitors Compounds of formula I in which R1, R2, R3, each X, L, Y, Cy, Lp, D and n have the meanings as set out in the specification, and corresponding compounds in which the unsubstituted...	05/22/2007
7163918	Iodothyronine compositions The present invention relates to compositions comprising thyroxine (T4) and triiodothyronine (T3). More specifically, the invention relates to thyroxine (T4) and triiodothyronine (T3) compositions that include a peptide carrier and thyroxine (T4) and triiodothyronin...	01/16/2007
7060708	Active agent delivery systems and methods for protecting and administering active agents The present invention relates to active agent delivery systems and more specifically to compositions that comprise amino acids, as single amino acids or peptides, covalently attached to active agents and methods for administering conjugated active agent compositions...	06/13/2006
7034015	Aminobenzoephenones The invention relates to a novel class of aminobenzophenones derivatives, to pharmaceutical preparations comprising said compounds, to dosage units of such preparations, to methods of treating patients comprising administering said compounds, and to the use of said ...	04/25/2006
6852738	Acyl sulfamides for treatment of obesity, diabetes and lipid disorders A class of acyl sulfamides comprises compounds that are potent ligands for PPAR gamma and generally have antagonist or partial agonist activity. The compounds may be useful in the treatment, control or prevention of obesity, non-insulin dependent diabetes mellitus (...	02/08/2005
6849626	Aza-amino acid derivatives (factor Xa inhibitors 15) The invention relates to semicarbazides of the general formula I where R1, R2, R3, R4 and I have the meaning indicated in claim 1. The compounds of the formul...	02/01/2005
6767922	IL-8 receptor antagonists This invention relates to novel compounds of Formula (I) to (VII), and compositions thereof, useful in the treatment of disease states mediated by the chemokine, Interleukin-8 (IL-8). ...	07/27/2004
6740682	Meta-benzamidine derivatives as serine protease inhibitors The novel compound 3-amidinobenzoyl-D-phenylglycine-3-phenylanilide is useful as a serine protease inhibitor. ...	05/25/2004
6703379	Benzene derivatives and pharmaceutical use thereof The present invention provides an AP-1 activation inhibitor, NF-kappa B activation inhibitor, inflammatory cytokine production inhibitor, matrix metalloprotease production inhibitor, inflammatory cell adhesion molecule expression inhibitor, anti-inflammat...	03/09/2004
6534542	(2-hydroxy)ethyl-thioureas useful as modulators of 򳄫 adrenergic receptors Compounds of formula (i) and of formula (ii) ##STR1## wherein the symbols have the meaning disclosed in the specification, specifically or selectively modulate 򳄫 and/or 򳄬 adrenergic receptors in preference over ³...	03/18/2003
6444702	Aminoadamantane derivatives as therapeutic agents The present invention provides novel aminoadamantane derivatives, methods of making the derivatives, compositions including the novel aminoadamantane derivatives, and methods for the treatment and prevention of neurological diseases using the derivatives ...	09/03/2002
6323227	Substituted N-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides This invention relates to compounds of formula ##STR1## which inhibit Factor Xa, to pharmaceutical compositions containing the compounds, and to the use of the compounds for the treatment of patients suffering from conditions which can be ameliorated by t...	11/27/2001
6225334	Glyoxylic acid derivatives The invention concerns novel glyoxylic acid derivatives, a process for their preparation and their use as pesticides....	05/01/2001
6218536	1,2-bis-adducts of stable nitroxides with substituted ethylenes and stabilized compositions 1,2-Bis-adducts of stable hindered nitroxide compounds with substituted ethylenes are prepared by reacting two equivalents of nitroxyl compound with an ethylenically unsaturated compound such as styrene or an acrylate ester. These adducts are very effecti...	04/17/2001
6187955	Guanidine derivatives and process for their production A guanidine derivative represented by formula (1), (2), (3) or its acid addition salt and a production process thereof ##STR1## wherein each of A and B is a C2 -C8 alkylene, D is a single bond, --CO-- or a C1 -C6	02/13/2001
6143790	L-N⁶ -(1-iminoethyl)lysine derivatives useful as nitric oxide synthase inhibitors There is disclosed a novel amino glycol derivatives of L-N6 -(1-iminoethyl)lysine, pharmaceutical compositions containing these novel compounds, and to their use in therapy, in particular their use as nitric oxide synthase inhibitors....	11/07/2000
6140361	Use of 2-deoxystreptamine as a molecular scaffold for the preparation of functionally and spatially diverse molecules and pharmaceutical compositions thereof 2-Deoxystreptamine is an aminocyclitol whose structural stability and abundant functionality make it an attractive scaffold for the combinatorial generation of small molecules. The ability to selectively functionalize the various positions of 2-deoxystrep...	10/31/2000
6124270	Use of a cationic amphipathic compound as a transfection agent, vaccine additive or drug A cationic amphipathic compound of formula (I), ##STR1## wherein A is a single bond, an NH--R' grouping or (a), wherein --R'-- is a straight or branched, optionally substituted, saturated or unsaturated C1-22 aliphatic chain optionally int...	09/26/2000
6080767	Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides The compounds according to the invention are substituted N-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides of formula I herein which exhibit useful pharmacological activity and accordingly are incorporated into pharmaceutical compositions and used ...	06/27/2000
6077970	Carboxylic acid esters of 2-hydroxy-5-isoalkyl-beta-methylstyrene The present invention relates to carboxylic acid esters of 2-hydroxy-5-isoalkyl-beta-methylstyrenes wherein the said isoalkyl substituent comprises 8-18 carbon atoms....	06/20/2000
6054457	Benzamide derivatives and their use as vasopressin antagonists This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkoxy, etc., R2 is lower...	04/25/2000
6011063	Ortho-substituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic, and medicament comprising them Ortho-substituted benzoylguanidines of the formula I ##STR1## in which R(1) to R(5) have the meanings given in the claims, are suitable as antiarrhythmic pharmaceuticals having a cardioprotective component for infarct prophylaxis and for infarct trea...	01/04/2000
5837873	Intermediates of retroviral protease inhibiting compounds A retroviral protease inhibiting compound of the formula A--X--B is disclosed. Also disclosed are a composition and method for inhibiting a retroviral protease and for treating an HIV infection. Also disclosed are processes and intermediates useful for th...	11/17/1998
5798383	Aryloxycycloalkenyl and aryloxyiminocycloalkenylhydroxyureas The prevent invention provides a compound of formula (I): ##STR1## wherein Ar is (a) phenyl, naphthyl and biphenyl, each optionally substituted with C1-4 alkyl, C1-4 haloalkyl, C1-4 hydroxyalkyl, C1-4 alkox...	08/25/1998
5723655	Amine compound and detergent composition containing the same The present invention relates to an amine compound represented by the following general formula (1): ##STR1## wherein R1 and R2 represent individually a linear or branched C1 -C24 alkyl or alkenyl group whi...	03/03/1998
5705681	Diquaternary compounds useful as bleach activators Diquaternary ammonium esters useful as bleach activators are disclosed as are bleach compositions comprising such an ester and peroxygen compound yield peroxide in solution....	01/06/1998
5698740	Hole-transport material A hole-transport material having excellent hole-transport capability and durability, suitable for use in an organic EL device and as an organic photoconductive material, has the formula (1)....	12/16/1997
5662827	Diquaternary compounds useful as bleach activators, and compositions containing them Disclosed are bleaching compositions comprising diquaternary ammonium esters which are useful as bleach activators with a peroxygen compound to yield peroxide in solution....	09/02/1997
5635571	Polymerizable macromonomers and polymers prepared therefrom Polyoxazolines having the structural formula: ##STR1## wherein R is phenylene or alkylene containing 2 to 18 carbon atoms, R2 is C1-4 alkyl and R1 is selected from the group consisting of C1-12 alkyl, vinyl...	06/03/1997
5631401	Inhibitors of protein farnesyltransferase and squalene synthase The present invention provides a compound of the formula ##STR1## or a pharmaceutically acceptable salt thereof, which are useful in inhibiting protein farnesyltransferase and the farnesylation of the oncogene protein Ras or inhibiting de novo squale...	05/20/1997
5606092	Monoazo compounds and method for dyeing or printing fiber materials using the same A monoazo compound of the following formula, ##STR1## wherein D is phenylene or naphthylene; X is halogeno, pyridinio or ##STR2## B is --OR3, --SR4, ##STR3## in which R3, R4, R5 and R	02/25/1997
5514642	Cyclohexenone oxime ethers, their preparation and their use Cyclohexenone oxime ethers of the formula I ##STR1##...	05/07/1996
5457108	5-oxo-dibenzo[a,d]cyclohepta-1,4-dienes The invention relates to substituted 5-oxo-di-benzo[a,d]cyclohepta-1,4-dienes of the formula (I) ##STR1## processes for their preparation and their use as retroviral agents....	10/10/1995
5446067	Oxime ethers and fungicides containing them Oxime ethers of the formula ##STR1## wherein m, G, R, R1, X, Y, and Z are as defined herein and fungicides containing these compounds....	08/29/1995
5440060	Surface-active compounds based on alkoxylated fatty amines The demands on the properties of pigments, in particular in the areas of emulsion paints and printing inks, which are continuously becoming more specific made it necessary to develop selective and environmentally safe dispersing and emulsifying agents and...	08/08/1995
5405997	Antiarrhythmic methanesulfonamides Methanesulfonamides are structurally depicted by Formula I' ##STR1## or its pharmacologically acceptable salts where R3 is a C1-7 alkyl substituted with C3-7 cycloalkyl, or a C1-10 alkyl substituted with on...	04/11/1995
5403850	Derivatives of P-substituted phenyl ester of pivalic acid A derivative of general formula: ##STR1## wherein Y is --SO2 --or ##STR2## (i) R1 and R2, which may the same or different, each represent, (1) --H, (2) C1-16 alkyl or (3) the formula ##STR3## wherein X ...	04/04/1995
5399746	Diquaternary bleach activators and compositions containing them Diquaternary ammonium esters useful as bleach activators are disclosed, as are bleach compositions comprising such an ester and a peroxygen compound which yields peroxide in solution....	03/21/1995

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Class 560/251 - Plural nitrogens in alcohol moiety