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| Number | Title | Issue Date |
| 7423012 | Phosphinyloxy, oxime and carboxylic acid derivatives which are useful as carboxypeptidase U inhibitors The present invention relates to compounds of Formula I, and pharmaceutically acceptable salts or solvates thereof, or solvates of such salts, which compounds inhibit carboxypeptidase U and thus can be used in the preventio... | 09/09/2008 |
| 7354895 | Phosphinyloxy, oxime and carboxylic acid derivatives which are useful as carboxypeptidase U inhibitors The present invention relates to compounds of Formula I, and pharmaceutically acceptable salts or solvates thereof, or solvates of such salts, which compounds inhibit carboxypeptidase U and thus can be used in the preventio... | 04/08/2008 |
| 7345188 | Process for preparing benzhydrylthioacetamide The present invention is directed to an improved process for preparing modafinil wherein benzhydrylthioacetate is prepared in high yield and purity by the reaction of a haloacetate with the reaction product of thiourea and benzhydrol. The reaction employing the halo... | 03/18/2008 |
| 7321049 | Synthesis of [C] and [H] substituted methacrylic acid, [C] and [H] substituted methyl methacrylate and/or related compounds The present invention is directed to labeled compounds of the formulae wherein Q is selected from the group consisting of —S—, —S(═O)—, and —S(═O)2—, Z is selec... | 01/22/2008 |
| 7301045 | Method for preparing ester condensate The present invention provides a method for preparing ester or thioester that can conduct catalytic esterification reaction with an equimolar amount of carboxylic acid and alcohol, or catalytic thioesterification reaction with carboxylic acid and an equimolar amount... | 11/27/2007 |
| 7297817 | Thio-substituted arylmethanesulfinyl derivatives The present invention is related to chemical compositions, processes for the preparation thereof and uses of the composition. Particularly, the present invention relates to compositions of compounds of Formula (A): wherein ... | 11/20/2007 |
| 7271283 | High refractive index, UV-curable monomers and coating compositions prepared therefrom Disclosed herein are high refractive index monomers that are curable by ultraviolet light. These monomers may be a component of curable compositions useful in the preparation of optical articles. Also disclosed is a method of synthesizing the monomers. ... | 09/18/2007 |
| 7057068 | Process for the preparation of modafinil A process for the preparation of 2-[(diphenylmethyl)sulfinyl]acetamide (I) comprising the oxidation of sodium 2-[(diphenylmethyl)sulfenyl]acetate to the corresponding sulfoxide and the derivatization of the latter to amide ... | 06/06/2006 |
| 6992105 | Dipeptide derivatives Compounds of the formula wherein R, R1, COOR2, R3–R7, alk, and X have meaning as defined, such being useful as dual inhibitors of angiotensin converting enzyme and neutral e... | 01/31/2006 |
| 6911521 | Polyhydroxyalkanoate that comprises unit having substituted or unsubstituted (phenylmethyl) sulfanyl structure in side chain thereof and process for producing the same A polyhydroxyalkanoate that comprises a unit represented by the following chemical formula (1): wherein R1 is a substituent of an aromatic ring selected from the group consisting of H, CH3, C2H | 06/28/2005 |
| 6803480 | Diphenylmethane derivatives The invention relates to novel diphenylmethane derivatives, processes for their preparation and their use in medicaments, in particular for the indications of arteriosclerosis and hypercholesterolaemia. ... | 10/12/2004 |
| 6767920 | 3, 7 or 3 and 7 thia or oxa prostanoic acid derivatives as agents for lowering intraocular pressure The present invention provides a method of treating ocular hypertension or glaucoma which comprises administering to an animal having ocular hypertension or glaucoma therapeutically effective amount of a compound represented by the general formula I; | 07/27/2004 |
| 6720445 | Acetyloxymethyl esters and methods for using the same Novel acetyloxymethyl esters are disclosed. Methods of treating an illness, including cancer, hemological disorders and inherited metabolic disorders, and treating or ameliorating other conditions using these compounds are also disclosed. The compounds are effective... | 04/13/2004 |
| 6703422 | Sulfide and disulfide compounds and compositions for cholesterol management and related uses The present invention relates to novel sulfide and disulfide compounds, compositions comprising sulfide and disulfide compounds, and methods useful for treating and preventing cardiovascular diseases, dyslipidemias, dysproteinemias, and glucose metabolism... | 03/09/2004 |
| 6683200 | N-substituted-N'-substituted urea derivatives and pharmaceutical compositions containing the derivatives N-Substituted-N'-substituted urea derivatives represented by the following formula, analogs thereof or pharmaceutically acceptable salts thereof are herein provided. These compounds show a TNF- production inhibitory activity. ##STR1##... | 01/27/2004 |
| 6649639 | Antipicornaviral compounds, compositions containing them, and methods for their use Picornaviral 3C protease inhibitors, obtainable by chemical synthesis, inhibit or block the biological activity of the picornaviral 3C protease. These compounds, as well as pharmaceutical compositions that contain these compounds, are suitable for treatin... | 11/18/2003 |
| 6638977 | Plasminogen activator inhibitor antagonists Compounds and pharmaceutical compositions useful as plasminogen activator inhibitor (PAI) antagonists are provided. In particular, methods of antagonizing PAI with substituted and unsubstituted aryl and heteroaryl ethers and thioethers are provided.... | 10/28/2003 |
| 6545050 | Aryl sulphonamide amino acid esters and analogues The present invention relates to novel amino acid esters of arylsulphonamides and analogues, to processes for their preparation and to their use for the prophylaxis and treatment of neurodegenerative disorders, in particular for the treatment of cerebral ... | 04/08/2003 |
| 6462081 | 5-thia-ω-substituted phenyl-prostaglandin E derivatives, process for producing the same and drugs containing the same as the active ingredient The present invention relates to 5-thia-ω-substituted phenylprostaglandin E derivatives of the formula (I) ##STR1## (wherein, all the symbols are as defined in the specification), process for producing them and pharmaceutical compositions comprising them... | 10/08/2002 |
| 6444850 | Fungicidial compounds having a fluorovinyloxphyenyl moiety and process for the preparation thereof A fungicidal compound of formula (I) having a fluorovinyloxyphenyl moiety and stereoisomers thereof are useful for protecting crops from fungal diseases: ##STR1## wherein: X is CH or N; Y is O or S; Z is O or NH; R1 is hydrogen or CF3 | 09/03/2002 |
| 6410775 | APL immunoreactive peptides, conjugates thereof and methods of treatment for APL antibody-mediated pathologies aPL analogs that (a) bind specifically to B cells to which an aPL epitope binds and are disclosed. Optimized analogs lack T cell epitope(s) are useful as conjugates for treating aPL antibody-mediated diseases. Conjugates comprising aPL analogs and nonimmu... | 06/25/2002 |
| 6331554 | Antipicornaviral compounds, compositions containing them, and methods for their use Picornaviral 3C protease inhibitors of formula I, obtainable by chemical synthesis, that inhibit or block the biological activity of the picornaviral 3C protease are described. ##STR1## These compounds, as well as pharmaceutical compositions that contain ... | 12/18/2001 |
| 6258977 | Alkyl3-oxoalkanoates An alkyl 3-oxoalkanoate, a process for preparation and use for the synthesis of fatty hydroxylated amino acids, fatty amino alcohols and ceramides.... | 07/10/2001 |
| 6201020 | Ortho-diphenol compounds, methods and pharmaceutical compositions for inhibiting parp This invention relates to compounds, pharmaceutical compositions, and methods of using compounds of the formula: ##STR1## A is O or S; R is C1 -C10 straight or branched chain alkyl, C2 -C10 straight or branched ... | 03/13/2001 |
| 6054457 | Benzamide derivatives and their use as vasopressin antagonists This invention relates to new benzamide derivatives having a vasopressin antagonistic activity, etc, and represented by general formula (I): ##STR1## wherein R1 is aryl optionally substituted with lower alkoxy, etc., R2 is lower... | 04/25/2000 |
| 6043275 | 3,7-dithiaprostanoic acid derivative A 3,7-dithiaprostanoic acid derivative of the formula (I) ##STR1## (wherein, R1 is OH, C1~6 alkyloxy, NR6 R7 (R6, R7 are H, C1~6 alkyl.); R2 is H, OH; R3 is single bond, C1~... | 03/28/2000 |
| 6028131 | Antioxidants containing phenol groups and aromatic amine groups The invention relates to compounds of the formula I ##STR1## in which R is C1 -C18 alkyl, C5 -C8 cycloalkyl, C7 -C9 phenylalkyl, --CH2 --A--R2 or a group of the f... | 02/22/2000 |
| 5981556 | 1,3-diazolino and 1,3-diazolidino heterocycles as useful nitric oxide synthase inhibitors 1,3-diazolino and 1,3-diazolidino heterocycle derivatives useful as nitric oxide synthase inhibitors.... | 11/09/1999 |
| 5977123 | Oximether and acrylic acid derivatives and their use as fungicides The invention relates to novel oximether and acrylic acid derivatives of the formula (I) ##STR1## in which Z, G, Ar, E, R1 and R2 have the meanings as given in the specification, to processes for their preparation and to their u... | 11/02/1999 |
| 5952386 | Dihalopropene compounds, insecticides containing them as active ingredients, and intermediates for their production The present invention provides dihalopropene compounds of the general formula: ##STR1## wherein R1 is C1 -C10 alkyl or the like; L is C(.dbd.O)NH or the like; R2, R3 and R4 are indepen... | 09/14/1999 |
| 5892099 | 3,7-dithiaprostanoic acid derivative A 3,7-dithiaprostanoic acid derivative of the formula (I) ##STR1## (wherein R1 is OH, C1-4 alkoxy, NR6 R7 (wherein R6, R7 are H, C1-4);R2 is H, OH; R3 is (i)alkyl, alkenyl, ... | 04/06/1999 |
| 5872282 | Allosteric modifiers of hemoglobin A family of compounds has been found to be useful for right-shifting hemoglobin towards a low oxygen affinity state. The compounds are capable of acting on hemoglobin in whole blood. In addition, the compounds can maintain the oxygen affinity in blood dur... | 02/16/1999 |
| 5756838 | Method of asymmetrically synthesizing optically active compounds using supported phase chiral sulfonated BINAP catalyst The present invention relates to water soluble chiral sulfonated 2,2'-bis(diphenylphosphino)-1,1'-binaphthyl and its use as organometallic catalysts for asymmetric synthesis of optically active compounds. Asymmetric reactions of the present invention incl... | 05/26/1998 |
| 5693848 | , ω-polymethacrylate dicarboxylic acids, their synthesis and use as dicarboxylic acid components for the synthesis or modification of polyesters, polyurethanes or polyepoxides ,ω-polymethacrylate dicarboxylic acids of the general formula ##STR1## wherein R1 is an optionally halogenated alkyl group with 1 to 22 carbon atoms, wherein the R1 group can assume different meanings in the polymer molecule, R | 12/02/1997 |
| 5686633 | Inks, particularly for ink jet printing Inks, particularly inks for ink jet printing, contain at least one compound of the formula I ##STR1## as a stabilizer. The symbols R1, R2, R3, R4, R3 ' and R4 ' are as defined in claim... | 11/11/1997 |
| 5663128 | Liquid antioxidants as stabilizers Products are described which can be obtained by reacting components a), b), c) and d), where component a) is a compound of the formula I or a mixture of compounds of the formula I, component b) is a compound of the formula II or a mixture of compounds of ... | 09/02/1997 |
| 5639903 | Sulfonium salt compounds and initiators of polymerization The present invention is related to sulfonium salt compounds useful as an initiator of cationic polymerization and represented by a following general formula (I): ##STR1## wherein R1 is benzyl, phenyl, etc., R2, R3 an... | 06/17/1997 |
| 5625067 | Cyclopentane ether derivatives, processes for their production, and their pharmaceutical use The invention relates to cyclopentane ether derivatives of Formula I ##STR1## their salts with physiologically compatible bases, as well as the -, ଲ- or γ-cyclodextrin clathrates, and also the liposome-encapsulated compounds of Formula ... | 04/29/1997 |
| 5536870 | Process for preparing olefins A process for preparing olefin compounds of the formula ##STR1## where A is aryl, substituted aryl, heteroaryl, substituted heteroaryl, benzyl, substituted benzyl, vinyl or substituted vinyl and R2, R3 and R4 are hydr... | 07/16/1996 |
| 5534651 | Process for preparing γ-mercaptocarboxylic acid derivatives γ-Mercaptocarboxylic acids and their derivatives, in particular esters and amides, are prepared from γ-butyrolactones via the corresponding thiolactones. The thiolactones are obtained by reaction of a γ-lactone with thiocarboxylates in polar solvents a... | 07/09/1996 |
