Celebrity Inventors
Comic actor Danny Kaye received patent D166,807 for the co-design of "Blowout Toy or the Like". It's similar to one of those toys that unravels when you blow into at a birthday party except Kaye's has three blowouts going in different directions, not just one.
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| Number | Title | Issue Date |
| 7402577 | Androstane 17-beta-carboxamides as androgen receptor modulators Compounds of structural formula as herein defined are disclosed as useful in a method for modulating the androgen receptor in a tissue selective manner in a patient in need of such modulation, as well as in a method of activating the function of the androgen recepto... | 07/22/2008 |
| 7371741 | Estradiol derivatives and pharmaceutical compositions using same Compositions and methods for treating mammalian disease characterized by undesirable angiogenesis by administering compounds of the general formula: wherein the variables are defined in the specification. ... | 05/13/2008 |
| 7199115 | 17α-fluorosteroids, pharmaceutical compositions containing 17α-fluorosteroids and a method of making them New 17α-fluorosteroid compounds of formula (I) are disclosed: wherein R1 denotes H or methyl; R2 and R3 each denote H, Cl or methyl; and either a double bond or a single bond is ... | 04/03/2007 |
| 6953785 | Estra-1,3,5(10)-triene derivatives Provided is steroid sulfatase inhibitors comprising, as the active ingredient, an estra-1,3,5(10)-triene derivative which is represented by formula (I): {wherein R1 and R2 are the same or differen... | 10/11/2005 |
| 6638923 | Estra-1,3,5(10),16-tetraene derivatives Estra-1,3,5(10),16-tetraene derivatives represented by the following formula (I): ##STR1## (wherein R1 is as defined by the present specification.... | 10/28/2003 |
| 6610866 | Stereoselective synthesis of 24-hydroxylated compounds useful for the preparation of aminosterols, vitamin D analogs, and other compounds A method is described for stereoselectively reducing an unsaturated alkyl ketone substituent attached to a fused ring base. In this method, the unsaturated alkyl ketone reacts with a chiral oxazaborolidine reagent. This reaction stereoselectively reduces ... | 08/26/2003 |
| 6596885 | 19-Nor steroids having a thiocarbonated chain in position 11beta, their preparation process and the intermediates of this process, their use as medicaments and compositions Novel compounds having a formula selected from the group consisting of ##STR1## wherein the substituents are defined as in the specification which are intermediates for the production of vinyl compounds having a remarkable anti-estrogenic and anti-prolife... | 07/22/2003 |
| 6437157 | 20-substituted steroids A compound selected from the group consisting of a compound of the formula ##STR1## wherein R1 and R2 are individually selected from the group consisting of alkyl of 1 to 12 carbon atoms and aralkyl of 7 to 15 carbon atoms or taken t... | 08/20/2002 |
| 6410760 | Process to prepare androst-4-en-17-carboxylic acid The process of the present invention transforms a steroidal ketone of formula (III) ##STR1## to androst-4-en-17ଲ-carboxylic acid (IV) ##STR2## by reaction with K2 SO5.KHSO.sub.4.K.sub.2 SO4.... | 06/25/2002 |
| 6399595 | Steroid sulfatase inhibitors and methods for making and using the same Novel sulfatase inhibitor compounds useful in the treatment of estrogen dependent illnesses are disclosed. These compounds generally comprise a steroid nucleus substituted at the C17 position. Methods for synthesizing these compounds and using them in the... | 06/04/2002 |
| 6376687 | Steroid sulfatase inhibitors and methods for making and using the same Novel sulfatase inhibitor compounds useful in the treatment of estrogen dependent illnesses are disclosed. These compounds generally comprise a steroid nucleus substituted at the C17 position. Methods for synthesizing these compounds and using them in the... | 04/23/2002 |
| 6288050 | Steroid sulfatase inhibitors and methods for making and using the same Sulfatase inhibitor compounds useful in the treatment of estrogen dependent illnesses are disclosed. These compounds generally comprise a steroid nucleus substituted at the C17 position. Methods for synthesizing these compounds and using them in the thera... | 09/11/2001 |
| 6262043 | Estra-1,3,5(10),16-tetraene derivatives Estra-1,3,5(10),16-tetraene derivatives represented by the following formula (I): ##STR1## (wherein R1 represents hydroxy, alkoxy, or NR2 R3 (wherein R2 and R3 are the same or different, and each repr... | 07/17/2001 |
| 6251887 | 17ଲ-aryl(arylmethyl)oxy(thio)alkyl-androstane derivatives The invention relates to 17ଲ-aryl(arylmethyl)oxy(thio)alkyl-androstane derivatives having general formula (I), wherein R1 is (H,OR), (H,OSO3 H) or NOR; with R being H, (C1-6)alkyl or (C1-6)acyl; each of R | 06/26/2001 |
| 6117994 | Intermediates for 16ଲ-methyl steroids A new process for the preparation of 16ଲ-methyl-steroids of the formula ##STR1## and novel intermediates.... | 09/12/2000 |
| 6080735 | Estra-1,3,5(10)-trien derivatives, processes for their preparation and pharmaceutical compositions containing these compounds This invention is relating to new estra-1,3,5(10)-trien-sulfamates carrying at the 3-position an R--SO2 --O--group, with R being an R1 R2 N--group in which R1 and R2, independently of each other, repr... | 06/27/2000 |
| 5969168 | Androstanes for inducing hypothalamic effects The invention relates to novel, androstane steroids which are the ligand semiochemicals which bind to neuroepithelial receptors. The steroids are useful as ligands to neuroepithelial receptors in the human vomeronasal gland to stimulate autonomic and hypo... | 10/19/1999 |
| 5925774 | Estrenes for inducing hypothalamic effects The invention relates to estrene steroids, which bind to neuroepithelial receptors. The steroid is preferably administered in the form of a pharmaceutical composition containing one or more pharmaceutically acceptable carriers.... | 07/20/1999 |
| 5880115 | Steroid sulfatase inhibitors and methods for making and using the same Sulfatase inhibitor compounds having the formula: ##STR1## wherein X, Y, R1, R2 and R3 are as defined in the specification. The compounds are useful in the treatment of estrogen dependent illnesses. Methods for synthe... | 03/09/1999 |
| 5792759 | 17-hydroxyiminoalkyl and 17-hydroxyiminomethylalkenyl cyclopentaneperhydrophenanthrene derivatives active on the cardiovascular system, a process for their preparation and pharmaceutical compositions containing the same Novel 17-hydroxyiminoalkyl and 17-hydroxyiminomethylalkenyl steroids of the general formula (I) ##STR1## where A, R1 and R2 are defined in the specification are disclosed. The compounds have cardiovascular activity. Pharmaceutic... | 08/11/1998 |
| 5723455 | Antiandrogenic agents and related pharmaceutical compositions and methods of use Novel antiandrogenic agents are provided. An exemplary group of compounds has the structural formula (I) ##STR1## wherein R1 through R10, a and b are as defined herein. Pharmaceutical compositions and methods for using the compo... | 03/03/1998 |
| 5650526 | Process for the preparation of an oxoetiocholenic acid The invention is drawn to a process for the preparation of oxoetiocholenic acid of the formula I ##STR1## by reacting a compound of the formula II ##STR2## with a halonitrile in the presence of a base followed by formation of a 3-ketone gro... | 07/22/1997 |
| 5633392 | Estrenes for inducing hypothalamic effects The invention relates to estrene steroids, which bind to neuroepithelial receptors. The steroid is preferably administered in the form of a pharmaceutical composition containing one or more pharmaceutically acceptable carriers.... | 05/27/1997 |
| 5618806 | 17 and 17ଲ-substituted estra-1,3,5(10)-triene-3-carbboxlic acid Invented are 17 and 17ଲ-substituted acyl-3-carboxy aromatic A ring analogues of steroidal synthetic compounds. Representative of such compounds include the following ##STR1## wherein Z is or ଲ ##STR2## in which A ... | 04/08/1997 |
| 5561124 | 17--acyl steroids which inhibit 5--reductase The invention relates to substituted 17-acyl steroidal 5-reductase inhibiting compounds. The invention also relates to pharmaceutical compositions containing these compounds and their use for reducing prostate size and treating prostate aden... | 10/01/1996 |
| 5523428 | Process for the production of 1-methyl-3-keto-Ɗ1,4 steroids A process for the production of 1-methyl-3-keto-Ɗ1,4 steroids of general formula I ##STR1## in which St symbolizes the radical of asteroid molecule, where a 3-keto-Ɗ1,4 steroid of general formula II ##STR2## in which... | 06/04/1996 |
| 5496813 | Spontaneously dispersible concentrates and aqueous microemulsions with steryl retinates having anti-tumor activity There are described spontaneously dispersible agents containing sterolester and/or sterolphosphor compounds having a pronounced antitumour activity. Novel sterolesters and sterolphosphor compounds, their use for treating tumors, and processes for their pr... | 03/05/1996 |
| 5438134 | Process for the production of unsaturated 17 -cyanomethyl-17 ଲ- h The unsaturated 17-cyanomethyl-17ଲ-hydroxy steroids of the formula I, ##STR1## in which R1 =Me, Eth; R2 =H, Me; R3 =H, OH, an acetoxy or alkoxy group; R4 =H, R5 =OH, an acetoxy, alko... | 08/01/1995 |
| 5436401 | 22-oxacholecalciferol derivative and process for preparing the same A 22-oxacholecalciferol derivative represented by formula (I): ##STR1## wherein R1 represents a hydrogen atom or a hydroxyl group; and R2 and R3, which may be the same or different, each represent a lower alkyl group ... | 07/25/1995 |
| 5273971 | 13-alkyl-11ଲ-phenylgonanes There are provided 13-alkyl-11beta-phenyl-gonanes of formula I ##STR1## wherein Z is an oxygen atom or N--OH; R2 is alpha- or beta-position methyl or ethyl; R1 is selected from heteroaryl radicals, cycloalkyl radicals, cycloalkenyl r... | 12/28/1993 |
| 5272140 | 11-aryl steroid derivatives The invention relates to 11-aryl steroid derivatives, having the structure ##STR1## wherein: R1, R2, R3, and R4 are as described in the specification and to processes for their preparation and to pharmaceutical... | 12/21/1993 |
| 5140106 | Process for the production of 3-deoxy-4-ene steroids A process for the production of 3-deoxy-4-ene steroids of the general formula I ##STR1## is described, in which R1, R2 and R3 mean a hydrogen atom or a methyl group, R4 represents a lower alkyl group, a phe... | 08/18/1992 |
| 5137882 | Steroidal 3-acetic acid derivatives as 5-alpha-reductase inhibitors Invented are 3-acetic acid-steroidal compounds, pharmaceutical compositions containing the compounds, and methods of using these compounds to inhibit steroid 5-reductase including using these compounds to reduce prostate size and to treat prostatic... | 08/11/1992 |
| 5086047 | Novel steroids A compound selected from the group consisting of a compound of the formula ##STR1## wherein R is selected from the group consisting of hydrogen, alkyl, alkylthio and haloalkyl of 1 to 6 carbon atoms, alkenyl and alkynyl of 2 to 6 carbon atoms, option... | 02/04/1992 |
| 5064822 | Novel 3-keto-19-nor-Ɗ4,9 -steroids Novel 3-keto-19-nor-Ɗ4,9 -steroids of the formula ##STR1## wherein R1 is selected from the group consisting of naphthyl, phenylphenyl, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms optionally containing additiona... | 11/12/1991 |
| 5041433 | 11-keto or hydroxy 3,5-diene steroids as inhibitors of steriod 5--reductase Invented are carboxyl and carboxyl alkyl ester substituted 11-keto and hydroxy analogues of synthetic steroidal compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase.... | 08/20/1991 |
| 5032586 | 7-keto or hydroxy 3,5-diene steroids as inhibitors of steroid 5-alpha reductase Invented are carboxyl and carboxyl alkyl ester substituted 7-keto and hydroxy analogues of synthetic steroidal compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5--reductase. ... | 07/16/1991 |
| 4996335 | Soft steroids having anti-inflammatory activity The invention provides novel soft steroidal anti-inflammatory agents, pharmaceutical compositions containing said agents, and methods of administering same to mammals in the treatment of inflammation. Preferred compounds of the invention include haloalkyl... | 02/26/1991 |
| 4954446 | Aromatic steroid 5--reductase inhibitors Invented are substituted acrylate analogues of steroidal synthetic compounds, pharmaceutial compositions containing the compounds, and methods of using these compounds to inhibit steroid 5--reductase including using these compounds to reduce prosta... | 09/04/1990 |
| 4946834 | Phosphonic acid substituted steroids as steroid 5-reductase inhibitors Invented are substituted acrylate analogues of steroidal synthetic compounds, pharmaceutical compositions containing the compounds, and methods of using these compounds to inhibit steroid 5-reductase. Also invented are intermediates used in prepari... | 08/07/1990 |
