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Behavior Modification Wristwatch
A wristwatch including a watch band and a watch body having an octagon shaped perimeter and being red in color and having the word STOP thereon to resemble a stop sign.
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| Number | Title | Issue Date |
| 6388108 | Aminosterol compounds and uses thereof Newly isolated aminosterol compounds and pharmaceutical compositions based on the aminosterol compounds are described. Methods for the treatment of various disorders, for example, a microbial infection, are also described.... | 05/14/2002 |
| 6028066 | Prodrugs comprising fluorinated amphiphiles The present invention describes, inter alia, novel prodrugs comprising fluorinated amphiphiles, compositions comprising the novel prodrugs, and methods of use of the prodrugs and compositions.... | 02/22/2000 |
| 5972922 | Steroids which inhibit angiogenesis Novel angiostatic Ɗ4,9(11) -steroids (I), ##STR1## C21 -oxygenated steroids (II) and other known steroidal compounds have been found to be useful in treating angiogenesis in mammals who have a need for the same. These steroids ... | 10/26/1999 |
| 5637691 | Steroid derivatives, pharmaceutical compositions containing them, and their use as antibiotics or disinfectants Compounds having a broad range of antimicrobial activity generally have a structure including asteroid nucleus with a cationic, preferably polyamine, side chain (X) and an anionic side chain (Y). The invention is also directed to compounds of the Formula ... | 06/10/1997 |
| 5428181 | Bisphosphonate derivative A compound represented by the general formula: ##STR1## wherein A-O-denotes a residue of a compound having an estrogenic activity; R1 denotes H or a C1 -C6 alkyl group; X denotes a single bond, a C1 -C... | 06/27/1995 |
| 5391776 | Steroid derivatives Asteroid derivative of the general formula: ##STR1## wherein X--O-- represents a residue of steroid compound and --A-- represents --CO[NH(CHR1)y --(Y)p --CO]m NH--, --CO--(R2)x --(Z) | 02/21/1995 |
| 5183815 | Bone acting agents Described are new agents for treating bone disorders associated with a reduction in bone mass and abnormalities in bone resportion or bone formation including osteoporosis. Paget's disease, bone metastases and malignant hypercalcemia. The agents are hydro... | 02/02/1993 |
| 5026882 | Phosphinic acid substituted steroids as inhibitors of steroid 5-reductase The invention relates to 3-phosphinic acid steroidal compounds, pharmaceutical compositions containing these compounds, and methods of using these compounds to inhibit steroid 5-reductase.... | 06/25/1991 |
| 4975537 | Ɗ9(11) -angiostatic steroids Disclosed are Ɗ9(11) -steroids of the formula ##STR1## which have been found to be angiostatic and therefore are useful in the control of embryogenesis, inflammatory conditions, tumor growth as well as other abnormalities.... | 12/04/1990 |
| 4678609 | Process for the preparation of corticosteroid-21-phosphoric acids and their salts and the corticosteroid-21-phosphoric acid triesters Steroid-21-phosphoric acids and pharmaceutically usable salts thereof of the formula III ##STR1## (in which U=H or CH3, V=H, OH, O or Hal; W=H or OH and Y=H or F) are obtained in a very pure state by reacting I ##STR2## (in which... | 07/07/1987 |
| 4603128 | Mineralocorticoid hormone antagonists 7-acylthio-4-pregnene-3,20-diones, active as mineralocorticoid hormone antagonists, of the formula: ##STR1## in which R1 is hydrogen, hydroxyl or acyloxy --OR2, R2 is an acyl group derived from a straight or br... | 07/29/1986 |
| 4525303 | Process for preparation of steroids A novel process for preparing a steroid of the following formula (to be referred to as compound .circle.13 ) is provided. ##STR1## This compound is known to have marked anti-inflammatory and anti-rheumatoid arthritic activity with very much reduced ... | 06/25/1985 |
| 4444689 | 17-Acyloxy-5ଲ-corticoids and 17-acyloxy-5-corticoids 17-Acyloxy-5ଲ-pregnanes (I) and 17-acyloxy-5-pregnanes (IV) have an excellent activity split providing high topical anti-inflammatory activity with very low systemic side effects.... | 04/24/1984 |
| 4427591 | Reduced A ring-Ɗ9(11) -corticoids 17-Acyloxy-5ଲ-pregnanes (I) and 17-acyloxy-5-pregnanes (IV) have an excellent activity split providing high topical anti-inflammatory activity with very low systemic side effects.... | 01/24/1984 |
| 4336200 | 17-Acyloxy-5ଲ-corticoids 17-Acyloxy-5ଲ-pregnanes (I) and 17-acyloxy-5-pregnanes (IV) have an excellent activity split providing high topical antiinflammatory activity with very low systemic side effects.... | 06/22/1982 |
| 4318853 | 9ଲ,11ଲ-Epoxy-5ଲ-corticoids 17-Acyloxy-5-pregnanes (I) and 17-acyloxy-5-pregnanes (IV) have an excellent activity split providing high topical anti-inflammatory activity with very low systemic side effects.... | 03/09/1982 |
| 4275061 | Steroids and process for preparing the same The present invention relates to 2-chloro-6ଲ-fluoropregna-1,4-diene-3,20-diones having good anti-inflammatory activity, to processes for their preparation and pharmaceutical compositions thereof.... | 06/23/1981 |
| 4268453 | Process for the manufacture of cholestene derivatives and novel intermediates in their manufacture The present disclosure is directed to 6-lower alkoxy-25,26-(lower alkyl or lower alkylene)methylene dioxy-3,5-cyclocholest-22-ene derivatives which are useful in the manufacture of 25,26-dihydroxycholecalciferol.... | 05/19/1981 |
| 4267173 | Use of 6ଲ-fluoro-7-halogenocorticoids as topical anti-inflammatories and pharmaceutical formulations useful therefor Described is the use of 6ଲ-fluoro-7-halogeno-1,4-pregnadiene-17,21-diol-3,20-di ones and their esters as topical anti-inflammatory agents, and pharmaceutical formulations thereof useful therefor. Preferred compounds are 6ଲ,9&... | 05/12/1981 |
| 4263290 | Novel 19-nor-steroids Novel 19-nor-steroids of the formula ##STR1## wherein R1 and R2 taken together form a cycloalkyl of 3 to 8 carbon atoms or are individually selected from the group consisting of hydrogen, alkyl of 1 to 4 carbon atoms and alkenyl... | 04/21/1981 |
| 4201778 | 6-Acyloxy-1,4,6-pregnatrienes, their use as anti-inflammatory agents, methods for their manufacture, and 6-oxo-1,4-pregnadiene intermediates Novel 6-acyloxy-3,20-dioxo-1,4,6-pregnatrienes and 6-acyloxy-3,20-dioxo-4,6-pregnadienes, useful anti-inflammatory agents, are prepared by reaction of the corresponding 3,6,20-trioxo-1,4-pregnadiene or 3,6,20-trioxo-4-pregnene with an acyl halide or ... | 05/06/1980 |
| 4196203 | Novel corticoids Compounds of the formula ##STR1## wherein X is ଲ-CH2 OH or CO and R2 is F, Cl or CH3, and their physiologically acceptable 21-esters are useful for the treatment of allergic diseases of the respiratory tract and... | 04/01/1980 |
| 4189440 | 2-Bromo-6ଲ-fluoro-3-keto-Ɗ1,4 -steroids of the pregnane series Pregnane series steroids are disclosed having good anti-inflammatory and anti-rheumatoid arthritic activity with a decreased degree of side effects, e.g., weight loss and sodium retention. The compounds have the formula ##STR1## where X is a ket... | 02/19/1980 |
| 4124707 | 7-Halogeno-3,20-dioxo-1,4-pregnadienes, methods for their manufacture, their use as anti-inflammatory agents, and pharmaceutical formulations useful therefor Novel 3,20-dioxo-7-halogeno-1,4-pregnadienes are described and their use as anti-inflammatory agents. Preferred are 7-bromo- and 7-chloro- derivatives, particularly 7-bromo- and 7-chloro-1,4-pregnadienes-11ଲ,17�... | 11/07/1978 |
| 4092310 | Difluorosteroids and processes for their manufacture A novel group of 18,18-difluorosteroids of the general formula ##STR1## wherein St, R1 and R2 have the meanings given hereinafter is produced by a chemically novel process characterized in that a corresponding 18-oxo compound is... | 05/30/1978 |
| 4076737 | Aldehydes of the pregnane series and derivatives thereof The derivatives of 1-dehydro-6,9-difluoro-16-methyl-corticosterone having an aldehyde group in 21-position instead of the hydroxyl group, and derivatives of such aldehydes having a 2-chlorine atom, the corresponding hydrates, as ... | 02/28/1978 |
| 4024131 | 16-Methyl-9-halo steroid esters, ethers and preparation thereof New 16-methyl-9-halo corticosteroid esters and ethers having high topical anti-inflammatory potency and low systemic activity and the manner in which they can be produced are described.... | 05/17/1977 |
| 4012510 | Novel methylene steroids Methylene steroids of the formula ##STR1## wherein X is H, F or CH3 ; Y is hydroxymethylene, alkanoyloxymethylene or carbonyl; R1 is H, OH or alkanoyloxy; and R2 is H, OH or esterified OH, possess topical anti-inflamm... | 03/15/1977 |
| 4008313 | Novel corticoids Corticoids of the formula ##STR1## wherein X is ଲ-hydroxymethylene or carbonyl, and 21-esters thereof with physiologically acceptable acids possess topical anti-inflammatory activity with relatively little systemic activity.... | 02/15/1977 |
| 3998701 | Process for the preparation of 17-acyl esters of 17, 21-dihydroxysteroids of the pregnane series and novel products A process is disclosed for making 17-monoesters of 17 , 21-dihydroxy steroids by acylating a 17 , 21-dihydroxy steroid phosphate and then subjecting the intermediate 17-acyloxy-21-phosphate to dephosphorylation using an acid phosphatase to a... | 12/21/1976 |
| 3971772 | Steroidal[16,17-b]1,4-dioxanes and Steroidal[16,17-b]1,4-dioxins A series of novel steroidal [[16,17-b]1,4-dioxanes and steroidal [ 16,17-b]1,4-dioxins having useful anti-inflammatory properties is disclosed herein.... | 07/27/1976 |
| 3966778 | Production of 21-phosphate corticords having unprotected hydroxyl radicals at least at the 17- and 21-position There is disclosed a process for preparing 17-hydroxy corticoid 21-phosphate which comprises reacting a compound selected from the group consisting of 17,21-dihydroxy corticoid and 11, 17,21-trihydroxy corticoid with pyrophosphoryl te... | 06/29/1976 |
| 3963707 | Novel N-nitroso compounds, compositions containing such compounds, processes for their preparation and methods of treatment therewith, and novel intermediates This invention relates to novel N-halogenoalkyl-N-nitroso carbamates and N4 halogenalkyl-N4 -nitroso allophanates of steroid compounds, having an anti-tumor activity, and to the preparation thereof. The invention is also concerned wi... | 06/15/1976 |
| 3944584 | Steroidal (16,17-d)cyclohexenes A series of novel steroidal[ 16, 17-d]cyclohexenes having a 9-fluoro group is disclosed herein for use as anti-inflammatory agents.... | 03/16/1976 |
| 3939187 | 15,-Sulfonyloxy-12ଲ-hydroxypregnanes and process for the preparation thereof 15-Sulfonyl-12ଲ-hydroxypregnanes of the formula ##SPC1## Wherein Ac is lower-acyl and R is alkyl, cycloalkyl, aralkyl or aryl, which are useful as intermediates for the production of digoxigenin, are produced by the selective sulfonic acid es... | 02/17/1976 |
| 3933799 | 11ଲ-Halo-9,12-unsubstituted-C19 -steroids 11ଲ-Halo-9,12-unsubstituted-C19 -steroids having hormonal activity and a process for preparing same by reacting the corresponding 11-hydroxy steroid with a compound of the formula ##EQU1## where R1 and R... | 01/20/1976 |
