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Mountable Printable Placard With Headband

A resilient headband in a shape for being mounted on the head of the user. The headband is equipped with a longitudinal slotted member for holding a placard.

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Class 549/289 - The other cyclo of the bicyclo ring system is a six-membered carbocyclic ring to which chalcogen is directly attached


Subclass of Class 549 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the other cyclo of the bicyclo ring system
No. of patents: 134
Last issue date: 12/06/2011


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NumberTitleIssue Date
8071794Long wavelength thiol-reactive fluorophores
Reactive fluorescent dyes compositions and methods of using same are disclosed. Squaraine nucleus, Nile Red nucleus, benzodioxazole nucleus, coumarin nucleus or aza coumarin nucleus dyes are disclosed having thiol-reactive groups. Squaraine nucleus, Nile Red nucleus...
12/06/2011
7897792Coumarin derivative having antitumor activity
The present invention provides a compound represented by general formula (1) below or a pharmaceutically acceptable salt thereof: wherein: X is selected from heteroaryl etc., Y1 and Y2 are selected fro...
03/01/2011
7709664Coumarin derivatives useful as TNFα inhibitors
Novel compounds composition capable of inhibiting TNFα and having anti immunoinflammatory and autoimmune properties useful in a pharmaceutical composition, such as for a drug containing this as an active ingredient; and a therapeutic method with the use of these no...
05/04/2010
7507837Process for performing an isolated Pd(II)-mediated oxidation reaction
There is disclosed a process for performing an isolated Pd(II) mediated oxidation reaction electrochemically. The inventive process is performed on an electrode array device having a plurality of separately addressable electrodes. Preferably, the Pd(II) mediated oxi...
03/24/2009
7439265Irciniastatins a and b
The Indo-Pacific marine sponge Ircinia ramosa has been found to contain two powerful (GI50 0.001 to
10/21/2008
7435455Dihydrocoumarin derivative, liquid crystal composition containing the same, and liquid crystal display device
A dihydrocoumarin ring-containing compound of the invention is represented by the following formula (1): wherein R represents hydrogen or an alkyl; A1 to A3 each represents 1,4-cyclohexylene or 1,4-phe...
10/14/2008
7304168Photo-caged fluorescent molecules
A class of photo-caged and cell permeable fluorescent molecules having high uncaging cross sections, robust fluorescence enhancement, and flexible chemistry for bioconjugation. Some of the photo-caged fluorescent molecules are derived from 6-chloro-7-hydroxy-coumari...
12/04/2007
7282575Functional peptide nucleic acid monomer and process for producing the same
A compound represented by the general formula (I) below: In the formula, A is as defined in the specification and B denotes where n is an integer of 1 to 4, ...
10/16/2007
7259185Stable warfarin sodium liquid formulation and method of making same
A stable liquid composition comprising warfarin sodium, glycerin, an alcohol such as ethanol, and a pH buffer such as a phosphate buffer providing a pH above 7 is provided. The stability of the composition is characterized by the amount of warfarin sodium in the com...
08/21/2007
7259265Coumarin compounds and method for preparing and using the same
4-Substituted coumarin compounds having the general formula of where R is H, CHO, OCH3, X, NO2, an alkyl having C1-10, —OCH2O—, an aryl being mono- or poly-substitu...
08/21/2007
7226945Estrogen receptor-β ligands
A method for treating a disease associated with the estrogen receptor-β, comprising the step of administiering a therapeutically-effective amount of a compound that satifies the equation: KiαA/KiβA>25, optionally having general structure (I)...
06/05/2007
7094378Method and apparatus for inactivation of biological contaminants using photosensitizers
Methods and apparatuses for treating fluids to inactivate microorganisms which may be present therein, said fluid containing one or more components selected from the group consisting of protein, blood and blood constituents are provided. The methods comprise adjusti...
08/22/2006
7064207Androgen receptor antagonists
The present invention is directed to a new class of 6-sulfonamido-quinolin-2-one and 6-sulfonamido-2-oxo-chromene derivatives to their use as androgen antagonists, and to relieve conditions associated with inappropriate activation of the androgen receptor. ...
06/20/2006
7057048Androgen receptor antagonists
The present invention is directed to a new class of 6-sulfonamido-quinolin-2-one and 6-sulfonamido-2-oxo-chromene derivatives to their use as androgen antagonists, and to relieve conditions associated with inappropriate activation of the androgen receptor. ...
06/06/2006
7026491Coumarin derivatives useful as TNFα inhibitors
Novel compounds composition capable of inhibiting TNFα and having antiimmunoinflammatory and autoimmune properties useful in a pharmaceutical composition, such as for a drug containing this as an active ingredient; and a therapeutic method with the use of these nov...
04/11/2006
6900340Preparation of isocoumarin derivatives and intermediates for the synthesis thereof
A method of preparing optically active isocoumarin-3-yl-acetic acid derivatives represented by Formula (I): wherein a specific isocoumarin-ketene derivative is subjected to an addition reaction with an optically active...
05/31/2005
6900239Tumor chemopotentiation using isocoumarin derivatives
A method for enhancing the efficacy of chemotherapy in the treatment of cancer in animals, particularly humans, is provided wherein isocoumarin derivatives that exhibit unique chemopotentiation properties are employed in a combination treatment with chemotherapy.
05/31/2005
6800768Non-nucleosidic coumarin derivatives as polynucleotide-crosslinking agents
Novel coumarin derivatives comprising a coumarin moiety linked to a non-nucleosidic backbone moiety are disclosed. The resulting molecules are typically used as photoactivate crosslinking groups when incorporated into polynucleotides as replacements for one or more ...
10/05/2004
6770764Trypsin substrate and diagnostic device, and method of using same
A compound of the formula (I) wherein R1 is a protecting group for Nα, R2 is a protecting group for NG, and R3 is aryl, and wherein the compound of formula (I) is a trypsin su...
08/03/2004
6752862Color fading/discoloration preventive agent
Disclosed are a color fading/discoloration preventive agent containing as its active ingredient a coumarin analog represented by general formula (1) below, a glycoside of that analog, or a plant extract containing the coumarin analog or its glycoside:
06/22/2004
6734313Synthesis of spiro esters, spiro ortho carbonates, and intermediates
Ortho esters and ortho carbonates can be produced by alkylating esters and carbonates with, for example, the hexafluorophosphate salt of a trialkyl oxonium ion. The spiro species are useful intermediates in the synthesis of complex organic molecules. Synthetic pathw...
05/11/2004
6716996Process for preparing substituted coumarins
The present invention relates to a process for preparing substituted coumarins. More particularly, the present invention relates to a process for preparing substituted coumarins using polyaniline salts as catalysts. ...
04/06/2004
6670383Pyranocoumarin compounds as a novel pharmacophore with anti-TB activity
The present invention relates to compounds and compositions useful in treating or preventing conditions and diseases related to Mycobacterium infection, and methods of use directed thereto....
12/30/2003
66171247-alkoxycoumarins as cytochrome p450 substrates
Coumarin derivatives as substrates for cytochrome P450 enzyme....
09/09/2003
6613918Synthesis of spiro ortho esters, spiro ortho carbonates, and intermediates
Ortho esters and ortho carbonates can be produced by alkylating esters and carbonates with, for example, the hexafluorophosphate salt of a trialkyl oxonium ion. The spiro species are useful intermediates in the synthesis of complex organic molecules. Synt...
09/02/2003
6538022Compounds for deactivating phospholamban function on Ca-ATPase (phopholamban inhibitors)
This invention relates to determining the three-dimensional structure of the cytosolic domain of phospholamban (PLB) and its active site from NMR data of sufficiently high resolution for the three-dimensional structure determination. The invention also re...
03/25/2003
6455579Pyran derivatives
Disclosed are pyran derivatives, which have distinctive sensitivity to visible light and distinctive luminous ability. The derivatives are useful in photopolymerization, electroluminescence, and dye lasers, and are obtainable through a step of reacting a ...
09/24/2002
6426420Process for producing isocoumarines and intermediates for the same
Provided is a process for producing an isocoumarin-3-yl-acetic acid derivative, characterized by reacting a homophthalic acid derivative represented by a formula: ##STR1## (wherein Rc, R2 and R are mainly protecting groups) with a ...
07/30/2002
6420130Optical molecular sensors for cytochrome P450 activity
The invention provides a compound, useful as an optical probe or sensor of the activity of at least one cytochrome P450 enzyme, and methods of using the compound to screen candidate drugs, and candidate drugs identified by these methods. The optical probe...
07/16/2002
64204011,2,5, thiadiazolidin-3-one 1,1-dioxide derivatives
Substituted derivatives of 1,2,5-thiadiazolidin-3-one 1,1-dioxides, oligomers containing them, and methods of using them....
07/16/2002
6387258Method of purifying statins from a fermentation broth
A process for purifying statin compounds from a fermentation broth by extraction and crystallization is disclosed. A fermentation broth is subjected to a pretreatment procedure which involves an alkaline pretreatment and an alkaline purification. Followin...
05/14/2002
6372739Compounds and methods for modulation of estrogen receptors
Compounds that modulate gene expression through the estrogen receptor (ER) are disclosed having the following structure, as well as pharmaceutical compositions containing the same: ##STR1## wherein R1, R2, R3, n and p are ...
04/16/2002
6344330Pharmacophore recombination for the identification of small molecule drug lead compounds
The present invention is directed to novel methods for identifying small molecule ligands that are capable of binding with high affinity to a biological target molecule of interest. High affinity binding ligands identified by the described methods find us...
02/05/2002
6344334Pharmacophore recombination for the identification of small molecule drug lead compounds
Method for identifying a drug lead compound that inhibits binding of target bioogical molecules (TBM) by contacting TBM with members of a library of candidate cross-linked target binding fragments (CXBF), each CXBF having at least two candidate target bin...
02/05/2002
6331562Compounds and methods for modulation of estrogen receptors
Compounds that modulate gene expression through the estrogen receptor (ER) are disclosed having the following structure, as well as pharmaceutical compositions containing the same: ##STR1## wherein R1, R2, R3, n and p are ...
12/18/2001
6310248Process and intermediates
The invention relates to a process for the enantioselective preparation of tolterodine and analogues and salts thereof comprises the steps of: a) enantioselectively reducing the carbonyl function in a compound of formula (II): ##STR1## wherein R1
10/30/2001
6291456Compounds and methods for modulation of estrogen receptors
Compounds that modulate gene expression through the estrogen receptor (ER) are disclosed having the following structure, as well as pharmaceutical compositions containing the same: ##STR1## wherein R1, R2, R3, n and p are ...
09/18/2001
6258839Isolation of naturally occuring isoflavanone and some clinical uses thereof
A compound of general formula I ##STR1## in which the 2-3 bond in ring C could be double or single bond. Ring B and its substituents may be attached at position 2 (at J) in ring C. The key feature in the modifications is that the prenylation must not cycl...
07/10/2001
6215006Process for the preparation of 3-isochromanoes by cyclization of o-chloromethylphenylacetic acids
The present invention relates to a process for the preparation of a 3-isochromanone of the formula (I) ##STR1## by reaction of an o-chloromethylphenylacetic acid of the formula (II) ##STR2## at a temperature of 100 to 250° C. in the presence or absence o...
04/10/2001
6100292Ketone derivatives and their medical applications
This invention relates to ketones represented by the following formula ##STR1## and to drugs in which such a ketone or pharmacologically acceptable salt thereof is an effective component. The ketones of the present invention encourage the production of pl...
08/08/2000
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