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| Number | Title | Issue Date |
| 7816542 | Compounds and compositions as TPO mimetics The invention provides a novel class of compounds, pharmaceutical compositions comprising such compounds and methods of using such compounds to treat or prevent diseases or disorders associated with abnormal or deregulated TPO activity, particularly diseases or diso... | 10/19/2010 |
| 7781599 | Process for production of aromatic compounds A problem of the present invention is to provide an economical process with minimized toxicity for producing an aromatic compound having a variety of substituents such as various alkyl groups, and the problem is solved by a process for production of an aromatic comp... | 08/24/2010 |
| 7217732 | Cannabinoid receptor agonists A compound of the formula or a pharmaceutically acceptable salt thereof, wherein: R1, R2, R3, R4, R5, R6, L1, L2 | 05/15/2007 |
| 7217706 | Propanolamine derivatives This invention relates to new propanolamine derivatives or salts thereof represented by the following formula [I]: Wherein each symbol is as defined in the specification or salts thereof which have gut selective sympatho... | 05/15/2007 |
| 7173129 | Sulfonamide-substituted chalcone derivatives and their use to treat diseases The invention relates to compounds, pharmaceutical compositions and methods of using compounds of the general formula or its pharmaceutically acceptable salt or ester, wherein the substituents are defined in the ... | 02/06/2007 |
| 7071180 | Certain arylaliphatic and heteroaryl-aliphatic piperazinyl pyrazines and their use in the treatment of serotonin-related diseases The invention relates to compounds of the general formula (I): wherein Ar is optionally substituted aryl or heteroaryl; A is (i) —O—, —S—, —SO2... | 07/04/2006 |
| 6969612 | Reagent and method for measuring a concentration of protein The object of the present invention is to measure a concentration of protein stably at a temperature not higher than 25° C., which is a possible ambient temperature at home, and further to expand the measurable concentration range while preventing an obstruction du... | 11/29/2005 |
| 6960611 | Sulfonyl-containing 2,3-diarylindole compounds, methods for making same, and methods of use thereof The present invention relates to sulfonyl-containing 2,3-diarylindole, especially to new compounds of general Formula, to a preparation method for their preparation, to pharmaceutical compositions containing said compound, and to the medical use thereof in the treat... | 11/01/2005 |
| 6960688 | Use of compounds for the elevation of pyruvate dehydrogenase activity The use of compounds of formula (I), and salts thereof; and pharmaceutically acceptable in vivo cleavable prodrugs of said compound of formula (I); and pharmaceutically acceptable salts of said compound or said prodrugs; in formula (I), Ring C is phenyl or a carbon ... | 11/01/2005 |
| 6951848 | Functionalized heterocycles as modulators of chemokine receptor function and methods of use therefor Disclosed are novel compounds having the formula or a physiologically acceptable salt, amide, ester or prodrug thereof. The compounds can be used to modulate (antagonize, agonize) chemokine receptor function. Also disc... | 10/04/2005 |
| 6875770 | Indole derivative having heterocycle and mono- or diazaindole derivative There is provided a compound represented by the general formula (1): wherein Het represents an optional substituted heterocylic group A1 and A2 each independently represent —CH═, etc.; A3... | 04/05/2005 |
| 6867200 | (Hetero)aryl-bicyclic heteroaryl derivatives, their preparation and their use as protease inhibitors The present invention provides novel compounds of the Formula (I): A-B, its prodrug forms, or pharmaceutically acceptable salts thereof, wherein A represents a saturated, unsaturated, or a partially unsaturated bicyclic heterocyclic ring structure, and B represents ... | 03/15/2005 |
| 6858642 | Indole derivatives The invention relates to 1-(R1)-2-(R2)-3-(Y-X—NH-A- or Z-A-)-4,5,6,7-R)0.4-indoles, and their acid addition salts where the compounds are basic, wherein A is C1-4 alkylene, X is >CH2, >C═O or >C═S, and the... | 02/22/2005 |
| 6825352 | Preparation and use of ortho-sulfonamido arylhydroxamic acids as matrix metalloproteinase inhibitors Ortho-sulfonamido aryl hydroxamic acids are provided which are useful, inter alia, for the inhibition of matrix metalloproteinases and the treatment of conditions associated with overexpression of MMPs. ... | 11/30/2004 |
| 6787550 | Indole derivatives and their use for the treatment of osteoporosis amongst other applications A compound of formula (1) or a salt thereof, or a solvate thereof, wherein; R1 and R2 each independently represents C1-6alkoxy or halo; R3 and R4 | 09/07/2004 |
| 6787535 | Indole derivatives with 5HT6 receptor affinity This invention relates to compounds which have generally 5-HT6 receptor affinity and which are represented by Formula I: wherein one of R5, R6 or R7 is a group of general Formula B, where... | 09/07/2004 |
| 6774242 | Method for arylating aza-heterocycles with activated aromatic compounds in the presence of caesium carbonate The invention concerns a process for the preparation of N-aryl-aza-heterocycles of the general formula I by reaction of aza-heterocycles with activated aryl halides with use of caesium carbonate without addition of furth... | 08/10/2004 |
| 6740128 | Agent for coloring fibers The object of the invention is a preparation for dyeing fibers, especially hair, which is prepared before use by mixing an acidic component (A1), containing at least an enamine of formula (I) or its acid addition salt of Formula (Ia) | 05/25/2004 |
| 6673797 | Heterocyclic indole derivatives and mono- or diazaindole derivatives There is provided a compound represented by the ##STR1## general formula (1): wherein Het represents an optionally substituted heterocyclic group; A1 and A2 each independently represent --CH.dbd., etc.; A3 represents -... | 01/06/2004 |
| 6669739 | Agent for coloring fibers and method for temporarily coloring fibers The object of the present invention is a preparation for coloring fibers, which is prepared before use by mixing an acidic component (A1), containing at least one enamine of Formula (I)/(Ia) with a component (A2), containing a Schiff's base of Formula (II... | 12/30/2003 |
| 6620824 | Process for the synthesis of gonadotropin releasing hormone antagonists The present invention relates to a process for preparing a compound of gonadotropin releasing hormone antagonists having a Formula I, ##STR1## in an efficient way, which involves preparation of key intermediates: 2-arylindole core; a chiral aziridine, in ... | 09/16/2003 |
| 6605634 | Aryl and heteroaryl substituted fused pyrrole anti-inflammatory agents The present invention comprises a new class of novel aryl and heteroaryl substituted fused pyrrole compounds useful for the prophylaxis and treatment of diseases or conditions, such as TNF-, IL-1ଲ, IL-6 and/or IL-8 mediated diseases, and othe... | 08/12/2003 |
| 6525083 | N-substituted indoles useful in the treatment of diabetes Certain N-substituted indoles having aryloxyacetic acid, substituents are agonists or partial agonists of PPAR gamma, and are useful in the treatment, control or prevention of non-insulin dependent diabetes mellitus (NIDDM), hyperglycemia, dyslipidemia, h... | 02/25/2003 |
| 6506758 | Indole derivatives useful A.O. for the treatment of osteoporosis A compound of formula (I): ##STR1## or a salt thereof, or a solvate thereof, wherein: A represents an optionally substituted aryl group or an optionally substituted heterocyclyl group; Ra represents --CO--NRs Rt wherein Rs... | 01/14/2003 |
| 6495546 | Propanolamine derivatives Propanolamine derivatives represented by the following formula (I): ##STR1## These derivatives may be 댣 agonists and exert sympathomimetic, anti-ulcerous, anti-pancreatitis, lipolytic and anti-urinary incontinence and anti-pollakiuria ac... | 12/17/2002 |
| 6479480 | Phenylindole derivatives as 5-ht2a receptor ligands Compounds according to Formula (I) or a salt thereof are selective antagonists of the human 5-HT2A receptor useful for treatment of adverse conditions of the central nervous system: ##STR1##... | 11/12/2002 |
| 6458966 | Dye intermediate and method Various classes of dyes are provided having acid, ester or amide groups for covalent linking to biomolecules. The dyes may be prepared by use of a compound of formula (I) ##STR1## where R1 comprises a linker and a carboxy including acid, salt, ... | 10/01/2002 |
| 6252042 | Compounds for detecting phosphoric acid esters Complexes, especially for the detection and separation of phosphoric-ester-containing compounds, are disclosed. The complexes according to the invention comprise at least one chelating agent, at least one central atom or central ion coordinated by the che... | 06/26/2001 |
| 6242609 | Method for manufacturing a color coupler used in a silver halide photographic light-sensitive material A method for manufacturing a color coupler used in a silver halide photographic light-sensitive material using an ammonium trihalide. Said method for manufacturing the color coupler comprising the following step: a step for halogenating a coupling position of ... | 06/05/2001 |
| 6218419 | Aminoiminoquinone and aminoquinone alkaloid compounds and methods of use The subject application concerns novel compounds with useful biological properties. For example, these compounds can be used as antinflammatory, anti-proliferative, immunomodulatory, and/or neuroprotective agents. Specific examples of the compounds of the... | 04/17/2001 |
| 6180643 | Aryl and heteroaryl substituted fused pyrrole antiinflammatory agents The present invention comprises a new class of novel aryl and heteroaryl substituted fused pyrrole compounds useful for the prophylaxis and treatment of diseases or conditions, such as TNF-, IL-1ଲ, IL-6 and/or IL-8 mediated diseases, and othe... | 01/30/2001 |
| 6169206 | 4-(n,n-dialkylamino)aniline compound, photographic processing composition containing the same and color image-forming method 4-(N,N-Dialkylamino)aniline compounds of the following general formula (I): ##STR1## wherein R1 represents an alkyl group, an aryl group or a heterocyclic group, R2 to R5 each represent a hydrogen atom or a substituent, an... | 01/02/2001 |
| 6133305 | 3-(substituted)-2-indolinones compounds and use thereof as inhibitors of protein kinase activity The present invention relates to novel 3-(substituted)-2-indolinones compounds and physiologically acceptable salts and prodrugs thereof which modulate the activity of protein kinases and therefore are expected to be useful in the prevention and treatment... | 10/17/2000 |
| 6110957 | Synthetic methods for the preparation of indolylquinones and mono- and bis-indolylquinones prepared therefrom The present invention relates to novel synthetic methods for the preparation of indolylquinones. The methods of the present invention are directed to synthetic reactions involving indoles and halo-quinones in solvent and in the presence of a metal carbona... | 08/29/2000 |
| 6090839 | Antidiabetic agents The instant invention is concerned with aryl and heteroaryl oxyacetic acid type compounds which are useful antidiabetic compounds. Compositions and methods for the use of the compounds in the treatment of diabetes and related diseases and for lowering tri... | 07/18/2000 |
| 5985910 | 3- [4- (2- Phenyl-Indole-1-ylmethyl) Phenyl]- Acrylamides as estrogenic agents The present invention relates to new 3-[4-(2-Phenyl-Indole-1-ylmethyl)-Phenyl]-Acrylamide compounds which are useful as estrogenic agents, as well as pharmaceutical compositions and methods of treatment utilizing these compounds, the compounds having the ... | 11/16/1999 |
| 5932725 | Chromene compound The present invention relates to a novel chromene compound having favorable photochromic properties, developing a color of a high density, exhibiting a small degree of initial color and permitting the color to quickly fade. The novel chromene compound has... | 08/03/1999 |
| 5932743 | Methods for the solid phase synthesis of substituted indole compounds The present invention relates to novel substituted indole compounds of formula (I) ##STR1## having pharmacological activity, to processes for their preparation, to solid phase methods for preparing libraries of the compounds, to utilizing librar... | 08/03/1999 |
| 5919947 | Traceless solid phase synthesis of indole derivatives The present invention relates to a traceless solid phase process for the preparation of an indole derivative, which comprises the following steps: (1) reaction of an optionally substituted 2-iodoaniline derivative via the nitrogen atom of the NH2 mo... | 07/06/1999 |
| 5886191 | Amidinoindoles, amidinoazoles, and analogs thereof The present application describes amidinoindoles, amidinoazoles, and analogs thereof of formula I: ##STR1## wherein W, W1, W2, and W3 are selected from CH and N, provided that one of W1 and W2 is... | 03/23/1999 |
