U.S. patents available from 1976 to present.
U.S. patent applications available from 2005 to present.

Icon_funbox Quotables

"Transmission of documents via telephone wires is possible in principle, but the apparatus required is so expensive that it will never become a practical proposition."

Dennis Gabor, British physicist

Newsletter  PatentStorm News

Make the Most of Our Site

See this month's Top Inventors and Most Cited Patents.

Stay on top of the latest innovations by subscribing to an RSS feed.

Registered users: Manage your profile.

 

Class 548/475 - Chalcogen or nitrogen attached directly to the ring nitrogen of the five membered hetero ring by nonionic bonding


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the ring nitrogen of the five-membered
No. of patents: 99
Last issue date: 09/09/2008


1      
NumberTitleIssue Date
7423155N-sulfonyldicarboximide containing tethering compounds
Compounds having two reactive functional groups are described that can be used as a tethering compound to immobilize an amine-containing material to a substrate. The first reactive functional group can be used to provide attachment to a surface of a substrate. The s...
09/09/2008
7402678Multifunctional amine capture agents
Multifunctional compounds having acylsulfonamide amine-reactive groups are described that can be used for the capture of amine containing materials. ...
07/22/2008
7351838N-sulfonyldicarboximide containing tethering compounds
Compounds having two reactive functional groups are described that can be used as a tethering compound to immobilize an amine-containing material to a substrate. The first reactive functional group can be used to provide attachment to a surface of a substrate. The s...
04/01/2008
7208566Imide-linked maleimide and polymaleimide compounds
The invention is based on the discovery that a remarkable improvement in the performance of maleimide thermosets can be achieved through the incorporation of imide-extended mono-, bis-, or polymaleimide compounds. These imide-extended maleimide compounds are readily...
04/24/2007
7015356Process for producing dicarboxylic acids
A carboxylic acid is produced by oxidative cleavage of a cycloalkane with oxygen and performs a reaction in the presence of a catalyst including an imide compound and a metallic compound, the imide compound having a cyclic imide skeleton represented by the following...
03/21/2006
6964976Amino alcohol derivatives
Compounds of formula (I) which exhibit excellent immune suppression activity, pharmacologically acceptable salts thereof, esters thereof or other derivatives: wherein R1 and R2 are a hydrogen atom...
11/15/2005
6410748Alicycli c group-containing monomer
A monomer represented by the following general formula (m-1): ##STR1## wherein R is a group having an alicyclic skeleton, R2 s may be the same or different and are individually hydrogen atom, halogen atom or monovalent organic group, X1
06/25/2002
6262302N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting ଲ-amyloid peptide release and/or its synthesis by use of such compounds
Disclosed are compounds which inhibit ଲ-amyloid peptide release and/or its synthesis, and, accordingly, have utility in treating Alzheimer's disease. Also disclosed pharmaceutical compositions comprising a compound which inhibits ଲ-amyloid pep...
07/17/2001
6232258Oxygenation catalyst and process for producing a ketone using the same
A substrate is contacted with oxygen in the presence of the imide compound shown by the following formula (1) (N-hydroxyphthalimide) and a strong acid, or the imide compound, the strong acid and a co-catalyst (e.g., a transition metal compound) to oxygena...
05/15/2001
6160128Tritioacetylating reagents and processes for preparation thereof
Novel acetylating and tritioacetylating reagents suitable for preparation of nonlabelled and radiolabelled organic compounds. N-acetoxynaphthalimide, N-tritioacetoxyphthalimide, N-tritioacetoxysuccinimide, N-tritioacetoxynaphthalimide and processes of ...
12/12/2000
6153652N-(aryl/heteroaryl/alkylacetyl) amino acid amides, pharmaceutical compositions comprising same, and methods for inhibiting ଲ-amyloid peptide release and/or its synthesis by use of such compounds
Disclosed are compounds which inhibit ଲ-amyloid peptide release and/or its synthesis, and, accordingly, have utility in treating Alzheimer's disease. Also disclosed pharmaceutical compositions comprising a compound which inhibits ଲ-amyloid pep...
11/28/2000
5977182O-benzyl oxime ether derivatives and their use as pesticides
Compounds of formula (I), wherein Y is hydrogen, C1 -C4 alkyl, C1 -C4 alkoxy, OH, CN, NO2, Si(CH3)3, CF3 or halogen, and T is a group (a) or (b), and wherein the remaining ...
11/02/1999
5929217Reactive dyes with a benzo-fused heterocycle as anchor
Reactive dyes of the formula I ##STR1## where a is 1 or 2, b is 0 or 1, Z1 is hydrogen, C1 -C6 -alkyl, C1 -C6 -alkoxy, halogen, nitro, amino, hydroxysulfonyl, C1 -C6 -alkoxycarbo...
07/27/1999
5919790Hydroxamate inhibitors of interleukin-1ଲ converting enzyme
The present invention relates to compounds that are inhibitors of interleukin-1ଲ converting enzyme that have the Formula II ##STR1## This invention also relates to a method of treatment of stroke, inflammatory diseases, septic shock, reperfusio...
07/06/1999
5872191Process for producing a polyoxyalkylene derivatives substituted with succinimidyl group
A process for producing a polyoxyalkylene derivative substituted with succinimidyl group which comprises reacting a polyoxyalkylene compound having carboxyl group at ends with N-hydroxysuccinimide in an inert solvent in the presence of dicyclohexylcarbodi...
02/16/1999
5763617Cephalosporins
A syn isomer in (R) or (S) form or a mixture thereof of a compound of the formula ##STR1## syn isomer, in the (R) or (S) form or in the form of an (R,S) mixture, in the form of an integral salt or their salts with organic or mineral acids wherei...
06/09/1998
5760165Bisallyloxyimides
Monoallyloxyimides, diallyloxyimides and polyallyloxyimides of general Formula I. ##STR1## wherein: X is an integer from 1 to 4 inclusive; R1, R2, and R3 are independently selected from the group comprising hydrogen, ...
06/02/1998
5719294Process for preparing N-cyclohexylthiophthalimide
The preparation of N-cyclohexylthiophthalimide from cyclohexylsulphenyl chloride and phthalimide can be reproduced more reliably if the cyclohexylsulphenyl chloride is prepared in sire by chlorinating dicyclohexyl disulphide....
02/17/1998
5663336Substituted diaminophthalimides and analogues
A process for the synthesis of compounds of formula I ##STR1## wherein Ar1, Ar2, A1, A2, R and X are as defined in the description, exhibit valuable pharmaceutical properties and are effective especially ag...
09/02/1997
5656654Arylidene and heteroarylidene oxindole derivatives and process for their preparation
Arylidene and heteroarylidene oxindole derivatives of formula (I) ##STR1## wherein, subject to provisos, Y is a bicyclic ring system chosen from naphthalene, tetralin, quinoline and isoquinoline; R is hydrogen or an oxo (.dbd.O) group when Y is tetralin; ...
08/12/1997
5650234Electrophilic polyethylene oxides for the modification of polysaccharides, polypeptides (proteins) and surfaces
Several poly(ethylene glycol) mixed carbonates and their preparation are closed. These carbonates are synthesized by conversion of polyethylene glycol first to the chloroformate then by reaction with the hydroxyl group of N-hydroxybenzotriazole or 2-hydr...
07/22/1997
5646300(1H-indol-1-yl)-2-(amino)acetamides and related (1H-indol-1-yl)-(aminoalkyl)amides, pharmaceutical composition and use
There are disclosed neuroprotective compounds having the formula ##STR1## wherein the moieties are defined in the specification, and processes for making them....
07/08/1997
5637702Sulfur compounds
Sulfur compounds of the formula ##STR1## where n is 0 or 2, R1 and R2 are hydrogen, C1 -C6 -alkyl, C1 -C6 -alkoxy, halogen, nitro, amino, hydroxysulfonyl, C1 -C6 ...
06/10/1997
5616726Optically active aminoalcohol derivatives and method of producing same
An object of the present invention is to provide a safe method of commercially producing optically active aminoalcohol derivatives, which serve as intermediates for the synthesis of medicinal chemicals such as the immunopotentiating anticancer agent besta...
04/01/1997
5612460Active carbonates of polyalkylene oxides for modification of polypeptides
Poly(ethylene glycol)-N-succinimide carbonate and its preparation are disclosed. Polyethylene glycol (PEG) is converted into its N-succinimide carbonate derivative. This form of the polymer reacts readily with amino groups of proteins in aqueous buffers. ...
03/18/1997
5580987Process for preparing 1-aminoacetamidopyrroles
There is disclosed a process for the preparation of 1-aminoacetamidopyrroles and 1-amino-2-(substituted)-pyrroles and related compounds of the formula ##STR1## wherein all substituents are defined herein, which are useful as glycine partial agon...
12/03/1996
5534533Carboxylate derivatives exhibiting phospholipase A2 inhibitory activity
Novel carboxylate derivatives exhibiting phospholipase A2 inhibitory activity are disclosed, Specifically, the following compounds of the formula and pharmaceutically acceptable salts thereof are disclosed: ##STR1## wherein A is hydroxy, a...
07/09/1996
5508412Phthalimides useful as intermediate compounds
Unsaturated cyclohexenone oxime ethers I ##STR1## (Q.dbd.H, alkylcarbonyl, benzoyl, alkali metal or alkaline earth metal ion, substituted or unsubstituted ammonium ion, phosphonium ion, sulfonium ion, sulfoxonium ion, an equivalent of a transition me...
04/16/1996
5491232Sulfur compounds useful for preparation of dyes
Sulfur compounds of the formula ##STR1## where n is 0 or 2, R1 and R2 are hydrogen, C1 -C6 -alkyl, C1 -C6 -alkoxy, halogen, nitro, amino, hydroxysulfonyl, C1 -C6 ...
02/13/1996
5491144Substituted diaminophthalimides and analogues
Compounds of formula I ##STR1## wherein Ar1, Ar2, A1, A2, R and X are as defined in the description, exhibit valuable pharmaceutical properties and are effective especially against diseases responsive to th...
02/13/1996
5414089Long chain carboxylic acid imide ester
Provided is a long chain carboxylic acid imide ester (I) represented by the following general formula (I) ##STR1## wherein W is a divalent long chain hydrocarbon group which may optionally be interrupted by one or more groups each independently selec...
05/09/1995
5346879Plant growth regulator containing a phthalimide derivative
Plant growth regulators comprising, as an active ingredient, a substituted dicarboxylic acid derivative having the formula: ##STR1## wherein R1, R2, R3 and R4 are the same as defined in the present specific...
09/13/1994
5324844Active carbonates of polyalkylene oxides for modification of polypeptides
Poly(ethylene glycol)-N-succinimide carbonate and its preparation are disclosed. Polyethylene glycol (PEG) is converted into its N-succinimide carbonate derivative. This form of the polymer reacts readily with amino groups of proteins in aqueous buffers. ...
06/28/1994
5304655N'-substituted N-amino-3,4,5,6-tetrafluorophthalimides, and processes for their preparation
Compounds of the formula ##STR1## in which X is the radical ##STR2## where R1 and R2 are in each case a hydrogen atom, an alkyl-(C1 -C10) group, aryl group, alkyl(C1 -C6)-CO ...
04/19/1994
5292759O-benzyloxime ethers and crop protection agents containing these compounds
O-Benzyloxime ethers of the formula I ##STR1## where 5 X is substituted or unsubstituted CH2, NOalkyl Y is O, S, NR5 R1, R2, R5 are H, alkyl Z1, Z2 are H, halogen, methyl, methoxy, cy...
03/08/1994
5288749Tertiary and secondary amines as alpha-2 antagonists and serotonin uptake inhibitors
The present invention provides tertiary and secondary amine compounds of the formula ##STR1## and the pharmaceutically acceptable salts thereof which are antagonists for alpha-2 adrenoreceptors and which inhibit serotonin (5-hydroxytryptamine, 5...
02/22/1994
5281617N-succinimidyl and N-phthalimidyl esters of 2-phenylalkanoic acid derivatives as inhibitors of human leukocyte elastase
N-succinimidyl and N-phthalimidyl esters of phenylalkanoic acid derivatives which are useful as inhibitors of HLE or HNE....
01/25/1994
5274115N'-substituted N-amino-3,4,5,6-tetrafluorophthalimides
Compounds of the formula ##STR1## in which X is the radical ##STR2## where R1 and R2 are in each case a hydrogen atom, an alkyl-(C1 -C10) group, aryl group, alkyl(C1 -C6)-CO ...
12/28/1993
5252689N-hydroxysuccinimide-blocked isopropenyl-alpha, alpha-dimethylbenzyl isocyanate and self-cross linking copolymers thereof
A novel, one component self-crosslinking resin and a process for its preparation are provided. The resin is the copolymer of: (I) N-hydroxysuccinimide-blocked meta-isopropenylalpha, alpha-dimethylbenzyl isocyanate; (II) a hydroxy group-containing ethylenically...
10/12/1993
5238950Inhibitors of platelet-derived growth factor
A method of inhibiting the binding of PDGF using compounds of the formula I ##STR1## useful in the treatment of atherosclerosis, cancer, retinal detachment, pulmonary fibrosis, arthritis, psoriasis and glomerulonephritis, and restenosis following ang...
08/24/1993
1      
 
Sign InRegister
Username  
Password   
forgot password?