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| Number | Title | Issue Date |
| 7745639 | Mitotic kinesin inhibitors The present invention relates to dihydropyrazole compounds that are useful for treating cellular proliferative diseases, for treating disorders associated with KSP kinesin activity, and for inhibiting KSP kinesin. The invention also related to compositions which com... | 06/29/2010 |
| 7705161 | Process for producing nitrogenous 5-membered cyclic compound A method of the intramolecular and intermolecular cyclization of an N-acylhydrazone for obtaining a pyrazoline skeleton or pyrazolidine skeleton under ordinary conditions with high stereoselectivity and in high yield. An N-acylhydrazone represented by the following ... | 04/27/2010 |
| 7482470 | Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes The present invention provides novel pyrazoles that are useful as cannabinoid receptor antagonists and pharmaceutical compositions thereof and methods of using the same for treating obesity, diabetes, and/or cardiometabolic disorders. ... | 01/27/2009 |
| 7465809 | Heterocycle derivatives useful as selective androgen receptor modulators (SARMs) The present invention is directed to novel heterocycle derivatives, pharmaceutical compositions containing them and their use in the treatment of disorders and conditions modulated by the androgen receptor. ... | 12/16/2008 |
| 7407972 | Inhibitors of factor Xa and other serine proteases involved in the coagulation cascade The present invention provides compounds of Formula (I): wherein A, B, C, G, and W1 have any of the values defined in the specification, and pharmaceutically acceptable salt thereof, that are useful to treat thro... | 08/05/2008 |
| 7320995 | Benzimidazoles and benzothiazoles as inhibitors of map kinase The present invention provides kinase inhibitors of Formula I: wherein W represents inter alia imidazol, oxazol, pyrazol, thiazol as triazol, which are substituted by phenyl or thienyl. The disclosed compounds inhibit p-38 kinase and are useful in the treatment of m... | 01/22/2008 |
| 7262223 | Amidine derivatives for treating amyloidosis The present invention relates to the use of amidine compounds in the treatment of amyloid-related diseases. In particular, the invention relates to a method of treating or preventing an amyloid-related disease in a subject comprising administering to the subject a t... | 08/28/2007 |
| 7122571 | Substituted hydrazones as inhibitors of cyclooxygenase-2 Compounds useful as inhibitors of cyclooxygenase-2 activity have the formulae I or Ia: wherein: Q1, Q2, n, m, X, Y and R are as defined herein. | 10/17/2006 |
| RE38963 | Pyrazoline derivatives, their preparation and application as medicaments The present invention relates to new pyazoline derivatives of formula and to physiologically acceptable salts thereof, to the method for their preparation and to their application as medicaments. ... | 01/31/2006 |
| 6974810 | 4,5-Dihydro-1H-pyrazole derivatives having potent CB1-antagonistic activity The present invention relates to a group of novel 4,5-dihydro-1H-pyrazole derivatives which are potent cannabinoid (CB1) receptor antagonists with utility for the treatment of diseases connected with disorders of the cannabinoid system. The compounds have... | 12/13/2005 |
| 6965032 | Substituted dihydro 3-halo-1h-pyrazole-5-carboxylates and their preparation and use This invention relates to a compound of Formula I, a method for its preparation and its use in the preparation of a compound of Formula II wherein R1, R2, R3, X and n are as defined in the disclosure. This invention also discloses pr... | 11/15/2005 |
| 6958403 | Procedure for the preparation of racemic and enantiomerically pure derivatives of 1,5 diaryl-3-trifluorromethyl-Δ-pyrazolines Procedure for preparation of compounds with the general formula 1, which include the racemic mixtures (±)-1, and the enantiomerically pure compounds (−)-1 and (+)-1, wherein R1 and R3, like or different, represent an atom of hydrogen, chlori... | 10/25/2005 |
| 6852750 | Benzenedicarboxylic acid derivatives New benzenedicarboxylic acid derivative compounds; pharmaceutical compositions, diagnostic methods, and diagnostic kits that include those compounds; and methods of using those compounds for inhibiting NAALADase enzyme activity, detecting diseases where NAALADase le... | 02/08/2005 |
| 6846935 | Procedure for the preparation of racemic and enantionmerically pure derivatives of 1,5-diaryl-3-trifluoromethyl-Δ2-pyrazolines Procedure for preparation of compounds with the general formula 1, which include the racemic mixtures (±)-1, and the enantiomeric ally pure compounds (−)-1 and (+)-1, wherein R1 and R3, like or different, represent an atom of hydrogen, chlor... | 01/25/2005 |
| 6573287 | 2,1-oxazoline and 1,2-pyrazoline-based inhibitors of dipeptidyl peptidase IV and method Dipeptidyl peptidase IV (DP 4) inhibiting compounds are provided having the formula ##STR1## where n is 0 or 1; X is H or CN; Y is N, NH or O; Z is CH2 when Y is O or N--H, with Y--Z forming a single bond, and Z is CH when Y is N, with Y--Z for... | 06/03/2003 |
| 6476060 | 4,5-dihydro-1H-pyrazole derivatives having CB1-antagonistic activity The present invention relates, among many things, to novel 4,5-dihydro-1H-pyrazole compounds which can be potent antagonists of the cannabis CB1 -receptor. The compounds have the formula (I) ##STR1## wherein R and R1 are the same or ... | 11/05/2002 |
| 6353117 | Pyrazoline derivatives, their preparation and application as medicaments The present invention relates to new pyazoline derivatives of formula ##STR1## and to physiologically acceptable salts thereof, to the method for their preparation and to their application as medicaments.... | 03/05/2002 |
| 6242609 | Method for manufacturing a color coupler used in a silver halide photographic light-sensitive material A method for manufacturing a color coupler used in a silver halide photographic light-sensitive material using an ammonium trihalide. Said method for manufacturing the color coupler comprising the following step: a step for halogenating a coupling position of ... | 06/05/2001 |
| 6184243 | N-linked ureas and carbamates of heterocyclic thioesters This invention relates to neurotrophic low molecular weight, small molecule N-linked ureas and carbamates of heterocyclic thioesters having an affinity for FKBP-type immunophilins, and their use as inhibitors of the enzyme activity associated with immunop... | 02/06/2001 |
| 6004903 | 2-Anylocyclohexanediones having improved herbicidal properties Benzoyl derivatives of the formula I ##STR1## where Z is a 5-membered or 6-membered heterocyclic, saturated or unsaturated radical containing one to three hetero atoms selected from the group consisting of oxygen, sulfur and nitrogen, Q is a cyclohex... | 12/21/1999 |
| 5908938 | Process for the preparation of 1-phenylpyrazoline-3-carboxylic acid derivatives There is described a process for the preparation of 1-phenylpyrazoline-3-carboxylic acid derivatives of the formula III by means of base-catalyzed reaction of hydrazones of the formula I with olefins of the formula II ##STR1## where Ph, R1 | 06/01/1999 |
| 5886015 | Benzyloxy substituted aromatics and their use as fungicides and insecticides Compounds with fungicidal and insecticidal properties having formula ##STR1## wherein A is N or CH; V is O or NH; m and n are independently 0 and 1 provided that m+n is not 2, and U and W are independently O or N; such that when U and W are both N and n i... | 03/23/1999 |
| 5849732 | Phenol compound having antioxidative activity and the process for preparing the same Disclosed are a phenol compound represented by the formula (1): ##STR1## wherein R0 represents H, alkyl or alkyloxy; R1 represents alkyl; R2 represents alkyl or alkyloxy; OR3 represents OH; R4 re... | 12/15/1998 |
| 5750690 | Asymmetric hydrogenation process using ruthenium-diphosphine complexe A process for the asymmetric hydrogenation of a compound of the formula ##STR1## wherein each R, independently, is alkyl, arylmethyl, aryl, alkoxy, arylmethoxy or aryloxy or both R's, taken together, are methylene, ethylene or 1,2-phenylene and n is ... | 05/12/1998 |
| 5728839 | Metal complexes with heterocycles carbenes A complex of the formula La Mb Xc !n (A)n I as described in the application useful as homogenous catalysts.... | 03/17/1998 |
| 5670456 | Compounds N-carbamoyl-2-carboxyaryl-heterocyclic and hydrazinecarboximidamidehydrazone derivatives, intermediates and processes for their preparation, agricultural compositions containing them and their use as agricultural chemicals, in particular herbicides.... | 09/23/1997 |
| 5641783 | Substituted amino alcohol compounds Disclosed are compounds having a straight or branched aliphatic hydrocarbon structure of formula I: ##STR1## In formula I, n is an integer from one to four and m is an integer from four to twenty. Independently, R1 and R2 are hy... | 06/24/1997 |
| 5591764 | N-acylated pyrazolines N-sulfenylated and N-acylated pyrazoline arthropodicides, compositions containing them and methods for controlling arthropods by applying compounds of the invention to them or to their environment. The pyrazolines are selected from those of Formulae I to ... | 01/07/1997 |
| 5543433 | Azine-substituted phenylacetic acid derivatives and fungicides containing these Compounds of the formula I ##STR1## where X is hydrogen, halogen, alkyl, alkoxy, trifluoromethyl, cyano or nitro, Y is an amino, methylamino or dimethylamino group, Z is a group CHCH3, CHOCH3 or NOCH3, R is hydrogen or alk... | 08/06/1996 |
| 5506191 | Heterocyclic hydrazines and hydrazones N-carbamoyl-2-carboxyaryl-heterocyclic and hydrazinecarboximidamide-hydrazone derivatives, intermediates and processes for their preparation, agricultural compositions containing them and their use as agricultural chemicals, in particular herbicides.... | 04/09/1996 |
| 5491162 | N-acylated pyrazolines, compositions and use N-sulfenylated and N-acylated pyrazoline arthropodicides, compositions containing them and methods for controlling arthropods by applying compounds of the invention to them or to their environment. The pyrazolines are selected from those of Formulae I to ... | 02/13/1996 |
| 5472984 | 1,2-ethanediol derivative and salt thereof and cerebral function-improving agent comprising the same This invention relates to a 1,2-ethanediol derivative and a salt thereof, a process for producing the same, and a cerebral function-improving agent comprising the same. The cerebral function-improving agent of this invention is useful for treating cerebro... | 12/05/1995 |
| 5232615 | Heterocyclic nitrogen compound Mannich base derivatives of polyolefin-substituted amines for oleaginous compositions The novel polymers of the present invention are prepared by reacting a heterocyclic nitrogen compound containing at least one --N(H)-- group in the ring, an aldehyde N-containing polymer adduct (e.g., an ashless nitrogen-containing dispersant or polyolefi... | 08/03/1993 |
| 5208251 | Styryl pyrazoles, isoxazoles and analogs thereof having activity as 5-lipoxygenase inhibitors, pharmaceutical compositions and methods of use therefor The present invention is 3,5-substituted, isoxazoles, pyrazoles, isothiazoles, and analogs thereof having 5-lipoxygenase or cyclooxygenase inhibiting activity or as a sunscreen.... | 05/04/1993 |
| 5187290 | Acylaminoalkanoyl urethanes or thiourethanes Compounds of the formula ##STR1## wherein Z is oxygen or sulfur are disclosed. These compounds are useful as hypotensive agents due to their angiotensin converting enzyme inbitition activity and depending upon the definition of X may also be useful a... | 02/16/1993 |
| 5153358 | Process for the preparation of alpha-alkylated alpha-amino acids and alpha-halogenated alpha-amino acids A novel process for the preparation of -alkylated -amino acids and -halogenated -amino acids is disclosed. These -alkylated -amino acids and -halogenated -amino acids are useful as intermediates for ... | 10/06/1992 |
| 5152824 | Sulfamidosulfonamide derivatives and herbicides A sulfamidosulfonamide derivative of the formula (1) and an agriculturally suitable salt thereof: ##STR1## wherein Q is ##STR2## X is an oxygen atom or a sulfur atom; and G is ##STR3## which are useful as herbicide.... | 10/06/1992 |
| 5103007 | Lipids Lipid derivatives represented by the formula: ##STR1## wherein R1 stands for an optionally substituted higher alkyl group, R2 stands for an optionally substituted lower alkyl group or an optionally substituted nitrogen-containin... | 04/07/1992 |
| 5091405 | Insecticidal pyrazolines Pyrazolines and their intermediates, including all geometric and stereoisomers of the pyrazolines and intermediates, agricultural compositions containing the pyrazolines, and methods for use as insecticides.... | 02/25/1992 |
| 5068241 | Pesticidal substituted pyrazoline derivatives, compositions and use Pesticidal substituted pyrazoline derivatives of the formula ##STR1## in which R1 represents optionally substituted phenyl or optionally substituted alkyl, R2 represents hydrogen, optionally substituted phenyl, optionally substi... | 11/26/1991 |
