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| Number | Title | Issue Date |
| 8188295 | Method for producing difluoromethyl-substituted pyrazole compounds The present invention relates to a process for preparing 3-difluoromethyl-Substituted pyrazole compounds of the formula (I) in which R1 is H, halogen, nitro, C1-C8-alkyl, C1-C | 05/29/2012 |
| 8134012 | Synergistic fungicidal active compound combinations The novel active compound combinations comprising a carboxamide of the general formula (I) (group 1) in which A, R1 and R2 are as defined in the description, and the active... | 03/13/2012 |
| 8124787 | Process for the production of pyrazoles A process for the production of a compound of formula (I), which comprises a) reacting a compound of formula (II), wherein R1 and R2 are both independently C1-C6 alkyl, with methylhydrazine in the presence of water and a w... | 02/28/2012 |
| 8124786 | Mental-catalyzed process for preparation of substituted pyrazolecarboxamides The present invention provides a metal-catalyzed process for preparation of substituted pyrazolecarboxamides of formula (I) as fungicidally active compounds from 2-alkylhaloaromatics and heterocyclylamides. ... | 02/28/2012 |
| 8115012 | Process for preparing difluoromethylpyrazolyl carboxylates The present invention relates to a process for preparing difluoromethyl-substituted pyrazol-4-ylcarboxylates of the formula I in which R1 is C1-C8-alkyl, C... | 02/14/2012 |
| 8101780 | Crystalline form of 3-(difluormethyl)-1-methyl-N-(3′,4′,5′-trifluor[1,1′-biphenyl]-2-yl)-1H-pyrazol-4-carboxamide The present invention relates to a new crystalline form of 3-(Difluormethyl)-1-methyl-N-(3′,4′,5′-trifluor[1,1′-biphenyl]-2-yl)-1H-pyrazol-4-carboxamide. The invention also relates to processes for the production of this crystalline form and formulations for... | 01/24/2012 |
| 7977494 | Method for producing substituted pyrazolecarboxylic acid chlorides The present invention relates to a process for preparing substituted pyrazolyl chlorides by chlorinating aldehydes of the formula (II) under free-radical conditions. ... | 07/12/2011 |
| 7968729 | 1-phenyl-1H-pyrazole-based compounds Methods useful for preparing compounds of formula I: and salts thereof are disclosed. Also disclosed are intermediates useful in the preparation of such compounds. ... | 06/28/2011 |
| 7968728 | Method for producing carboxamides The present invention relates to a novel process for preparing known fungicidally active 1,3-dimethyl-5-fluoro-1H-pyrazole-4-carboxamides from the corresponding acid fluoride and aniline derivatives in the presence of alkylpyridine derivatives as an acid acceptor. | 06/28/2011 |
| 7939673 | Process for preparing 3-dihalomethyl-pyrazole-4-carboxylic acid derivatives The invention relates to a process for preparing 3-dihalomethylpyrazole-4-carboxylic acid derivatives of the formula (I) by reacting α-fluoroamines of the formula (III) in the presence of Lewis acids with acrylic acid derivatives of the formula (II) to give vinamid... | 05/10/2011 |
| 7919632 | Method for producing carboxamides The present invention relates to a novel process for preparing known fungicidally active 1,3-dimethyl-5-fluoro-1H-pyrazole-4-carboxamides from the corresponding acid fluoride and aniline derivatives in the absence of an acid acceptor. ... | 04/05/2011 |
| 7906656 | Iodopyrazolyl carboxanilides This invention relates to novel intermediates used in the preparation of iodopyrazolylcarboxanilides of the formula (I) in which R1, R2, R3, R4, R5, R6 and Z... | 03/15/2011 |
| 7872146 | Process for the preparation of a carboxamide derivative Process for the preparation of a carboxamide derivative of formula (I) or a salt thereof Intermediates for preparing this compound are also provided. ... | 01/18/2011 |
| 7863460 | Process for producing 1-substituted-3-fluoroalkylpyrazole-4-carboxylate In a process for producing 1-substituted-3-fluoroalkyl-pyrazole-4-carboxylate (3) by a reaction of 2-alkoxymethylenefluoroacylacetate (1) and hydrazine (2), the reaction is conducted in the presence of a base and water, to produce 1-substituted-3-fluoroalkylpyrazole... | 01/04/2011 |
| 7820830 | Process for the production of carboxanilides The present invention relates to a novel process for the preparation of a compound of general formula (I): wherein R1 is H or C1-4 alkyl and R2 is difluoromethyl or trifluoromethyl, which comprises reacting a compound of general form... | 10/26/2010 |
| 7714144 | Method for the production of 5-fluoro-1,3-dialkyl-1H-pyrazol-4-carbonyl fluorides The present invention relates to a novel process for preparing known 5-fluoro-1,3-dialkyl-1H-pyrazole-4-carbonyl fluorides which can be used as starting materials for active fungicidal ingredients by a halex reaction. ... | 05/11/2010 |
| 7678924 | Process for the preparation of pyrazoles The present invention relates to a process for the preparation of compounds of formula I wherein R1 is C1-C4haloalkyl; R2 is C1-C6alkyl and R3 is ... | 03/16/2010 |
| 7659408 | Pyrazole carboxamides as inhibitors of 11-β-hydroxysteroid dehydrogenase-1 Pyrazole carboxamides of structural formula I are selective inhibitors of the 11β-hydroxysteroid dehydrogenase-1. The compounds are useful for the treatment of diabetes, such as noninsulin-dependent diabetes (NIDDM), hyperglycemia, obesity, insulin resistance, dysl... | 02/09/2010 |
| 7622595 | Substituted 1-dihydropyrazoles, their preparation and use This invention provides compounds of Formula I, methods for their preparation and use for preparing compounds of Formula II wherein R1, R2, R3, R5, R... | 11/24/2009 |
| 7605273 | Aryl-substituted pyrazole-amide compounds useful as kinase inhibitors The present invention relates to compounds having the formula, and pharmaceutically-acceptable salts, prodrugs, solvates, isomers, and/or hydrates thereof, wherein Q is an optionally-substituted phenyl, pyridyl, pyridazinyl... | 10/20/2009 |
| 7528260 | Method for preparing -phenylpyrazole-1-carboxamides A method is disclosed for preparing compounds of Formula 1 by combining compounds of Formulae 2 and 3 and a sulfonyl chloride. Also disclosed are compounds of Formula 3, which are useful as starting materials for this metho... | 05/05/2009 |
| 7504518 | Process for producing blocked isocyanate compound Disclosed is a process for producing a blocked isocyanate compound represented by general formula (III): wherein R1, R2, Q1, and Q2 are as defined in the specification, characterized by comprising reacting a pyrazole compo... | 03/17/2009 |
| 7501527 | Method for the production of fluoromethyl-substituted heterocycles The present invention relates to a process for preparing fluoromethyl-substituted heterocycles of the formula (I) in which R1, R2, R3 and A are each as defined in th... | 03/10/2009 |
| 7442801 | Pyrazole compound A pyrazole compound of formula (a): wherein R1 represents C1-C4 alkyl or trifluoromethyl, R2 represents C1-C4 alkyl, R3 represents hydrogen or C1-C6 alkyl; R4 represents halogen a... | 10/28/2008 |
| 7425640 | Substituted 5-carboxyamide pyrazoles and [1,2,4]triazoles as antiviral agents The present invention provides compounds of formula I wherein X, Y, R1-R7 are as defined herein. Compositions containing these compounds, and methods for inhibiting HCV RNA-dependent RNA polymerase and treating hepatitis C and related disorders... | 09/16/2008 |
| 7417152 | 4-bromo-5-(2-chloro-benzoylamino)-1H-pyrazole-3-carboxylic acid amide derivatives and related compounds as bradykinin Breceptor antagonists for the treatment of inflammatory diseases Disclosed are compounds of formula I and II that are bradykinin B1 receptor antagonists and are useful for treating diseases, or relieving adverse symptoms associated with disease conditions, in mammals mediated by bradykinin B1 receptor. Certa... | 08/26/2008 |
| 7378448 | Diphenylether amide derivatives as opioid receptor antagonists A compound of the formula (I) wherein the variables X1, X2, B, D, R1 to R7 including R3′, p, y, q, and z, are as defined or a pharmaceutically acceptable salt, solvate, enantiomer, racemate, diastereomer or mi... | 05/27/2008 |
| 7378409 | Substituted cycloalkylamine derivatives as modulators of chemokine receptor activity The present application describes modulators of MCP-1 of formula (I): or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma, multiple sclerosis, artherosclerosis, and rheumatoid arthritis. | 05/27/2008 |
| 7358214 | Pyrazolyl carboxanilides for controlling unwanted microorganisms This invention relates to novel pyrazolylcarboxanilides of the formula (I) in which R1, G and n are as defined in the disclosure, to a plurality of processes for preparin... | 04/15/2008 |
| 7358371 | Process for the preparation of 1,5—carboxylic acid derivatives The present invention comprises a process for the preparation of compounds that possess an affinity for the cannabinoid receptor in the human brain. These compounds are useful as immunomodulators and psychotropic agents in the treatment of thymic disorders, vomiting... | 04/15/2008 |
| 7354929 | Cannabinoid receptor ligands and uses thereof Compounds of Formula (I) that act as cannabinoid receptor ligands and their uses in the treatment of diseases linked to the mediation of the cannabinoid receptors in animals are described herein ... | 04/08/2008 |
| 7348350 | Pyrazolyl biphenyl carboxamides and the use thereof for controlling undesirable microorganisms Novel pyrazolylbiphenylcarboxamides of the formula (I) in which R1, R2, X, m, Y and n are each as defined in the description, a plurality of processe... | 03/25/2008 |
| 7345058 | Pyrazoles Provided herein are compounds of the formula (I): as well as pharmaceutically acceptable salts thereof, wherein the substituents are as those disclosed in the specification. These compounds, and the pharmaceutical compositi... | 03/18/2008 |
| 7335780 | Method for preparing 3-halo-4,5-dihydro-1H-pyrazoles This invention relates to a method for preparing 3-halo-4,5-dihydro-1H-pyrazole compound of Formula (I), comprising contacting with HX1 a different 4,5-dihydro-1H-pyrazole compound of Formula (II), wherein X1 is halogen and L, R, k and X2 ... | 02/26/2008 |
| 7329633 | Disubstituted pyrazolylcarboxanilides This invention relates to novel pyrazolylcarboxanilides of formula (I) in which R, R1, R2 and R3 are as defined in the disclosure, to a plurality of processes for preparing these ... | 02/12/2008 |
| 7319150 | Method for preparing styryl pyrazole, isoxazole and isothiazole derivatives The invention concerns a method for synthesizing styryl isoxazole, styryl pyrazole and styryl isothazole derivatives in a synthesis step followed by a recrystallization in a basic alcohol medium. ... | 01/15/2008 |
| 7304070 | Aadenosine receptor antagonists Disclosed are novel A2B adenosine receptor antagonists having the structure of Formula I or Formula II: The compounds are particularly useful for treating asthma, inflammatory gastrointestinal tract di... | 12/04/2007 |
| 7291647 | Guanylhydrazone compounds, compositions, methods of making and using The present invention relates to compounds having the formula: salts thereof; compositions comprising one or more of the compounds and/or salts thereof; methods of using; and methods of m... | 11/06/2007 |
| 7288554 | Ortho-substituted aryl amides for controlling invertebrate pests Disclosed are compounds of Formula I, their N-oxides and agriculturally suitable salts (I) wherein J is a phenyl ring, a 5- or 6-membered heteroaromatic ring or an aromatic 8-, 9- or 10-membered fused carbobicyclic or heterobicyclic ring system wherein each ring or ... | 10/30/2007 |
| 7247628 | Cannabinoid receptor ligands and uses thereof Compounds of Formula (I) that act as cannabinoid receptor ligands and their uses in the treatment diseases, conditions and/or disorders herein. ... | 07/24/2007 |
