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Patent No. 6205950

Pet Toilet-Like Water Disk and Food Storage

One pet-friendly inventor patented "a device for watering pets, e.g., a dog or cat." The device, he helpfully noted, "has the general shape of a toilet."

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Class 548/359.5 - At least three ring hetero atoms in the tricyclo ring system


Subclass of Class 548 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the tricyclo ring system contains at least
No. of patents: 51
Last issue date: 01/31/2012


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NumberTitleIssue Date
8106218Pharmaceutical compounds
Tricyclic pyrazole derivatives of the following formula (I) having affinity for the cannabinoidergic CB1 and/or CB2 receptors: wherein: A represents a group selected from one of the follow...
01/31/2012
7485730Pharmaceutical compounds
Tricyclic pyrazole derivatives of the following formula (I) having affinity for the cannabinoidergic CB1 and/or CB2 receptors: wherein: A represents a group selected from one of the follow...
02/03/2009
7425572Use of dioxindoindazoles and dioxoloindazoles for treating glaucoma
Novel dioxinoindazole compounds and dioxoloindazole compounds are disclosed. Also disclosed are methods for the lowering and controlling of normal or elevated intraocular pressure as well as a method for the treatment of glaucoma using compositions of one or more of...
09/16/2008
7320986Fused tri and tetra-cyclic pyrazole kinase inhibitors
Compounds having the formula (I) are useful for inhibiting protein kinases. Also disclosed are methods of making the compounds, compositions containing the compounds, and methods of treatment using the compounds....
01/22/2008
7291612Immunomodulatory compounds
The present invention relates to novel heterocyclic compounds, to methods for their preparation, to compositions containing them, and to methods and use for clinical treatment of medical conditions which may benefit from immunomodulation, including rheumatoid arthri...
11/06/2007
7253292Synthesis of cyclopentadiene derivatives
A process for preparing cyclopentadiene derivatives comprising the steps of: a) coupling a five membered heterocycle ring with a five or six membered heterocycle ring; b) reacting the obtained compound with a carbonilating system: c) reducing the obtained compound.
08/07/2007
7081456Immunomodulatory compounds
The present invention relates to novel heterocyclic compounds, to methods for their preparation, to compositions containing them, and to methods and use for clinical treatment of medical conditions which may benefit from immunomodulation, including rheumatoid arthri...
07/25/2006
6906080Pyrazolecarboxylic acid tricyclic derivatives, preparation and pharmaceutical compositions containing same
The subject of the invention is tricyclic derivatives of pyrazolecarboxylic acid of formula: in which R1 represents a C3-C15 carboxyl radical or an NR2R3 group. Th...
06/14/2005
6881749Pyranoindazoles and their use for the treatment of glaucoma
Pyranoindazoles are disclosed. Also disclosed are methods for the lowering and controlling of normal or elevated intraocular pressure as well as a method for the treatment of glaucoma using compositions containing one or more of the compounds of the present inventio...
04/19/2005
6838193Organic light-emitting diode
This invention features a dipyrazolo-pyridine compound of formula (I): each of R1, R2, R3, and R4, independently, is H, alkyl, alkenyl, cycloalkyl, aryl, or heteroaryl; and e...
01/04/2005
6696476Pyranoindazoles and their use for the treatment of glaucoma
Pyranoindazoles are disclosed. Also disclosed are methods for the lowering and controlling of normal or elevated intraocular pressure as well as a method for the treatment of glaucoma using compositions containing one or more of the compounds of the prese...
02/24/2004
6642249Immunomodulating compounds
The present invention relates to a novel heterocyclic compound, a pharmaceutical composition comprisining said compound, a method and use of said compound for clinical treatment of medical conditions which may benefit from immunomodulation, e.g. rheumatoi...
11/04/2003
6583089Tricyclic benzoylcyclohexanedione derivatives
Tricyclic benzoylcyclohexanedione derivatives of the formula I ##STR1## where X, Y, R1, R2, R3, R4, R5, R9, and m are defined herein, and their agriculturally useful salts. Process for prep...
06/24/2003
6518294Fused pyrazolyl compounds
A fused pyrazolyl compound of the following formula: ##STR1## wherein each of Ar1, Ar2, and Ar3, independently, is phenyl, thienyl, pyrrolyl, or furyl, optionally substituted with halo, alkyl, carboxyl, alkoxycarbonyl, thi...
02/11/2003
6462036Tricyclic pyrazole derivatives
This invention relates to certain 3-aryl or 3-heteroaryl pyrazoles with 4,5(3,4)-bicyclic ring fusion which are inhibitors of protein kinase activity, of which some are novel compounds, to pharmaceutical compositions containing these pyrazoles and to proc...
10/08/2002
6436967Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
This invention is in the field of antiinflammatory pharmaceutical agents and specifically relates to prodrugs of compounds which selectively inhibit cyclooxygenase-2. The use of non-steroidal antiinflammatory drugs (NSAIDs) in treating pain and the swelli...
08/20/2002
6391905Condensed 4,5,6,7-tetrahydrobenzo[C]thiopenes as enhancer for cell differentiation induction factor action
A compound represented by the formula: ##STR1## wherein X represents a sulfur atom or an oxygen atom; Y represents an optionally oxidized sulfur atom or an oxygen atom; Z represents a bond or a divalent hydrocarbon group; R1 represents an optio...
05/21/2002
6297238Therapeutic agents
This invention realtes to compounds formula I ##STR1## and pharmaceutically acceptable salts thereof, which are inhibitors of protein kinase activity, pharmaceutical compositions thereof and provesses for their preparation....
10/02/2001
6245796Tricyclic pyrrole or pyrazole derivative
A tricyclic pyrrole or pyrazole derivative represented by the following general formula (I), or a pharmaceutically acceptable salt thereof, which shows strong affinity and selectivity for the 5-HT2C receptor and is useful for the treatment of c...
06/12/2001
6034252Substituted thienocycloalkylpyrazoles: dopamine receptor subtype specific ligands
Disclosed are compounds of the formula: ##STR1## or the pharmaceutically acceptable salts thereof wherein wherein: R1, R2, and and R4 independenlty represent hydrogen, halogen, alkyl, cyano, alkoxycarbonyl, trifluorom...
03/07/2000
5985799Tricyclic herbicidal heterocycles
Compounds of Formula (I), and their N-oxides and agriculturally-suitable salts, are disclosed which are useful in controlling undesired vegetation, wherein J is Formula (II), Q is represented by Q-1 through Q-4 and X, Y, Z, R1-19, m, n, p, q, a...
11/16/1999
5932598Prodrugs of benzenesulfonamide-containing COX-2 inhibitors
Prodrugs of COX-2 inhibitors are described as being useful in treating inflammation and inflammation-related disorders....
08/03/1999
5886016Benzopyranopyrazolyl derivatives for the treatment of inflammation
A class of benzopyranopyrazolyl derivatives is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula I ##STR1## wherein A, wherein X, m, n, p, B, R1, R2
03/23/1999
5827799Compounds and herbicides containing same as active components
An object of the invention is to provide herbicides which are completely selective to crops such as paddy rice, soybeans and cotton and have an excellent herbicidal activity on weeds. The invention relates to ether compounds of the general formula (I) ##S...
10/27/1998
5686480Fused tricyclic heteroaromatic derivatives as dopamine receptor subtype ligands
A class of fused tricyclic heteroaromatic compounds of formula (I), or a salt thereof or a prodrug thereof containing a fused pyrazole ring are ligands for dopamine receptor subtypes within the body and are therefore of use in the treatment and/or prevent...
11/11/1997
5670532Pyrazolyl derivatives for the treatment of inflammation
A class of benzopyranopyrazolyl derivatives is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula I ##STR1## wherein A is --(CH2)m --X--(CH...
09/23/1997
5565482Heteroarylpyranopyrazolyl derivatives for the treatment of inflammation
A class of benzopyranopyrazolyl derivatives is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula I ##STR1## wherein A is --(CH2)m --X--(CH...
10/15/1996
5547975Benzopyranopyrazolyl derivatives for the treatment of inflammation
A class of benzopyranopyrazolyl derivatives is described for use in treating inflammation and inflammation-related disorders. Compounds of particular interest are defined by Formula I ##STR1## wherein A is --(CH2)m --X--(CH...
08/20/1996
5500438Arthropodicidal anilides
Substituted anilides of the formula ##STR1## wherein Q is one of ##STR2## and R1 to R5, Y, Z and Z1 are as defined in the text, arthropodicidal compositions containing such compounds; and a method for contr...
03/19/1996
5424308Condensed pyrazole 3-oxo-propanenitrile derivatives
Condensed pyrazole 3-oxo-propanenitrile derivatives of formula (I) ##STR1## wherein X represents a --CH(R4)-- group, an oxygen atom or a --S(O)n -- group where n is 0, 1 or 2; R1 represents C1 -C6
06/13/1995
5369121Arthropodicidal pyrazolines, pyrazolidines and hydrazines
Compounds of Formula I ##STR1## wherein Q, W, R1 and m are as defined in the text; these compounds being useful in controlling agronomic and nonagronomic arthropods....
11/29/1994
5276039Substituted indazole arthropodicides
Indazole arthropodicides, compositions containing them and a method for controlling arthropods employing these indazoles as the active ingredient. The indazoles have the following general formula wherein Q, X, Y, R1 and m are as defined in the ...
01/04/1994
5258511Pyrazoloazepinones and methods of using such pyrazoloazepinones to dye synthetic fibers and to pigment pastes, paints, printing inks, colored paper and colored macromolecular substances
Heterocyclic compounds of the formula ##STR1## in which R represents hydrogen, substituted or unsubstituted alkyl, substituted or unsubstituted cycloalkyl, substituted or unsubstituted aryl, substituted or unsubstituted hetaryl, A represents C--R
11/02/1993
5206258Use of heteroaryl-3-oxo-propanenitrile derivatives in treating clinical wherein myelopoiesis suppression occurs
Heteroaryl-3-oxo-propanenitrile derivatives of formula (I) ##STR1## wherein X represents an oxygen atom or a --CH(R4)--, --O--CH(R4)--,--S(O)n --, --S(O)n --CH(R4)--, --CH(R4)--O--, --...
04/27/1993
5171862Process and indazole intermediates for the preparation of oxophthalazinyl acetic acids and analogs thereof
Oxophthalazinyl acetic acids having benzothiazole side chains are prepared by reacting an oxophthalazinyl thioacetamide acetate with hydrogen sulfide and a nitrophenyl compound having a reactive group such that the benzothiazole side chain may be formed b...
12/15/1992
5166152Tricyclic 3-oxo-propanenitrile derivatives
Compounds having the general formula (I) ##STR1## wherein X represents an oxygen atom or a --S(O)n --group, wherein n is zero, 1 or 2; R represents C1 -C6 alkyl, pyridyl or substituted or unsubstituted phenyl; R2...
11/24/1992
5108485Herbicidal 2-(2-imidazolin-2-yl)-benzazoles
There are provided o-carboxy-(5-oxo-2-imidazolin-2-yl)benzoheterocyclic compounds wherein the fused heterocyclic ring system is a 5-membered ring containing one, two or three nitrogen atoms, derivatives of said benzoheterocyclic compounds and a method for...
04/28/1992
4960784Insecticidal substituted indazoles
Certain substituted indazoles, including all geometric and stereoisomers thereof, agricultural compositions containing the indazoles and use of the indazoles as insecticides....
10/02/1990
4816467Heteroaryl 3-oxo-propanenitrile derivatives, pharmaceutical compositions and use
The invention relates to compounds having the general formula (I) ##STR1## and the pharmaceutically acceptable salts thereof, which possess immunomodulating activity and are useful e.g. in the treatment of neoplastic diseases and acute and chronic in...
03/28/1989
4803193Heat-sensitive recording material using chromeno compound
In a heat-sensitive recording material comprising on a substrate a recording layer containing a colorless or pale-colored basic dye and an electron accepting reactant material, the heat-sensitive recording material which is characterized in that the basic...
02/07/1989
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