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| Number | Title | Issue Date |
| 8013169 | Naphthylmethylimidizoles as therapeutic agents Disclosed herein is a compound of the formula (a): Therapeutic methods, compositions and medicaments related thereto are also disclosed. ... | 09/06/2011 |
| 7902377 | Method for preparing medetomidine and its salts The invention provides an improved, highly efficient method for preparing Medetomidine, and its salts, in particular its pharmaceutically acceptable salts. The method utilizes the high reactivity of halogenated imidazoles towards transmetalation with Grignard reagen... | 03/08/2011 |
| 7728147 | Detomidine hydrochloride crystallization method A method of isolating detomidine (I) hydrochloride as a crystalline salt is provided. The method comprises hydrogenating in the presence of a catalyst of compound of formula (II) in aqueous solution comprising hydrochloric acid, concentrating the solution by distill... | 06/01/2010 |
| 7563906 | Indazole derivatives An object of the present invention is to create a novel indazole derivative useful as a drug and to find a novel pharmacological action of the derivative. The compound of the present invention is represented by the formula [I] and has an excellent Rho kinase inhibit... | 07/21/2009 |
| 7371871 | Inhibitors of glutaminyl cyclase The present invention relates to compounds that act as inhibitors of QC including those represented by the general formulae 1 to 9: and combinations thereof for the treatment of neuronal disorders, especially Alzheimer's di... | 05/13/2008 |
| 7365196 | Sulphonamido-substituted bridged bicycloalkyl derivatives A class of compounds is disclosed, comprising sulphonamido-substituted bridged bicycloalkyl structures. The compounds are inhibitors of gamma-secretase, and hence are useful in the treatment of and/or prevention of Alzheimer's disease. ... | 04/29/2008 |
| 7351835 | Organic molecular cataylst having binaphthol skeleton and processes for producing the same and application thereof A novel organic molecular catalysts represented by the following formula (1) or (2): and a method for carrying out asymmetric reactions/asymmetric synthesis using these organic molecular catalysts. ... | 04/01/2008 |
| 7321044 | Synthesis of oxygen-substituted benzocycloheptenes as valuable intermediate products for the production of tissue-selective estrogens The invention relates to intermediate products and a new process for the production of benzocycloheptene C. The process for the production of its new intermediate products according to the invention starts from eco... | 01/22/2008 |
| 7223871 | Process for preparing substituted imidazole derivatives and intermediates used in the process The invention relates to a process for preparing substituted imidazole derivatives of formula (I) and acid addition salts thereof in which formula Y is —CH2— or —CO—, R1 is H, halo o... | 05/29/2007 |
| 7211595 | Farnesyltransferase inhibitors Substituted imidazoles and thiazoles having the formula are useful for inhibiting farnesyltransferase. Also disclosed are farnesyltransferase-inhibiting compositions and methods of inhibiting farnesyltransferase in a p... | 05/01/2007 |
| 7125725 | Biaryl-type compounds, CD color fixing agent and method for determination of absolute configuration A novel achiral biaryl-type compound and a circular dichroism(CD) color fixing agent are provided. Furthermore, a method for determining an absolute configuration of a chiral compound is carried out by introducing the above achiral biaryl-type compound into the chir... | 10/24/2006 |
| 7002022 | N-Aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF Described are compunds of formula (I), wherein W is O or S; X is NR8; Y is CR9R10—(CH2)n wherein R9 and R10 are independently of each other hydrogen or lower alkyl, and n is an integer of from and i... | 02/21/2006 |
| 6727098 | Biaryl-type compounds, CD color fixing agent and method for determination of absolute configuration A novel achiral biaryl-type compound and a circular dichroism (CD) color fixing agent are provided. Furthermore, a method for determining an absolute configuration of a chiral compound is carried out by introducing the above achiral biaryl-type compound into the chi... | 04/27/2004 |
| 6683115 | 댢-adrenergic receptor agonists Disclosed are multibinding compounds which are 댢 adrenergic receptor agonists and are useful in the treatment and prevention of respiratory diseases such as asthma, bronchitis. They are also useful in the treatment of nervous system injury and prem... | 01/27/2004 |
| 6683191 | Method for synthesis of substituted azole libraries The invention relates to methods of synthesizing libraries of diverse and complex 2-substituted azole compounds of the general formula (I) or (II) ##STR1## wherein X, R2 and the ring components ##STR2## are as described herein, novel interm... | 01/27/2004 |
| 6673941 | Disubstituted imidazoles useful in the treatment of bacterial infections Compounds of formula (I) and formula (II) are disclosed which are useful in the treatment bacterial infections: ##STR1## wherein: R1 is C1-4 alkyl, Ar or 2-thienyl or 3-thienyl; R2 is C1-4 alkyl or Ar; and ... | 01/06/2004 |
| 6646162 | Compounds and compositions for delivering active agents Compounds and compositions for the delivery of active agents are provided. Methods of administration and preparation are provided as well.... | 11/11/2003 |
| 6638321 | Cationic oxidation bases, their use for oxidation dyeing of keratin fibres, dyeing compositions and dyeing methods The invention relates to novel monobenzene oxidation bases containing at least one cationic group Z, Z being chosen from aliphatic chains containing at least one quaternized unsaturated ring, to their use for the oxidation dyeing of keratin fibers, to dye... | 10/28/2003 |
| 6593497 | 댢-adrenergic receptor agonists The present invention is directed to multibinding compounds which are 댢 adrenergic receptor agonists and are therefore useful in the treatment and prevention of respiratory diseases such asthma, bronchitis, and the like. They are also useful in the... | 07/15/2003 |
| 6559172 | Disubstituted imidazoles useful in the treatment of bacterial infections Novel disubstituted imidazoles are disclosed which are useful in the treatment of bacterial infections, particularly through the inhibition of FAB I.... | 05/06/2003 |
| 6545163 | Process to prepare 1-aryl-2-(1-imidazolyl) alkyl ethers and thioethers A process is disclosed for the preparation of imidazole derivatives, in particular, 1-aryl-2-(1-imidazolyl) alkyl ethers and thioethers, and more particular for the preparation of tioconazole. The preferred process involves alpha bromination of thiophene ... | 04/08/2003 |
| 6541669 | 댢-adrenergic receptor agonists Disclosed are multibinding compounds which are 댢 adrenergic receptor agonists and are useful in the treatment and prevention of respiratory diseases such as asthma, bronchitis. They are also useful in the treatment of nervous system injury and prem... | 04/01/2003 |
| 6509366 | Substituted imidazoles as selective modulators of Bradykinin B2 receptors Disclosed are compounds of the formula: ##STR1## or the pharmaceutically acceptable non-toxic salts thereof wherein Y, R1, R2, R3, R4, R5, R6, R7 R7 ' are variables de... | 01/21/2003 |
| 6420375 | Fused ring compounds, process for producing the same and use thereof To provide a novel compound of the formula: ##STR1## [wherein A1 ix a 5 or 6-membered ring which may be substituted by a group not containing a cyclic group, A2 is an aromatic ring which may be substituted, X is a divalent group, Y i... | 07/16/2002 |
| 6379398 | Cationic compounds, their use for the oxidation dyeing of keratin fibres, dye compositions and dyeing processes Dibenzenic ortho-phenylenediamines comprising at least one cationic group Z, Z being chosen from quaternized aliphatic chains, aliphatic chains comprising at least one quaternized saturated ring, and aliphatic chains comprising at least one quaternized un... | 04/30/2002 |
| 6340371 | Cationic ortho-phenylenediamines, their use for the oxidation dyeing of keratin fibers, dye compositions and dyeing processes Monobenzenic ortho-phenylenediamines comprising at least one cationic group Z, Z being chosen from aliphatic chains, comprising at least one quaternized unsaturated ring, to their use for the oxidation dyeing of keratin fibers, to dye compositions contain... | 01/22/2002 |
| 6313132 | Therapeutically active diarylpropylamines; their pharmaceutically acceptable salts; a method for their preparation and method for their use The invention relates to novel compounds of Formula (I) wherein R1, R2, R3, R4, R5, R6, R7 and Ar are as defined in claim 1, their salts with physiologically acceptable acids and, whe... | 11/06/2001 |
| 6297239 | Inhibitors of prenyl-protein transferase The present invention is directed to compounds which inhibit a prenyl-protein transferase (FTase) and the farnesylation of the oncogene protein Ras. The invention is further directed to chemotherapeutic compositions containing the compounds of this invent... | 10/02/2001 |
| 6288071 | 1-ethylene-2-alkylene-1,4-cyclohexadiene pesticides Pesticidally active cyclohexadienyl derivative compounds of the formula I that are esters, oximes or amides are claimed. These compounds may be used as fungicides, acaricides and insecticides in plant protection.... | 09/11/2001 |
| 6270533 | Cationic oxidation bases, their use for oxidation dyeing of keratin fibres, dyeing compositions and dyeing methods The invention relates to novel dibenzene oxidation bases containing at least one cationic group Z, Z being chosen from quaternized aliphatic chains, aliphatic chains containing at least one quaternized saturated ring and aliphatic chains containing at lea... | 08/07/2001 |
| 6265428 | Substituted phenyl compounds and derivatives thereof that modulate the activity of endothelin Methods, compositions, and compounds for modulating the activity of an endothelin peptide are provided. The methods use compositions that contain compounds of formula (1): ##STR1## where X and Y are selected from groups that include O, S, and NH; and ... | 07/24/2001 |
| 6262101 | Immunotherapeutic agents Cyano and carboxy derivatives of substituted styrenes are inhibitors of tumor necrosis factor , nuclear factor .kappa.B, and phosphodiesterase and can be used to combat cachexia, endotoxic shock, retrovis replication, asthma, and inflammatory condi... | 07/17/2001 |
| 6172239 | Substituted 1-phenyl-3-pyrazolecarboxamides active on neurotensin receptors, their preparation and pharamaceutical compositions containing them The invention relates to compounds of the formula ##STR1## The compounds have agreat affinity for the neurotensin receptors.... | 01/09/2001 |
| 6166060 | 1H-4(5)-substituted imidazole derivatives The present invention provides, in its principal aspect, compounds of the general formula: ##STR1## when A is --NHCO--, --N(CH3)--CO--, --NHCH2 --, --N(CH3)--CH2 --, --CH.dbd.CH--, --COCH2 --, CH... | 12/26/2000 |
| 6124484 | Recovery of triarylmethyl halide protecting groups cleaved during oligonucleotide synthesis The present invention provides a method for the preparation of triarylmethyl protecting group reagents. The reagents are prepared from reaction effluent from the cleavage step of oligonucleotide synthetic regimes.... | 09/26/2000 |
| 6107311 | Dihydrobenzofuran and related compounds useful as anti-inflammatory agents A compound having the structure: ##STR1## wherein (a) n is from 1 to about 3; (b) X is selected from the group consisting of O, S, SO, or SO2 ; (c) Y is independently hydrogen or straight, branched or cyclic alkyl having from 1 to about 4 carbo... | 08/22/2000 |
| 6103749 | Aryl imidazole compounds having phosphodiesterase IV inhibitory activity Novel compounds which are effective PDE IV inhibitors are disclosed. These compounds have the general structure of: ##STR1## where R1, R2, R3, R4, X1, X2 and Z are described herein. Th... | 08/15/2000 |
| 6103733 | Method for increasing HDL cholesterol levels using heteroaromatic phenylmethanes An HDL cholesterol level inducing compound and a method of administering the compound having the structural formula I. ##STR1## wherein n is 1 or 2; R1 is a heteroaromatic substituent independently selected from a five-membered heteroaroma... | 08/15/2000 |
| 6063930 | Substituted imidazole compounds useful as farnesyl-protein transferase inhibitors The present invention is directed to compounds which inhibit farnesyl-protein transferase (FTase) and the farnesylation of the oncogene protein Ras. The invention is further directed to chemotherapeutic compositions containing the compounds of this invent... | 05/16/2000 |
| 6057322 | Basically-substituted benzoylguanidines, a process for preparing them, their use as a medicament or diagnostic agent, and a medicament containing them Compounds of the formula I ##STR1## and the pharmaceutically tolerated salts thereof, are described. A process for their preparation and their use as medicaments in cardiovascular diseases are also described.... | 05/02/2000 |
