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| Number | Title | Issue Date |
| 7893278 | CIS-imidazolines The present invention relates to compounds of the formula and the pharmaceutically acceptable salts and esters thereof, a process for their manufacture, medicaments containing them as well as the use of these compounds as p... | 02/22/2011 |
| 7524970 | Compounds A compound of formula (I): wherein X represents O or S; R1 represents C1-6 alkyl, C3-8 cycloalkyl, C3-8 cycloalkylmethyl or C | 04/28/2009 |
| 7425638 | Cis-imidazolines The present invention provides compounds according to formula I having the designations provided herein, and pharmaceutically acceptable salts and esters thereof. These compounds inhibit the interaction of MDM2 protein with... | 09/16/2008 |
| 7291642 | Bradykinin-B1 antagonists, process for their preparation and their use as medicaments The present invention provides bradykinin-B1 antagonists of the formula in which A, Ar, G, Q, R1 and R4 are as defined in claim 1, their enantiomers, their diastereomers, their mixtures and ... | 11/06/2007 |
| 7235516 | Semiconductor cleaning composition comprising an ethoxylated surfactant A substrate surface cleaning liquid medium and a cleaning method using the cleaning liquid medium are capable of removing finely particulate contaminants more efficiently than conventional techniques from substrates for devices in the production of semiconductor dev... | 06/26/2007 |
| 7141677 | Peroxyoxalate chemiluminescence compound and system An unstable, methyl-substituted (1,1 oxaly diimidazole) molecule capable of accelerating the rate at which a material attains maximum chemiluminescence when reacted hydrogen peroxide in the presence of a fluorophore and a method to synthesize such molecules. ... | 11/28/2006 |
| 7132421 | CIS-imidazoles The present invention provides compounds according to formula I and pharmaceutically acceptable salts and esters thereof, having the designations provided herein and which inhibit the interaction of MDM2 protein with a p53-like peptide and have antiproliferative act... | 11/07/2006 |
| 7022847 | Method for the production of 2-(2-ethoxyphenyl)-substituted imidazotriazinones The invention relates to a method for the production of 2-phenyl-substituted imidazotriazinones of general formula (I), comprising the reaction of compounds of formula (II) with compounds of formula (III) and subsequent reaction with iodine or bromine, then with a m... | 04/04/2006 |
| 6974801 | Inhibitors and methods of use thereof New triterpenoid derivatives with various substituents at the C-17 position of 2-cyano-3,12-dioxooleana-1,9(11)-dien-28-oic acid (CDDO) were synthesized. Among them, 2-cyano-3,12-dioxooleana-1,9(11)-dien-28-onitrile (CNDDO), 1-(2-cyano-3,12-dioxooleana-1,9(11)-dien-... | 12/13/2005 |
| 6759511 | Compound used as an amino-protecting group, process for preparing the same, and synthetic method of a peptide using the same The present invention relates to a carbonic acid ester compound of the following formula (1): in which X, Y, and Ar are defined in the specification, which can be easily combined with the amino group of an amino acid or ... | 07/06/2004 |
| 6747148 | Sulfonamide derivatives as inhibitors of bone resorption and as inhibitors of cell adhesion Sulfonamide derivatives, their physiologically tolerable salts and their prodrugs according to the present invention are vitronectin receptor antagonists and inhibitors of cell adhesion, as well as inhibit bone resorption by osteoclasts. These derivatives, salts and... | 06/08/2004 |
| 6734302 | Cis-imidazolines The present invention provides compounds according to formula I and formula II and pharmaceutically acceptable salts and esters thereof, having the designations provided herein and which inhibit the interaction of MDM2 protein with a p53-like peptide and have antipr... | 05/11/2004 |
| 6605608 | Amino acid derivatives and drugs containing the same as the active ingredient The present invention relates to the compounds of the formula (I) and salts thereof (all the symbols are the same meanings as described in the specification). ##STR1## The compounds of the formula (I) possess inhibitory activity of N-type calcium cha... | 08/12/2003 |
| 6495522 | Substituted alpha-hydroxy acid caspase inhibitors and the use thereof The present invention is directed to novel substituted -hydroxy acid thereof, represented by the general Formula I: ##STR1## where R1 -R5, X and Z are defined herein. The present invention also relates to the discovery that co... | 12/17/2002 |
| 6465677 | Method for the preparation of N-neohexyl--aspartyl-L-phenylalanine methyl ester from imidazolidin-4-one intermediates The synthesis of N-[N-(3,3-dimethylbutyl)-L--aspartyl]-L-phenylalanine 1-methyl ester via conversion under reducing conditions of novel imidazolidinone(s) is disclosed.... | 10/15/2002 |
| 6451824 | Sulfonylaminocarboxylic acids Compounds of formula (I) ##STR1## are suitable for the production of pharmaceuticals for the prophylaxis and therapy of disorders in the course of which an increased activity of matrix-degrading metalloproteinases is involved.... | 09/17/2002 |
| 6410744 | Carbonyldiimidazoles, their ester derivatives and method for their production Carbonyldiimidazoles of the formulae Ia, Ib, Ic or mixtures thereof ##STR1## where R1 is C1-4 -alkyl and R2 is hydrogen or methyl, and tert-butyl esters derived therefrom are described.... | 06/25/2002 |
| 6380237 | Diphenylimidazolines The invention relates to novel diphenylimidazolines of the formula (I) ##STR1## in which Ar1, Ar2 and R are each as defined in the description, and a plurality of processes for their preparation and to their use for controlling animal pes... | 04/30/2002 |
| 6191157 | Hetero-linked phenylglycinolamides The hetero-linked phenylglycinolamides are prepared by reaction of the corresponding hetero-linked phenylacetic acids with appropriate phenylglycinols. The hetero-linked phenylglycinolamides are suitable as active compounds in medicaments.... | 02/20/2001 |
| 6136942 | Latent amino groups and isocyanate groups comprising polyurethane prepolymers, method for their production and their use A one-component polyurethane composition is described that comprises a latent curing agent bonded to the prepolymer, from which curing agent aldehyde is liberated upon curing. Said aldehyde comprises two phenyl groups. By the specific design of the polyur... | 10/24/2000 |
| 6093816 | Cationic lipids The present invention is directed to new cationic lipids and intermediates in their synthesis that are useful for transfecting nucleic acids or peptides into prokaryotic or eukaryotic cells. The lipids comprise one or two substituted histidine residues, o... | 07/25/2000 |
| 5972940 | Arginine analogues having nitric oxide synthase inhibitor activity A compound selected from the group consisting of a compound of the formula wherein A is selected from the group consisting of hydrogen, alkyl of 1 to 6 carbon atoms and --NO2, E is --O-- or a covalent bond, n is an integer from 1 to 12, R1... | 10/26/1999 |
| 5919792 | Integrin antagonists This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as vitronectin receptor antagonists. The vitronectin receptor antagonist compounds of the present invention are v댣 antagonists, ... | 07/06/1999 |
| 5883125 | Benzyloxy substituted aromatics and their use as fungicides and insecticides Compounds with fungicidal and insecticidal properties having formula I ##STR1## wherein A is N or CH; V is O or NH; m and n are integers 0 and 1 provided that m+n is 1; X is independently selected from hydrogen, halo, (C1 -C4)alkyl, ... | 03/16/1999 |
| 5807748 | N-terminal protein sequencing reagents and methods which form amino acid detectable by a variety of techniques Novel alkoxythiocarbonylimidazoles provide new reagents for the N-terminal sequencing of small polypeptide samples. These reagents form an alkoxy thiourea derivative which is cleaved with acid to remove the N-terminal amino acid as a stable thiazolinone w... | 09/15/1998 |
| 5756758 | Peptide intermediates The invention relates to compounds which can be reacted with a carboxyl function with formation of an ester bond, whereby a protective group and, in particular, an anchor group for the carboxyl function is provided. The invention further relates to esters... | 05/26/1998 |
| 5719240 | Compounds containing cyclic amidine and uretdione groups, a process for their preparation and the use thereof A compound containing cyclic amidine groups and uretdione groups, having the formula: ##STR1## wherein X is O or NR2, R is the hydrocarbon radical of isophorone diisocyanate: ##STR2## R1 is a substituted (cyclo)alkylen... | 02/17/1998 |
| 5693310 | Amide complexes Compounds of general Formula I ##STR1## wherein R3 is a saturated, unsaturated, straight- or branched-chain or cyclic aliphatic hydrocarbon residue of up to 16 carbon atoms or, if R4 is a hydrogen atom, a cycloalkyl group or an ... | 12/02/1997 |
| 5686435 | Vitamin D amide derivatives The invention pertains to vitamin D amide derivatives of formula (I). These novel 1-hydroxy vitamin D derivatives and their 20-epi analogues comprise compounds of formula (I) and corresponding 5,6-trans isomers, where Y represents an alkylene or al... | 11/11/1997 |
| 5637730 | Sodium enalapril complex and the use thereof to make sodium enalapril A process for making pure sodium enalapril is provided which includes the step of decomplexing essentially pure sodium enalapril-sodium iodide complex to yield essentially pure sodium enalapril.... | 06/10/1997 |
| 5597855 | Poly(pentaerythrityl diphosphonate) and its use in self-extinguishing thermoplastic compositions Poly(Pentaerythrityl diphosphonate) of formula (I): ##STR1## wherein n is an integer having a value comprised within the range of from 3 to 100. The poly(pentaerythrityl diphosphonate) of formula (I) is useful as a flame retardant additive for thermo... | 01/28/1997 |
| 5591863 | Imidazolium hardeners for hydrophilic colloids This invention is related to improved hardeners for proteinaceous materials. More specifically this invention is related to improved imidazolium hardeners for crosslinking a proteinaceous material for use in a photographic film. The improved hardeners are... | 01/07/1997 |
| 5584888 | Perhydrolysis-selective bleach activators Bleaching compositions, laundry and automatic dishwashing detergent compositions comprising particular neutral or anionically charged substituted bleach activators are provided. More specifically, the invention relates to compositions which provide enhanc... | 12/17/1996 |
| 5585486 | Peptidic ketones as interleukin-1ଲ-converting enzyme inhibitors Disclosed are compounds of the formula (I) and pharmaceutically acceptable salts thereof: ##STR1## wherein R1 is (CR5 R6)n, (CR5 R6)n,-aryl, (CR5 R6) | 12/17/1996 |
| 5560862 | Multiple-substituted bleach activators Bleaching compositions, laundry and automatic dishwashing detergent compositions comprising multiple-substituted bleach activators which have at least one quaternary nitrogen atom, are provided. More specifically, the invention relates to compositions whi... | 10/01/1996 |
| 5552554 | Imidazole and triazole carboxylates, and processes for preparing 2,4-oxazolidinediones Processes are described for preparing 2,4-oxazolidinediones having Formula (I) ##STR1## wherein: R1 is phenyl optionally substituted with 1-2 halogens; or 4-phenoxy, 4-(1-phenethyloxy) or 4-benzyloxy each optionally substituted with R... | 09/03/1996 |
| 5552556 | Perhydrolysis-selective bleach activators Bleaching compositions, laundry and automatic dishwashing detergent compositions comprising particular neutral or anionically charged substituted bleach activators are provided. More specifically, the invention relates to compositions which provide enhanc... | 09/03/1996 |
| 5550280 | Hindered aromatic ester compounds useful as anti-viral agents Compounds of the formula ##STR1## wherein X is O or S; Y is O or S; R1 is hydrogen, halogen, C1 -C4 alkyl or C1 -C4 alkoxy; R2 is hydrogen, halogen, C1 -C4 alkyl, C | 08/27/1996 |
| 5550159 | Peptide mimics useful as platelet aggregation inhibitors This invention relates to compounds having the following formula ##STR1## or pharmaceutically acceptable salt thereof which are useful in the inhibition of platelet aggregation, to pharmaceutical compositions of such phenylamidines derivatives, and t... | 08/27/1996 |
| 5503776 | N-acylcarnosines and their use as antioxidants An N-acylamino acid compound represented by the general formula (1): R--CO--(NH--X--CO)n --OR1 (1) wherein (NH--X--CO) is an amino acid residue, X in (NX--X--CO) is variable with the kind of amino acid to be used, R--CO ... | 04/02/1996 |
