Quotables
"There is no likelihood man can ever tap the power of the atom."
Robert Millikan, Nobel Prize winner in physics
PatentStorm News
Make the Most of Our Site
See this month's Top Inventors and Most Cited Patents.
Stay on top of the latest innovations by subscribing to an RSS feed.
Registered users: Manage your profile.
| Number | Title | Issue Date |
| 7414046 | Gyrase inhibitors and uses thereof The present invention relates to compounds of the formula I: or a pharmaceutically acceptable derivative or prodrug thereof. The compounds are useful as inhibitors of bacterial gyrase activity. The present invention also re... | 08/19/2008 |
| RE40245 | Gyrase inhibitors and uses thereof The present invention relates to compounds of the formula I: or a pharmaceutically acceptable derivative or prodrug thereof. The compounds are useful as inhibitors of bacterial gyrase activity. The present invention also relates ... | 04/15/2008 |
| 7348333 | Cycloalkyl derivatives as inhibitors of bone resorption and vitronectin receptor antagonists There are described cycloalkyl derivatives of the formula (I) R1—Y-A-B-D-E-F-G (I) in which R1, Y, A, B, D, E, F and G have the meaning indicated herein, their preparation and their use as medicaments. The compounds a... | 03/25/2008 |
| 7176312 | Kinase inhibitor scaffolds and methods for their preparation General methods for the solution phase as well as solid phase synthesis of various substituted heteroaryls has been demonstrated. These substituted heteroaryls can be further elaborated by aromatic substitution with amines at elevated temperature or by anilines, bor... | 02/13/2007 |
| 6933390 | Process for the arylation of aza-heterocycles with activated aromatics in presence of caesium carbonate The invention concerns a process for the preparation of N-aryl-aza-heterocycles of the general formula I by reaction of aza-heterocycles with activated aryl halides with use of caesium carbonate without addition of fur... | 08/23/2005 |
| 6632809 | Gyrase inhibitors and uses thereof The present invention relates to compounds of the formula I: ##STR1## or a pharmaceutically acceptable derivative or prodrug thereof. The compounds are useful as inhibitors of bacterial gyrase activity. The present invention also relates to methods for tr... | 10/14/2003 |
| 6407105 | Compounds and methods for use thereof in the treatment of cancer or viral infections Benzimidazole derivatives and salts and prodrugs thereof are disclosed, together with methods for the treatment of cancers or viral infections in warm blooded animals by administration of these compounds. Such compounds may be used in combination with a c... | 06/18/2002 |
| 6204264 | Benzimidazole derivative, hair growth promoter and external composition for skin using the same A benzimidazole derivative or a salt thereof expressed by the following Formula (I): ##STR1## wherein one of A and B is a hydrocarbon group of C10-30 expressed by R1 and the other is --(CH2)n --NR2 R | 03/20/2001 |
| 5919792 | Integrin antagonists This invention relates to certain novel compounds and derivatives thereof, their synthesis, and their use as vitronectin receptor antagonists. The vitronectin receptor antagonist compounds of the present invention are v댣 antagonists, ... | 07/06/1999 |
| 5693661 | Anti-viral compounds Certain vinyl acetylene benzimidazole compounds which inhibit the growth of picornaviruses, such as rhinoviruses, enteroviruses, cardioviruses, polioviruses, coxsackieviruses of the A and B groups, echo virus and Mengo virus.... | 12/02/1997 |
| 5599830 | Sulphorous derivatives of imidazole and their use as medicaments The invention relates to the products: ##STR1## in which: R1 =alkyl, alkenyl, alkynyl, alkylthio, R2B, R3B representing: hydrogen, mercapto, formyl, acyl, carboxy nitro, cyano, --PO3 (R)2, R representing h... | 02/04/1997 |
| 5554633 | Substituted amines as tachykinin receptor antagonists Compounds of formula (I), and salts and prodrugs thereof, wherein Q is optionally substituted phenyl or benzhydryl; X and Y are each H or together form a group=O; Z is O, S or NR9, where R9 is H or C1-6 alkyl; R1 | 09/10/1996 |
| 5405862 | Low free formaldehyde methylolhydantoin compositions Compositions of dimethyloldimethylhydantoin, monomethyloldimethylhydantoin, and dimethylhydantoin having less than 0.1% by weight of free formaldehyde based upon 100% by weight of total composition; and wherein the weight ratio of dimethyloldimethylhydant... | 04/11/1995 |
| 5298403 | Labeled drug hapten analogues for immunoassays The invention is directed to labeled drug hapten analogues comprising: (A) a label, of the type used in immunoassays, having an amine or sulfhydryl group; (B) a drug hapten nucleus selected from barbiturates or hydantoins and (C) a linking chain linking the 3-posit... | 03/29/1994 |
| 4948901 | Benzamide protease inhibitors Compounds of the formula ##STR1## where HET is a heterocyclic group, n is an integer of 0 to 2 and R1 is hydrogen or lower alkyl are protease inhibitors useful as anti-plasmin and antithrombin agents.... | 08/14/1990 |
| 4948891 | Benzamide protease inhibitors Compounds of the formula ##STR1## where Het is a heterocyclic group, n is an integer of 0 to 2 and R1 is hydrogen or lower alkyl are protease inhibitors useful as anti-plasmin and anti-thrombin agents.... | 08/14/1990 |
| 4942245 | Benzimidazole Derivatives Benzimidazole derivatives of the following formula, ##STR1## wherein R1 indicates hydrogen atom, lower alkyl group having carbon atoms of 1 to 6 or dimethylaminopropyl group, R2 indicates hydrogen atom or lower alkanoyl group ha... | 07/17/1990 |
| 4874864 | Benzamide protease inhibitors Compounds of the formula ##STR1## where HET is a heterocyclic group, n is an integer of 0 to 2 and R1 is hydrogen or lower alkyl are protease inhibitors use as anti-plasmin and anti-thrombin agents.... | 10/17/1989 |
| 4745125 | Antiulcer benzimidazoles Antiulcer amino-benzimidazole compounds substituted on the nitrogen; these compounds correspond to the following general formula: ##STR1## in which the various substituents are defined hereinbelow.... | 05/17/1988 |
| 4284584 | Process for the preparation of acyl cyanides Acyl cyanides of the formula ##STR1## in which R represents alkyl or substituted alkyl of from 1 to 8 carbon atoms, cycloalkyl or substituted cycloalkyl of from 3 to 12 carbon atoms, aryl or substituted aryl; or an optionally substituted 5-membered o... | 08/18/1981 |
| 4011236 | N-(Benzimidazol-2-yl)arylcarboxamides as ultraviolet (UV) light absorbers This invention relates to compositions containing N-(benzimidazol-2-yl)arylcarboxamides as ultraviolet (UV) light absorbers. The compounds are useful to protect UV sensitive materials, particularly plastic compositions, or ingredients thereof such as dyes... | 03/08/1977 |
| 3980796 | Substituted 2-alkoxycarbonylamine-5-(6)-phenylmercapto-benzimidazoles Substituted 2-alkoxycarbonylamine-5(6)-phenylmercapto-benzimidazoles are described as well as a process for their manufacture. The compounds are chemotherapeutics being especially suitable for the control of parasites of humans and animals, for example fo... | 09/14/1976 |
| 3932448 | 2-(Alkoxycarbonylamino)-1-benzimidazolecarboxylic acid esters with hydroxyaliphatic acids and derivatives thereof Substituted 2-alkoxycarbonylamino-1-benzimidazoles having the formula: ##SPC1## Wherein R is a lower alkyl radical, such as --CH3, and A is various organic radicals, hereinafter defined, such as: ##EQU1## are useful as fungicides and mite ... | 01/13/1976 |
