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| Number | Title | Issue Date |
| 8076489 | 5-hydroxy-benzothiazole derivatives having beta-2-adrenoreceptor agonist activity Compounds of formula (I) in free or salt or solvate form, wherein T has the meaning as indicated in the specification, are useful for treating conditions that are prevented or alleviated by activation of the β2-adrenoreceptor. Pharmaceutical compositions... | 12/13/2011 |
| 7700782 | Compounds 569 The present invention provides compounds of formula (I) wherein Ra, Rb, R1, R2, R3, R4, R5, R6 and R29 are as defined in the... | 04/20/2010 |
| 7402598 | Arylethanolamine β-adrenoreceptor agonist compounds The present invention relates to compounds of formula (I) as defined herein and salts or solvates thereof. Processes for preparing these compounds and pharmaceutical formulations containing them are also disclosed, as well as methods for the prophylaxis of treatment... | 07/22/2008 |
| 7323564 | Preparation of thiazoles The present invention is directed to a process for preparing a compound having the formula: wherein R is a range of organic groups and X is a leaving group. The process may include reacting a compound of the form... | 01/29/2008 |
| 7235668 | Process for the preparation of thioalkylamine derivatives The present invention relates to a novel process for the preparation of compounds of the formula (I) by reacting in a first step amino alcohols of the formula (II) | 06/26/2007 |
| 6992228 | Method for producing bisphenol catalysts and bisphenols This disclosure relates to a method for producing and using catalysts in the production of bisphenols, and in particular to a method for producing catalysts which contain poly-sulfur mercaptan promoters, and using these catalysts in the production of bisphenol-A and... | 01/31/2006 |
| 6946173 | Catheter balloon formed of ePTFE and a diene polymer A catheter balloon formed of a polymeric material such as expanded polytetrafluoroethylene (ePTFE) bonded to a second layer formed of a low tensile set polymer and/or impregnated with a low tensile set polymer. In a presently preferred embodiment, the low tensile se... | 09/20/2005 |
| 6943170 | N-cycloalkylglycines as HIV protease inhibitors This invention relates generally to N-cycloalkylglycines of the Formula (I): or a stereoisomeric form, a mixture of stereoisomeric forms, or a pharmaceutically acceptable salt thereof, which are useful as HIV protease ... | 09/13/2005 |
| 6900218 | Pyruvate derivatives Certain known and novel pyruvate derivatives are particularly active in restoring or preserving metabolic integrity in oxidatively competent cells that have been subjected to oxygen deprivation. These pyruvate-derived compounds include, but are not limited to oximes... | 05/31/2005 |
| 6710045 | Heterocyclic fluoroalkenyl thioethers and the use thereof as pesticides (IV) The present invention relates to novel heterocyclic fluoroalkenyl thioethers of the formula (I) in which m represents integers from 3 to 10, n represents 0, 1 or 2 and Het represents the following, i... | 03/23/2004 |
| 6683101 | Bicyclic cyclohexylamines and their use as NMDA receptor antagonists Described are heterocycle-substituted cyclohexylamines of formula (I), and their pharmaceutically acceptable salts thereof. The compounds of the formula (I) are antagonists of NMDA receptor channel complexes useful for treating cerebral vascular disorders... | 01/27/2004 |
| 6624186 | Ion channel modulating agents comprising novel benzimidazolone derivatives The present invention relates to ion channel modulating agents. More particularly, the present invention relates to a particular class of chemical compounds that has proven useful as modulators of SKCa, IKCa and BKCa chann... | 09/23/2003 |
| 6548667 | Sulfonamide derivative as a matrix metalloproteinase inhibitor The present invention provides a novel sulfonamide derivative of general formula (I) useful as an inhibitor of matrix metalloproteinase (MMP), its isomers, pharmaceutically acceptable salts thereof and a process for preparing the same. Since the sulfonami... | 04/15/2003 |
| 6544931 | Substituted heteroaryloxyacetanilides and their use as herbicides The invention relates to novel substituted heteroaryloxyacetanilides of the general formula (I), ##STR1## in which n, R, X, and Z are to intermediates for their preparation and to their use as herbicides.... | 04/08/2003 |
| 6358983 | Heterocyclically substituted -hydroxycarboxylic acid derivatives, method for producing the same and their use as endothelin receptor antagonists The present invention relates to carboxylic acid derivatives of the formula I ##STR1## the substituents having the meanings explained in the description, preparation and use as endothelin receptor antagonists.... | 03/19/2002 |
| 6340372 | Compositions for dyeing keratin fibers containing S-oxide-thiazolo-azoles and/or S,S-dioxide-thiazolo-azoles; their use for dyeing as couplers, method of dyeing A compostion for the dyeing of keratinous fibres comprising, in a medium appropriate for dyeing keratinous fiber contains: as coupler, at least one compound of formula: ##STR1## in which R1 denotes in particular hydrogen, halogen, aryloxy, alkoxy, a... | 01/22/2002 |
| 6268313 | Dihalopropene compounds, insecticidal/acaricidal agents containing same, and intermediates for their production The dihalopropene compounds of the general formula [I] have excellent insecticidal/acaricidal activity, so that they are satisfactorily effective for the control of noxious insects, mites and ticks.... | 07/31/2001 |
| 6204380 | Production pyridazine herbicides Carboxylic acid ester derivatives of formula (1): ##STR1## wherein R is C1 -C6 alkyl, R2 and R3 are independently hydrogen or C1 -C3 alkyl, and Q is optionally substituted phenyl, can be ea... | 03/20/2001 |
| 6130217 | Compounds enhancing antitumor activity of other cytotoxic agents This invention relates to certain heterocyclic compounds and their pharmaceutically acceptable salts, which are useful for sensitizing multidrug-resistant tumor cells to anticancer agents and multidrug resistant forms of malaria, tuberculosis, leishmania ... | 10/10/2000 |
| 6080869 | Benzothiazolone derivatives A compound of formula I, including optical isomers thereof, wherein X represents --SO2 NH-- or --NHSO2 --, p, q and r independently represent 2 or 3, Y represents thienyl optionally substituted by alkyl or halogen, or phenylthio- or phenyl opt... | 06/27/2000 |
| 6069160 | Heteroatom-containing benzocyclopentane-oxazolidinones The invention relates to heteroatom-containing benzocyclopentaneoxazolidinones, to processes for their preparation and their use as medicaments, especially as antibacterial medicaments.... | 05/30/2000 |
| 5980779 | Liquid crystalline compound and use thereof A process for producing a liquid crystalline compound represented by the following general formula (A): ##STR1##... | 11/09/1999 |
| 5914408 | Olefin polymerization catalysts containing benzothiazole A novel metallocene catalyst for the polymerization of olefin (co)polymers is of the general formula: Benzothiazole--E--M--Xm Ln where, M is a transition metal of Groups 3-10 of the Periodic Table; E is sulfur or oxygen; E being bond to the tr... | 06/22/1999 |
| 5892051 | Additives for lubricants Compounds of formula I, R--S--CH2 CH(OH)CH2 --S--R4 (I), where R is tert-alkyl of 4 to 20 carbon atoms and 4 is benzothiazolyl, --(CH2)m --S--CH2 CH(OH)CH2 --S--(C1 | 04/06/1999 |
| 5886014 | Benzimidazole derivatives, their preparation and their therapeutic use Compounds of formula (I): ##STR1## wherein: X represents an optionally substituted benzimidazole group; Y represents an oxygen or sulfur atom; Z represents a 2,4-dioxothiazolidin-5-ylidenylmethyl, 2,4-dioxothiazolidin-5-ylmethyl, 2,4-dioxooxaz... | 03/23/1999 |
| 5863915 | Substituted 4-arylbutyric acid derivatives as matrix metalloprotease Inhibitors for matrix metalloproteases, pharmaceutical compositions containing them, and a process for using them to treat a variety of physiological conditions. The compounds of the invention have the generalized formula ##STR1## wherein R... | 01/26/1999 |
| 5846989 | Benzothiazolone derivatives A compound of formula I, including optical isomers thereof, ##STR1## wherein X represents --SO2 NH-- or --NHSO2 --, p, q and r independently represent 2 or 3, Y represents thienyl optionally substituted by alkyl or halogen, or phenyl... | 12/08/1998 |
| 5763465 | 7-(2-aminoethyl) benzothiazolones There are disclosed compounds of formula I, Ar--CH2 CH2 --NH--CR1 R2 --X--Y I in which Ar represents a group, ##STR1## X represents a C1-12 alkylene chain optionally interrupted or terminated b... | 06/09/1998 |
| 5750711 | Dicarboxylic acid derivatives The dicarboxylic acid derivatives according to the invention have the following structure ##STR1## wherein X denotes O, S, (CF2)m, C(CF3)2 or CF2 --CF(CF3) (m=1 to 10), and R stems fro... | 05/12/1998 |
| 5728833 | Process for the preparation of fluoroalkenylthio heterocyclic derivatives A process for the preparation of a compound of formula (I): HetSCH2 CH2 CH.dbd.CF2 (I) wherein Het is an optionally substituted 5- or 6-membered heterocyclic ring, which comprises reacting a compound of formula ... | 03/17/1998 |
| 5716756 | Sulfonic acid esters, radiation-sensitive mixtures prepared therewith and their use Sulfonic acid esters are used as (a) compounds for forming a strong acid on irradiation in radiation-sensitive, positive or negative working mixtures also comprising (b) either a compound with at least one acid-decomposable C--O--C or C--O--Si bond (for p... | 02/10/1998 |
| 5688820 | Aminoalkyl benzoxazolinones and benzothiazolinones The invention relates to a compound selected from those of formula (I): ##STR1## in which R1, R2, R3, X and n are as defined in the description, the optical isomers thereof, and the addition salts thereof with a pharm... | 11/18/1997 |
| 5688811 | Aminoalkyl benzoxazolinones and benzothiazolinones The invention relates to a compound selected from those of formula (I): ##STR1## in which R1, R2, R3, X and n are as defined in the description, the optical isomers thereof, and the addition salts thereof with a pharm... | 11/18/1997 |
| 5681843 | Parabanic acid derivatives Parabanic acid derivatives, pharmaceutically acceptable salts thereof, and therapeutic agents containing said compounds as an effective component are useful pharmaceuticals for the treatment of diabetic complications such as diabetic neuropathy, diabetic ... | 10/28/1997 |
| 5648370 | 7-(2-aminoethyl) benzothiazolones There are disclosed compounds of formula I, Ar--CH2 CH2 --NH--CR1 R2 --X--Y I in which Ar represents a group, ##STR1## X represents a C1-12 alkylene chain optionally interrupted or terminated b... | 07/15/1997 |
| 5602196 | Bisphenol ester derivatives Stabilisers of formula I ##STR1## wherein R1 and R2 may be C1 -C5 alkyl, the substituents R3 to R8 may be hydrogen, the variable n may be 1 or 2, and, when n is 1, A may be an alkoxy r... | 02/11/1997 |
| 5594145 | Process for the preparation of 2(3H)-benzothiazolones The process for the preparation of 2(3H)-benzothiazolones which are optionally substituted on the benzene ring by reacting a 2-aminobenzothiazole which is optionally substituted on the benzene ring with a diazotization agent in the presence of aqueous hyd... | 01/14/1997 |
| 5576343 | Aromatic amidine derivatives and salts thereof An anticoagulant agent which comprises, as an active ingredient, an aromatic amidine derivative represented by the following general formula (1) or a salt thereof: ##STR1## wherein the group represented by ##STR2## is a group selected from ... | 11/19/1996 |
| 5539121 | 2-formylmercaptobenzothiazole There is disclosed a novel formylating agent, 2-formylmercaptobenzothiazole.... | 07/23/1996 |
| 5534634 | Process for preparing trifluoroethyl sulfur compounds from thiolates and 1-chloro-2,2,2-trifluoroethane Process for preparing trifluoroethyl sulfur compounds from thiolates and 1-chloro-2,2,2-trifluoroethane. The invention relates to the preparation of trifluoroethyl sulfur compounds of the formula RSCH2 CF3 by reacting 1-chloro-2,2,2-... | 07/09/1996 |
