Bizarre Patents
Decorative Jeweled Wheel Cover
An improved wheel is provided wherein decorative items such as gem stones are embedded in either the wheel surface, a special mounting section attached to the wheel surface, or to a spoke strap that wraps around each spoke and positions embedded gem stones on the outside surface of the spoke.
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| Number | Title | Issue Date |
| 7855296 | Method for synthesizing 2-carbomethoxytropinone Disclosed is a method of making (−)-cocaine efficient for use on a large scale. The cocaine is created by reacting an aqueous solution of (+)-2-carbomethoxytropinone (2-CMT) bitartrate, sodium amalgam and an acid that forms a highly soluble sodium salt to form (âˆ... | 12/21/2010 |
| 7429601 | Esters of hydroxyl-substituted nitrogen heterocycles, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions The present invention relates to new compounds of general formula 1 wherein X− and the groups A, B, R, R1, R2, R3, R3′, R4, R4′, Rx | 09/30/2008 |
| 7407970 | 8-aza-bicyclo[3.2.1]octane derivatives and their use as monoamine neurotransmitter re-uptake inhibitors This invention relates to novel 8-aza-bicyclo[3.2.1]octane derivatives useful as monoamine neurotransmitter re-uptake inhibitors. In other aspects the invention relates to the use of these compounds in a method for therapy and to pharmaceutical compositions c... | 08/05/2008 |
| 7358244 | Azabicycloalkane compounds This invention provides compounds of formula I: wherein R1, R2, R3, R4, R5, R6 and R7 are as defined in the specification, or a pharmaceutically acc... | 04/15/2008 |
| 7321039 | Industrial process for preparing tropenol The invention relates to a new industrially useable process for preparing tropenol, optionally in the form of the acid addition salts thereof. ... | 01/22/2008 |
| 7199132 | Tropane analogs and methods for inhibition of monoamine transport New tropane analogs that bind to monoamine transporters are described, particularly, 8-aza, 8carbo and 8-oxo tropanes having 6- or 7-hydroxyl or ketone substituents. The compounds of the present invention can be racemic, pure R-enantiomers, or pure S-enantiomers. Ce... | 04/03/2007 |
| 7192969 | Ester derivatives This invention relates to compounds which exhibit selective muscarinic M3 receptor antagonism, have little side effects, are suitable for inhalation therapy and are useful as treating agents of respiratory system diseases, of the general formula (I); ... | 03/20/2007 |
| 7186731 | 2-cyanopyrrolidinecarboxamide compound A compound of the formula (I) or a pharmaceutically acceptable salt thereof: [wherein X1 and X2 each is independently lower alkylene; X | 03/06/2007 |
| 7148236 | Modulators of acetylcholine receptors The present invention relates to compounds that modulate neurotransmission by promoting the release of neurotransmitters such as acetylcholine, dopamine and norepinephrine. More particularly, the present invention relates to thio-bridged aryl compounds that are capa... | 12/12/2006 |
| 7094788 | Esters of hydroxyl-substituted nitrogen heterocycles, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions The present invention relates to new compounds of general formula 1 wherein X− and the groups A, B, R, R1, R2, R3, R3′, R4, R4′, ... | 08/22/2006 |
| 7094784 | High affinity ligands for nociceptin receptor ORL-1 Novel compounds of the formula or a pharmaceutically acceptable salt or solvate thereof, wherein: the dotted line represents an optional double bond; X1 | 08/22/2006 |
| 7041674 | Carbamic acid esters with anticholinergic activity A compound of formula 1 wherein X−, A, R1, R2, R3, and R4 may have the meanings given in the claims and in the specification, processes for preparing them, their... | 05/09/2006 |
| 7012142 | Process for preparation of bicyclic and polycyclic molecules The present application is directed to a method of synthesis of a bicyclic or polycyclic compound of formula I or formula II: in which E, G, Y, n, m, R, R1, R2, R3, R6, R | 03/14/2006 |
| 6891042 | Industrial process for preparing tropenol The invention relates to a new industrially useable process for preparing tropenol, optionally in the form of the acid addition salts thereof. ... | 05/10/2005 |
| 6790857 | Benzoylecgonine compositions and methods for producing them This invention provides a method for preparing a benzoylecgonine composition comprising the steps of: (a) contacting benzoylmethylecgonine and propylene glycol in the presence or absence of water to form a reaction mixture; (b) maintaining the reaction... | 09/14/2004 |
| 6747153 | Industrial process for preparing tropenol The invention relates to a new industrially useable process for preparing tropenol, optionally in the form of the acid addition salts thereof. ... | 06/08/2004 |
| 6610849 | Process for the manufacture of tropenol A process for preparing tropenol (I) ##STR1## or an acid addition salt thereof, the process comprising: (a) reducing a scopine ester of formula (II) ##STR2## wherein R is C1 -C4 -alkyl or C1 -C4 -alkylen... | 08/26/2003 |
| 6486323 | Process for producing optically active tropinonemonocarboxylic acid derivative An optically active tropinonemonocarboxylic acid ester derivative useful as an intermediate for synthesis of optically active tropane derivatives was obtained by reacting succindialdehyde with an organic amine and acetonedicarboxylic acid ester to obtain ... | 11/26/2002 |
| 6353106 | Process for the production of trifluoromethyltropanone cyanohydrin A process for the preparation of a compound of formula (I), the process comprising the steps of (i) adding a solution of a compound of formula (II) in aqueous hydrochloric acid to an aqueous solution of sodium cyanide at a temperature in the range -5 to 1... | 03/05/2002 |
| 6353105 | Tropane analogs and methods for inhibition of monoamine transport New tropane analogs that bind to monoamine transporters are described, particularly, 8-aza, 8carbo and 8-oxo tropanes having 6- or 7-substituents. The compounds of the present invention can be racemic, pure R-enantiomers, or pure S-enantiomers. Certain pr... | 03/05/2002 |
| 6350758 | Tropane derivatives and method for their synthesis A compound of formula (I) wherein R1 -R6 have any of the values defined in the specification are described, as well as pharmaceutical compositions comprising a compound of formula (I), and methods for preparing and using compounds of... | 02/26/2002 |
| 6323343 | Process for the preparation of 8-azabicyclo(3.2.1)octane derivatives A process for preparing a compound of formula (IV), wherein R1 is C1-4 alkyl, CH2 (C1-3 haloalkyl), benzyl, CH2 (C2-5 akenyl or CH2 (C2-5 alkynyl), which comprises red... | 11/27/2001 |
| 6262066 | High affinity ligands for nociceptin receptor ORL-1 Novel compounds of the formula ##STR1## or a pharmaceutically acceptable salt or solvate thereof, wherein: the dotted line represents an optional double bond; X1 is optionally substituted alkyl, cycloalkyl, aryl, heteroaryl or heterocycloalkyl; X | 07/17/2001 |
| 6239142 | 4-oxo-4,7-dihydro-thieno[2,3-b]pyridine-5carboxamides as antiviral agents The invention provides a compound of formula I: ##STR1## wherein R1, R2, R3, and R4 have any of the values defined in the specification, or a pharmaceutically acceptable salt thereof, as well as processes and in... | 05/29/2001 |
| 6228867 | Antagonists of gonadotropin releasing hormone There are disclosed compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men an... | 05/08/2001 |
| 6200957 | Antagonists of gonadotropin releasing hormone There are disclosed compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both men an... | 03/13/2001 |
| 6005110 | Process for the production of endotropine A process for the production of endotropine by catalytically reducing tropanone with hydrogen with Raney nickel or Raney copper. This process is conducted with tropanone in an aqueous solution absent of organic solvents, in a closed system, at atmospheric... | 12/21/1999 |
| 5990312 | Method for the preparation of esters of anhydroecgonine The present invention discloses compounds of the formula any mixture thereof, or a pharmaceutically acceptable salt thereof; wherein R, R3, and R4 each have the meanings set forth in the specification. The compounds possess valuable pharm... | 11/23/1999 |
| 5952505 | Process for preparing pure enantiomers of tropic acid esters Precursors of anticholinergically active quaternary compounds can be synthesized from optically active tropic acid by acetylation, conversion into the acid chloride, reaction with amino alcohols of formula (I) ##STR1## (as the methanesulphonate; Q an... | 09/14/1999 |
| 5804685 | Deazapurine derivatives: a new class of CRF1 specific ligands Disclosed are compounds of the formula ##STR1## wherein Ar represents an aryl or heteroaryl group; and R1, R2, R3, R4, and R5 represent organic or inorganic substituents, which compounds are highly se... | 09/08/1998 |
| 5780437 | Antagonists of gonadotropin releasing hormone There are disclosed compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both m... | 07/14/1998 |
| 5770180 | Bridge-substituted tropanes for methods of imaging and therapy Disclosed are bridge-substituted analogs of tropanes and benztropines as well as methods for: imaging of cocaine receptors; treatment of cocaine abuse; and imaging and treatment of Parkinson's disease.... | 06/23/1998 |
| 5677311 | Aminobenzoic acid derivatives To provide a compound which exhibits a serotonin antagonism and an acetylcholine release accelerating activity at a well-balanced activity ratio. An aminobenzoic acid derivative represented by the general formula (I) or (II) or a pharmacologically accepta... | 10/14/1997 |
| 5663345 | Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same The present invention relates to a novel class of benzoylecgonine, ecgonine and ecgonidine derivatives which are useful for preventing and treating immunoregulatory disorders, neuromuscular. disorders, joint disorders, connective tissue disorders, circula... | 09/02/1997 |
| 5622973 | Treatment of osteoporosis with substituted piperidines, pyrrolidines and hexahydro-1H-azepines in combination with bisphosphonates The present invention is directed to certain novel compounds identified as di- and tri-substituted piperidines, pyrrolidines, and hexahydro-1H-azepines of the general structural formula: ##STR1## wherein R1, R4, R5, A... | 04/22/1997 |
| 5583142 | Analgesic and nootropic drugs Compounds of general formula: ##STR1## where: Ar=phenyl or beta-naphtyl, or aromatic heterocyclic 6-membered ring containing one or two nitrogen atoms; R1 =one or more substituents of the Ar nucleus, preferably in para position, and select... | 12/10/1996 |
| 5559123 | Derivatives of benzoylecgonine, ecgonine and ecgonidine and methods for preparing and using same The present invention relates to a novel class of benzoylecgonine, ecgonine and ecgonidine derivatives which are useful for preventing and treating immunoregulatory disorders, neuromuscular disorders, joint disorders, connective tissue disorders, circulat... | 09/24/1996 |
| 5416092 | 3-azabicyclo[3.2.1]-oct-8-yl-terminated non-peptidyl -succinamidoacyl aminodiols as anti-hypertensive agents Non-peptidyl compounds characterized generally as -succinamidoacyl aminodiols having a 3-azabicyclo[3.2.1]-oct-8-yl-type group at the N-terminus are useful as renin inhibitors for the treatment of hypertension.... | 05/16/1995 |
| 5389643 | Aminobenzoic acid derivatives useful for treating gastro-intestinal conditions An aminobenzoic acid derivative represented by the following general formulas (I), (I-2) or (I-3), or a pharmacologically acceptable salt thereof, which exhibits a serotonin antagonism and an acetylcholine release accelerating activity at a well-balanced ... | 02/14/1995 |
| 5376667 | Derivatives of benzoylecgonine, ecgonine and their multiple pharmacological properties The present invention relates to a novel class of benzoylecgonine, ecgonine and ecgonidine derivatives which are useful for preventing and treating immunoregulatory disorders, neuromuscular disorders, joint disorders, connective tissue disorders, circulat... | 12/27/1994 |
