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Patent No. 5678617

Method and apparatus for making a drink hop along a bar or counter

A method for generating a drink which appears to hop from a remote spot on the bar or counter and take one or more leaps, before landing in a patron's glass.

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Class 546/106 - The nitrogen is part of a substituent which contains additional nonionically bonded nitrogen


Subclass of Class 546 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the nitrogen is a member of a group containing
No. of patents: 65
Last issue date: 03/22/2011


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NumberTitleIssue Date
7910739Acetylcholinesterase dual inhibitors
The invention provides compounds of formula: which have a tacrine moiety connected to an heterocyclic moiety through a linker. Through careful selection of the substituents and the linker, the activity and selectivity towar...
03/22/2011
7605265Heterodimers and methods of using them
Novel heterodimers of tetrahydroacridines and tetrahydroquinolinones are disclosed. The heterodimers are capable of acting as both acetylcholinesterase inhibitors and N-methyl-D-aspartate (NMDA) receptor antagonists. The heterodimers may be used to improve cognitive...
10/20/2009
72301059-aminoacridine derivatives and process for the preparation thereof
The present invention relates to a new 9-aminoacridine derivative which exhibits prominent antitumor activity and low toxicity. ...
06/12/2007
6869974Pharmaceutical compounds
Compounds or their salts having general formulas (I) and (II): wherein s is an integer equal to 1 or 2, A is the radical of a drug that satisfies certain pharmacological tests, C and C1 are bivalent radicals, and precursors of the radicals B and B1
03/22/2005
68219835-(9-acridinylamino)-toluidine compounds
This invention relates to 9-anilinoacridine compounds, and more particularly to their synthesis and their use in pharmaceutical compositions for treating diseases. ...
11/23/2004
66209369-aminoacridine derivatives and process for the preparation thereof
The present invention relates to new 9-aminoacridine derivatives of general formula (I), wherein A is hydrogen or (II) (wherein X is oxygen or sulfur, R1, R2, R3, R4 and R5 are independently hydrogen, ...
09/16/2003
6489336Nitrogen-containing tricyclic compounds and drugs containing the same
A phenothiazine, acridan, acridone oxime, acridone hydrazone and dibenzodiazepine derivative represented by formula (I) ##STR1## effective against diseases in which histamine, leukotrienes, etc. participate and effective in preventing or treating diseases...
12/03/2002
6262104Diarylalkenylamine derivatives
Compounds, or solvates or salts thereof, of formula (I): ##STR1## selective delta opioid agonists and antagonists and may be of therapeutic utility as analgesics, immunosuppressants to prevent rejection in organ transplant and skin graft, anti-allergic an...
07/17/2001
6262265Non-hydrolyzable analogs of heroin metabolites suitable for use in immunoassay
Novel chemical analogs are disclosed for the essential heroin metabolite 6-O-acetyl morphine (6MAM). The analogs optionally can be made to contain protein reactive groups, and can be used to form protein conjugates, fluorescently labeled compounds, and so...
07/17/2001
62487509-hydroxyamino tetrahydroacridine and related compounds
There are disclosed compounds having the formula ##STR1## wherein n is 1-4; X is hydrogen, loweralkyl, cycloalkyl, loweralkoxy, halogen, hydroxy, nitro, trifluoromethyl, formyl, loweralkylcarbonyl, arylcarbonyl, --SH, loweralkylthio, --NHCOR2 o...
06/19/2001
6242459Substituted bis-acridines and related compounds as CCR5 receptor ligands, anti-inflammatory agents and anti-viral agents
This invention relates to substituted bis-acridines and related compounds which are ligands, in particular, antagonists of the CCR5 receptor. In addition, this invention relates to the treatment and prevention of disease states mediated by CCR5, including...
06/05/2001
6207673Covalent conjugates of topoisomerase I and topoisomerase II inhibitors
The present invention provides covalent conjugates of topoisomerase I and topoisomerase II inhibitors. Such compounds have a structure according to formula I: TI --L--TII (I) wherein: TI is a topoisomerase I inhibitor such as ...
03/27/2001
6197825Azulenyl nitrone spin trapping agents, methods of making and using same
The present invention relates to chromotropic nitrone spin trapping agents, methods of making these agents, compositions comprising same, and methods of their use. In particular, azulenyl nitrones of the present invention are effective agents for trapping...
03/06/2001
6194403Tacrine derivatives for treating Alzheimer's disease
A series of tacrine derivatives has be synthesized and disclosed. These tacrine derivatives were claimed to be new and be useful for the treatment of Alzheimer's disease alone or in combination with other drugs for Alzheimer's disease. These tacrine deriv...
02/27/2001
6187787Bis(9-aminoacridine) DNA intercalating agents having antitumor activity
A series of bis-acridinyl DNA intercalating agents with anticancer cell activity represented by formula (I), where Z is a linear arrangement of multiple aromatic rings, containing at least three aromatic rings, or at least two alicyclic rings, said rings ...
02/13/2001
6093725Frangible compounds for pathogen inactivation
Compounds and methods for inactivating pathogens in materials are described, including compositions and methods for inactivating pathogens in biological materials such as red blood cell preparations and plasma. The compounds and methods may be used to tre...
07/25/2000
6083988Azulenyl nitrone spin trapping agents, methods of making and using same
The present invention relates to chromotropic nitrone spin trapping agents, methods of making these agents, compositions comprising same, and methods of their use. In particular, azulenyl nitrones of the present invention are effective agents for trapping...
07/04/2000
60751449-hydroxyamino tetrahydroacridine and related compounds
There are disclosed compounds having the formula ##STR1## wherein n is 1-4; X is hydrogen, loweralkyl, cycloalkyl, loweralkoxy, halogen, hydroxy, nitro, trifluoromethyl, formyl, loweralkylcarbonyl, arylcarbonyl, --SH, loweralkylthio, --NHCOR2
06/13/2000
5939428Alkyl N-›3-(acridin-9-yl)amino-5-hydroxymethyl! phenylcarbamates
The invention provides a compound of the following formula: ##STR1## wherein R1 is C1-6 alkyl; or phenyl; R2 is hydrogen; an acyl group of the formula --CORa wherein Ra is C1-6 alkyl or phe...
08/17/1999
5886185Polyamine-linked acridine dimers
A series of novel polyamine-linked acridine dimers and derivatives thereof are described. The polyamine-linked acridine dimers and derivatives are potential anti-cancer agents....
03/23/1999
56727079-aminoacridine derivatives possessing psychotropic, antiamnestic and lipid-regulative activity
"Derivatives of 9-aminoacridine characterized by psychothropic, antiamnestic and lipid-regulating activities". New chemical compounds derived of 9-aminoacridine with a general formula are presented: ##STR1## where R=H or CH3 R1 ...
09/30/1997
5602142DNA-affinic hypoxia selective cytotoxins
Hypoxia selective cytotoxins having the structural formula ##STR1## wherein D, E, F and G, independently, are carbon or nitrogen, with the proviso that three or more of D, E, F and G are carbon; R1 and R2, independently, are sel...
02/11/1997
5569763Hydrazone compound and the use thereof
Hydrazone compound useful as an excellent organic nonlinear optical material and a highly sensitive coloring chelation agent, represented by the following formula (1): ##STR1## wherein Ar is a substituted or an non-substituted 2-imidazolyl group, a ...
10/29/1996
55367284-acylaminopyridine derivative
A novel 4-acylaminopyridine derivative represented by the following formula (I) is disclosed. ##STR1## The 4-acylaminopyridine derivative of the present invention is useful as a medicine for treating disturbances of memory such as senile dementia and...
07/16/1996
5512667Trifunctional intermediates for preparing 3'-tailed oligonucleotides
Oligonucleotides having a low molecular weight tail molecules joined to the 3' terminus of the oligonucleotide via a linking molecule of the structure: Z is ##STR1## wherein ##STR2## m and m' are positive integers less than 11, n is 0 or 1...
04/30/1996
5478837Use of quinacrine in preventing adhesion formation
Compositions and methods for prevention of adhesion formation, whereby an effective amount of quinacrine as active agent is administered for a period of time sufficient to permit tissue repair. The active agent is preferably administered in conjunction wi...
12/26/1995
53548643-(9-acridinylamino)-5-hydroxymethylaniline derivatives as anticancer agents
The present invention provides a compound having the structure: ##STR1## wherein R1 and R2 are independently the same or different and are hydrogen, an acetyl group; an acyl group having the formula --CO(CH2)n
10/11/1994
5312820Substituted carbamoyl and oxycarbonyl derivatives of biphenylmethylamines
Carbamoyl and oxycarbonyl derivatives of biphenylmethylamines of structure I are angiotensin-II antagonists with balanced AT1 and AT2 activity useful in the treatment of hypertension and related disorders and ocular hypertension. ...
05/17/1994
5294715Acridine-intercalator based hypoxia selective cytotoxins
Hypoxia selective cytotoxins of the general formula ##STR1## wherein n is from 1 to 5, and NO2 is in at least one of the 2, 4 or 5-positions of the imidazole. Such compounds have utility as radiosensitizers and chemosensitizers....
03/15/1994
5204348Heterocyclic compounds and anticancer-drug potentiaters conaining them as effective components
Novel heterocyclic compounds, which are represented by the following general formula, useful as anticancer drug potentiaters having a potentiating effect on the incorporation of anticancer drugs into cancer cells, the compounds each synthesized by, for ex...
04/20/1993
51207451-dimethylcarbamoyl-3-substituted-5-substituted-1H-1,2,4-triazoles
This invention relates to 1-dimethylcarbamoyl-3-substituted-5-substituted-1H-1,2,4-triazoles of the formula ##STR1## wherein the substituents are as defined herein, compositions containing those compounds and methods of use....
06/09/1992
5100904Prolinal compounds which are useful in treating amnesia
A novel prolinal derivatives of the general formula: ##STR1## [wherein A represents alkylene or alkenylene group of from 1 to 8 carbon atom(s) or a saturated hydrocarbon ring of from 3 to 7 carbon atoms, R represents hydrogen atom, phenyl group, benzyl gr...
03/31/1992
5089615Compound, 5,6,7,8-tetrahydro-1-(1,2,3,4-acridin-9-yl)-2H-3,1-benzoxazine-2,4-(1H)d ione
There are described compounds of the formula ##STR1## where X is hydrogen, loweralkyl, loweralkoxy or halogen; R when present is hydrogen, loweralkyl or aryloweralkyl; R1 is hydrogen, loweralkyl or arylloweralkyl; and R2 when present is h...
02/18/1992
4999358(1,2,3,4-tetrahydro-9-acridinimino)cyclohexane carboxylic acid and related compounds
There are described compounds of the formula, ##STR1## where X is hydrogen, loweralkyl, loweralkoxy or halogen; R when present is hydrogen, loweralkyl or arylloweralkyl; R1 is hydrogen, loweralkyl or arylloweralkyl; and R2 when present is...
03/12/1991
49854309-acylamino-tetrahydroacridine derivatives and memory enhancing agent containing said derivative as active ingredient
There are disclosed a 9-acylamino-tetrahydroacridine derivative represented by the following formula (I): ##STR1## wherein R ##STR2## are as defined in the specification, its optical antipode or pharmaceutically acceptable acid addition sa...
01/15/1991
4952589Pyridine compounds
This invention relates to aminoalkylphenoxyalkyl substituted heterocycles. These compounds antagonize the action of histamine on histamine H2 -receptors in the brain. A compound of the invention is 2-[3-[3-(piperidinomethyl)phenoxy]propylamino]...
08/28/1990
4916135N-heteroaryl-4-quinolinamines
There are described compounds of the formula ##STR1## where --R is ##STR2## --R3 and R3 being independently --H, loweralkyl, --CHO, --CH.dbd.CH2, --CH.dbd.CH--loweralkyl, --CH.dbd.CHCO2 C2 ...
04/10/1990
4851536Cyclohexylquinolines as inhibitors of interleukin 1
There are disclosed compounds of the formula ##STR1## wherein X is O, S, SO, SO2 or CR1 R2 ; R1 and R2 are each independently hydrogen, lower alkyl, carboxyl, lower alkoxy carbonyl, lower cycloalkyl, ...
07/25/1989
48393649-Amino-3,4-dihydroacridines and related compounds useful for enhancing memory
There are disclosed compounds having the formula ##STR1## wherein n is 1, 2 or 3; X is hydrogen, loweralkyl, loweralkoxy, halogen, hydroxy, nitro, trifluoromethyl, NHCOR2 where R2 is loweralkyl, or NR3 R4 w...
06/13/1989
4834769Compositions for the dyeing of leather
Dye compositions containing (a) at least one blue sulpho group-containing triphendioxazine dye and (b) at least one blue sulpho group-containing anthraquinone dye and preferably (c) lignine sulphonic acid or a salt of it and optionally (d) a non-ionic ble...
05/30/1989
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