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Patent No. 6049912

Mountable Printable Placard With Headband

A resilient headband in a shape for being mounted on the head of the user. The headband is equipped with a longitudinal slotted member for holding a placard.

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Class 546/103 - Chalcogen bonded directly to ring carbon of the six-membered hetero ring


Subclass of Class 546 - Organic compounds -- part of the class 532-570 series
Definition: Compounds in which chalcogen (i.e., oxygen, sulfur, selenium,
No. of patents: 117
Last issue date: 11/09/2010


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NumberTitleIssue Date
7829714Method for measuring aromatase activity
The present invention relates to compounds useful for measuring aromatase activity. The invention further provides methods for measuring aromatase activity and for screening test agents which modulate aromatase activity. A kit is also provided for use in such screen...
11/09/2010
7579468Methods of modulating neurotrophin-mediated activity
Disclosed are compositions which modulate the interaction with nerve growth factor and precursors thereof with neurotrophic receptors. Also disclosed are methods of using the compositions of the invention, including methods of administration. ...
08/25/2009
7351807Cyanine-sulfenates for dual phototherapy
Dye-sulfenate derivatives and their bioconjugates for dual phototherapy of tumors and other lesions. The compounds comprise sulfenates having the formula, t,0080 where E is selected from the group consisting of somatostatin receptor binding molecules, heat se...
04/01/2008
7338533Methods of fire retarding textiles with aqueous suspensions of pentabromobenzyl acrylate
A process for the fire retardation of textile materials comprising applying to the textile materials aqueous suspensions of finely ground pentabromobenzyl acrylate particles, suspending agents chosen from xanthan gums, anionic purified suspending agents, nonionic pu...
03/04/2008
7312209Acridone inhibitors of IMPDH enzyme
Compounds having the formula (I), wherein R3 is selected from H, OH and NH2; R30 is selected from ═O and ═S; W is —C(═O)—, —S(═O)—, or —S(O)2—; or W...
12/25/2007
7214684Methods for the treatment of allergic rhinitis
Methods are disclosed utilizing DCL, a metabolic derivative of loratadine, for the treatment of allergic rhinitis, and other disorders, while avoiding the concomitant liability of adverse side-effects associated with other non-sedating antihistamines. ...
05/08/2007
7211582Methods for treating urticaria using descarboethoxyloratadine
Methods are disclosed utilizing DCL, a metabolic derivative of loratadine, for the treatment of allergic rhinitis, and other disorders, while avoiding the concomitant liability of adverse side-effects associated with other non-sedating antihistamines. ...
05/01/2007
7160896Therapeutic acridone and acridine compounds
The present invention pertains to acridone and acridine compounds of formula (I), wherein either: (a) K is ═O, L is —H, alpha single bond, beta is a double bond, gamma is a single bond (acridones); or, (b) K is a 9-substituent, L is absent, alpha is a double bon...
01/09/2007
7144843Pest controllers
An objective of the present invention is to provide a harmful organism control agent that possesses excellent control effect against harmful organisms and can be safely used. The present invention provides a compound of formula (1) or a salt thereof. The present inv...
12/05/2006
70676684-quinolinol derivatives and fungicides containing the same as an active ingredient used for agriculture and horticulture
A new agricultural and horticultural fungicide having an excellent control effect is provided. 4-Quinolinol derivatives represented by the following formula: or agriculturally and horticulturally acceptabl...
06/27/2006
7022855Halogen-substituted quinoline derivatives and ectoparasite control agent
An objective of the present invention is to provide an ectoparasite control agent for homothermic animals, which has high control effect and is safe. The compounds according to the present invention are compounds represented by formula (I) and salts thereof:
04/04/2006
6936638Ligands of adenine nucleotide translocase (ANT) and compositions and methods related thereto
Compounds which have utility in the treatment of conditions associated with altered mitochondrial function. The compounds have the following structure (I): including stereoisomers, prodrugs, and pharmaceutically accept...
08/30/2005
6900322Method for stereochemically controlled production of isomerically pure highly substituted azacyclic compounds
A method for stereochemically controlled production of azacyclic compounds of general formula (I) in which the substituents have the meanings given in the specification. The invention also relates to intermediate produ...
05/31/2005
6872828Compounds for generating chemiluminescence with a peroxidase
Novel compounds comprising a C—C double bond substituted at one carbon with two sulfur atom-containing groups are disclosed. The compounds are useful in methods and compositions for generating chemiluminescence rapidly by reaction with a peroxidase enzyme and a pe...
03/29/2005
6858733Compounds for generating chemiluminescence with a peroxidase
Novel compounds comprising a C—C double bond substituted at one carbon with two sulfur atom-containing groups are disclosed. The compounds are useful in methods and compositions for generating chemiluminescence rapidly by reaction with a peroxidase enzyme and a pe...
02/22/2005
68219835-(9-acridinylamino)-toluidine compounds
This invention relates to 9-anilinoacridine compounds, and more particularly to their synthesis and their use in pharmaceutical compositions for treating diseases. ...
11/23/2004
6706722Heteroaryl derivatives and their use as medicaments
The invention relates to novel acridine derivatives of formula 1, to their preparation and to their use as medicaments, in particular for treating tumors. ...
03/16/2004
66802824-Quinolinol derivatives and agrohorticultural bactericides containing the same as active ingredient
A new agricultural and horticultural fungicide having an excellent control effect is provided. 4-Quinolinol derivatives represented by the following formula: ##STR1## or agriculturally and horticulturally acceptable acid addition salts thereof....
01/20/2004
6630481Viologen linked acridine based molecule and process for the preparation thereof
The present invention provides a series of novel bifunctional molecules based on viologen linked acridine, bisacridine and bisacridinium salts of the general formula 1 (1a, 1b, 1c and 1d) and or pharmaceutically acceptable derivatives thereof, which can b...
10/07/2003
6608066Tissue factor antagonists and methods of use thereof
The invention includes pharmaceutically active compounds and methods of treatment and pharmaceutical compositions that utilize or comprise one or more such compounds. Compounds of the invention are particularly useful for treating or prophylaxis of undesi...
08/19/2003
6489336Nitrogen-containing tricyclic compounds and drugs containing the same
A phenothiazine, acridan, acridone oxime, acridone hydrazone and dibenzodiazepine derivative represented by formula (I) ##STR1## effective against diseases in which histamine, leukotrienes, etc. participate and effective in preventing or treating diseases...
12/03/2002
6417178Amyloid binding nitrogen-linked compounds for the antemortem diagnosis of alzheimer's disease, in vivo imaging and prevention of amyloid deposits
Amyloid binding compounds which are derivatives of Chrysamine G, pharmaceutical compositions containing, and methods using such compounds to identify Alzheimer's brain in vivo and to diagnose other pathological conditions characterized by amyloidosis, suc...
07/09/2002
6410732Processing and synthetic intermediates for preparing N-arylacridancarboxylic acid derivatives
Synthetic processes and intermediates are disclosed for the preparation of N-arylacridancarboxylic acid derivatives. The derivatives are esters, thioesters, amides and sulfonimides. A key feature of the processes is the preparation of N-aryl substituted i...
06/25/2002
6248891Synthesis of acridine derivative multidrug-resistant inhibitors
Synthesis of the MDRI of formula (I) from intermediates of acridone acid of formula (II) and aminophenethyl isoquinoline of formula (III), via steps including coupling and conversion to yield the MDRI of formula (I)....
06/19/2001
6242459Substituted bis-acridines and related compounds as CCR5 receptor ligands, anti-inflammatory agents and anti-viral agents
This invention relates to substituted bis-acridines and related compounds which are ligands, in particular, antagonists of the CCR5 receptor. In addition, this invention relates to the treatment and prevention of disease states mediated by CCR5, including...
06/05/2001
6229015Acridone derivatives and method of preparation of 8-hydroxy imidazoacridinone derivatives
A process of preparing a compound of formula (I): ##STR1## wherein R1 and R2 are alkyl groups of 1 to 4 carbon atoms and n is from 2 to 5, comprises reacting a 1-chloro-7-(protected hydroxy)-4-nitroacridin-9(10H)-one of formula (IV-P...
05/08/2001
6168776Alkyl, alkenyl and alkynyl Chrysamine G derivatives for the antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition
Amyloid binding compounds which are non-azo derivatives of Chrysamine G, pharmaceutical compositions containing, and methods using such compounds to identify Alzheimer's brain in vivo and to diagnose other pathological conditions characterized by amyloido...
01/02/2001
6133259Alkyl, alkenyl and alkynyl chrysamine G derivatives for inhibition of cell degeneration and toxicity associated with amyloid deposition
Amyloid binding compounds which are non-azo derivatives of Chrysamine G, pharmaceutical compositions containing, and methods using such compounds to identify Alzheimer's brain in vivo and to diagnose other pathological conditions characterized by amyloido...
10/17/2000
6126870Chemiluminescent labeling compounds
Chemiluminescent labeling compounds and chemiluminescent labeled conjugates are provided. The compounds comprise an acridan ring bearing an exocyclic double bond and further contain a labeling substituent which permits attachement to compounds of interest...
10/03/2000
6117869Compounds for and methods of inhibiting matrix metalloproteinases
The present invention relates to compounds of Formula I that inhibit matrix metalloproteinases and to a method of inhibiting matrix metalloproteinases using the compounds ##STR1## More particularly, the present invention relates to a method of treati...
09/12/2000
6111109Process for the preparation of N-[2-(dimethylamino)ethyl]acridine-4-carboxamide
A process for producing an acridine carboxamide of formula (I): ##STR1## wherein each of R1, R2, R5 and R6, which may be the same or different, is H or an organic subsituent, x is from 1 to 6 and Y is N(R)2...
08/29/2000
6066632Heterocyclic compounds
The present invention relates to novel N-substituted azaheterocyclic compounds of the general formula ##STR1## wherein X, Y, Z, R1, R2 and r are as defined in the detailed part of the present description, or salts thereof, to me...
05/23/2000
6063847Thrombin receptor antagonists
Heterocyclic-substituted tricyclics of the formula ##STR1## or a pharmaceutically acceptable salt thereof, wherein: the single dotted line represents an optional double bond; the double dotted line represents an optional single bond; n is 0-2; Q is option...
05/16/2000
6045727Compounds, compositions and methods for generating chemiluminescence with phosphatase enzymes
Novel heterocyclic compounds which generate chemiluminescence on reaction with a phosphatase enzyme are provided as well as a process for their preparation and intermediates useful therein. The compounds comprise a nitrogen, oxygen or sulfur-containing he...
04/04/2000
6022970Process for preparing 2-anilinoacridones
An improved process for the preparation of optionally substituted 2-anilinoacridones from optionally substituted 2,5-dianilinoterephthalic acids, comprises: (a) cyclizing 2,5-dianilinoterephthalic acid to give an intermediate product mixture which contain...
02/08/2000
6018047Acridinium compounds as chemiluminogenic label
New acridinium compounds are provided which comply with formula 1, wherein A is a divalent organic moiety, such as an alkylene chain, X is a group which can be transformed together with C-9 of the acridine into a dioxetane by reaction with hydrogen peroxide, such a...
01/25/2000
5834462Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives
Novel tricyclic heterocyclic sulfonamide derivatives and sulfonic ester derivatives which have each an antitumor action and are represented by the following general formula (I) and processes for producing the same are provided. These compounds have each a...
11/10/1998
5721254N-substituted azaheterocyclic carboxylic acids and esters thereof
The present invention relates to novel N-substituted azaheterocyclic carboxylic acids and esters thereof in which a substituted alkyl chain forms part of the N-substituent or salts thereof, to methods for their preparation, to compositions containing them...
02/24/1998
5693649N-substituted azaheterocyclic carboxylic acids and esters thereof
The present invention relates to novel N-substituted azaheterocyclic carboxylic acids and esters thereof in which a substituted alkyl chain forms part of the N-substituent or salts thereof, to methods for their preparation, to compositions containing them...
12/02/1997
5688788N-substituted azaheterocyclic carboxylic acids and esters thereof
The present invention relates to novel N-substituted azaheterocyclic carboxylic acids and esters thereof in which a substituted alkyl chain forms part of the N-substituent or salts thereof, to methods for their preparation, to compositions containing them...
11/18/1997
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