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| Number | Title | Issue Date |
| 7427614 | Prostaglandin analogs Compounds comprising or a pharmaceutically acceptable salt or a prodrug thereof is disclosed herein. A, X, J, E, and Z are as described herein. These compounds are useful for treating diseases. ... | 09/23/2008 |
| 7399760 | Pyrimidinedione derivatives Pyrimidinedione derivatives of the general formula (I), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them are useful for the tre... | 07/15/2008 |
| 7351849 | Process for producing optically active β-amino acid derivatives The present invention is to provide a method for producing the desired optically active β-amino acid derivatives of high optical purities in high yields, without requiring a step of deprotection. More particularly, the present invention relates to a method for prod... | 04/01/2008 |
| 7279582 | Retroviral protease inhibiting compounds A compound of the formula: is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed. ... | 10/09/2007 |
| 7101873 | Pyrimidinedione derivatives Pyrimidinedione derivatives of the general formula (I), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts and pharmaceutically acceptable compositions containing them are useful for the tre... | 09/05/2006 |
| 7094778 | Heterocyclylalkylamines as muscarinic receptor antagonists This invention relates to compounds which are generally muscarinic M2/M3 receptor antagonists and which are represented by Formula I: wherein X, Y, and Z are O, S or NR5, and the other substituents are... | 08/22/2006 |
| 7087676 | Blocked polyisocyanates Blocked polyisocyanates and one-component stoving systems containing these blocked polyisocyanates, and the preparation thereof and their use for the preparation of lacquers, paints, adhesives and elastomers, wherein blocked polyisocyanates are prepared by reacting ... | 08/08/2006 |
| 7074852 | Blocked polyisocyanates Blocked polyisocyanates and one-component stoving systems containing these blocked polyisocyanates, and the preparation thereof and their use for the preparation of lacquers, paints, adhesives and elastomers. The blocked polyisocyanates are derived from polyisocyana... | 07/11/2006 |
| 7057038 | Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids One aspect of the present invention relates to a method for the kinetic resolution of racemic and diastereomeric mixtures of chiral compounds. The critical elements of the method are: a non-racemic chiral tertiary-amine-containing catalyst; a racemic or diastereomer... | 06/06/2006 |
| 7053085 | EP receptor agonist, compositions and methods thereof This invention relates to potent selective agonists of the EP4 subtype of prostaglandin E2 receptors, their use or a formulation thereof in the treatment of glaucoma and other conditions, which are related to elevated intraocular pressure in the eye of a ... | 05/30/2006 |
| 7038039 | Process for selectively producing 1-phosphorylated sugar derivative anomer and process for producing nucleoside A desired isomer is selectively prepared by phosphorolyzing and isomerizing an anomer mixture of a 1-phosphorylated saccharide derivative while crystallizing one of the isomers to displace the equilibrium. Furthermore, using the action of a nucleoside phosphorylase,... | 05/02/2006 |
| 6946460 | Azole or triazole derivatives, method for preparing same and use thereof as fungicides The invention concerns novel azole or triazole derivatives of formula (I), wherein X, Ar1, Ar2, Ar3, A, B, and R1 are as defined herein, their preparation method and their use as fungicides. | 09/20/2005 |
| 6900161 | Azole or triazole derivatives, method for preparing same and use thereof as fungicides The invention concerns novel azole or triazole derivatives of formula (Ia) or (Ib), wherein: X, Ar1, Ar2, Ar3, A, B and R1 are such as defined in the description, the method for preparing same and their use as fungicides. ... | 05/31/2005 |
| 6858727 | Intermediate of carbapenem antibiotics and process for the preparation thereof There is disclosed an azetidinone compound of the formula (I): wherein R is hydrogen, or a hydroxy protecting group, R1 and R2 are each independently alkyl of 1-15 carbon atoms, benzyl or cyclized... | 02/22/2005 |
| 6841668 | Polyoxometalate catalysts for the preparation of sterically hindered N-substituted aryloxyamines Sterically hindered N-substituted aryloxyamines are prepared by the Keggin polyoxometalate or the transition metal substituted polyoxometalate (TMS-POM) catalyzed decomposition of diazonium salts in the presence of a sterically hindered nitoxyl radical. These compou... | 01/11/2005 |
| 6759402 | Cyclic felbamate derived compounds The present invention relates to novel felbamate derivatives and their use to treat neurological diseases such as epilepsy and to treat tissue damage resulting form ischemic events. The felbamate derivatives are modified to prevent the formation of metabolites that ... | 07/06/2004 |
| 6743914 | Kinetic resolutions of chiral 2-and 3-substituted carboxylic acids One aspect of the present invention relates to a method for the kinetic resolution of racemic and diastereomeric mixtures of chiral compounds. The critical elements of the method are: a non-racemic chiral tertiary-amine-containing catalyst; a racemic or diastereomer... | 06/01/2004 |
| 6664253 | Neurokinin antagonists The invention relates to new compounds of formula I ##STR1## or the pharmaceutically acceptable salts thereof, wherein R1, R2, R3, R4, X and Ar1 have the meanings given in the specification, as well as... | 12/16/2003 |
| 6562967 | Kinetic resolutions of chiral 2-and-3-substituted carboxylic acids One aspect of the present invention relates to a method for the kinetic resolution of racemic and diastereomeric mixtures of chiral compounds. The critical elements of the method are: a non-racemic chiral tertiary-amine-containing catalyst; a racemic or d... | 05/13/2003 |
| 6562966 | Kinetic resolutions of chiral 2- and 3-substituted carboxylic acids One aspect of the present invention relates to a method for the kinetic resolution of racemic and diastereomeric mixtures of chiral compounds. The critical elements of the method are: a non-racemic chiral tertiary-amine-containing catalyst; a racemic or d... | 05/13/2003 |
| 6472529 | Retroviral protease inhibiting compounds A compound of the formula: ##STR1## is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.... | 10/29/2002 |
| 6469000 | 1,3-diheterocyclic metalloprotease inhibitors Disclosed are compounds which are inhibitors of metalloproteases having the following structure: ##STR1## where Ar, W, X, Y, Z, R1 and R2 have the meanings described in the specification and optical isomers, diastereomers, and enanti... | 10/22/2002 |
| 6407232 | Ionic metal complex and process for synthesizing same The invention relates an ionic metal complex represented by the general formula (1): ##STR1## wherein M is an element of groups 3-15 of the periodic table; Aa+ represents a metal ion, onium ion or proton; X1 represents O, S or N... | 06/18/2002 |
| 6365587 | Substituted aryl hydroxamic acids as metalloproteinase inhibitors The present application describes novel substituted aryl hydroxamic acids of formula I: ##STR1## or pharmaceutically acceptable salt forms thereof, wherein ring A is a 5-8 membered ring containing from 0-1 additional heteroatoms selected from N, O, a... | 04/02/2002 |
| 6355796 | Processes and intermediate compounds for the preparation of 2-(N,N-disubstituted) amino-4-(perfluoroalkyl)-1, 3- oxazin-6-one and 6-(perfluoroalkyl) uracil compounds An improved process and intermediate compounds for the preparation of 2-(N,N-disubstituted)amino-4-(perfluoroalkyl)-1,3-oxazin-6-one compounds having the structural formula I ##STR1## and an improved process for the preparation of 6-(perfluoroalkyl)uracil... | 03/12/2002 |
| 6340751 | Process for the preparation of 4-substituted azetidinone derivatives Disclosed is a process for the preparation of a 4-substituted azetidinone derivative, which comprises reacting an azetidinone derivative and an amide compound in the presence of a magnesium compound such as those represented by the following formulas (II)... | 01/22/2002 |
| 6265400 | Cyclic carbamates and isoxazolidines as IIb/IIIa antagonists The present invention relates generally to cyclic carbamates and isoxazolidines or Formula (I) ##STR1## or their pharmaceutically acceptable salts thereof, which are useful as antagonists of the platelet glycoprotein IIb/IIIa fibrinogen receptor comp... | 07/24/2001 |
| 6251897 | 6-phenyltetrahydro-1,3-oxazin-2-one derivative and pharmaceutical composition containing the same A 6-phenyltetrahydro-1,3-oxazin-2-one derivative having the formula (I): ##STR1## wherein, R1 is an unsubstituted or substituted C1 to C8 alkyl group; an unsubstituted or substituted C3 to C7 cycloalkyl ... | 06/26/2001 |
| 6235901 | Oxazoline or oxazine acetoacetate aqueous coating compositions A novel compound having the formula: ##STR1## wherein R is an alkyl group containing 1-5 carbon atoms or an aryl, substituted aryl, substituted or unsubstituted heteroaryl, alkyl-aryl, alkylether-aryl or O; R1 and R2 are hydrogen or ... | 05/22/2001 |
| 6166010 | Azine derivatives The invention relates to the use of azine derivatives, some of which are known, of the formula ##STR1## in which A represents substituted phenyl, or represents in each case optionally substituted naphthyl, pyridyl, thienyl or pyrazolyl; B represents ... | 12/26/2000 |
| 6159902 | Herbicides The invention relates to 1,3-oxazin-4-one derivatives of formula (I): ##STR1## and to their use as herbicides.... | 12/12/2000 |
| 6080857 | Method of preparation of ଲ-amino acids A method for the preparation of ଲ-amino acid compounds is provided. The method includes contacting an amine nucleophile with an ,ଲ-unsaturated amide compound in the presence of a chiral Lewis acid complex. The chiral Lewis acid complex ... | 06/27/2000 |
| 6046135 | 1,3-oxazin-4-one derivatives as herbicides 1,3-Oxazin-4-one derivatives of formula (I): ##STR1## wherein Q represents --C(.dbd.O)--, --CH(OH)-- or --C(OR11)(OR11)--, in which R11 represents lower alkyl; or the two groups --OR11, together with the ca... | 04/04/2000 |
| 6028224 | Fluoxetine process from benzoylpropionic acid A synthesis of fluoxetine is disclosed. The process begins with a lower alkyl ester of 3-benzoylpropionic acid, which is reduced in the presence of a chiral ligand to produce the corresponding γ-hydroxy ester, and the ester is cleaved. The free acid is t... | 02/22/2000 |
| 6028032 | 1,3-oxazin-4-one derivatives as herbicides 1,3-oxazin-4-ones of formula (I), ##STR1## wherein R1 represents phenyl optionally substituted; R2 represents: a straight- or branched-chain alkyl having from one to ten carbon atoms which is substituted by one or more groups R | 02/22/2000 |
| 5977025 | 1,3-oxazin-4-one derivative, herbicide containing same, and intermediate for preparing same This invention provides 1,3-oxazin-4-one derivatives represented by following general formula (I): ##STR1## in which R1 represents a phenyl group which may be substituted; R2 represents a hydrogen atom or a lower alkyl group; R | 11/02/1999 |
| 5977359 | Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present The invention relates to compounds of the formula ##STR1## in which: A is a divalent radical selected from: A1) --O--CO-- A2) --CH2 --O--CO-- A3) --O--CH2 --CO-- A4) --O--CH2 --CH | 11/02/1999 |
| 5972237 | Use of heterocyclic compounds as activators for inorganic peroxy compounds Heterocyclic compounds I R1 --X--L (I) where L is a cyclic carbamate residue, a lactonoxy residue or a lactam residue, X is an oxygen-containing group ##STR1## where A is a linker, and R1 is an ... | 10/26/1999 |
| 5932521 | Herbicidal 1,3-oxazin-4-one derivatives and intermediates thereto Novel 1,3-oxazin-4-one derivatives of the formula ##STR1## wherein R1 to R5 are hydrocarbyl radicals which are optionally substituted, and herbicidal compositions comprising the same as active ingredients and their use in contro... | 08/03/1999 |
| 5914332 | Retroviral protease inhibiting compounds A compound of the formula: ##STR1## is disclosed as an HIV protease inhibitor. Methods and compositions for inhibiting an HIV infection are also disclosed.... | 06/22/1999 |
