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Class 544/9 - Polycyclo ring system having the thiadiazine ring as one of the cyclos


Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the thiadiazine ring is one of the cyclos
No. of patents: 44
Last issue date: 08/28/2007


1    
NumberTitleIssue Date
7262190Benzothiazine and benzothiadiazine compounds
The invention relates to compounds of formula (I): wherein: R1 represents hydrogen, alkyl or cycloalkyl, R2 represents hydrogen, halogen or hydroxy, A ...
08/28/2007
7262189Benzothiazine and benzothiadiazine derivatives, method for preparing same and pharmaceutical compositions containing same
Compounds of formula (I): wherein: R1 represents aryl or heteroaryl, R2 represents hydrogen, halogen or hydroxy, X represents oxygen or sulphur, ...
08/28/2007
7253161Benzothiazine and benzothiadiazine derivatives method for preparing same and pharmaceutical compositions containing same
Compounds of formula (I): wherein: R1 represents aryl or heteroaryl, R2 represents hydrogen, halogen or hydroxy, A represents CR4R5
08/07/2007
7253163Benzothiazine and benzothiadiazine compounds
Compounds of formula (I): wherein: R1 represents a heterocycle, R2 represents hydrogen, a halogen or hydroxy, A represents CR4R5 ...
08/07/2007
7253162Benzothiazine and benzothiadiazine compounds
Compounds of formula (I): wherein: R1 represents hydrogen, a halogen or alkyl, R1a represents hydrogen or alkyl, R2 ...
08/07/2007
7244843Modulators of serotonin receptors
The present invention provides modulators of serotonin receptors, pharmaceutical compositions containing such modulators and methods for treating various diseases, conditions and disorders associated with modulation of serotonin receptors such as, for example: metab...
07/17/2007
7196194Dye-forming coupler, silver halide photographic light-sensitive material and azomethine dye compound
A yellow dye-forming coupler represented by formula (I): wherein Q represents a group of nonmetallic atoms that form a 5- to 7-membered ring in combination with the —N═C—N(R1)—; R1 and...
03/27/2007
6943158Diazinopyrimidines
Compounds of formula I are p38 inhibitors: or a pharmaceutically acceptable salt thereof, wherein R1 is hydrogen or alkyl; R2 alkyl, h...
09/13/2005
6943159Compounds and their use as positive AMPA receptor modulators
The invention provides novel compounds represented by general formula (I) wherein the bond represented by the broken line may be a single, double bond or absent; and if the bond is absent, then the nitrogen is substitu...
09/13/2005
6906063Platelet ADP receptor inhibitors
Novel compounds of formulae (I) to (VIII), which more particularly include sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives whi...
06/14/2005
6878711Indole derivatives as PDE5-inhibitors
Compounds of the general structural formula and use of the compounds and salts and solvates thereof, as therapeutic agents. ...
04/12/2005
6683028Cyclic guanidine derivatives and their use as pesticides
The invention relates to novel guanidine derivatives of the formula (I) ##STR1## in which A, R1, R2, R3 and Z are as defined in the description, to a process for their preparation and to their use for controlling animal ...
01/27/2004
6667306Platelet ADP receptor inhibitors
The invention relates to novel compounds of formula (I) containing fused heterocyclic ring systems which are effective platelet ADP receptor inhibitors: ##STR1## In formula (I), W is carbon or nitrogen, wherein at least one W is a carbon; and Y is ni...
12/23/2003
6635635Benzothiadiazine compounds
Compound of formula (I): ##STR1## wherein: R1 represents hydroxy, RCO--O-- or RCO--NRa --, R2 represents hydrogen, halogen, or hydroxy, R'CO--O or R'CO--NR'a --, R and R', which may be identical or differ...
10/21/2003
6624159Heterocycle carboxamides as antiviral agents
The present invention provides a compound of formula I ##STR1## which is useful as antiviral agents, in particular, as agents against viruses of the herpes family....
09/23/2003
6541469CRF receptor antagonists and methods relating thereto
CRF receptor antagonists are disclosed which have utility in the treatment of a variety of disorders, including the treatment of disorders manifesting hypersecretion of CRF in a warm-blooded animals, such as stroke. The CRF receptor antagonists of this in...
04/01/2003
6518422Process for the synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4] benzothiadiazine
Process for the industrial synthesis of (3aS)-5,5-dioxo-2,3,3a,4-tetrahydro-1H-pyrrolo[2,1-c][1,2,4]benzothiadiazi ne of formula (I): ##STR1## by enantioselective catalytic hydrogenation of 5,5-dioxo-2,3-dihydro-1H-pyrrolo[2,1-c][1,2,4]benzothiadiazin...
02/11/2003
5846969Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives
A sulfonamide derivative or a sulfonic ester derivative represented by the following general formula (I): ##STR1## {G represents an aromatic 5- or 6-membered ring; L represents O or --N(R1)-- (R1 represents hydrogen or lower alk...
12/08/1998
5817820Quinolone derivatives and processes for the preparation thereof
The present invention relates to optical isomers of quinoline compounds of Formula (IA) or Formula (IA'), their pharmaceutically acceptable salts and their intermediates: ##STR1## In the above formulae, A represent nitrogen or ##STR2## in w...
10/06/1998
5728693Arthropodicidal oxadiazine-thiadiazine-or triazine-carboxanilides
Arthropodicidal compounds, compositions and use of compounds having the formula ##STR1##...
03/17/1998
5602126Arthropodicidal anilides
Substituted anilides of formula (I), wherein Q is one of (Q-1), (Q-2) and (Q-3), and R1 to R5, Y, Z and Z1 are as defined in the text, arthropodicidal compositions containing such compounds; and a method for controlling ar...
02/11/1997
5536719Benzothiadiazine compound
A compound of formula (I): ##STR1## in the form of its S enantiomer, its addition salts with a pharmaceutically acceptable acid or base and medicinal product containing the same are useful for the treatment or prevention of pathologies associate...
07/16/1996
54038371,2,4-thiadiazino[3,4-b]benzothiazole derivatives, and medicinal products containing them
This invention relates to compounds of formula (I): ##STR1## wherein R is a polyfluoroalkoxy, polyfluoroalkyl, alkoxy or alkyl radical and R1 is a hydrogen atom or an alkyl radical; salts thereof; the preparation thereof; and drugs contain...
04/04/1995
5356862Herbicidal sulfonylureas
The invention relates to herbicidal sulfonylurea compounds, agriculturally suitable compositions thereof and a method for their use as general or selective preemergent or postemergent herbicides or plant growth regulants....
10/18/1994
5210209Pyrazolo(1,5-a)benzimidazole couplers
The invention provides a method for the production of a pyrazolo(1,5-a)benzimidazole of the general formula (A): ##STR1## wherein R is a substituted or unsubstituted alkyl or aryl group, and R1 -R4 =R, H, halogen, OR, COOR, CONHR, SO...
05/11/1993
5166348Bornyl and isobornyl esters of carboxylic acids of condensed tetrahydroquinoxalines
Bornyl and isobornyl esters of carboxylic acids of condensed tetrahydroquinoxalines having the general formula ##STR1## where R1 is CH3 or C2 H5 ##STR2## where R2 is ##STR3## The p...
11/24/1992
5162317Pyridinium salt and pharmacological composition containing the same
A pyridinium salt useful as an antiulcer agent, defined by formula (I) is disclosed. It includes a sulphenamide compound and a pyridinium compound. J is benzimidazole, K is --S-- or --SSR-- and Z is hydroxy or alkoxy. ##STR1##...
11/10/1992
5130313Serotonin antagonists, their preparation and medications containing them
This invention relates to compounds of formula: ##STR1## in which R1 denotes a 1,2,3,6-tetrahydro-1-pyridyl radical substituted in the 4-position by an optionally substituted phenyl, optionally substituted 3-indolyl or 3-(5-hydroxyindolyl)...
07/14/1992
4943570Benzimidazolesulfonamides and imidazopyridinesulfonamides, and their application as drugs
Benzimidazole-2-sulfonamide and imidazopyridine-2-sulfonamide derivatives corresponding to the general formula: ##STR1## and their pharmaceutically acceptable salts in which: Z1 to Z4 represent a nitrogen atom or a substituted o...
07/24/1990
4906628N-phenylpyridone type III phosphodiesterases
Phosphodiesterase (type III) inhibitors having the formula: ##STR1## which are useful in stimulating cardiac activity and in treating congestive heart failure and bronchoconstriction, pharmaceutical compositions including these inhibitors, and method...
03/06/1990
4861773Heterocyclic compounds
The invention relates to thiadiazinone derivatives that have utility as cardiac stimulants. A compound of the invention is 7-(1H-imidazol-1-yl)-9,9a-dihydroindeno[1,2-e][1,3,4]-thiadiazin-2(3H)-one ....
08/29/1989
4769456Sulfenamide derivatives and their production
The compound of the formula ##STR1## wherein R1 is hydrogen, methoxy or trifluormethyl, R2 and R3 are the same or different and are each hydrogen or methyl, R4 is a fluorinated lower alkyl having 2 to 5 car...
09/06/1988
4741765Herbicidal sulfonamides
Benzenesulfonamide compounds such as N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4 -oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide and N-[(4-methoxy-6-methyl-pyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl- 4-oxo-1-phe...
05/03/1988
4716161Phenylpiperazine derivatives and their acid addition salts
A phenylpiperazine derivative according to the present invention has the following general formula [I]: ##STR1## wherein R1, R2 and R3 are independently hydrogen or alkoxy group having 1 to 3 carbon atoms, or R1
12/29/1987
4678499Herbicidal sulfonamides
Benzenesulfonamide compounds such as N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4 -oxo-1-phenyl-indeno[1,2-C]-pyrazole-5-sulfonamide and N-[(4-methoxy-6-methyl-pyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl- 4-oxo-1-ph...
07/07/1987
4636499Sulphenamides
Novel compounds of the formula IIIa ##STR1## wherein R1a, R2a, R3a and R4a are the same or different and are hydrogen, an alkyl, alkoxy optionally completely or predominantly substituted by fluorine or chlo...
01/13/1987
4616013Fused thiadiazines
This invention relates to thiadiazinone derivatives which have inotropic and vasodilator activity. A specific compound of this invention is 7-acetamido-9,9a-dihydroindeno[1,2-e][1,3,4]thiadiazine-2(3H)-one....
10/07/1986
46123111,2,4-benzothiadiazine oxide derivatives
1,2,4-Benzothiadiazine oxide derivatives of the general Formula I ##STR1## in which R1 represents an unsubstituted or substituted aryl radical; R2 and R5, which may be the same or different, and represent hydrogen, halogen...
09/16/1986
41713611-Substituted-3-amino-6,7-dialkoxy-1H-1,2,4-benzothiadiazine-1-oxides
1-Substituted-3-amino-6,7-dialkoxy-1H-1,2,4-benzothiadiazine-1-oxides, useful as hypotensive agents....
10/16/1979
4035374Imidazolyl alkylaminopyridone and pyridinethione compounds
Heterocyclic compounds which are inhibitors of histamine activity, in particular, inhibitors of H-2 histamine receptors. A specific compound of this invention is 2-[2-(4-methyl-5-imidazolylmethylthio)ethylamino]-4-pyrimidone....
07/12/1977
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