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Patent No. 5823572

Self Defense Weapon With Memo

A self defense weapon formed as a memo pad and which is easily held by a person's fingers, therefore making it possible to provide protection from a mugger and also to quickly and easily write a record or a message without failure of missing or forgetting significant information under a stressful situation.

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Class 544/66 - Plural nitrogens in the six-membered hetero ring


Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the six-membered ring contains at least
No. of patents: 129
Last issue date: 12/27/2011


1        
NumberTitleIssue Date
8084603Naphthalenetetracarboxylic acid derivatives and their use as semiconductors
The present invention relates to naphthalenetetracarboxylic acid derivates, to a process for their preparation and to their use, especially as an n-type semiconductor. ...
12/27/2011
7384936Carboxamidine derivatives and their use in the treatment of vascular diseases
The invention relates to carboxamidine derivatives to pharmaceutical compositions containing the same and the use thereof in the preparation of pharmaceutical compositions for the treatment of vascular diseases. ...
06/10/2008
7229988Dialkylhydroxybenzoic acid derivatives containing metal chelating groups and their therapeutic uses
The present invention provides novel dialkylhydroxybenzoic acid derivatives containing metal chelating groups and the use of the novel compounds as therapeutics for treating and/or preventing various medical dysfunctions and diseases arising from reactive oxygen spe...
06/12/2007
7105661Process for manufacturing morpholino-nucleotides, and use thereof for the analysis of and labelling of nucleic acid sequences
The invention relates to the use of morpholino-nucleosides of formula: in which R1 represents a nucleic base and R2 represents a group corresponding to one of the following formulae:
09/12/2006
7087598Diamide invertebrate pest control agents containing a non-aromatic heterocyclic ring
This invention provides compounds of Formula I, their N-oxides and agriculturally suitable salts wherein A and B are independently O or S; J is an optionally substituted 5- or 6-memebered nonaromatic heterocyclic ring; K is taken together with the two contiguous lin...
08/08/2006
7081526Process for manufacturing morpholino-nucleotides, and use thereof for the analysis of and labelling of nucleic acid sequences
The invention relates to the use of morpholino-nucleosides of formula: in which R1 represents a nucleic base and R2 represents a group corresponding to one of the following formulae:
07/25/2006
6956129Polyhalogen-substituted cinnamic acids and cinnamic acid derivatives and a process for the preparation of polyhalogen-substituted cinnamic acids and cinnamic acid derivatives
Polyhalogenated cinnamic acids and cinnamic acid derivatives are prepared by reacting diazonium salts accessible from polyhalogenated anilines with acrylic acid or acrylic acid derivatives in the presence of a homogeneous, palladium-containing catalyst at about −5...
10/18/2005
6943158Diazinopyrimidines
Compounds of formula I are p38 inhibitors: or a pharmaceutically acceptable salt thereof, wherein R1 is hydrogen or alkyl; R2 alkyl, h...
09/13/2005
69169334-pyridinyl-n-acyl-l-phenylalanines
Compounds of Formula I have activity as inhibitors of binding between VCAM-1 and cells expressing VLA-4 and are useful for treating disease whose symptoms and or damage are related to the binding of VCAM-1 to cells expressing VLA-4. ...
07/12/2005
6867298Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
The present invention relates to copper-catalyzed carbon-heteroatom and carbon-carbon bond-forming methods. In certain embodiments, the present invention relates to copper-catalyzed methods of forming a carbon-nitrogen bond between the nitrogen atom of an amide or a...
03/15/2005
6838560Process for manufacturing morpholino-nucleotides, and use thereof for the analysis of and labelling of nucleic acid sequences
The invention relates to the use of morpholino-nucleosides of formula: in which R1 represents a nucleic base and R2 represents a group corresponding to one of the following formulae: ...
01/04/2005
6790955Processes for the preparation of aminophenylsulfonyl-ureas and intermediate products for the processes
The invention relates to the preparation of compounds (I) in which A═H or acyl and R1, R2, R3, R, n, X, Y and Z are as defined in claim 1 by halogenation and rearrangement of compounds ...
09/14/2004
6737525Electrophilic fluorination
N-fluorotriazinium salts, especially those of the following Formula I, are electrophilic fluorinating agents useful in fluorinating, preferably in a nitromethane solvent, carbanionic species and/or activated aromatic compounds: ...
05/18/2004
6734304Method for producing asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives
The invention relates to a novel process for preparing known asymmetrical 4,6-bis(aryloxy)pyrimidine derivatives. ...
05/11/2004
6683028Cyclic guanidine derivatives and their use as pesticides
The invention relates to novel guanidine derivatives of the formula (I) ##STR1## in which A, R1, R2, R3 and Z are as defined in the description, to a process for their preparation and to their use for controlling animal ...
01/27/2004
6639070N-substituted perhydrodiazine
N-substituted perhydro-2,3-diazines of the formula I ##STR1## in which the variables Z, R, m and RA are as defined in claim 1, a process for their preparation and the use of the compounds of the formula I as starting materials for preparing her...
10/28/2003
6635637Cyclic oxyguanidine protease inhibitors
Cyclic oxyguanidine compounds, including compounds of Formulae I and II: ##STR1## wherein R1, R3 -R6, R21 -R26, L, Y, Z, and A are set forth in the specification, as well as hydrates, solvates or phar...
10/21/2003
6624159Heterocycle carboxamides as antiviral agents
The present invention provides a compound of formula I ##STR1## which is useful as antiviral agents, in particular, as agents against viruses of the herpes family....
09/23/2003
6579982Pyrimidine-2,4,6-trione metalloproteinase inhibitors
The present invention relates to pyrimidine-2,4,6-trione metalloproteinase inhibitors of the formula ##STR1## wherein X, Y, Ar1, Z, R1, R2 and R3 are as defined in the specification, and to pharmaceutical compos...
06/17/2003
6552187Process for the preparation of herbicidal derivatives
##STR1## A process for the preparation of compounds of formula (I), which process comprises reacting a compound of formula (II), in an inert organic solvent, optionally in the presence of a base, with a compound of formula (IV), (IVa) or (IVb), and option...
04/22/2003
6541469CRF receptor antagonists and methods relating thereto
CRF receptor antagonists are disclosed which have utility in the treatment of a variety of disorders, including the treatment of disorders manifesting hypersecretion of CRF in a warm-blooded animals, such as stroke. The CRF receptor antagonists of this in...
04/01/2003
65182661- Aryl-3-thioalkyl pyrazoles, the synthesis thereof and the use thereof as insecticides
The present invention is directed to novel pyrazole derivatives and their use as pesticidal agents. The pyrazole derivatives have Formula I: ##STR1## or a salt thereof, where R1 represents R5 O, R5 SO2, R5...
02/11/2003
6476016Cyclic oxyguanidine pyrazinones as protease inhibitors
Cyclic oxyguanidine pyrazinone compounds are described, including compounds of the Formula I: ##STR1## wherein R3, R4, R5, W, and A are as set forth in the specification, as well as hydrates, solvates or pharmaceutically ...
11/05/2002
6432948USE OF 7-(2-OXA-5,8-DIAZABICYLCO[4.3.0]NON-8-YL)-QUINOLONE CARBOXYLIC ACID AND NAPHTHYRIDON CARBOXYLIC ACID DERIVATIVES FOR THE TREATMENT OF HELIOBACTER PYLORI INFECTIONS AND ASSOCIATED GASTRODUODENAL DISEASES
The invention relates to the use of quinolone- and naphthyridonecarboxylic acid derivatives, which are substituted in the 7-position by a 2-oxa-5,8-diazabicyclo[4.3.0]-non-8-yl) radical, and their pharmaceutically utilizable hydrates and/or salts for the ...
08/13/2002
6410482(Het) arylsulfonylureas having an amino function, their presentation and their use as herbicides and plant growth regulators
(Het)Arylsulfonylureas having an imino function, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## in which A is a (hetero)aromatic or heterocyclic bridge linked to the group...
06/25/2002
6384029Optically active pyridyl-4h-1,2,4-oxdadiazine derivative and its use in the treatment of vascular diseases
The invention relates to (-)-5,6-dihydro-5-(1-piperidinyl)-methyl-3-(3-pyridyl)-4H-1,2,4-oxadiazine to the therapeutical use thereof and to phamaceutical compositions containing the compounds as active ingredient....
05/07/2002
6346522Pesticides
Compounds of formula (I) or pesticidally acceptable salts thereof, compositions containing them and methods of use. ##STR1##...
02/12/2002
63425991,3,4-oxadiazine derivatives and their use as pesticides
The invention relates to a novel process of preparing (1,3,4)-oxadiazine derivatives of formula (I) and to their usefulness as pesticides in particular as anthelminticides, insecticides, acaricides, and nematicides....
01/29/2002
6288081Use of 7-(1-aminomethyl-2-oxa-7-aza-bicyclo[3.3.0]oct-7-yl)-quinolone carboxylic acid and naphthyridone carboxylic acid derivatives for treating Helicobacter pylori infections and the gastroduodenal diseases associated therewith
The invention relates to the use of quinolone- and naphthyridonecarboxylic acid derivatives which are substituted in position 7 by a 1-aminomethyl-2-oxa-7-azabicyclo[3.3.0]oct-7-yl radical, and of their salts for the therapy of Helicobacter pylori infecti...
09/11/2001
6251899Methoximinomethyloxadiazines
A compound of the formula (I) ##STR1## wherein Z represents a moiety selected from the group consisting of cycloalkyl having 3 to 7 carbon atoms in the cycloalkyl moiety or cycloalkylalkyl having 3 to 7 carbon atoms in the cycloalkyl moiety and 1 to 4 car...
06/26/2001
6232309Insecticidal heterocyclic compounds
Insecticidal heterocyclic compounds of the formula: ##STR1## wherein A represents a five-membered or six-membered heteroaryl group containing one to three hetero atoms selected from the group consisting of S, O and N, said heteroaryl group being unsubstit...
05/15/2001
6214825Aza-heterocycloakenes, pesticidal compositions containing them, pesticidal methods of using them, and processes for preparing them
Aza-heterocycloalkenes of the formula (I): ##STR1## wherein Z, G, Ar, E, y1, A and Y2 are as described herein are useful for combating pests, particularly fungi. Processes for preparing the compounds of formula (I) are also disclosed...
04/10/2001
6197766Insecticidal dihydrooxadiazine compounds
Insecticidal dihydrooxadiazine compounds having the formula: ##STR1## wherein X is O, N or S; R is a substituted or unsubstituted phenyl or C4 -C5 heterocyclic group; R2, R3, R4, and R5 are one ...
03/06/2001
6175007Substituted aromatic phoshonic acid derivatives
Phosphonic acid compounds I ##STR1## wherein Eth is optionally substituted 1,2-ethynediyl, ethanediyl or ethene-1,2-diyl; Y1 is oxygen or sulfur; Y2 is oxygen, sulfur or --N(R6)--; Y3 is oxygen, sulfur or --N(R7...
01/16/2001
61273641,3,4-oxadiazine derivatives and their use as pesticides
The invention relates to novel (1,3,4)-oxadiazine derivatives of formula (I), to a process and intermediates for their preparation, and to their usefulness as pesticides, in particular as anthelminthics, insecticides, acaricides, and nematicides....
10/03/2000
6121278Di-n-heterocyclic compounds, methods, and compositions for inhibiting parp activity
A compound of formula I: ##STR1## or a pharmaceutically acceptable salt, hydrate, ester, solvate, prodrug, metabolite, stereoisomer, or mixtures thereof, wherein: Y represents the atoms necessary to form a fused 5- to 6-membered, aromatic or non-arom...
09/19/2000
6103716Pyrido(3,2,1-ij)-1,3,4-benzoxadiazine
A novel compound having antibacterial activity according to the the formula ##STR1## The compound of the present invention may be prepared from (9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7H-pyrido [3,2,1-ij]-1,3,4-benzadiazine-6-...
08/15/2000
6083942Pesticidal hetero-substituted oxadiazine compounds
Pesticidal substituted oxadiazines having the formula: ##STR1## wherein R is a substituted or unsubstituted heterocyclic group, pesticidal compositions containing these oxadiazines, and methods for their use....
07/04/2000
6080856Preparation of arthropodicidal oxadiazines
A method for making arthropodicidal oxadiazines and intermediates which are racemic or enantiomerically enriched at their chiral center, the method for making the oxadiazines comprising reaction of an intermediate selected from ##STR1## wherein:...
06/27/2000
60691142-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators
Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepa...
05/30/2000
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