Class 544/6 - Spiro

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which contain a spiro ring system.
No. of patents: 116
Last issue date: 07/10/2007

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Number	Title	Issue Date
7241021	Emergency information lighting system An emergency information lighting system (100/200/300), comprising a primary light source (110/210/310) and a housing (112/212/312) for the primary light source (110/210). The housing (112/212/312) includes a first wall (120/220...	07/10/2007
7199118	Benzothiazine derivatives, their preparation and use This invention relates to novel benzothiazine derivatives of Formula I useful as modulators of the AMPA sensitive glutamate receptors, pharmaceutical compositions comprising such compounds and their use in therapy. ...	04/03/2007
7122662	Tricyclic compound having spiro union This invention relates to tricyclic compounds having spiro union represented by the following formula (I) or its salt which is useful as a drug, and in particular, as an inhibitor for activated blood coagulation factor X, which can be administered orally and which e...	10/17/2006
7051290	Graphical interface for receiving eyeglass prescription information A high volume lens curing system is described. The high volume lens curing system is configured to cure multiple eyeglass lenses in a continuous manner. The lens curing system includes a computer-implemented method configured to collect prescription information, sav...	05/23/2006
7014925	Heterogeneous spiro compounds in organic light emitting device elements A family of non-polymeric heterogeneous spiro compounds having visible light emissive, hole-transport, electron transport or bipolar-transport properties may be used in organic light emitting devices (OLEDs), as an emissive layer in the OLEDs and/or in one or more o...	03/21/2006
7001910	Thiazolidinedione derivatives as antidiabetic agents The present invention refers to compounds of the general formula (I), to their possible pharmaceutically acceptable salts and tautomeric forms. The present invention also refers to a process for their production and to their use as antidiabetic and *hypoglycemic age...	02/21/2006
6916806	Medicinal composition containing 1,3-thiazine derivative A compound of the formula (I) having a binding activity to the cannabinoid type 2 receptor: wherein R1 is optionally substituted heterocyclic group or the like; R2 and R2 each is indepe...	07/12/2005
6916807	Triaryl-oxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors The present invention relates to triaryl-oxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors of the formula wherein said ring X is a 5-7 membered heterocyclic ring, and wherein A, Y, B, G, and W are as ...	07/12/2005
6900201	N-substituted-heteroaryloxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors The present invention relates to N-substituted-heteroaryloxy-aryl-spiro-pyrimidine-2,4,6-trione metalloproteinase inhibitors of the formula wherein ring X is a 5-7 membered heterocyclic ring, and wherein A, Y, B, and G...	05/31/2005
6849732	Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation The invention relates to compounds of the formula 1: wherein: Z is O or S; V is a divalent radical which together with C* and N forms a ring having six ring atoms, where each of said ring atoms other than C* and...	02/01/2005
6756371	Phthalazinone derivatives as PDE4 inhibitors The compounds of formula (I) in which R1, R2, A, B and Ar have the meanings as given in the description are novel effective PDe4 inhibitors ...	06/29/2004
6743798	Substituted pyrazole derivatives condensed with six-membered heterocyclic rings The present invention relates to novel substituted pyrazole derivatives of the general formula (I) in which R1, R2, R3 and A are each as defined, and to processes for their preparation an...	06/01/2004
6683709	Photochromic pyran compounds Photochromic pyran compounds and their use in synthetic resin objects of all types, especially for ophthalmic applications, particularly spiro compounds having a fluorene structure derived from naphthopyrans, which are known as spirofluorenopyrans. By int...	01/27/2004
6667306	Platelet ADP receptor inhibitors The invention relates to novel compounds of formula (I) containing fused heterocyclic ring systems which are effective platelet ADP receptor inhibitors: ##STR1## In formula (I), W is carbon or nitrogen, wherein at least one W is a carbon; and Y is ni...	12/23/2003
6472398	Spiropiperidine derivatives as melanocortin receptor agonists Certain novel spiropiperidine derivatives of structural formula Ia wherein the substituents are as defined herein are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). T...	10/29/2002
6451804	Heteroalkylamino-substituted bicyclic nitrogen heterocycles The invention provides compounds represented by the formula: ##STR1## wherein R1, R2, R3, R4, and n are as defined in the Summary of the Invention; and individual isomers, racemic or non-racemic mixtures of isom...	09/17/2002
6444819	Benzylpiperazinyl and piperidinyl ethanone derivatives: dopamine receptor subtype specific ligands Disclosed are compounds of the formula: ##STR1## or pharmaceutically acceptable addition salts thereof wherein: Y represents oxygen or sulfur; Z is nitrogen or CH; R1, R2 and R3 independently represent organic or inorganic subs...	09/03/2002
6407232	Ionic metal complex and process for synthesizing same The invention relates an ionic metal complex represented by the general formula (1): ##STR1## wherein M is an element of groups 3-15 of the periodic table; Aa+ represents a metal ion, onium ion or proton; X1 represents O, S or N...	06/18/2002
6369057	Quinoxalines, processes for their preparation and their use Compounds of the formula I or Ia ##STR1## in which n and the substituents R1, R5 and x have the meaning mentioned have an antiviral activity....	04/09/2002
6191127	Substituted heterocycles and their use in medicaments Compounds of Formula I ##STR1## wherein X and R1-6, are as defined herein, tautomeric forms thereof, and isomeric forms thereof, and salts thereof, are suitable for treating diseases that are induced by the action of nitrogen monooxide at ...	02/20/2001
6100246	Spiro-piperidine derivatives as inhibitors of nitric oxide synthase There are provided novel compounds of formula (I) ##STR1## wherein A represents a benzo ring; a six membered heterocyclic aromatic ring containing 1 to 3 nitrogen atoms; or a five membered heterocyclic aromatic ring containing 1 to 3 heteroatoms whic...	08/08/2000
6060469	Spiro-piperidine derivatives and their use as tachykinin antagonists The present invention relates to compounds of formula (I), ##STR1## wherein R1 represents halogen, hydroxy, C1-6 alkyl group optionally substituted by one or three fluorine atoms, C1-6 alkoxy group optionally substitu...	05/09/2000
6013652	Spiro-substituted azacycles as neurokinin antagonists Disclosed are spiro-substituted azacycles of formula I are tachykinin receptor antagonists useful in the treatment of inflammatory diseases, pain or migraine, and asthma. In particular compounds of formula I are shown to be neurokinin antagonists....	01/11/2000
6011150	Azetidinone compound and process for preparation thereof There is disclosed an azetidinone compound of the formula [I]: ##STR1## wherein Ring B is a benzene ring which may have substituent(s), R1 is a hydroxy-substituted lower alkyl group which may have substituent(s), X is oxygen atom and the l...	01/04/2000
6002000	Chemiluminescent compounds and methods of use Methods are disclosed for determining an analyte in a medium suspected of containing the analyte. One method comprises providing (1) combining a medium suspected of containing the analyte and a novel chemiluminescent compound, (2) combining a means for ch...	12/14/1999
5994350	3-spiro-indolin-2-one derivatives as vasopressin and/or oxytocin receptor ligands The subject of the invention is indolin-2-one derivatives of formula: ##STR1## in which: W represents a --CH2 -- or --SO2 -- group; Cy forms, with the carbon to which it is bonded, a non-aromatic, saturated or unsaturated C3	11/30/1999
5981523	Compounds and methods for treating multiple sclerosis This invention provides thiomorpholinone compounds useful for treating multiple sclerosis of formula I wherein: R1 and R2 are each independently selected from C1 -C8 alkyl; C2 -C8 alkenyl; C	11/09/1999
5945413	Aspartyl protease inhibitors This invention relates to a novel class of compounds that are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of aspartyl protease inhibitors characterized by specific structural and physicochemical features. This ...	08/31/1999
5929072	1H-2,1,3-benzothiadiazine-2,2-dioxide compounds or derivatives thereof A pharmaceutical compound having the formula: ##STR1## in which n is 1 or 2, m is 1 or 2, p is 1 to 6, q is 0 or 1 to 3, R1 and R2 are each hydrogen or C1-4 alkyl, R3, R4 and R5 are each hydroge...	07/27/1999
5922748	Indole derivatives as 5-HT agonists Compounds of formula (I) ##STR1## wherein R and R1 are hydrogen, C1-4 alkyl or are linked to form a ring, A is a cycloalkyl or alkyl-cycloalkyl group, n is an integer from 0 to 3, W is an optionally substituted 5-or 6-membered hetero...	07/13/1999
5874382	Cyclic sulfonamide herbicides Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C1 -C3 alkyl); N(C1 -C3...	02/23/1999
5783579	Spiro-substituted azacyclic-substituted piperazino derivatives as neurokinin antagonists The invention relates to compounds of the formula ##STR1## wherein Z, Rc, y, m, u, Ar2, n, X, Rc', I and Ar2 are as described herein. These compounds are neurokinin antagonists. These compounds are useful i...	07/21/1998
5760029	Spirocycle integrin inhibitors This invention relates to novel heterocycles, including (S)-2-phenylsulfonylamino-3-8-(2-pyridinylaminomethyl)-!-1-oxa-2-azaspi ro-4,5!-dec-2-en-3-yl!carbonylamino! propionic acid, which are useful as antagonists of the ଱v ଲ	06/02/1998
5728693	Arthropodicidal oxadiazine-thiadiazine-or triazine-carboxanilides Arthropodicidal compounds, compositions and use of compounds having the formula ##STR1##...	03/17/1998
5726126	1-(3-heterocyclyphenyl)-S-triazine-2,6,6-oxo or thiotrione herbicidal agents There is provided a 1-(3-heterocyclylphenyl)-s-triazine-2, 4,6-oxo or thiotrione compound having the structural formula I ##STR1## Further provided are a composition and a method comprising that compound for the control of undesirable plant species....	03/10/1998
5696145	1-benzyl-1,3-dihydroindol-2-one derivatives, their preparation and the pharmaceutical compositions in which they are present The present invention relates to 1-benzyl-1,3-dihydroindol-2-one derivatives of the formula ##STR1## to their preparation and to the pharmaceutical compositions in which they are present. These derivatives have an affinity for the vasopressin and ...	12/09/1997
5679805	Photochromic spironaphthopyran compounds A naphthopyran compound represented by the formula: ##STR1## wherein A and B are each selected from the following group: a substituted divalent cyclic radical, a substituted divalent aromatic radical, and a substituted divalent fused heterocyclic rad...	10/21/1997
5597819	Phenothiazine cytokine inhibitors New benzothiazine derivatives corresponding to the general formula I: ##STR1## in which: X represents halogen, n represents 0, 1, or 2, B represents the following formula: ##STR2## in which: R1 & R2 together with the carbons to ...	01/28/1997
5591848	Spiroconjugated charge-transfer dyes for optical applications New intramolecular charge-transfer organic dyes are described. The design of these molecules is based on the phenomenon of spiroconjugation, and it provides a modular approach to the preparation of unique materials with interesting optical properties. In ...	01/07/1997
5589489	Cyclic amide derivatives for treating asthma Compounds of formula I ##STR1## wherein Q1, Q2, Q3, and Q4 have any of the meanings given in the specification, their N-oxides, and their pharmaceutically acceptable salts are nonpeptide antagonists of neur...	12/31/1996

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Class 544/6 - Spiro