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| Number | Title | Issue Date |
| 7312211 | Pryanone compounds useful as reversible inhibitors of cysteine proteases Disclosed are cathepsin S, K, F, L and B reversible inhibitory compounds of the formulas (Ia) and (Ib) where R2, R3, R4, R6, R8 and Y are defined herein. The compounds are useful for treating autoimmune and othe... | 12/25/2007 |
| 7300934 | Benzamide nitriles Compounds of the formula (I) wherein m, n, A, R1, R2, R3, R4, R5 and R6 are as described herein, together with methods for making the compounds an... | 11/27/2007 |
| 7101874 | Antimicrobial dihydrothiazine and dihydrothiopyran oxazolidinones The present invention provides a compound of formula I or a pharmaceutically acceptable salt thereof wherein Y is —S(═O)n—, —S(═NR8)—, or —S(═NR8)(═O)—; Z is ... | 09/05/2006 |
| 6881735 | Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them The present invention relates to compounds of the formula I wherein A1, A2, R1, R2, R3, X and n are as defined in the claims, which are valuable pharmaceutically a... | 04/19/2005 |
| 6784167 | 17-beta-hydroxysteroid dehydrogenase-II inhibitors 17-beta-hydroxysteroid dehydrogenase-II inhibitors having the structural formula wherein the phenyl group labeled A and the group —C(R4)(R6)Y are oriented cis to each other; W represents O or S; R... | 08/31/2004 |
| 6770596 | Fused tricyclic compounds, process for their preparation, and herbicidal compositions containing them Novel fused tricyclic compounds represented by formula (I) are described. Q, Y, —L—X—, A, A′, B, E, D, n and m are as defined in the disclosure. Also described are the processes for the manufacture of these compounds and agriculturally suitable compositions ... | 08/03/2004 |
| 6605609 | Thizaine oxazolidinone The present invention provides a thizaine oxazolidinone useful as antimicrobial.... | 08/12/2003 |
| 6448396 | Compounds useful as neuro-protective agents The present invention provides a process of preparing a compound of the formula IV ##STR1## wherein: R1 and R2 are each individually -(C1 -C6)alkyl, -(C1 -C6)alkoxy or phenyl, R3... | 09/10/2002 |
| 6387896 | Bicyclic oxazolidinones as antibacterial agents The present invention provides compounds of formula I useful as antimicrobial agents ##STR1## wherein W, X, Y, R1, R2 and n are as defined in thereof.... | 05/14/2002 |
| 6200378 | Thiazine indigo pigments, solid solutions thereof and their preparation A compound according to the formula (I) ##STR1## wherein R1 and R2 are independently the atoms necessary to complete the formation of a substituted or unsubstituted aromatic or aliphatic carbocyclic or heterocyclic ring system and R | 03/13/2001 |
| 5925642 | Pyridopyrimidines The invention concerns compounds of formula (I) in which the substituents and symbols have the meanings given in the specification. These compounds are advantageous as resistance modulators. ##STR1##... | 07/20/1999 |
| 5854277 | Thiophenebutanoic acid derivatives as matrix metalloprotease inhibitors Inhibitors for matrix metalloproteases, pharmaceutical compositions containing them, and a process for using them to treat a variety of physiological conditions. The compounds of the invention have the generalized formula ##STR1## wherein each T... | 12/29/1998 |
| 5679670 | Sulfonamides useful as carbonic anhydrase inhibitors Sulfonamides and pharmaceutical compositions containing the compounds useful in controlling intraocular pressure are disclosed. Methods for controlling intraocular pressure through administration of the compositions are also disclosed.... | 10/21/1997 |
| 5674894 | Amidine derivatives useful as platelet aggregation inhibitors and vasodilators The current invention discloses novel amidine derivatives with nitric oxide donating property that can inhibit platelet aggregation and promote vasodilation in a single compound.... | 10/07/1997 |
| 5625072 | Retroviral protease inhibiting compounds A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.... | 04/29/1997 |
| 5597928 | Retroviral protease inhibiting compounds A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.... | 01/28/1997 |
| 5591860 | Retroviral protease inhibiting compounds A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.... | 01/07/1997 |
| 5583233 | Retroviral protease inhibiting compounds A retroviral protease inhibiting compound of the formula: ##STR1## is disclosed.... | 12/10/1996 |
| 5523403 | Tropone-substituted phenyloxazolidinone antibacterial agents A novel class of phenyloxazolidinone antibacterial agents which have, as their salient structural feature, an appended substituted tropone moiety, are described. Intermediates and processes for the preparation of these antibiotics are also disclosed. Thes... | 06/04/1996 |
| 5512569 | Aminoalkyl benzothiazolinones The invention relates to the compounds of formula (I): ##STR1## in which R1 and R2 are as defined in the description, the optical isomers thereof, and an addition salt thereof with a pharmaceutically-acceptable acid or base, and... | 04/30/1996 |
| 5489589 | Amino acid derivatives of paclitaxel The present invention concerns water-soluble amino acid derivatives of paclitaxel, their use as antitumor agents, and pharmaceutical compositions containg the compounds.... | 02/06/1996 |
| 5478945 | Thiazoline derivatives A thiazoline derivative represented by the formula: ##STR1## [wherein R1 is cyano, carbamoyl, thiocarbamoyl, morpholinothiocarbonyl, alkylthioimidoyl, amidino, substituted amidino or imidazolin-2-yl, R2 is alkyl or aralkyl, R | 12/26/1995 |
| 5458814 | Substituted naphthopyrans Described are novel reversible photochromic naphthopyran compounds, examples of which are compounds having certain substituents at the number 5 and 6 carbon atoms of the naphtho portion of the naphthopyran and at the 2-position of the pyran ring. Certain ... | 10/17/1995 |
| 5420273 | Condensed heterocyclic compounds The invention relates to compounds of the formula ##STR1## wherein R1 is hydrogen, acyl, lower-alkyl or --CHO, --CH2 OR10, --COR7 or OR13 ; R2, R3 and R4 are, ind... | 05/30/1995 |
| 5352689 | Rhizoxin derivatives and their use as anti-tumor agents Rhizoxin and rhizoxin-2-ene derivatives of formula ##STR1## in which: n is 1 to 25; A is an extra bond or oxygen, X is oxygen, sulfur, nitrogen or carbonyl; and R is hydrogen, carboxylic acyl having from 1 to 25 carbon atoms, alkoxycarbonyl group hav... | 10/04/1994 |
| 5300522 | Condensed heterocyclic compounds and pharmaceutical use thereof The invention relates to compounds of the formula ##STR1## wherein R1 is hydrogen. acyl, lower-alkyl or --CHO, --CH2 OR10, --COR7 or OR13 ; R2, R3 and R4 are, ind... | 04/05/1994 |
| 5256657 | Succinamide derivative matrix-metalloprotease inhibitors Compounds having the structural formula ##STR1## wherein X is HONH or HO and especially wherein the carbon atom bearing CH2 R1 has the R-configuration, the carbon atom bearing CH2 R2 has the S-configuration... | 10/26/1993 |
| 5246927 | Benzazole derivatives, processes for their preparation containing such compounds and the use thereof The invention relates to new benzazole derivatives of the formula I ##STR1## wherein X is oxygen or sulphur, R1 is lower alkyl, lower alkenyl or cycloalkyl, R2 and R3 independently of one another are each hydrogen, lo... | 09/21/1993 |
| 5179092 | Compound effective as cerebral insufficiency improver A compound having the formula (I): ##STR1## wherein A is --CH2 --, --O--, or --S--; R1 is CH3 or OCH3 ; R2 is hydroxy or carboxy which may be optionally esterized or amidated; R3 is H ... | 01/12/1993 |
| 5164387 | Condensed heterocyclic compounds The invention relates to compounds of the formula ##STR1## wherein R1 is hydrogen, acyl, lower alkyl or --CHO, --CH2 OR10, --COR7 or OR13 ; R2, R3 and R4 are, ind... | 11/17/1992 |
| 5104985 | Labdane process Novel labdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure utilizing compounds or compositions thereof are disclosed.... | 04/14/1992 |
| 5103007 | Lipids Lipid derivatives represented by the formula: ##STR1## wherein R1 stands for an optionally substituted higher alkyl group, R2 stands for an optionally substituted lower alkyl group or an optionally substituted nitrogen-containin... | 04/07/1992 |
| 5098931 | 7-substituted HMG-CoA reductase inhibitors Novel HMG-CoA reductase inhibitors are useful as antihypercholesterolemic agents and are represented by structural formulae (I) and (II): ##STR1##... | 03/24/1992 |
| 5093336 | 6- and 7-deoxyforskolin and derivatives thereof Novel forskolin derivatives, intermediates and processes for the preparation thereof, and methods for treating cardiac failure and memory deficit utilizing compounds or compositions thereof are disclosed.... | 03/03/1992 |
| 5081245 | Carboxylic acid derivatives A compound represented by the formula: ##STR1## wherein R represents a hydrogen atom or a lower alkyl group; R1 represents a higher alkyl group which may be substituted; R2 represents a hydrogen atom or a lower alkyl group, a lower alkano... | 01/14/1992 |
| 5051504 | Doubled triphenylmethane dyes having bis acylpiperazine linkage Triphenylmethane dyes of the formula ##STR1## where each R1 is independently of the others hydrogen or substituted or unsubstituted C1 -C6 -alkyl, or two R1 radicals together with the nitrogen atom joining ... | 09/24/1991 |
| 5047549 | Derivatives of pravastatin for inhibiting cholesterol biosynthesis Derivatives of pravastatin are provided which are useful in inhibiting cholesterol biosynthesis and in preparing radiolabeled compounds useful in the radioimmunoassay (RIA) of pravastatin and derivatives thereof. The pravastatin derivatives have the struc... | 09/10/1991 |
| 5030646 | Novel tricyclic indole compound The invention relates to compounds of general formula: ##STR1## in which A, B, G, D which may be identical or different, each denote a hydrogen atom or a halogen atom, a lower alkoxy group or alternatively a lower alkyl group optionally substituted w... | 07/09/1991 |
| 5000777 | Imidazole derivatives 1,5-substituted imidazole derivatives of formula I ##STR1## the stereochemically isomeric forms thereof, and the salts thereof, have useful herbicidal properties. The substituents R1, R2, R3, R4, X1 | 03/19/1991 |
| 4999350 | (RS)-2-(2,3-dihydro-5-hydroxy-4,6,7-trimethylbenzofuranyl) acetic acids and 2-(2,3-dihydro-5-acyloxy-4,6,7-trimethylbenzofuranyl) acetic acids and esters thereof, useful as mucoregulator and anti-ischemic drugs The present invention relates to (RS)-2-(2,3-dihydro-5-hydroxy-4,6,7-trimethylbenzofuranyl) acetic acids and 2-(2,3-dihydro-5-acyloxy-4,6,7-trimethylbenzofuranyl) acetic acids and esters thereof, the process for producing them and their relevant ther... | 03/12/1991 |
