Class 544/58.5 - Additional hetero ring containing

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which include an additional hetero ring.
No. of patents: 166
Last issue date: 02/12/2008

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Number	Title	Issue Date
7329752	Carbamate compounds as 5-HTreceptor agonists The invention provides novel benzoimidazolone-carboxamide-derived carbamate 5-HT4 receptor agonist compounds of formula (I): wherein R1, R2, R3, R4, a, and b...	02/12/2008
7122231	Ink jet recording element An ink jet recording element comprising a support having thereon an image-receiving layer, the ink jet recording element containing finely divided particulate material and a metal(oxy)hydroxide complex, Mn+(O)a(OH)b(Ap−)...	10/17/2006
7109186	HIV integrase inhibitors The present invention describes novel compounds of Formula I which inhibit HIV integrase. The invention also describes compositions and treatments of AIDS or ARC by using these compounds ...	09/19/2006
7105215	Ink jet recording element An ink jet recording element comprising a support having thereon an image-receiving layer, the ink jet recording element containing a metal(oxy)hydroxide complex, Mn+(O)a(OH)b(Ap−)c•xH2O, wherein ...	09/12/2006
7041669	1,4-benzofused urea compounds useful in treating cytokine mediated diseases Disclosed are 1,4-disubstituted benzo-fused urea compounds of formula (I): wherein Ar, X, A, L, and Q of formula(I) are defined herein. The compounds inhibit production of cytokines involved in inflammatory processes an...	05/09/2006
6982264	Substituted alcohols useful in treatment of Alzheimer's disease The invention relates to substituted alcohol compounds of the formula (I): wherein X, R1, R2, R3, RN, R20 and RC are defined herein. The compounds are u...	01/03/2006
6670363	Azole compounds as therapeutic agents for fungal infections The present invention relates to the derivatives of specially substituted azole compounds which have improved antifungal activity as compared to known compounds such as fluconazole and itraconazole and the processes for the preparation thereof. This inven...	12/30/2003
6573267	Useful aroyl aminoacyl pyrrole compounds This invention is directed to aroyl aminoacyl pyrroles pharmaceutically useful as agents and modulators for the treatment of central nervous system disorders and a method for the treatment of central nervous system disorders including, but not limited to,...	06/03/2003
6506748	Aromatic heterocyclic compounds as antiinflammatory agents Disclosed are novel aromatic heterocyclic compounds of the formula(I) wherein Ar1,Ar2,L,Q and X are described herein. The compounds are useful in pharmaceutic compositions for treating diseases or pathological conditions involving in...	01/14/2003
6506478	Inkjet printable media An ink receptive media suitable for use in a passport is disclosed. A media in accordance with the present invention comprises a substrate, and an image receptive layer comprising a plurality of particles. In a preferred embodiment, the image receptive la...	01/14/2003
6498178	Inhibitors of IMPDH enzyme The present invention relates to compounds which inhibit IMPDH. This invention also relates to pharmaceutical compositions comprising these compounds. The compounds and pharmaceutical compositions of this invention are particularly well suited for inhibit...	12/24/2002
6476016	Cyclic oxyguanidine pyrazinones as protease inhibitors Cyclic oxyguanidine pyrazinone compounds are described, including compounds of the Formula I: ##STR1## wherein R3, R4, R5, W, and A are as set forth in the specification, as well as hydrates, solvates or pharmaceutically ...	11/05/2002
6458950	Compounds and pharmaceutical compositions containing the same A compound shown by the formula II, wherein Het is a mono- or polycyclic heterocyclic group comprising one or more hetero atoms selected from the group consisting of N, O and S which may be the same or different from each other; R1 is hydrogen,...	10/01/2002
6410482	(Het) arylsulfonylureas having an amino function, their presentation and their use as herbicides and plant growth regulators (Het)Arylsulfonylureas having an imino function, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## in which A is a (hetero)aromatic or heterocyclic bridge linked to the group...	06/25/2002
6407103	Indeno [1,2-c] pyrazol-4-ones and their uses The present invention relates to the synthesis of a new class of indeno[1,2-c]pyrazol-4-ones of formula (I): ##STR1## that are potent inhibitors of the class of enzymes known as cyclin dependent kinases, which relate to the catalytic subunits cdk1-9 and t...	06/18/2002
6331538	7-substituted quinazolin-2,4-diones useful as antibacterial agents The invention is a series of 7-substituted quinazolin-2,4-diones useful as antibacterial agents, processes for the preparation of the compounds, and a pharmaceutical composition containing one or more of the compounds....	12/18/2001
6319921	Aromatic heterocyclic compound as antiinflammatory agents Disclosed are novel aromatic heterocyclic compounds of the formula (I) wherein Ar1, Ar2, L, Q and X are described herein. The compounds are useful in pharmaceutic compositions for treating diseases or pathological conditions involvin...	11/20/2001
6310080	Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors Selected amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, rela...	10/30/2001
6294542	Pyrimidinone compounds, pharmaceutical compositions containing the compounds and the process for preparing the same The present invention relates to a novel pyrimidinone compounds and the pharmaceutical acceptable salts thereof having remarkable antagonistic action against angiotensin II receptor, thereby, being useful in treating cardiovascular disease caused by bindi...	09/25/2001
6288059	Acylated hetero-alicyclic derivatives A compound of formula (I), a pharmaceutically acceptable salt or ester or other derivative thereof: ##STR1## R1 is optionally substituted cycloalkyl or optionally substituted saturated heterocyclic group. R2 is optionally substituted...	09/11/2001
6265408	Sulphonamide derivatives and their use in the treatment of CNS disorders Sulphonamide compounds according to formula (I) or pharmaceutically acceptable salts thereof: ##STR1## wherein: Ar is naphthyl, phenyl or thienyl optionally substituted by one or more substituents selected from the group consisting of C1-6 alky...	07/24/2001
6200378	Thiazine indigo pigments, solid solutions thereof and their preparation A compound according to the formula (I) ##STR1## wherein R1 and R2 are independently the atoms necessary to complete the formation of a substituted or unsubstituted aromatic or aliphatic carbocyclic or heterocyclic ring system and R	03/13/2001
6121260	Method of treating conditions susceptible to modulation of NPY receptors with diarylimidazole derivatives Certain diaryl imidazoles act as partial agonists or antagonists for NPY receptors, in particular NPY 5 receptors. They are of use, for example in treating loss of appetite. Such compounds bear aryl groups in the 2 position. Many of the compounds are nove...	09/19/2000
6090753	Pyridazin-3-one derivatives, their use, and intermediates for their production Novel pyridazin-3-one derivatives of formula [1] are provided, which are useful as active ingredients of herbicides, wherein R1 is haloalkyl; R2 and R3 are the same or different and are hydrogen, alkyl, haloalkyl, or alkox...	07/18/2000
6069114	2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepa...	05/30/2000
6013648	CB₂ Receptor agonist compounds The use of human CB2 receptor-specific agonists of formula (I) or (I') for preparing immunomodulating drugs is disclosed. In formulae (I) and (I'), R1 is a group selected from --CH2 CHR10 NR6 R11...	01/11/2000
5965565	Piperidines promote release of growth hormone The present invention is directed to certain piperidines, pyrrolidines, and hexahydro-1H-azepines of the general structural formula: ##STR1## wherein B is selected from: ##STR2## and R1, R1a, R2a, R3a,...	10/12/1999
5948784	Quinazoline derivatives Disclosed are quinazoline derivatives represented by formula (I): wherein R1 represents hydrogen, lower alkyl, alkenyl, or aralkyl; R2, R3, R4, and R5 represent hydrogen, lower alkyl, lower alkoxy, lo...	09/07/1999
5908852	1,3,5 trisubstituted pyrazole compounds for treatment of inflammation A class of 1,3,5-substituted pyrazoles is described for the treatment of inflammation, including treatment of pain and disorders such as arthritis. Compounds of particular interest are of Formula I ##STR1## wherein R1, R2, R	06/01/1999
5854241	Pyrido3,2,1-I,J!3,1!benzoxazine derivatives Disclosed are pyrido3,2,1-i,j!3,1!benzoxazine compounds of the formula (I): ##STR1## wherein z represents a radical having the formula: ##STR2## wherein B represents --CH2 --, --O-- or a direct bond; and the other variables i...	12/29/1998
5756533	Amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors Selected amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, rela...	05/26/1998
5698690	Hydroxamic acid derivatives with tricyclic substitution The invention provides hydroxamic acid derivatives of the general formula ##STR1## wherein Bz represents benzyl; R1 represents cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl; R2 represents a saturated 5- to 8-membered monocy...	12/16/1997
5674894	Amidine derivatives useful as platelet aggregation inhibitors and vasodilators The current invention discloses novel amidine derivatives with nitric oxide donating property that can inhibit platelet aggregation and promote vasodilation in a single compound....	10/07/1997
5648367	Aminoalkyloximes Novel aminoalkyloximes, precursors and processes for the preparation thereof, and methods of treating depression and obsessive compulsive disorders are described....	07/15/1997
5614625	Hydroxamic acid derivatives with tricyclic substitution The invention provides hydroxamic acid derivatives of the general formula ##STR1## wherein R1 represents cyclopropyl, cyclobutyl, cyclopentyl or cyclohexyl; R2 represents a saturated 5- to 8-membered monocyclic or bridged N-hete...	03/25/1997
5612337	Substituted morpholine derivatives and their use as therapeutic agents The present invention relates to compounds of formula (I), wherein R1 is hydrogen, halogen, C1-6 C alkyl, C1-6 alkoxy, CF3, NO2, CN, SRa, SORa, SO2 Ra, CO2	03/18/1997
5602101	Antithrombotic agents This invention relates to L-Arginine aldehyde derivatives, pharmaceutical formulations containing those compounds and methods of their use as thrombin inhibitors, coagulation inhibitors and thromboembolic disorder agents....	02/11/1997
5578574	Antithrombotic agents This invention relates to L-arginine aldehyde derivatives, having the formula I ##STR1## where X and Y have the values defined in the description, as well as pharmaceutical formulations containing those compounds and methods of their use as thro...	11/26/1996
5541340	Method of preparing 1,2,3,3a,8,8a-hexahydro-3a,8(and 1,3a,8)-Di(and Tri)methylpyrrolo[2,3,-b] indoles There are described compounds of the formula ##STR1## where (a) X is O or S; (b) R is H, loweralkyl, ##STR2## where Y is O or S; R2 is alkyl, cycloalkyl, bicycloalkyl, cycloalkenyl, aryl, arylloweralkyl, heteroaryl or heteroaryllower...	07/30/1996
5532237	Indole derivatives with affinity for the cannabinoid receptor Disclosed are indole derivatives having activity on the cannabinoid receptors and the methods of their preparation. The compounds are useful for lowering ocular intra ocular pressure and treating glaucoma because of the activity on the cannabinoid recepto...	07/02/1996

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Class 544/58.5 - Additional hetero ring containing