Class 544/52 - Double bonded divalent chalcogen containing

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds which include a double bonded divalent chalcogen
No. of patents: 142
Last issue date: 03/25/2008

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Number	Title	Issue Date
7348426	Substituted bicyclic heterocycles, process for their preparation and their use as antiobesity and hypocholesterolemic agents The present invention relates to novel antiobesity and hypocholesterolemic compounds, their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates...	03/25/2008
7253164	Bicyclic compounds and compositions as PDF inhibitors This invention is directed to novel bicyclic compounds, to the uses of these compounds in various medicinal applications, including treating disorders amenable to treatment by peptidyl deformylase inhibitors such as treatment of bacterial infections, and to pharmace...	08/07/2007
7235549	Benzamide, heteroarylamide and reverse amides The present invention relates to novel to P2X7 inhibitors of formula I and to processes for their preparation, intermediates useful in their preparation, pharmaceutical compositions containing them, an...	06/26/2007
7205408	Quinolines and nitrogenated derivative thereof substituted in 4-position by a piperidine-containing moiety and their use as antibacterial agents Piperidine derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly in man. ...	04/17/2007
7202196	Selective herbicide comprising a tetrazolinone derivative The invention relates to novel herbicidal synergistic active compound combinations comprising a known tetrazolinone derivative and known herbicidally active compounds and/or safeners, which compositions can be used with particularly good results for the selective co...	04/10/2007
7141564	Nitrogen-containing bicyclic heterocycles for use as antibacterials Cyclohexane and cyclohexene derivatives and pharmaceutically acceptable derivatives thereof useful in methods of treatment of bacterial infections in mammals, particularly man. ...	11/28/2006
7141566	Benzoxazine and benzothiazine derivatives and the use thereof in medicaments The invention relates to compounds of formula (I), the tautomeric and isomeric forms and salts thereof, in addition to a method for production and use thereof in medicaments. ...	11/28/2006
7067513	Phenylpiperazines The invention relates to a novel group of phenylpiperazines having interesting pharmacological properties such as a high affinity for the dopamine D2 receptor and/or the serotonin reuptake site, and the ability to treat conditions related to disturbances ...	06/27/2006
7049312	Benzothiazinone and benzoxazinone compounds Q is —N=or CR2 X is S, O or NOR3 Y is —O—, —S—, —SO— or —SO2— R and R1 are each...	05/23/2006
6964973	Bicyclic androgen and progesterone receptor modulator compounds and methods The present invention is directed to compounds, pharmaceutical compositions, and methods for modulating processes mediated by AR and PR. More particularly, the invention relates to nonsteroidal compounds and compositions that are high affinity, high specificity agon...	11/15/2005
6949543	Amide derivative The invention relates to a novel amide derivative which is an N-({[4-(substituted thiazol-4-yl)phenyl]carbamoyl}methyl)amide derivative having a characteristic in that an aryl or heteroaryl group as an aromatic ring group is directly substituted on the N atom of ami...	09/27/2005
6900204	Antimicrobial agents and uses thereof The invention features compounds that act as antimicrobial agents and/or antimicrobial enhancer agents, compositions that include the antimicrobial enhancer agents of the invention, and methods for treating microbial infections using those compositions. ...	05/31/2005
6809095	Bicyclic compounds and their use in medicine; process for their preparation and pharmaceutical compositions containing them A method for preventing or treating complications of diabetes by administering a compound of formula (I) its tautomeric forms, its stereoisomers, its polymorphs, its pharmaceutically acceptable salts or its pharmaceuti...	10/26/2004
6740649	Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- α converting enzyme (TACE) The present application describes novel cyclic hydroxamic acids of formula I: or pharmaceutically acceptable salt forms thereof, wherein ring B is a 5-7 membered cyclic system containing from 0-2 heteroatoms selected fro...	05/25/2004
6716851	Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators or caspases and inducers of apoptosis and the use thereof The present invention is directed to substituted 2-aryl-4-arylaminopyrimidine and analogs thereof, represented by the general Formula I: wherein A, Ar1, Ar2, R1 and R3 are defi...	04/06/2004
6683101	Bicyclic cyclohexylamines and their use as NMDA receptor antagonists Described are heterocycle-substituted cyclohexylamines of formula (I), and their pharmaceutically acceptable salts thereof. The compounds of the formula (I) are antagonists of NMDA receptor channel complexes useful for treating cerebral vascular disorders...	01/27/2004
6573218	Fused-benzene derivatives useful as herbicides A compound of the formula (Ia): ##STR1## or its salts, in which the variables are as described in the disclosure; herbicidal compositions of said compounds, herbicidal processes using said compounds, defoliant processes using said compounds, and processes...	06/03/2003
6448246	Substituted 4H-1,4-benzothiazine-2-carboxamide: GABA brain receptor ligands Disclosed are 4H-1,4-Benzothiazine-2-carboxamides. These compounds are highly selective agonists, antagonists or inverse agonists for GABAa brain receptors or prodrugs of agonists, antagonists or inverse agonists for GABAa brain receptors. These compounds...	09/10/2002
6410484	6-Hydroxy-5,6-dihydrouracil compound and herbicidal composition containing thereof A 5,6-dihydrouracil compound given by the formula [I]: ##STR1## wherein, R1 represents C1-C2 haloalkyl group and Q represents Q1 of the formula below, etc.: ##STR2## wherein, R3 is hydrogen atom or halogen atom, R15 is C3-...	06/25/2002
6339084	Process for the production of thiazine-indigo pigments A process of forming the cis- or the trans-isomers of thiazine-indigo compounds comprising the step of reacting o-aminomercapto-carbocyclic or -heterocyclic compounds with a maleic acid or fumaric acid derivative in the presence of an aqueous system. The ...	01/15/2002
6339155	Process for producing 3-phenyluracil compounds The uracil compounds represented by the formula [V]: ##STR1## wherein R1 represents C1-C5 perfluoroalkyl group and Q represents an aromatic group, can be produced by making the amide compounds represented by the formula [II]: ##STR2## wher...	01/15/2002
6333413	Production of pyridazine herbicides Carboxylic acids of formula (1): ##STR1## wherein R2 and R3 are independently hydrogen or C1 -C3 alkyl, and Q is optionally substituted phenyl, can be easily converted by ring closing into pyridazin-3-one derivatives...	12/25/2001
6303542	Herbicidal 3-substituted-phenyl-1,2,3-benzotriazin-4-ones This invention relates to 3-substituted-phenyl-1,2,3-benzotriazin-4-ones which have activity as herbicides, to compositions which contain these compounds and to methods of use of these compounds....	10/16/2001
6300342	Antithrombotic phenylalkyl derivatives Antithrombotic phenylalkyl derivatives of the formula ##STR1## Exemplary compounds are: (a) 1-[3-(4-amidino-phenyl)propionyl]-6-(4-fluoro-phenylsulphonamido)-1,2,3,4- tetrahydro-quinoline, (b) 1-[3-(4-amidino-phenyl)propionyl]-6-butylsulphonamido-1,2,...	10/09/2001
6265401	Bicyclic compounds and their use in medicine, process for their preparation and pharmaceutical compositions containing them Compounds of formula (I) ##STR1## its tautomeric forms, its stereoisomers, its polymorphs, its pharmaceutically acceptable salts or its pharmaceutically acceptable solvates can be used to prevent or treat diabetes caused by insulin resistance or impa...	07/24/2001
6232310	Fused 1,4-thiazine-2-carbonitrile derivatives, their preparation and use The present invention relates to fused 1,4-thiazine-2-carbonitrile derivatives, compositions thereof and methods for preparing the compounds. The compounds are useful in the treatment of diseases of the central nervous system, the cardiovascular system, the pu...	05/15/2001
6204380	Production pyridazine herbicides Carboxylic acid ester derivatives of formula (1): ##STR1## wherein R is C1 -C6 alkyl, R2 and R3 are independently hydrogen or C1 -C3 alkyl, and Q is optionally substituted phenyl, can be ea...	03/20/2001
6200971	Bicyclic heterocyclic compounds The bicyclic heterocyclic compounds are prepared by reaction of correspondingly substituted carboxylic acids with amines, in particular with phenylglycinolamine. The bicyclic heterocyclic compounds according to the invention are suitable as active compoun...	03/13/2001
6191127	Substituted heterocycles and their use in medicaments Compounds of Formula I ##STR1## wherein X and R1-6, are as defined herein, tautomeric forms thereof, and isomeric forms thereof, and salts thereof, are suitable for treating diseases that are induced by the action of nitrogen monooxide at ...	02/20/2001
6127357	N-((phenyl, benzodioxinyl or N-heteroarylpiperazinyl)alkyl)-N-(N-heteroaryl)substituted carboxamides Piperazine derivatives of formula I ##STR1## and their pharmaceutically acceptable acid addition salts are 5-HT1A binding agents, particularly 5-HT1A antagonists and may be used, for example, as anxiolytics. In the formula A is ...	10/03/2000
6071860	2,4-Diamino-1, 3,5-triazines, their preparation, and their use as herbicides and plant growth regulators Compounds of the formula (I) and salts thereof ##STR1## where R1 to R5, A, Z, X, X', n and m are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepared analogously to known processes u...	06/06/2000
6069114	2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepa...	05/30/2000
6015774	Pyrazin-2-one derivatives, their use, and intermediates for their production Novel pyrazin-2-one derivatives of formula [1] are provided, ##STR1## which are useful as active ingredients of herbicides, wherein R1 is hydrogen or alkyl; R2 is haloalkyl; R3 is optionally substituted alkyl; alkenyl...	01/18/2000
6011031	Azolidinediones useful for the treatment of diabetes, dyslipidemia and hypertension: process for their preparation and pharmaceutical compositions containing them Novel antidiabetic compounds, their tautomeric forms, their derivatives, their analogues, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compositio...	01/04/2000
6011033	Phenylene derivatives This invention relates to a phenylene derivative represented by the following formula (1) or a salt thereof and also to a medicine containing it as an effective ingredient. ##STR1## wherein R1 represents H or halogen; A represents --CH.dbd...	01/04/2000
6008218	N-phenyl carbamate compounds, process for producing the same, and agricultural or horticultural bactericides This invention relates to An N-phenyl carbamate compound which is represented by the following formula (1): wherein R1 represents a hydrogen atom, an alkoxyalkyl group having 2 to 5 carbon atoms, an alkynyl group having 2 to 5 carbon atoms, an ...	12/28/1999
5981436	Substituted diazacyclohexanedi (thi) ones The invention relates to new substituted diazacyclohexanedi(thi)ones of the general formula (I) ##STR1## in which Q1, Q2, R1, R2, R3, R4, R5, R6 and R7...	11/09/1999
5919784	Heterocyclic aminomethyl compounds A compound of general formula (I): ##STR1## where A, X, R1, Y, n and Ar are defined in the description. Medicinal products containing the same are useful as D4 receptor Ligands....	07/06/1999
5885987	Phenylene derivatives This invention relates to a phenylene derivative represented by the following formula (1) or a salt thereof and also to a medicine containing it as an effective ingredient. ##STR1## wherein R1 represents H or halogen; A represents --CH.dbd...	03/23/1999
5883049	Hydantoin derivatives and herbicides containing said derivatives as active ingredient This invention provides with novel hydantoin derivatives, processes for preparing them, and herbicides containing said derivatives as active ingredient. The hydantoin derivative of this invention represented by the general formula (1): ##STR1## ...	03/16/1999

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Class 544/52 - Double bonded divalent chalcogen containing