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| Number | Title | Issue Date |
| 7414050 | Inhibitors of c-fms kinase The invention is directed to compounds of Formula I: wherein Z, X, J, R2 and W are set forth in the specification, as well as solvates, hydrates, tautomers and pharmaceutically acceptable salts thereof, that inhi... | 08/19/2008 |
| 6974869 | Piperizinones as modulators of chemokine receptor activity The present application describes modulators of CCR3 of formula (I): or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma and other allergic diseases. ... | 12/13/2005 |
| 6927215 | Heterocyclic fluoroalkenyl thioethers and the use thereof as pesticides (I) The present invention relates to novel heterocyclic fluoroalkenyl thioethers of the formula (I) in which X represents hydrogen, halogen or alkyl, m represents integer... | 08/09/2005 |
| 6878711 | Indole derivatives as PDE5-inhibitors Compounds of the general structural formula and use of the compounds and salts and solvates thereof, as therapeutic agents. ... | 04/12/2005 |
| 6727258 | Allosteric adenosine receptor modulators The present invention relates to compounds of formula (IA): the preparation thereof, pharmaceutical formulations thereof, and their use in medicine as allosteric adenosine receptor modulators for uses including protectio... | 04/27/2004 |
| 6683028 | Cyclic guanidine derivatives and their use as pesticides The invention relates to novel guanidine derivatives of the formula (I) ##STR1## in which A, R1, R2, R3 and Z are as defined in the description, to a process for their preparation and to their use for controlling animal ... | 01/27/2004 |
| 6531496 | O-aryl dithiazole dioxides The invention relates to new O-aryldithiazole dioxides, to two processes for their preparation, and to their use as pesticides in crop protection and in the protection of materials.... | 03/11/2003 |
| 6423718 | 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones useful as HIV reverse transcriptase inhibitors The present invention relates to 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones of formula I: ##STR1## or stereoisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as inhibitors of HIV reve... | 07/23/2002 |
| 6407232 | Ionic metal complex and process for synthesizing same The invention relates an ionic metal complex represented by the general formula (1): ##STR1## wherein M is an element of groups 3-15 of the periodic table; Aa+ represents a metal ion, onium ion or proton; X1 represents O, S or N... | 06/18/2002 |
| 6326368 | Aryloxy- and arylthiosubstituted pyrimidines and triazines and derivatives thereof The present invention provides novel compounds, and pharmaceutical compositions thereof, and methods of using same in the treatment of affective disorders, anxiety, depression, post-traumatic stress disorders, eating disorders, supranuclear palsey, irrita... | 12/04/2001 |
| 6124302 | 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones useful as HIV reverse transcriptase inhibitors The present invention relates to 4,4-disubstituted-3,4-dihydro-2(1H)-quinazolinones of formula I: ##STR1## or steroisomeric forms, stereoisomeric mixtures, or pharmaceutically acceptable salt forms thereof, which are useful as inhibitors of HIV ... | 09/26/2000 |
| 6075019 | Arylthio-dithiazindioxides and their use as pesticides The invention relates to novel S-aryl-dithiazine dioxides, to processes for their preparation and to the use in crop protection and in the protection of materials.... | 06/13/2000 |
| 6069114 | 2-amino-4-bicycloamino-1,3,5-Triazines, their preparation, and their use as herbicide and plant growth regulators Compounds of the formula (I) and their salts ##STR1## in which R1 to R6, Y1, to Y2, Y3, m and n are as defined in claim 1 are suitable as herbicides and plant growth regulators. They can be prepa... | 05/30/2000 |
| 5962437 | Lipid analogs for treating viral infections A method of treating viral infections, and in particular HIV-1, hepatitis B virus and herpes viruses, is disclosed. The method comprising administering to a subject in need of such treatment an infection-combating amount of a phospholipid or phospholipid ... | 10/05/1999 |
| 5874382 | Cyclic sulfonamide herbicides Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C1 -C3 alkyl); N(C1 -C3... | 02/23/1999 |
| 5824677 | Substituted amino alcohol compounds Disclosed are compounds having a straight or branched aliphatic hydrocarbon structure of formula I: ##STR1## In formula I, n is an integer from one to four and m is an integer from four to twenty. Independently, R1 and R2 are hy... | 10/20/1998 |
| 5786474 | N-fluorosulfonimides, process for their production, as well as their use as fluorinating agents N-fluorosulfonimides of general formula I (R1 --SO2)2 NF (I), in which R1 means a methyl group each or together a group --(CH2)n --with n=1, 2 or 3, especially N-flourome... | 07/28/1998 |
| 5728830 | Farnesyltransferase inhibitor The present invention relates to a farnesyltransferase inhibitor and an antitumor agent comprising, as an active ingredient, a piperazinedione derivative represented by formula (I): ##STR1## wherein R1 and R2 independently repre... | 03/17/1998 |
| 5571773 | (2-imidazolin-2-yl) fused heteropyridine compounds intermediates for the preparation of and use said compounds as herbicidal agents There are provided novel (2-imidazolin-2-yl) fused heteropyridine compounds, and intermediate compounds for the preparation thereof, and a method for controlling a wide variety of annual and perennial plant species therewith.... | 11/05/1996 |
| 5504095 | Aminobenzosultam derivatives as lipoxygenase inhibitors Aminobenzosultam derivatives, which are inhibitors of lipoxygenase, having the formula ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein Ar is cycloalkyl having five to seven carbon atoms, tetrahydropyranyl, pyrid... | 04/02/1996 |
| 5298499 | S-2-(substituted ethylamino)ethyl phosphorothioates Substituted phosphorothioate derivatives and pharmaceutical compositions thereof as potential antiradiation agents are disclosed.... | 03/29/1994 |
| 5212301 | Substituted fluorobenzenes Introduction of a fluoro substituent into an aromatic ring adjacent an electron donating group is difficult producing mixed isomers and low yields of desired products. A process for the introduction of a fluoro substituent into a substantially adjacent po... | 05/18/1993 |
| 5166342 | Dimethylfuryl-dihydro-1,3,5-dithiazines Dimethylfuryl-dihydro-1,3,5-dithiazines are useful flavorings having low taste threshold values. They impart a coffee or mocha taste, in particular to drinks, confectionery and bakery products.... | 11/24/1992 |
| 5158959 | Decahydroisoquinoline carboxylic acids What are disclosed are aminoacid compounds of the formula ##STR1## wherein n is 0 or 1, and salts thereof, said compounds and salts having hypotensive properties; methods for making the compounds; pharmaceutical compositions containing the compounds ... | 10/27/1992 |
| 5041667 | Process for producing chlorophenylhydrazine compounds A process for producing a chlorohenylhydrazine compound is disclosed, which comprises chlorinating at least one hydrogen atom on the phenyl nucleus in a beta-imidated phenylhydrazine compound and subsequently hydrolyzing the chlorinated compound. Said chl... | 08/20/1991 |
| 4954509 | Isoquinoline derivatives and their use as analgesics A compound, or a solvate or salt thereof, of formula (I): ##STR1## in which: RCO is an acyl group in which the group R contains a substituted or unsubstituted carbocyclic aromatic or heterocyclic aromatic ring and R1 R2 are inde... | 09/04/1990 |
| 4939251 | Novel spirolactones Novel 1-azaspiro[4.4] lactams are produced by reaction of at least one hydroxy-containing primary amino compound with a 4-ketodiacid compound or a 1,6-dioxaspiro[4.4]lactone. Molar excesses of amion compound result in production of spirodilactams, while l... | 07/03/1990 |
| 4929270 | Method of inducing chlorosis in a knapweed plant A method of selectively inducing chlorosis on a knapweed plant while spar other plants comprises applying a knapweed phytotoxic amount of the L,L isomer of the cyclodipeptide of the invention to a field at a period in time prior, during or subsequent to ... | 05/29/1990 |
| 4927831 | Spiro-isoquinoline-pyrrolidine tetrones and analogs thereof useful as aldose reductase inhibitors This invention relates to spiro-isoquinoline-pyrrolidine tetrones and their pharmaceutically acceptable salts thereof, to processes for their preparation, to methods for using the compounds, and to pharmaceutical preparations thereof. The compounds have p... | 05/22/1990 |
| 4895942 | Novel epoxy compounds Novel epoxyalkoxy-containing [4.4] spirodilactams having ring nitrogen atoms in the 1- and the 6- ring positions and having a substituent on each ring nitrogen atom, at least one of which substituents contains an epoxyalkyl moiety. Such epoxy compounds ar... | 01/23/1990 |
| 4838929 | Herbicidal sulfonamides Sulfonamides such as N-[(4,6-dimethoxypyrimidin-2-aminocarbonyl]-1,3-dihydro-6-methyl-3-oxofuro [3,4-c]pyridine-4-sulfonamide are useful as herbicides and plant growth regulants.... | 06/13/1989 |
| 4772309 | 5-acylamino-pyrazoles, composition containing them, and herbicidal and plant growth regulating method of using them A 5-Acylamino-pyrazole derivatives of the formula ##STR1## in which R1 represents hydrogen, halogen or nitro, R2 represents hydrogen, alkyl, alkenyl, alkinyl or optionally substituted cycloalkyl, R3 represents hydrogen or ... | 09/20/1988 |
| 4741765 | Herbicidal sulfonamides Benzenesulfonamide compounds such as N-[(4,6-dimethoxy-1,3,5-triazin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl-4 -oxo-1-phenyl-indeno[1,2-C]pyrazole-5-sulfonamide and N-[(4-methoxy-6-methyl-pyrimidin-2-yl)aminocarbonyl]-1,4-dihydro-3-methyl- 4-oxo-1-phe... | 05/03/1988 |
| 4742055 | 3- and 5-amino thiatriazines, and their pharmaceutical uses A class of 3- and 5-amino thiatriazine compounds exhibiting pharmacological activity, including anti-ulcerogenic and gastrointestinal cytoprotective activity, pharmaceutical compositions comprising these compounds, and methods for the treatment of gastroi... | 05/03/1988 |
| 4740231 | 1-aryl-5-alkoximinoalkylamino-pyrazoles, composition containing them, herbicidal and plant-growth regulating method of using them, and intermediates in the preparation of them 1-Aryl-5-alkoximinoalkylamino-pyrazoles of the formula ##STR1## in which R represents cyano or nitro, or represents an optionally substituted heterocyclic radical, R1 represents hydrogen or alkyl, R2 represents hydrogen or alkyl, or ... | 04/26/1988 |
| 4737184 | Herbicidal sulfonamides Novel N-(heterocyclicaminocarbonyl) substituted thiophene-, furan- and pyrrolesulfonamides, such as N-[(4-methoxy-6-methylpyrimidin-2-yl)aminocarbonyl]-6,7-dihydro-5H-thieno- [3,2-b]thiopyran-3-sulfonamide, 4,4-dioxide and N-[(4,6-dimethoxypyrimidin-2... | 04/12/1988 |
| 4723987 | Herbicidal sulfonamides Sulfonamides such as N-[(4,6-dimethoxypyrimidin-2-yl)aminocarbonyl]-1,3-dihydro-6-methyl-3-oxof uro[3,4-c]pyridine-4-sulfonamide are useful as herbicides and plant growth regulants.... | 02/09/1988 |
| 4713456 | Process for the preparation of 5-acylpyrimidines A process for the preparation of a 5-acylpyrimidine of the formula ##STR1## in which R is an organic radical comprising reacting a methyl ketone of the formula in a first stage with a formylating reagent in the presence of a base to form an enolketon... | 12/15/1987 |
| 4697011 | N-fluoro-N-perfluoromethyl sulfonamides N-fluoro-N-perfluoromethyl sulfonamide compounds are provided as fluorinating agents for the fluorination of organic compounds by either the direct electrophilic fluorination of organic compounds or by the fluorination of organic compound carbanions.... | 09/29/1987 |
| 4689414 | 2-(substituted imino)-6-aryl-3,6-dihydro-4-substituted-1,5(2H)-pyrimidinecarboxylic acids and analogs Cardiovascular activity is exhibited by compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof, wherein R1 is alkyl, cycloalkyl, aryl, heterocyclo, --(CH2)n --Y2, --(CH2 | 08/25/1987 |
