Class 544/304 - Alicyclic ring attached directly or indirectly to the diazine ring by nonionic bonding

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein an alicyclic ring is attached directly
No. of patents: 38
Last issue date: 10/10/2006

Number	Title	Issue Date
7119201	Triaryl-oxy-aryloxy-pyrimidine-2,4,6-trione metalloproteinase inhibitors The present invention relates to triaryl-oxy-aryloxy-pyrimidine-2,4,6-trione; metalloproteinase inhibitors of the formula wherein X, A, Y, B, G, W, and R1 are as defined in the specification, and to pharmace...	10/10/2006
7105670	Intermediates useful in the preparation of diaminothiazoles Disclosed are novel diaminothiazoles that are selective inhibitors of Cdk4. These compounds and their pharmaceutically acceptable salts and esters are anti-proliferative agents useful in the treatment or control of solid tumors, in particular breast, colon, lung and...	09/12/2006
7074925	N-substituted derivatives of 5-oxyiminobarbituric acid N-substituted derivatives of 5-oximinobarbituric add of the general formula where X is sulfur; R1 is selected from the group consisting of saturated or unsaturated alkyl, cycloalkyl, aryl and arylalkyl; and ...	07/11/2006
6833372	Non-peptide GnRH agents, Pharmaceutical compositions, and methods for their use Non-peptide GnRH agents that inhibit the effect of gonadotropin-releasing hormone are described. Such agents are useful for treating mammalian reproductive disorders and steroid hormone-dependent tumors as well as for regulating fertility, where suppression of gonad...	12/21/2004
6756374	Diaminothiazoles having antiproliferative activity Disclosed are novel diaminothiazoles of formula wherein R1, R2, R3, R4 and R5 are as herein disclosed. These compounds and their pharmaceutically acceptable salts an...	06/29/2004
6713486	Antiviral 2,4-pyrimidinedione derivatives and process for the preparation thereof 2,4-pyrimidinedione derivatives of formula (I) having high antiviral activity against wild-type and mutant HIV-1 and low toxicity are useful for treating AIDS (I) wherein: R1 is a C6-10 aryl or C3-10 heteroaryl group optionally havin...	03/30/2004
6706723	Pyrimidine-2,4,6-trione metalloproteinase inhibitors The present invention relates to pyrimidine-2,4,6-trione metalloproteinase inhibitors of the formula wherein X, Y, A, B and R1 are as defined in the specification, and to pharmaceutical compositions and method...	03/16/2004
6562542	Image-forming material and novel sulfonic acid ester derivative An image-forming material is described, comprising on an support an acid-generating agent selected from a sulfonic acid ester of a specific structure generating an acid by the action of heat and the polymer thereof, and a compound causing a light absorpti...	05/13/2003
6518425	Method of manufacture of 1,3-oxathiolane nucleosides Processes for the preparation of 1,3-oxathiolane nucleosides are provided that include efficient methods for the preparation of the 1,3-oxathiolane ring and subsequent condensation of the 1,3-oxathiolane with a pyrimidine or purine base. Using the process...	02/11/2003
6444682	Base analogues Nucleotide or base analogues having structure (3) or (4) ##STR1## wherein X.dbd.O or NH or S and each R6 is independently H or alkyl or alkenyl or alkoxy or aryl or a reporter moiety....	09/03/2002
6329379	Hepatitis C inhibitor tri-peptides Racemates, diastereoisomers and optical isomers of a compound of formula (I): ##STR1## wherein B is H, a C6 or C10 aryl, C7-16 aralkyl; Het or (lower alkyl)-Het, all of which optionally substituted with C1-6 alk...	12/11/2001
6254669	Bleed reduction agents for ink printing inks A compound of the Formula (1) and salts thereof: ##STR1## wherein: Ar, Ar1, J, J1, X, X1 W, W1, L and m are as defined in the description. The compounds of Formula (1) are useful as additives in inks, especially...	07/03/2001
6087498	Process for the preparation of unsymmetrical 4,6-bis(aryloxy) pyrimidine compounds There is provided a process for the preparation of unsymmetrical 4,6-bis(aryloxy)pyrimidine compounds. The unsymmetrical 4,6-bis(aryloxy)pyrimidine compounds are useful as pesticidal agents....	07/11/2000
5922727	Antiviral substituted pyrimidinedione homocarbocyclic nucleoside derivatives and methods for the preparation thereof and compositions containing the same as active ingredients The present invention relates to novel compound of general formula (I) and pharmaceutically acceptable salts thereof, and process for the preparation of such derivatives and to pharmaceutical compositions containing the same as active ingredients. ##...	07/13/1999
5849910	Process for the preparation of unsymmetrical 4,6-bis aryloxy-pyrimidine compounds This invention provides an improved process for the preparation of unsymmetrical 4,6-bis(aryloxy)pyrimidine compounds having the structural formula I ##STR1## The unsymmetrical 4,6-bis(aryloxy)pyrimidine compounds are useful as pesticidal agents...	12/15/1998
5747500	Antiviral 2, 4-pyrimidinedione derivatives Novel 2,4-pyrimidinedione compounds, and pharmaceutically acceptable salts thereof which possess good antiviral activities, and specifically represented by the following formula(I): ##STR1## wherein: R1 represents an unsubstituted or subst...	05/05/1998
5656745	Nucleotide analogs Nucleotide analogs characterized by the presence of an amidate linked amino acid or an ester linked group which is bonded to the phosphorus atom of phosphonate nucleotide analogs are disclosed. The analogs comprise a phosphoamidate or ester bond that is h...	08/12/1997
5599770	Herbicidal composition containing 2-benzyloxypyrimidine derivatives, processes for producing the derivatives and 2-benzyloxypyrimidine derivatives A herbicidal composition comprising a herbicidally effective amount of a 2-benzyloxypyrimidine derivative represented by the formula (I): ##STR1## wherein R1 and R2 are each independently H, a halogen, hydroxyl, C1 -C...	02/04/1997
5478928	2',3'-dideoxy-4'-thioribonucleosides and synthetic precursors thereof 2',3'-dideoxy-4'-thioribonucleosides useful as antiviral agents in the treatment and prevention of AIDS are disclosed. In accordance with one aspect of the invention there are provided compounds of the formula ##STR1## where X.dbd.H, N3 or...	12/26/1995
5420133	Quinazolinones substituted with phenoxyphenylacetic acid derivatives Phenoxyphenylacetic acids and derivatives of general structural formula I ##STR1## have endothelin antagonist activity and are therefore useful in treating cardiovascular disorders, such as hypertension, postischemic renal failure, vasospasm, cerebra...	05/30/1995
5360576	Chiral alkenylaryl 2,3-epoxyalkyl ethers, and the use thereof in liquid-crystalline mixtures Compounds of the formula (I) in which the symbols have the following meanings: R1 is straight-chain or branched (C3 -C2)alkenyl containing a terminal double bond, it being possible for one or two non-adjacent CH2	11/01/1994
5284820	Herbicidal substituted cycloalkenes Herbicidal substituted cycloalkenes of the formula ##STR1## in which A is a straight-chain or branched, optionally substituted alkanediyl group, X is O, S, N--R8 or CR9 R10, Y is O, S, NH or N-alkyl, Z is N or R11	02/08/1994
5270318	Heterocyclic compounds A compounds of formula (I): ##STR1## wherein R1 and R2 are independently hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, halogen, haloalkyl, alkoxy, alkenoxy, alkoxyalkyl, haloalkoxy, alkylthio, cyano, nitro, ami...	12/14/1993
5262385	Halogen-containing compounds, herbicidal composition containing the same as an active ingredient, and intermediary compounds therefor A compounds represented by the formula ##STR1## wherein X represents a fluorine atom, W represents an oxygen atom, sulfur atom or group --OCH2 --, Z1 and Z 2 each represent a nitrogen atom or group CH, but when Z1	11/16/1993
5262386	Pyrimidinyl- and triazinyl-salicylamides and their use and preparation Pyrimidinyl- and triazinyl-salicylamides of the formula I ##STR1## in which the meanings of the radicals are described in claim 1, and the salts of compounds of the formula I which have a free hydroxycarbonyl group have a herbicidal and plant-growth ...	11/16/1993
5246914	Salicyloyl (thio)ether derivatives, their preparation and intermediates for their preparation Salicyloyl(thio)ether derivatives of the formula I, ##STR1## where is oxygen or sulfur and Z is carbon or nitrogen, and the radicals R1 to R4 and A have the meanings given in the disclosure, and processes and intermediates for p...	09/21/1993
5246938	Heterocyclic compounds Compounds of formula (I): ##STR1## wherein R1, R2 and R3 are independently hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, alkylcycloalkyl, halogen, haloalkyl, alkoxy, alkenoxy, alkoxyalkyl, haloalkoxy, alkylthio, cyan...	09/21/1993
5232897	Herbicidal pyrimidine compounds, compositions containing the same and method of use Herbicidal pyrimidine compound having the formula ##STR1## wherein the substitutents A, R1, R2, X, Y1, Y2, Y3 and Z are as defined herein below....	08/03/1993
5225550	Process for the preparation of substituted acyclic nucleosides, and intermediates occurring therein It is possible, by using symmetrical formaldehyde acetals of the formula ##STR1## in which the substituents R1 -R3 have the specified meanings, advantageously to introduce the substituent ##STR2## into nitrogen-containing h...	07/06/1993
5178663	3-alkoxyalkanoic acid derivative, process for preparing the same and herbicide using the same Disclosed is a 3-alkoxyalkanoic acid compound represented by the following formula (I): ##STR1## wherein R1 represents a lower alkyl group, a lower alkenyl group, a lower alkynyl group, a cycloalkyl group, a halo-lower alkyl group or a ...	01/12/1993
5139563	Herbicidal compounds Compounds of formula I ##STR1## wherein A is nitrogen or a group CR5 ; each of R1, R2 and R5 is, independently, hydrogen, halogen, formyl, cyano, carboxy, azido or optionally substituted alkyl, alkenyl, alk...	08/18/1992
5112835	6-substituted acyclopyrimidine nucleoside derivatives and antiviral agents containing the same as active ingredient thereof 6-substitutted acyclopyrimidine nucleoside derivatives represented by the following general formula I: ##STR1## wherein R1 represents a hydrogen or halogen atom or a group of alkyl, alkenyl, alkynyl, alkylcarbonyl, arylcarbonyl, arylcarbon...	05/12/1992
4908379	Nitrogen-containing heterocyclic compounds and compositions for controlling and/or preventing pests and blights (diseases) A nitrogen-containing heterocyclic compound of the following formula: ##STR1## wherein D represents --N.dbd. or ##STR2## E represents .dbd.N--, ##STR3## G represents --N.dbd., ##STR4## with proviso that when G represents --N.dbd. ...	03/13/1990
4889552	2-Phenoxypyrimidine derivative and herbidical composition A 2-phenoxypyrimidine derivative having the formula: ##STR1## wherein R is a formyl group or --COOR1 wherein R1 is a hydrogen atom, a lower alkyl group, a 2-methylsulfonylethyl group, a diethoxypropyl group, a lower alkenyl grou...	12/26/1989
4469696	Substituted 2-amino-pyridine derivative compounds, their production and their medicinal use The invention relates to 4-,5-and 6-substituted 2-amino pyridines of Formula (I) and methods for their preparation. Also included in the invention are compositions containing said 2-amino pyridines of Formula (I) and the use of said compounds and composit...	09/04/1984
4427437	Use of 2-phenoxypyrimidines as herbicides A process of inhibiting the growth of, severely damaging, or killing plants which process comprises applying to the plant or to the growth medium thereof an effective amount of a composition comprising as active ingredient a compound of formula I: ##...	01/24/1984
4412856	Herbicidal heterocyclic and substituted phenyl phenylacetylene amines The novel compounds of the formula I are useful selective herbicides for postemergence application in crops of cereals, maize and rice. In formula I, ##STR1## A is an unsubstituted or substituted amino group, Q is a C2 -C6 alkyl...	11/01/1983
4060525	Five- or six-membered heterocyclic mono -and dialcohols New mono- or dialcohols of mononuclear, five-membered or six-membered, unsubstituted or substituted N-heterocyclic compounds which contain two NH-groups in the molecule, by reaction of mononuclear, five-membered or six-membered, unsubstituted or substitut...	11/29/1977

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Class 544/304 - Alicyclic ring attached directly or indirectly to the diazine ring by nonionic bonding