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Class 544/3 - Six-membered hetero ring consists of sulfur, nitrogen, and carbon


Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the six- membered hetero ring includes
No. of patents: 188
Last issue date: 10/14/2008


1          
NumberTitleIssue Date
7435731Substituted pyrazolo[3,4-d]pyrimadines and methods of using the same
Compounds of the formula Ia or Ib: wherein A, B, X, Y, Z, W, k, R1, R2, R3, R4 and R5 are those defined herein, and compositions comprising the same. The present invent...
10/14/2008
7411093Aminocycloalkanes as DPP-IV inhibitors
The present invention relates to compounds of formula (I) wherein R1 is as defined in the description and claims, and pharmaceutically acceptable salts thereof. The compounds are useful for the treatment and/or p...
08/12/2008
7371743Carboxylic acid amides, the preparation thereof and their use as medicaments
The present invention relates to new substituted carboxylic acid amides of general formula wherein A, B and R1 to R5 are defined as in claim 1, the tautomers, the enantiomers, the diastereomers,...
05/13/2008
7329288N-heteroaryl secondary para-phenylenediamine, a dye composition comprising such a para-phenylenediamine, a process for preparing this composition and use thereof
The present disclosure relates to a novel family of N-heteroaryl secondary para-phenylenediamines, to their preparation, to their use for dyeing the hair and to a dye composition for dyeing keratin fibers, for example, human keratin fibers such as the hair, comprisi...
02/12/2008
7323460N-(substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides useful as HIV integrase inhibitors
N-(Substituted benzyl)-8-hydroxy-1,6-naphthyridine-7-carboxamides are inhibitors of HIV integrase and inhibitors of HIV replication. The naphthyridine carboxamides are of Formula (I): wherein R1′, R
01/29/2008
7301028Mitotic kinesin inhibitors
The present invention relates to dihydropyrazole compounds that are useful for treating cellular proliferative diseases, for treating disorders associated with KSP kinesin activity, and for inhibiting KSP kinesin. The invention also related to compositions which com...
11/27/2007
7192948Bicyclic heterocycles as HIV integrase inhibitors
The invention encompasses a series cyclic bicyclic heterocyclic compounds of Formula I which are inhibitors of HIV integrase and prevent viral integration into human DNA. This action makes the compounds useful for treating HIV infection and AIDS. The invention also ...
03/20/2007
7157447Bicyclic heterocycles as HIV integrase inhibitors
The invention encompasses a series bicyclic pyrimidinone compounds of Formula I which inhibit HIV integrase and prevent viral integration into human DNA. This action makes the compounds useful for treating HIV infection and AIDS. The invention also encompasses pharm...
01/02/2007
7135467HIV integrase inhibitors
Compounds useful for treating HIV are disclosed having the general formula wherein R1, R2, and B are as defined in the specification. Compositions containing the compounds and methods for us...
11/14/2006
7115599Sulfonamide-substituted pyrazolopyridine compounds
This invention relates to compounds of the formula in which R1, R2, and R3 are as defined in the claims, to a process for preparing such compounds, to pharmaceutical compositions ...
10/03/2006
7108962Photographic processing composition and image-forming method using the same
A photographic processing composition, containing at least one compound of formula (I) or (II): A1-X-L-Y-A2  (I) wherein A1 and A2 each are a specific aryl or aromatic heterocyclic group; L is a...
09/19/2006
7037908HIV integrase inhibitors
The present invention relates to a series of pyrimidine compounds of Formula I which inhibit HIV integrase and to pharmaceutical compositions and methods of treatment for AIDS or ARC using these compounds ...
05/02/2006
6927216Cyclic sulfonyl compounds as inhibitors of metalloproteases
The present application describes novel cyclic sulfonyl derivatives of formula I: or pharmaceutically acceptable salt forms thereof, wherein ring B is a 5-7 membered cyclic system containing from 0-2 heteroatoms select...
08/09/2005
6924282Sodium salt of an HIV integrase inhibitor
A sodium salt of Compound A is disclosed, wherein Compound A is of formula: Compound A is an HIV integrase inhibitor useful for preventing or treating HIV infection, for delaying the onset of AIDS, and for treating AID...
08/02/2005
6921759Aza- and polyaza-naphthalenyl carboxamides useful as HIV integrase inhibitors
Aza- and polyaza-naphthalenyl carboxamide derivatives including certain quinoline carboxamide and naphthyridine carboxamide derivatives are described. These compounds are inhibitors of HIV integrase and inhibitors of HIV replication, and are useful in the prevention...
07/26/2005
6894005Herbicides
Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomer of those compounds, are suitable for use as herbicides. ...
05/17/2005
6894041Oxazolyl-acid amide derivatives useful as inhibitors of PDE4 isozymes
This application is directed to compounds useful as inhibitors of PDE4 in the treatment of diseases regulated by the activation and degranulation of eosinophils, especially asthma, chronic bronchitis, and chronic obstructuive pulmonary disease, of the formula:
05/17/2005
6887994C-nitroso compounds and use thereof
A C-nitroso compound having a molecular weight ranging from about 225 to about 1,000 (from about 225 to about 600 for oral administration) on a monomeric basis wherein a nitroso group is attached to a tertiary carbon, which is obtained by nitrosylation of a carbon a...
05/03/2005
6881840Benzothiazine dyes for imaging elements
This relates to a dye represented by Formulae II and IIA below: wherein; R1 represents a hydrogen, an aryl group containing 6 to 14 carbon atoms, or an alkyl group containi...
04/19/2005
6869945Pyrrolyl-and imidazolyl-acid amide derivatives useful as inhibitors of PDE4 isozymes
This application is directed to compounds useful as inhibitors of PDE4 in the treatment of diseases regulated by the activation and degranulation of eosinophils, especially asthma, chronic bronchitis, and chronic obstructuive pulmonary disease, of the formula:
03/22/2005
6849623Xanthine and phenazone-acesulfame-H complexes having improved taste, process for their preparation and their use
Complex compounds or adducts of xanthine derivatives, for example propentofylline or pentoxyfylline, or phenazone derivatives, for example phenazone, propylphenazone and aminophenazone, and acesulfame-H, in which the components are present in a molar ratio of 1:1 or...
02/01/2005
6828276Herbicidally active benzoylcyclohexanediones
There are described benzoylcyclohexanediones of the formula I, their preparation, and their use as herbicides and plant growth regulators. In this formula (I), C1, C2, C3 are cyclic radic...
12/07/2004
6787522Antibacterial agents
Compounds of formula (I) are antibacterials: wherein: R1 represents hydrogen, or C1-C6 alkyl or C1-C6 alkyl substituted by one or more halogen atoms; R2 ...
09/07/2004
6759544Antimicrobially active acesulfame complexes, process for their preparation and their use
Complex compounds containing acesulfame have good antimicrobial action, in particular antibacterial action, and are distinguished by the fact that they are complex compounds of metallic elements such as zinc, copper, silver, or nonmetallic quaternary ammonium cation...
07/06/2004
6753425Photographic processing composition containing bistriazinyl arylenediamine derivative
A processing composition for silver halide photographic light-sensitive materials, comprises a bis[2,6-diaminotriazin-4-yl]arylenediamine derivative having at least one of a sulfonic acid group, a carboxylic group and a hydroxyl group within the molecule. This proce...
06/22/2004
6627629N-ureidoheterocycloalkyl-piperidines as modulators of chemokine receptor activity
The present application describes modulators of CCR3 of formula (I): ##STR1## or pharmaceutically acceptable salt forms thereof, useful for the prevention of asthma and other allergic diseases....
09/30/2003
66080702,3-substituted indole compounds as anti-inflammatory and analgesic agents
This invention provides a compound of the following formula: ##STR1## or the pharmaceutically acceptable salts thereof wherein Z is OH, C1-6 alkoxy, --NR2R3 or heterocycle; Q is selected from the following: (a) an optionally substituted phenyl, (b) an opt...
08/19/2003
65967162-propane-sulphonamide derivatives
The present invention relates to the potentiation of glutamate receptor function using certain 2-propane-sulphonamide derivatives. It also relates to novel 2-propane-sulphonamide derivatives, to processes for their preparation and to pharmaceutical compos...
07/22/2003
6559155Pyrimidinone derivatives for the treatment of atherosclerosis
Pyrimidones of formula (I) are inhibitors of the enzyme LpPLA2 and thereof use in treating inter alia atherosclerosis, ##STR1## in which: R1 is COOH or a salt thereof, COOR10, CONR11R.sup.12, CN or CH...
05/06/2003
6531539Organosilicon compounds
The invention is directed to organosilicon compounds of the general formula ##STR1## prepared by reacting triazine compounds with functional groups (e.g., chlorine) and corresponding compounds (e.g., mercapto). The organosilicon compounds can be used in r...
03/11/2003
6525099N-substituted sulfonamide derivatives
The present invention provides certain N-substituted sulfonamide derivatives useful for potentiating glutamate receptor function in a mammal and therefore, useful for treating a wide variety of conditions, such as psychiatric and neurological disorders....
02/25/2003
65093543-arylphenyl sulfide derivative and insecticide and miticide
3-Arylphenyl sulfide derivatives represented by general formula (I): ##STR1## (wherein R is a C2 -C6 alkyl group, a C2 -C6 alkenyl group, a C2 -C6 alkynyl group or the like, B0 to B
01/21/2003
6500818Naphthalenecarboxamides as tachykinin receptor antagonists
Compounds having the following formula ##STR1## wherein L, M, R2, R3, R4, R5, R6, R7, X1 and X2 are as defined in the specification, pharmaceutically-acceptable salt t...
12/31/2002
6495686Pyrimido [4,5,b]indolizine derivatives and aza analogues thereof; CRF1 specific ligands
Disclosed are compounds of the formula: ##STR1## wherein Ar, R1, R2, R3, W, X, Y, and Z are substituents as defined herein, which compounds are highly selective partial agonists or antagonists at human CRF1 rece...
12/17/2002
6420360Sultam and sultone derived oxazolidinones
The present invention provides a compound of formula I ##STR1## These compounds are useful as antibiotic agents....
07/16/2002
6416762Anti-picornaviral ligands via a combinatorial computational and synthetic approach
The present invention provides structure-based combinatorial libraries of compounds containing the functional group minima of picornaviruses including poliovirus and rhinovirus. The libraries can be used to screen for therapeutical antiviral compounds, e....
07/09/2002
6416922Azomethine dye precursor, image-forming material, and image-forming method
The present invention related to an azomethine dye precursor represented by the following general formula (1) and the image-forming material and image-forming method using the azomethine dye precursor: wherein Ar represents an aryl group or a heterocyclic...
07/09/2002
6407232Ionic metal complex and process for synthesizing same
The invention relates an ionic metal complex represented by the general formula (1): ##STR1## wherein M is an element of groups 3-15 of the periodic table; Aa+ represents a metal ion, onium ion or proton; X1 represents O, S or N...
06/18/2002
6407098Fungicidal aza-heterocycloalkenes
The application relates to novel heterocycloalkenes, to a number of processes for their preparation and to their use as fungicide....
06/18/2002
6383230Cationic monobenzenic dyes, their use for the oxidation-dyeing of keratin fibers, dye compositions and dyeing processes
The invention relates to novel monobenzenic dyes including at least one cationic group Z, Z chosen from quaternized aliphatic chains, aliphatic chains including at least one quaternized saturated ring and aliphatic chains including at least one quaternize...
05/07/2002
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