Class 544/294 - Polycyclo-carbocyclic ring system having at least three cyclos

Subclass of Class 544 - Organic compounds -- part of the class 532-570 series
Definition: Compounds having a polycyclo ring system which contains
No. of patents: 87
Last issue date: 10/07/2008

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Number	Title	Issue Date
7432371	Nanofilm and membrane compositions Nanofilms useful for filtration are prepared from oriented amphiphilic molecules and oriented macrocyclic modules. The amphiphilic species may be oriented on an interface or surface. The nanofilm may be prepared by depositing or attaching an oriented layer to a subs...	10/07/2008
7321033	3-B-D-ribofuranosylthiazolo [4,5-] pyrimidine nucleosides and uses thereof The invention is directed to 3-β-D-ribofuranosylthiazolo[4,5-d]pyridimine nucleosides and pharmaceutical compositions containing such compounds that have immunomodulatory activity. The invention is also directed to the therapeutic or prophylactic use of such compou...	01/22/2008
7279575	Pyrimidylpyrrole derivatives active as kinase inhibitors Pyrimidylpyrrole derivatives of formula (I) and pharmaceutically acceptable salts thereof, as defined in the specification, process for their preparation and pharmaceutical compositions comprising them are disclosed; the compounds of the invention may be useful, in ...	10/09/2007
7226926	8-fluoroimidazo 1,2-a pyridine derivatives as ligands for GABA receptors A class of 8-fluoroimidazo[1,2-α]pyridine derivatives, substituted at the 3-position by an optionally substituted five-membered or six-membered heteroaromatic ring, being selective ligands for GABAA receptors, in particular having high affinity for the �...	06/05/2007
7205304	Sulfonyl-Derivatives as novel inhibitors of histone deacetylase This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, composition...	04/17/2007
7176310	Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents This invention is directed to compound of the following formula (I): wherein R1, R2, R3 and R4 are as described herein. These compounds and pharmaceutical compositions ...	02/13/2007
7125996	Fluorescent probes for use in protein kinase inhibitor binding assay The invention provides methods relating to a novel screening assay format that can be applied to broad members of the protein kinase gene family. The assay uses a series of labeled, active site probes described herein that can be displaced by an inhibitor agent. The...	10/24/2006
7087599	Estrogen receptor modulators The present invention relates to compounds and derivatives thereof, their synthesis, and their use as estrogen receptor modulators. The compounds of the instant invention are ligands for estrogen receptors and as such may be useful for treatment or prevention of a v...	08/08/2006
7087598	Diamide invertebrate pest control agents containing a non-aromatic heterocyclic ring This invention provides compounds of Formula I, their N-oxides and agriculturally suitable salts wherein A and B are independently O or S; J is an optionally substituted 5- or 6-memebered nonaromatic heterocyclic ring; K is taken together with the two contiguous lin...	08/08/2006
7018685	Fluorinated aromatic compounds and the use of the same in liquid crystal mixtures The invention relates to fluorinated aromatics of the formula (I) where X is CH2, C═O, CF2, O or S, Y is H or F, with the proviso that Y has to be F when X is CH2	03/28/2006
6972297	2-Hydroxy-mutilin carbamate derivatives for antibacterial use 2-(S)-hydroxymutilin carbamate derivatives of formula (I), in which R1 is a 5- or 6-membered optionally substituted heteroaryl group; and R2 is vinyl or ethyl, are useful in the treatment of bacterial infections	12/06/2005
6949557	Hydroanthracene based compounds as anticancer agents The invention relates to the use of novel anthracene based compounds for the inhibition or prevention of the growth or multiplication of cancer cells, and to therapeutic compositions containing such compounds. The invention relates more specifically to the use of hy...	09/27/2005
6872824	Pyrimidine spirobifluorene oligomer for organic light-emitting device A fluorene-based pyrimidine-containing conjugated oligomer applied in six different layers in an OLED, respectively, used as an electron-transport emitting layer, an emitting layer, a host in the emitting layer, the ETL, a host in the electron-transport emitting lay...	03/29/2005
6756375	10-Aryl-11h-benzo[b]fluorene derivatives and analogs for medicinal use The invention provides for a non-steroidal compound having the formula wherein Re and ′Re are OH, optionally independently etherified or esterified; Z is —CH2— or —CH2C...	06/29/2004
6737423	Substituted heterocyclo-norbornylamino derivatives, processes for their preparation, their use as medicaments or diagnostics, and medicaments comprising them Substituted heterocyclo-norbornylaminoderivatives having: a) an exo-configuration nitrogen and an endo-fused five-membered ring or six-membered ring of the formula (I) or b) an exo-configuration nitrogen and an exo-fused five-membered ring or six-membered ring of th...	05/18/2004
6492355	Adamantane derivatives The invention provides compounds of general formula ##STR1## in which m, A, R1 and Ar have the meanings defined in the specification; a process for their preparation; pharmaceutical compositions containing them; a process for preparing the phar...	12/10/2002
6399620	Cycloalkyl derivatives as inhibitors of bone resporption and vitronectin receptor antagonists There are described cycloalkyl derivatives of the formula (I) R1 --Y--A--B--D--E--F--G (I) in which R1, Y, A, B, D, E, F and G have the meaning indicated herein, their preparation and their use as medicaments. The compounds according to ...	06/04/2002
6288123	Therapeutic guanidines The present invention provides therapeutically useful substituted guanidines, and methods of treatment and pharmaceutical compositions that utilize or comprise one or more of such guanidines....	09/11/2001
6211189	Amino-spiro-quinazoline compounds There are provided novel compounds of formula (I) ##STR1## wherein A represents an aromatic carbocyclic ring or a 5- or 6-membered heterocyclic aromatic ring containing 1 to 3 heteroatoms which may be the same or different and are selected from O, N and S...	04/03/2001
6200981	Pyrimidin derivatives The invention relates to new pharmaceutically active compounds which are are P2-purinoceptor 7-transmembrane (TM) G-protein coupled receptor antagonists, compositions containing them and processes for their preparation....	03/13/2001
6174924	Therapeutic guanidines The present invention provides therapeutically useful substituted guanidines, and methods of treatment and pharmaceutical compositions that utilize or comprise one or more of such guanidines....	01/16/2001
6143791	Therapeutic guanidines The present invention provides therapeutically useful substituted guanidines, and methods of treatment and pharmaceutical compositions that utilize or comprise one or more of such guanidines....	11/07/2000
6107297	2,4-Dithi(oxo)-pyrimidin-5-yl compounds bearing a tricyclic substituent useful as P2 purinoceptor antagonists The invention relates to new pharmaceutically active compounds which are P2-purinoceptor 7-transmembrane (TM) G-protein coupled receptor antagonists, compositions containing them and processes for their preparation....	08/22/2000
6060591	Water-soluble fiber-reactive dyes, processes for their preparation, and their use The disclosed dyes (which are fiber-reactive and are useful for dyeing materials containing OH and/or carboxamide groups) are compounds of the formula (1) Fb--Zn (1) in which: Fb is the radical of vario...	05/09/2000
6015900	N-aminoalkylfluorenecarboxamides Disclosed are compounds of formula (I) or the pharmaceutically acceptable salts thereof wherein: ##STR1## G represents a group of the formula (a), (b) or (c) where Ra and Rb represent hydrogen, or organic or inorganic substituen...	01/18/2000
5703235	N-Aminoalkyl-2-anthracenecarboxamides; new dopamine receptor subtype specific ligands Disclosed are compounds of the formula: ##STR1## or the pharmaceutically acceptable acid addition salts thereof, wherein: R1, R2, R3, R4, R5, R6, R7, R8 and R	12/30/1997
5659033	N-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands Disclosed are compounds of the formula ##STR1## or the pharmaceutically acceptable salts thereof wherein: G represents a group of the formula ##STR2## where Ra and Rb represent hydrogen, or organic or inorganic substit...	08/19/1997
5646269	Method for oligonucleotide analog synthesis The present invention is directed to improved methods to synthesize oligonucleotide analogs having an acetal linkage, such as a 3',5'-formacetal (3' --O--CH2 --O-- 5'), 3',5'-thioformacetal (3' --S--CH2 --O-- 5') or an analogous 2',5...	07/08/1997
5512575	Methanoanthraceneyl methyl piperidinyl compounds Compounds of formula I or I', ##STR1## wherein X and Y are independently selected from hydrogen, halo, and (1-6C)alkoxy; R1 is selected from (A) (1-6C)alkyl; (B) phenyl and naphthyl or substituted versions thereof; (C) phenyl (1-3C)alkyl and na...	04/30/1996
5503666	Dyestuffs and their use in inks for ink-jet printing processes Novel dyestuffs have been found which are obtainable by reacting A) polyamines containing at least 2 primary or secondary amino groups with B) reactive compounds containing at least two groups which are reactive towards primary and secondary amines in an amount of ...	04/02/1996
5463031	Reactive dyestuffs Reactive dyestuffs of the formula ##STR1## in which the substituents have the meanings given in the description are highly suitable for the dyeing and printing of cellulose materials and nitrogen-containing materials. They produce dyeings and prints ...	10/31/1995
5455246	Piperidine derivatives Compounds of formula I, Ia or Ib and pharmaceutically acceptable salts thereof, useful in the treatment of neuropsychiatric disorders such as psychoses; pharmaceutical compositions comprising a compound of formula I and a pharmaceutically acceptable dilue...	10/03/1995
5420255	Process for the continuous reaction of halogenopyrimidines with amines A process for the continuous reaction of halogenopyrimidines with amines, a halogenopyrimidine and an aqueous amine solution or suspension being passed into a reactor and the reaction product being subsequently conducted away, is described, characterized ...	05/30/1995
5399674	Dyestuffs containing pyrimidine-carboxylic acid amide radical having fiber-reactive group, processes for their preparation and their use Fiber-reactive dyestuffs, processes for their preparation and their use Dyestuffs of the formula (1) are described ##STR1## The dyestuffs have fiber-reactive properties and dye materials containing hydroxy groups and/or containing carboxamide groups, in p...	03/21/1995
5342927	Reactive dyestuffs for the dyeing and printing of hydroxyl-or amino-containing materials Reactive dyestuffs of the formula ##STR1## in which X is ##STR2## and Z is a heterocyclic reactive group and the remaining groups have the meaning given in the description, are highly suitable for the dyeing and printing of hydroxyl- or ami...	08/30/1994
5300642	଱, ଱-disubstituted aromatics and heteroaromatics as cognition enhancers Cognitive defeciencies or neurological dysfunction in mammals are treated with ଱,଱-disubstituted aromatic or heteroaromatic compounds. The compounds have the formula: ##STR1## or a salt thereof wherein X and Y are taken together to form a...	04/05/1994
5256784	Nonlineaphores and polymers incorporating such nonlineaphores Nonlinear-optic (NLO) compositions containing functionalized merocyanine dyes, such that the molecules, comprising the NLO-active compositions have a functional group at each end of the molecule and each functional group differing in reactivity, thus perm...	10/26/1993
5173489	଱,଱-disubstituted aromatics and heteroaromatics as cognition enhancers Cognitive defeciencies or neurological dysfunction in mammals are treated with ଱,଱-disubstituted aromatic or heteroaromatic compounds. The compounds have the formula: ##STR1## or a salt thereof wherein X and Y are taken together to form a...	12/22/1992
5164499	Nitroaryl carbonyl compounds, nitrodihydroaryl carbonyl intermediates thereto, and processes Nitroaryl carbonyl Formula (IIA) compounds, their nitrodihydroaryl carbonyl Formula (I) intermediates, processes for preparing Formula (II) compounds, and a process for preparing Formula (I) compounds, wherein each process comprises the reaction of a nitr...	11/17/1992
5147882	Cyclophanes, pharmaceutical compositions containing these compounds and processes for preparing them Cyclophanes of the general formula ##STR1## wherein X1, X2, A, R and R1 to R4 are as defined herein, the enantiomers, diastereomers and addition salts thereof and, more particularly, for pharmaceutical use,...	09/15/1992

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Class 544/294 - Polycyclo-carbocyclic ring system having at least three cyclos