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| Number | Title | Issue Date |
| 7968710 | Prokineticin 1 receptor antagonists The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1... | 06/28/2011 |
| 7902358 | Prokineticin 1 receptor antagonists The present invention relates to certain novel compounds of Formula (I): and methods for preparing these compounds, compositions, intermediates and derivatives thereof and for the treatment of prokineticin 1 or prokinetin 1... | 03/08/2011 |
| 7230100 | Stereoselective method for the preparation of nucleosides A process for producing predominantly cis nucleosides or nucleoside analogues and derivatives of formula (A): wherein R1 is a pyrimidine base or a pharmaceutically acceptable derivative thereof and Q is oxygen, c... | 06/12/2007 |
| 7193080 | Dye-forming coupler, silver halide photographic light-sensitive material and azomethine dye compound A dye-forming coupler and compound of formula (I): wherein Q represents a residue that forms, together with —N—C═N—, a nitrogen-containing 6-membered ring; RA represents an aryl, heterocyclic, ... | 03/20/2007 |
| 6831174 | Processes for preparing substituted 1, 3-oxathiolanes with antiviral properties Disclosed are processes for preparing compounds of the formula (I) and pharmaceutically acceptable salts or esters thereof: wherein R2 is a purine or pyrimidine base or an analogue or derivative thereof; and... | 12/14/2004 |
| 6780992 | Heterocyclic compounds, process for their preparation and pharmaceutical compositions containing them and their use in the treatment of diabetes and related diseases The present invention relates to novel antidiabetic compounds, their tautomeric forms, their derivatives, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutically acceptable compo... | 08/24/2004 |
| 6630578 | Thioether derivatives, their method for production and use Novel dendritic molecules are provided which respond immediately by emission of light when stimulated with light or electric energy, and are useful, for example, as switching material of memory. The dendritic molecules have a core, a branch structure comp... | 10/07/2003 |
| 6372435 | Methods of surveying for CC (Beta) chemokine receptor variants and their association with HIV-1 transmission and/or disease progression The present invention provides methods of correlating genetic variants in the beta-chemokine receptor 5 (CCR5) locus, more specifically CCR5 promoter alleles and genotypes, with HIV-1 transmission and/or disease progression in individuals and populations.... | 04/16/2002 |
| 6258915 | Solid polyurethane hardeners having triazine groups, processes for preparing such compounds, and their use Solid polyurethane hardeners (curing agents) having triazine groups, are prepared by reacting polyaddition compounds with a second compound having a >C.dbd.N-- group. The polyaddition compounds are prepared by reacting a uretdione-functional polyisocyanat... | 07/10/2001 |
| 6251829 | Herbicidal benzoyloxy carboxylates and carboxamides This invention relates to herbicidal alpha-(2,4,5-trisubstituted)- and alpha-(2,5-disubstituted)-benzoyloxy-alpha-beta-, and/or beta-gamma-unsaturated-carboxylates and their derivatives, to compositions which contain these compounds, and to methods of use... | 06/26/2001 |
| 6136827 | Cyclic amine modulations of chemokine receptor activity The present invention is directed to cyclic amines of the formula I: ##STR1## (wherein R1, R2, R3, m and n are defined herein) which are useful as modulators of chemokine receptor activity. In particular, these compou... | 10/24/2000 |
| 6124308 | Optically active phenyl pyrimidine derivatives as analgesic agent A pyrimidine of formula (I) ##STR1## and its pharmaceutically acceptable acid addition salts are useful as analgesics, as anticonvulsants or in the treatment of irritable bowel syndrome or bipolar disorder.... | 09/26/2000 |
| 6090940 | Method for producing potassium oxonate A method for producing potassium oxonate which comprises dissolving allantoin in an aqueous potassium hydroxide solution or an aqueous potassium carbonate solution, and oxidizing said allantoin with an alkali metal hypohalogenite in the presence of potass... | 07/18/2000 |
| 6057444 | Process for the preparation of phenyldichloro-1,3,5-triazine compounds A process is described for the preparation of an aryl-1,3-5-triazine compound of formula (1). This process comprises reacting an aldehyde compound of formula (2) with biuret, compound of formula (3), in hydrochloric medium or with methyl sulfate (1st... | 05/02/2000 |
| 5968482 | -hydroxyketoalkyl derivatives as light protection filters The invention relates to the use of -hydroxyketoalkyl derivatives as light protection filters for cosmetic or pharmaceutical products, the -hydroxyketoalkyl group being linked, if appropriate via a spacer, to a chromophoric group which has a... | 10/19/1999 |
| 5962683 | Oxazoline compounds as stabilizers A description is given of compounds of the formula I ##STR1## where r is 0 or 1 and y is a number from the range 1-3; X is a direct bond or --NR8 --, --CO--, --CONH-- or --COO-- or a divalent aliphatic or mixed aromatic-aliphatic C1 | 10/05/1999 |
| 5874382 | Cyclic sulfonamide herbicides Compounds of Formula I and II, and their agriculturally-suitable salts, are disclosed which are useful for controlling undesired vegetation ##STR1## wherein X is a direct bond; O; S; NH; N(C1 -C3 alkyl); N(C1 -C3... | 02/23/1999 |
| 5804583 | Pyrimidinone derivatives fused to nitrogen heterocycles having a II antagonistic activity Derivatives of bicyclic heterocycles comprising a pyrimidone ring fused to another 5, 6, or 7 membered nitrogen heterocycle which is C-substituted, through a methylene bridge, by a biphenyl group.... | 09/08/1998 |
| 5658933 | Substituted heterocyclic carboxamide esters, their preparation and their use as pharmaceuticals The invention relates to compounds of the formula I, ##STR1## to a process for their preparation and to their use as pharmaceuticals. The compounds are employed, in particular, as ester prodrugs of prolyl hydroxylase inhibitors for inhibiting collage... | 08/19/1997 |
| 5567670 | Herbicides for citrus oil palm rubber and other plantation crops This invention provides herbicides for use in plantation and specialty crops; and further provides novel substituted heterocyclic compounds, their agriculturally suitable compositions, and methods of using these compounds as preemergent or postemergent he... | 10/22/1996 |
| 5389599 | Substituted heterocyclyltriazinediones The invention relates to new substituted heterocyclyltriazinediones of the general formula (I) ##STR1## in which R1 represents hydrogen or an in each case optionally substituted radical from the series comprising alkyl, alkenyl, alkinyl or... | 02/14/1995 |
| 5232924 | Heterocyclic compound having serotonine 2-receptor antagonistic activity A heterocyclic compound represented by formula (I): ##STR1## wherein R1 represents a hydrogen atom, an alkyl group, an aryl group which may be substituted with one or more substituents selected from the group consisting of a halogen atom, ... | 08/03/1993 |
| 5084459 | Tetrahydropyrimidines, their production and use There is provided a pest control composition containing a compound represented by the formula, ##STR1## wherein R1, R2, R3 and R4 are the same or different and independently mean a hydrogen atom, a hydrocar... | 01/28/1992 |
| 5043443 | Aminomethyloxooxazolidinyl arylbenzene derivatives Novel aminomethyloxooxazolidinyl arylbenzene derivatives, wherein the aryl includes the phenyl, substituted phenyl, pyridyl, and substituted pyridyl groups, such as (l)-N-{3-[4- (4'-pyridyl)phenyl]-2-oxooxazolidin-5-ylmethyl}acetamide, possess useful ... | 08/27/1991 |
| 5034528 | Compositions for the control of hyperlipidemia The invention provides pharmaceutical compositions comprising hypolipidemically active derivatives of 1,2,4-triazolidine-3,5-diones, 1,3,5-triazabicyclo[3.1.0]hexane-2,4-diones, and 1,3,5-triazine-2,4(1H,3H)-diones in a pharmaceutically acceptable carrier... | 07/23/1991 |
| 4975434 | Antiviral and anticancer cyclopentenyl cytosine Cyclopentenyl pyrimidine compounds have potent anti-viral, anti-tumor and differentiating activity. Of these compounds, cyclopentenyl cytosine has proved to be particularly effective in a variety of tumors, as well as having good antiviral activity and po... | 12/04/1990 |
| 4968690 | 3-deazaneplanocin, intermediates for it, and antiviral composition and method of treatment using it The new compound 3-deazaneplanocin A has been discovered to have potent anti-viral, anti-tumor activity and differentiating activity. A simple method for preparing 3-deazaneplanocin A has been developed involving nucleophilic substitution, which method ca... | 11/06/1990 |
| 4935423 | Substituted 1,2,4-triazinediones, processes for their preparation and their use A substituted, 1,2,4-triazinedione of the formula ##STR1## in which R1 stands for an unsubstituted or substituted heteroaromatic radicals bonded via carbon, X stands for one or more, identical or different radicals selected from the group ... | 06/19/1990 |
| 4783531 | Production of S-substituted isothioureas In the production of an S-substituted isothiourea including the functional group ##STR1## in which R1 is an alkyl, alkenyl, aryl or aralkyl radical, wherein a thiourea including the functional group ##STR2## is reacted with an et... | 11/08/1988 |
| 4725684 | Synthesis of urea cyanurate A process for producing urea cyanurate which comprises reacting an aqueous solution of urea with cyanuric acid at a temperature below the melting point of urea provides reaction conditions which minimize urea decomposition and are energy efficient. The ur... | 02/16/1988 |
| 4684728 | Solubilizing biologically active compounds with reactive hydrogen atoms A biologically active compound can be solubilized by reaction in different sequences to form a derivative carrying the active moiety, a linking group such as an optionally substituted diisocyanate radical, a polyether moiety such as a polyoxyethylene radi... | 08/04/1987 |
| 4666902 | Tetrahydropyridazinone derivatives, processes for their preparation and their use Tetrahydropyridazinones of the formula I ##STR1## wherein R denotes an optionally substituted carbocyclic or heterocyclic radical, R1 denotes hydrogen; alkyl; aralkyl, which is optionally substituted in the aryl part; or acyl, and R2 | 05/19/1987 |
| 4659819 | Production of S-substituted isothioureas In the production of an S-substituted isothiourea including the function group ##STR1## in which R1 is an alkyl, alkenyl, aryl or aralkyl radical, wherein a thiourea including the functional group ##STR2## is reacted with an eth... | 04/21/1987 |
| 4524205 | Process for the preparation of 1-amino-1,3,5-triazine-2,4(1H,3H)-diones A process for the preparation of a herbicidally active 1-amino-1,3,5-triazone-2,4 (1H,3H)-dione of the formula ##STR1## comprising in a first stage at a temperature from about 0° to 100° C. reacting an isocyanate of the formula with an isothio semi... | 06/18/1985 |
| 4518761 | Process for the preparation of mixed trimers from organic isocyanates, the mixed trimers obtained according to the process and the use thereof for the production of polyurethanes The present invention is directed to a new process for the preparation of mixed trimers by at least partly trimerizing the isocyanate groups of at least two organic isocyanates of a reactivity which differs in the sense of the trimerization reaction, in t... | 05/21/1985 |
| 4500345 | Isoxazolotriazindiones and plant growth inhibiting use thereof Certain isoxazolotriazinediones, useful for controlling the growth of unwanted plants.... | 02/19/1985 |
| 4476303 | Thiazolino-[3,2-a]-1,3,5-triazine-2-one-4-(one or thione) derivatives Compounds having the formula ##STR1## wherein R1 denotes hydrogen atom, halogen group atom or methyl radical, R2 denotes cyclohexyl radical, phenyl radical or phenyl radical substituted with methyl radical or nitro radical, and ... | 10/09/1984 |
| 4447635 | N-Substituted imido-dicarboxylic acid diaryl ester compounds and herbicide intermediates Novel N-substituted imido-dicarboxylic acid diaryl ester compounds of the general formula ##STR1## in which R1 represents an optionally substituted aliphatic, cycloaliphatic, araliphatic, aromatic, heterocyclic radical and R2 an... | 05/08/1984 |
| 4426523 | Preparation of 1-amino-1,3,5-triazine-2,4(1H, 3H)-diones Herbicidal 1-amino-1,3,5-triazine-2,4(1H, 3H)-diones of the general formula ##STR1## are obtained in good yields if an N-substituted O-aryl N-chlorocarbonyl carbamate of the general formula ##STR2## is reacted with an isothiosemicarbazone of the... | 01/17/1984 |
| 4356024 | Process for the preparation of 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds A process for the preparation of a 1-amino-1,3,5-triazine-2,4(1H, 3H)-dione compounds comprising the steps of reacting an N-substituted imido-dicarboxylic acid diaryl ester with an isothiosemicarbazone at a temperature of between 50° and 150° C. to form... | 10/26/1982 |
