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| Number | Title | Issue Date |
| 7473779 | Derivatives of amidines, their preparation, their use as medicaments and the pharmaceutical compositions containing them Novel derivatives of amidines of formula wherein the substituents are defined as in the specification which are useful for inhibiting activity on NO-synthase enzymes producing nitrogen mono oxide and/or trapping the reactiv... | 01/06/2009 |
| 7250521 | Method for production of Δ-pyrrolines 2,5-Bisaryl-Δ1-pyrrolines of the formula (I) in which Ar1 and Ar2 are as defined in the description can be prepared by reacting aroylpyrrolidinones ... | 07/31/2007 |
| 7226917 | Derivatives of N-[phenyl(pyrrolidine-2-yl)methyl]benzamide and N-[(azepan-2-yl)phenylmethyl]benzamide, preparation, and use in treatment of schizophrenia Compounds of formula (I) as defined herein: are useful for treating behavioral disorders associated with dementia, psychoses, in particular schizophrenia (deficient form and productive form) and acute or chronic ... | 06/05/2007 |
| 7217707 | Amide of R-2-(aminoaryl)-propionic acid for use in the prevention of leucocyte activation N-(2-aminoaryl-propionyl)-amides of formula (1) are described. The process for their preparation and pharmaceutical preparations thereof are also described. The amides of the invention are useful in the prev... | 05/15/2007 |
| 7153958 | Farnesyl transferase inhibiting benzoheterocyclic derivatives This invention comprises the novel compounds of formula (I) wherein r, s, t, X, Z, R1, R2, R3, R4, R5, R6 and R7 have defined meanings,... | 12/26/2006 |
| 7148238 | Phenyl-piperazine derivatives as serotonin reuptake inhibitors The invention provides compounds represented by the general formula I wherein the substituents are defined in the application. The compounds are useful in the treatment of an affective disorder, including depress... | 12/12/2006 |
| 7138407 | Phenyl-piperazine derivatives as serotonin reuptake inhibitors The invention provides compounds represented by the general formula I wherein the substituents are defined in the application. The compounds are useful in the treatment of an affective disorder, including depress... | 11/21/2006 |
| 6849203 | Photoisomerizable compounds The invention relates to photoisomerizable compounds of formula I wherein A, Z, L, R, R1, k, m and r are defined herein. ... | 02/01/2005 |
| 6680314 | Azacyclooctane and heptane derivatives, their preparation and use in therapy Compounds of formula (1) or (2), enantiomers thereof, mixtures thereof, and pharmaceutically acceptable salts thereof: ##STR1## wherein: n is 0, or 1; R is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, aryl or aralkyl; and R1 ... | 01/20/2004 |
| 6451789 | 1-aza-2-alky-6-aryl-cycloalkanes Compound of formula (I): ##STR1## wherein: n represents 0 or 1, R1 represents hydrogen, arylalkyl, alkyl, acyl, alkoxycarbonyl, arylalkoxycarbonyl or trifluoroacetyl, R2 represents alkyl, X represents oxygen, chlorine, OR3, SR | 09/17/2002 |
| 6436925 | Substituted benzamides, their production and their use as cysteine protease inhibitors Benzamides of the formula I ##STR1## and its tautomeric forms, possible enantiomeric and diastereomeric forms, E and Z forms, and possible physiologically tolerated salts, in which the variables have the following meanings: R1 --C1 -... | 08/20/2002 |
| 6420395 | Azacyclooctane and heptane derivatives, their preparation and use in therapy The present invention discloses compounds of formula (1) or (2), any of its enantiomers or any mixture thereof, or a pharmaceutically acceptable salt thereof; wherein n is 0, or 1; R is hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, cycloalky-alkyl, aryl ... | 07/16/2002 |
| 6399771 | Cyclic imines as pesticides The invention relates to novel cyclic imines of the formula (I) ##STR1## in which Ar1 and Ar2 each represent substituted phenyl and n represents 1, 2 and 3, to a plurality of processes for their preparation and to their use as pestic... | 06/04/2002 |
| 6352981 | Substituted AZA- and diazacycloheptane and -cyclooctane Aza- and diazacyclohexane and -cyclooctane compounds of the following formula: Ar1 --A--B--Ar2 (I) where Ar1, A, B and Ar2 have the meanings stated in the description have a high affinity for the dopamine D3 | 03/05/2002 |
| 6165230 | 1,4-diazacycloheptane derivatives and their use in hair oxidation dyes A 1,4-diazacycloheptane derivative and an oxidative hair colorant containing the derivative as a primary intermediate is presented. The 1,4-diazacycloheptane derivative is of the formula: ##STR1## where R1, R2, R3 and... | 12/26/2000 |
| 6140321 | Polymorphs of donepezil hydrochloride and process for production Donepezil hydrochloride, 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl]methylpiperidine hydrochloride, is provided here in the form of four polymorphs which are stable against heat and humidity in the pharmaceutical use. They can be industrially produce... | 10/31/2000 |
| 5985864 | Polymorphs of donepezil hydrochloride and process for production Donepezil hydrochloride, 1-benzyl-4-[(5,6-dimethoxy-1-indanon)-2-yl]methylpiperidine hydrochloride, is provided here in the form of four polymorphs which are stable against heat and humidity in the pharmaceutical use. They can be industrially produce... | 11/16/1999 |
| 5977357 | Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof A novel process for the preparation of compounds of formula I ##STR1## by aminolysis of a p-halophenyl alkyl ketone of formula II ##STR2## with a cyclic amine of formula III ##STR3## in water at a temperature of at least 130° C., in which ... | 11/02/1999 |
| 5912343 | Tertiary amines containing side-chain organolithium structures and method for the preparation thereof A compound comprising at least one cyclic amine, having an organolithium side-chain, defined according to formula (I) ##STR1## wherein Z is a lithium atom (Li); R1 is selected from the group consisting of organic groups containing from 1 t... | 06/15/1999 |
| 5795890 | Sulfonamide derivatives A sulfonamide derivatives of formula (I) ##STR1## a non-toxic salts, an acid addition salts or a solvates thereof which has an inhibitory effect on elastase.... | 08/18/1998 |
| 5276053 | Polycyclic amines useful as cerebrovascular agents A novel series of polycyclic amines, derivatives, methods of making the compounds, novel intermediates, compositions containing them, and methods for using them in the treatment and prevention of cerebrovascular disorders are disclosed.... | 01/04/1994 |
| 5223498 | Phenylamidine and phenylguanidine derivatives and their use as antidiabetic agents Compounds of formula I ##STR1## and their salts in which n=0 or 1, R1 and R2 are each aliphatic or cycloalkyl or NR1 R2 is an optionally substituted heterocyclic ring, R3 is alkyl, cycloalkyl or ... | 06/29/1993 |
| 5153228 | 9-amino-2-phenylbicyclo[3.3.1]nonanes and 9-amino-2-phenylbicyclo[3.3.1]non-2-enes and drugs containing them 9-Amino-2-phenylbicyclo-[3.3.1]nonanes and 9-amino-2-phenylbicyclo[3.3.1]non-2-enes of the formula I ##STR1## where R1 and R2 are identical or different and each is hydrogen, halogen, alkyl, alkoxy, dialkylamino, trifluoromethyl... | 10/06/1992 |
| 5071853 | Polycyclic amines useful as cerebrovascular agents A novel series of polycyclic amines, derivatives, methods of making the compounds, novel intermediates, compositions containing them, and methods for using them in the treatment and prevention of cerebrovascular disorders are disclosed.... | 12/10/1991 |
| 5041545 | 2-hydroxybenzophenone hydrazides and derivatives thereof Hydrazide functionalized 2-hydroxybenzophenone ultraviolet light and heat stabilizers and derivatives are disclosed having the general formula: ##STR1## wherein R1, R2, R3, R4, R5, R6, X, Y... | 08/20/1991 |
| 4910304 | Preparation of N-substituted cyclic amines N-substituted cyclic amines of the general formula I ##STR1## where A is an alkylene group or a --(CH2)n --[--O--(CH2)m ]r group which may be monosubstituted or polysubstituted by radicals R with... | 03/20/1990 |
| 4895841 | Cyclic amine compounds with activity against acetylcholinesterase A cyclic amine compound is defined by the formula: ##STR1## in which J is indanyl, indanonyl, indenyl, indenonyl, indanedionyl, tetralonyl, benzosuberonyl, indanolyl or a divalent group thereof, K is phenyl, an arylalkyl or cynnamyl, B is --(CHR22)r-... | 01/23/1990 |
| 4686220 | Substituted 2-[b-substituted-amino)-ethylamino]-1,4-naphthalenediones for treating asthma, allergic diseases and inflammation in warm-blooded animals This disclosure describes certain substituted piperazine-1,4-naphthalenediones useful as anti-asthmatic agents.... | 08/11/1987 |
| 4394156 | Novel N-phenyl-substituted N-heterocyclic compounds, their preparation and use in agents for regulating plant growth The present invention relates to novel active compounds having a plant growth-inhibiting and herbicidal action and their preparation and to agents containing these active ingredients, and their use. The novel active compounds are saturated and unsaturated 4-me... | 07/19/1983 |
| 4374991 | 2,6-Dimethylpiperidinyl-N-carbobutoxymethyl urea This invention relates to a method of using compounds of the formula: ##STR1## wherein R1 is hydrogen, alkyl or alkenyl; R2 is hydrogen, alkyl, cycloalkyl or mononuclear aryl or R1 and R2, taken together with ... | 02/22/1983 |
| 4357471 | Azaspiro compounds This invention relates to a method of using compounds of the formula: ##STR1## wherein R1 is hydrogen, alkyl or alkenyl; R2 is hydrogen, alkyl, cycloalkyl or mononuclear aryl or R1 and R2, taken together with ... | 11/02/1982 |
| 4051067 | Stabilization of unsaturated carboxylic acid esters with mixtures of polyalkyleneamines and arylenediamines A method of inhibiting polymerization of unsaturated carboxylic acid esters and improved unsaturated carboxylic acid ester compositions are described. The method comprises, and the compositions are prepared by, incorporating into the ester composition a c... | 09/27/1977 |
| 4046758 | 3-Halo-2,6-dinitro-4-trifluoromethylanilines 3-Halo-2,6-dinitro-4-trifluoromethylanilines having hydrocarbon substituents on the nitrogen atom. The hydrocarbon substituents can be alkyl, alkenyl, alkynyl or a portion of a heterocyclic group. The compounds are especially useful as intermediates for p... | 09/06/1977 |
| 4036977 | Polycyclophenylpyrrolidines, their compositions and use Compounds of the formula ##STR1## where R4 X is a polycyclocoupled group and R1 and R2 are H or simple hydrocarbon and R3 has the same value and additionally simple acyl, can be made by a variety of synthes... | 07/19/1977 |
| 4028415 | Diphenylpropylamines 1,1-DIPHENYL-2-HYDROXY-3-AMINOPROPANE DERIVATIVES ARE USEFUL FOR THEIR PSYCHOTROPIC ACTIVITY AND, IN PARTICULAR ARE USEFUL AS ANTIDEPRESSANTS.... | 06/07/1977 |
| 4022764 | 3-(Meta-oxyphenyl) hexahydroazepines The invention concerns novel hexahydroazepines of the formula ##STR1## and their pharmaceutically acceptable acid addition salts, wherein R is hydrogen, lower alkyl, benzyl or lower alkanoyl, R1 is hydrogen, lower alkyl, lower alkenyl, low... | 05/10/1977 |
| 4021550 | Hexahydroazepines as antiinflammatory agents The invention concerns hexahydroazepines of the formula ##STR1## and the pharmaceutically acceptable acid addition and quaternary ammonium salts thereof, wherein R4 is lower alkyl, R5 is lower alkyl, lower alkenyl, lower alkynyl... | 05/03/1977 |
| 3993763 | Tertiary aminoacids as anti-inflammatory agents New -(cyclic tert. aminophenyl)-aliphatic acids, e.g. those of the formula ##SPC1## R1 = h or alkyl R2 = h, alk(en)yl, cycloalk(en)yl or cycloalk(en)yl-alkyl A = hydroxylated lower alkylene And functional derivatives thereof, are a... | 11/23/1976 |
| 3989701 | Diamine-benzophenones and a process for the preparation thereof New compounds of the general formula (I) ##SPC1## wherein R1 and R2 each is a saturated or unsaturated, straight-chained or branched alkyl group, an aralkyl group, a saturated or unsaturated cycloalkyl group or an aryl group, or R | 11/02/1976 |
| 3989834 | Alkoxy anilides and pharmaceutical compositions This invention relates to ortho-alkoxy anilines having the amino group substituted with an amino lower alkyl carboxylic residue, as well as their physiologically-compatible acid-addition salts and their optically-active isomers.... | 11/02/1976 |
