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Class 514/490 - Ring attached directly to oxygen of N-C(=0)-0


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the ring is directly attached to
No. of patents: 120
Last issue date: 11/06/2007


1      
NumberTitleIssue Date
7291645Phenylalanine derivatives as alpha 4 integrin inhibitors
Disclosed are a series of phenylalanine derivatives, to compositions containing them, to processes for their preparation, and to their use in medicine. ...
11/06/2007
7276534Carbon-substituted diketopiperazine delivery systems
Compositions useful in the delivery of active agents are provided. These delivery compositions include (a) an active agent; and (b) a carrier of at least one mono-C-substituted or di-C-substituted diketopiperazine. Methods for preparing these compositions and admini...
10/02/2007
7252842Induced phase transition method for the production of microparticles containing hydrophilic active agents
Microparticles and a method for their production is described. The process of the present invention provides a simple, quick, and efficient one-pot process for the production of microparticles containing a hydrophilic active agent of various and uniform morphologies...
08/07/2007
7176201Modulation of anxiety through blockade of anandamide hydrolysis
Fatty acid amide hydrolase inhibitors of the Formula: are provided wherein X is NH, CH2, O, or S; Q is O or S; Z is O or N; R is an aromatic moiety selected from the group consisting of substituted or ...
02/13/2007
7166744Retinoid derivatives and methods for producing said compounds and anti-cancer pharmaceutical composition comprising said compounds
The present invention relates to a novel retinoid derivative compound represented by the formula I: wherein X, R1, R2 and R3 are as defined herein or pharmaceutically acceptalbe s...
01/23/2007
7025978Use of polysiloxanes containing quarternary amino groups as formulation auxiliary agents, and agents containing the same
The present invention relates to the use of polysiloxanes containing at least one quaternary ammonium group as formulation auxiliaries in formulations of pharmaceutically and veterinary active compounds, and to compositions comprising a) pharmaceuticall...
04/11/2006
6835748Treatment of ocular disorders
The present invention is in particular related to the use of rivastigmine in the manufacture of a medicament for the treatment of ocular disorders. ...
12/28/2004
6573297(2-substituted oxyphenyl)alkanamide derivative, hair growth promoter and external composition for skin using the same
A (2-substituted oxyphenyl)alkanamide derivative or a salt thereof expressed by the following Formula (I): ##STR1## wherein one of A and B is a hydrocarbon group of C3-30 expressed by R1 and the other is --(CH2)n-NR2
06/03/2003
6534541Treatment of ocular disorders
The present invention is in particular related to the use of rivastigmine in the manufacture of a medicament for the treatment of ocular disorders....
03/18/2003
6476067N-formyl hydroxylamine derivatives as antibacterial agents
Compounds of formula (I) are in the preparation of antibacterial agents, wherein: R1 represents hydrogen, C1 -C6 alkyl or C1 -C6 alkyl substituted by one or more halogen atoms; R2 represent...
11/05/2002
6461591Medical aerosol formulations
A pressure-liquefied propellant mixture for aerosols, comprising a fluorinated alkane, in particular 1,1,1,2-tetrafluoroethane and/or 1,1,1,2,3,3,3-heptafluoropropane, and carbon dioxide, makes possible an improvement of the wetting properties of pharmace...
10/08/2002
6395774Carbon-substituted diketopiperazine delivery systems
Compositions useful in the delivery of active agents are provided. These delivery compositions include (a) an active agent; and (b) a carrier of at least one mono-C-substituted or di-C-substituted diketopiperazine. Methods for preparing these compositions...
05/28/2002
6303569Trialkyl-lock-facilitated polymeric prodrugs of amino-containing bioactive agents
The present invention is directed to double prodrugs containing polymeric-based transport forms. These polymeric compounds comprise the formula: ##STR1## wherein: B is H, OH, OSiR13, a residue of an amine-containing target moiety or a resi...
10/16/2001
6277880Chemical compounds
Prodrugs, of generic formula I, are disclosed for use in antibody directed enzyme prodrug therapy (ADEPT). The prodrugs are substrates for carboxypeptidase G2 (CPG2) and yield more active cytotoxic drugs than known products of CPG2 catalysed reactions....
08/21/2001
6251938Phenylethylamine derivatives
This invention is directed to compounds of the following formula: ##STR1## wherein m is from 0-4; X is O or S; Y is halogeno; R1 is hydrogen or C1-4 alkyl; R2 is hydrogen, C1-4 alkyl or optionally substituted pr...
06/26/2001
6080784Protein kinase C modulators N
Compositions with protein kinase C-modulatory, anti-inflammatory and other activities are disclosed....
06/27/2000
6075048Pediatric method of use of bambuterol
New aqueous formulations of, and the paediatric use of, bambuterol, and of its pharmaceutically acceptable salts, are described....
06/13/2000
6034117Methods of treating and diagnosing sleep disordered breathing and means for carrying out the method
This invention relates to a method for treating snoring, sleep apnea and other form of sleep-disordered breathing, which comprises administration of a therapeutically effective dose of an acetyl choline esterase inhibitor (CEI) such as pyridostigmine or a...
03/07/2000
6005002Nitrogen mustard prodrugs with novel lipophilic protecting groups, and processes for their production
The invention provides compounds of formula (I) and (II) wherein X and Y are independently chlorine, bromine, iodine, a mesyl group CH3 SO3 or a tosyl group OSO2 phenyl (wherein phenyl is optionally substituted by 1, 2, 3,...
12/21/1999
5925674Cycloalkylcarboxanilides
This invention relates to cycloalkylcarboxanilides of the formula ##STR1## which are used to combat pests....
07/20/1999
5846997Liquid formulations
The present invention relates to water-emulsifiable liquid formulations of insecticidal active compounds, characterized in that they contain a) 2.5 to 30% of active compound, b) 5 to 77.5% of a mixture of benzyl acetate and an alcohol in the ratio 25-95% to 5-...
12/08/1998
5733935Hydroxylamine derivatives and fungicides containing the same
A hydroxylamine derivatives of formula (I): ##STR1## wherein R represents ##STR2## in which R1 and R2 represents alkyl group, alkenyl group, alkynyl group, cycloalkyl group, haloalkyl group, haloalkynyl group, alkoxy -...
03/31/1998
57287293-methoxy-2-phenylacrylic acid esters used as pest-control agents, especially as fungicides
3-Methoxy-2-phenyl-acrylic esters of the formula ##STR1## in which R represents optionally substituted alkyl, cycloalkyl or aryl and n represents a number 0 or 1, a process for their preparation and their use as pesticides....
03/17/1998
5709890Polyaspartic acid and its analogues in combination with insecticides
An insecticide composition is enhanced from the standpoint of its ability to be absorbed by insects, such as red fire ants, particularly dithiophosphate ester pesticides by the addition of a small amount of a water soluble non-aromatic polyorganic acid or...
01/20/1998
5700831Pesticidal hydrazide derivatives
A compound of the formula ##STR1## wherein R is a) phenyl; phenyl(C1 -C4 alkoxy); phenoxy; or benzyl; the phenyl ring of each substituent being optionally substituted with one or more of halogen, nitro, C1 -C8
12/23/1997
5646133Polyaspartic acid and its analogues in combination with insecticides
An insecticide composition is enhanced from the standpoint of its ability to be absorbed by insects, such as red fire ants, particularly dithiophosphate ester pesticides by the addition of a small amount of a water soluble non-aromatic polyorganic acid or...
07/08/1997
5602176Phenyl carbamate
The (S)-N-ethyl-3-[(1-dimethylamino)ethyl]-N-methyl-phenylncarbamate in free base or acid addition salt form is useful as pharmaceutical, particularly for systemic transdermal administration....
02/11/1997
5574029Method for treating anxiety
The present invention provides a method for treating anxiety in a human in need thereof, comprising administering an antianxiety amount of a muscarinic agonist compound of the general formula ##STR1## wherein X R43, R44, R4...
11/12/1996
5565490P-hydroxyaniline derivatives, their preparation and their use
p-Hydroxyaniline derivatives of the formula I ##STR1## where the substituents have the following meanings: R1 is hydrogen, or unsubstituted or substituted alkyl; R2 and R3 independently of one another are halogen, alkyl, ...
10/15/1996
5512565Cholesterol ester hydrolase inhibitors
The compounds of the formula: ##STR1## in which ##STR2## where R7 is hydrogen, alkyl, hydroxy, alkanoyloxy, hydroxyalkyl, hydroxycarbonyl, alkoxycarbonyl, phenyl or substituted phenyl, in which the substituent is alkyl, alkoxy, h...
04/30/1996
5391571Cholesterol ester hydrolase inhibitors
The compounds of the formula: ##STR1## in which R1 is alkyl of 4 or more carbon atoms, cycloalkyl, 1-adamantyl, 2-adamantyl, 3-noradamantyl, 3-methyl-1-adamantyl, 1-fluorenyl, 9-fluorenyl, cycloalkylalkyl, phenyl, substituted phenyl, ...
02/21/1995
5384328Oxysulfonyl carbamates
The present invention is directed to compounds of the following general Formula I, methods for using the compounds of Formula I, pharmaceutical compositions thereof, and processes for preparing the compounds. ##STR1## wherein X is oxygen or sulfur; w...
01/24/1995
5360783Water-based pesticidal composition
A water-based pesticidal composition contains 100 weight parts of substantially water-insoluble pesticide and 1.7-200 weight parts of a surface active agent. The surface active agent contains Component A and Component B at weight ratio of A/B=80/20-20/80....
11/01/1994
5290546Method for thermal vaporization of chemical
The present invention provides a cordless thermal vaporizer of the liquid type wherein the body of the vaporizer has a heater for heating a wick for drawing up a chemical solution from a bottle, and a socket disposed under the heater and removably fittabl...
03/01/1994
5214061Method of using p-acylaminophenoxycarbamates and derivatives as analgesics
This invention relates to p-acylaminophenoxycarbamates having the formula ##STR1## where R1 and R2 are each independently hydrogen, loweralkyl, aryl and arylloweralkyl; R3 is hydrogen, loweralkyl, arylloweralkyl; R
05/25/1993
5198012Phosphate activators for cyclohexenone herbicides
A biocide composition comprises an effective amount of a biocide and an effective amount of a biocide activator selected from the group consisting of an alkyl phosphate, an alkenyl phosphate, a hydroxyalkyl phosphate, a polyoxyalkylene alkyl ether phospha...
03/30/1993
5180420Water dispersible granules
The water dispersible granule of the present invention contains (a) a pesticidal active ingredient which is solid at room temperature, (b) an anionic surface active agent, and (c) a kaolin series clay having a volume median diameter of 2 μm or more, and ...
01/19/1993
5176914Fungicidal carbocyclic anilide carbamates
Fungicidal carbocyclic anilide carbamates of the formula ##STR1## in which X represents optionally alkyl-substituted cycloalkyl or optionally alkyl-substituted cycloalkenyl, Hal represents halogen, and Y1, Y2 and Y3 indepe...
01/05/1993
5122539Allosteric hemoglobin modifiers useful for decreasing oxygen affinity and preserving oxygen carrying capability of stored blood
Compounds of the general structural formula: ##STR1## wherein X, Y and Z may each be CH2, NH, or O, R2-6 are either hydrogen, halogen, or a substituted or unsubstituted C1, C2, or C3 alkyl group ...
06/16/1992
5114965Flubenzimine containing agents for combating pests
The foregoing invention relates to new soil pest combating agents which contain at least one conventional active agent, especially a carbamate, P-esters (phosphoric and phosphonic acid esters, including esteramides, as well as corresponding thiono-, thiol...
05/19/1992
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