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Patent No. 6637447

Beerbrella

A small umbrella which may be removably attached to a beverage container in order to shade the beverage container from the direct rays of the sun.

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Class 514/483 - Plural N-C(=X)-X groups


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the organic ingredient contains plural
No. of patents: 132
Last issue date: 12/28/2010


1        
NumberTitleIssue Date
7858659Redox therapy for tumors
The invention provides methods and compositions for treatment of tumors comprising administering to subject bearing a tumor an effective amount of at least one agent that decreases the [GSH]2/[GSSG] ratio in the malignant cells of said tumor, wherein said...
12/28/2010
7816403Method of inhibiting ATF/CREB and cancer cell growth and pharmaceutical compositions for same
There is provided a method for inhibiting ATF/CREB and cancer cell growth using disulfiram, administered in combination with heavy metals. It was found that disulfiram disrupts transcription factor DNA binding by forming mixed disulfides with thiols within the DNA-b...
10/19/2010
7705045Prodrugs built as multiple self-elimination-release spacers
This invention concerns multiple release spacers and spacer systems, which release multiple leaving groups following a single activation. It concerns compounds comprising a specifier linked to two or more of the same or different leaving groups (L in the figure) via...
04/27/2010
7495028R-bambuterol, its preparation and therapeutic uses
R-enantiomer of Bambuterol, its preparation and therapeutic uses are disclosed. A composition includes R-Bambuterol or its therapeutically acceptable salt. A composition of R-Bambuterol includes at least 80% by weight of the R-enantiomer and not more than 20% by wei...
02/24/2009
7368478Methods for inhibiting angiogenesis and tumor growth
Angiogenesis, tumor growth, and metalloproteinase 2 (MMP2) interaction with integrin-αvβ3 are inhibited by an inhibitor compound of formula: wherein G1 and G2 are each independe...
05/06/2008
7358397Preparation of halogenated 4-aminophenols
The present invention relates to halogenated 4-aminophenols and to halogenated 4-(phenyidiazenyl)phenols, to a process for their preparation and to the use of the halogenated 4-hydroxyphenols for preparing active ingredients, especially in pharmaceuticals and agroch...
04/15/2008
7279470Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
Use of compounds to inhibit hormone-sensitive lipase, pharmaceutical compositions comprising the compounds, methods of treatment employing these compounds and compositions, and novel compounds. The present compounds are inhibitors of hormone-sensitive lipase and may...
10/09/2007
7235585Enzyme activated self-immolative n-substituted nitrogen mustard prodrugs
This invention pertains to certain enzyme (CPG2) activated self-immolative nitrogen mustard prodrugs, which are useful in enzyme prodrug therapy (EPT), such as ADEPT and GDEPT, for the treatment of proliferative conditions, such as cancer, and which have the followi...
06/26/2007
7122576Carbamate compounds for use in preventing or treating bipolar disorder
This invention is directed to a method for preventing or treating bipolar disorder comprising administering to a subject in need thereof a therapeutically effective amount of an enantiomer of Formula (I) or enantiomeric mixture wherein one enantiomer of Formula (I) ...
10/17/2006
7115660Methods for inhibiting angiogenesis and tumor growth
Angiogenesis, tumor growth, and metalloproteinase 2 (MMP2) interaction with integrin-αvβ3 are inhibited by an inhibitor compound of formula (I): wherein G1 and G2 are each independently NH—C(O)—O—R1, —...
10/03/2006
7087643Carbamate compounds for use in preventing or treating neuropathic pain and cluster and migraine headache-associated pain
This invention is directed to a method for preventing or treating neuropathic pain and cluster and migraine headache-associated pain comprising administering to a subject in need thereof a therapeutically effective amount of a compound of Formula (I):
08/08/2006
7078460Room temperature curable organopolysiloxane composition for molding
A room temperature curable organopolysiloxane composition is provided which includes an organopolysiloxane, a curing agent, and a specific organic compound incorporating at least one sulfur atom within each molecule. By producing a molding matrix with this type of c...
07/18/2006
7078436Carbamate compounds for use in preventing or treating anxiety disorders
This invention is directed to a method for preventing or treating anxiety disorders comprising administering to a subject in need thereof a therapeutically effective amount of a compound selected from the group consisting of Formula (I) and Formula (II):
07/18/2006
7067517Use of compounds for decreasing activity of hormone-sensitive lipase
Use of compounds to inhibit hormone-sensitive lipase, pharmaceutical compositions comprising the compounds, methods of treatment employing these compounds and compositions, and novel compounds. The present compounds are inhibitors of hormone-sensitive lipase and may...
06/27/2006
7056919Synergistic combination of fungicides to protect wood and wood-based products and wood treated by such combination as well as methods of making the same
A wood treatment composition having a synergistic combination of fungicides which may include two or more compounds. These combinations are shown to be especially effective in providing resistance to decay, mold and mildew when wood is treated with these combination...
06/06/2006
7056947Aza-peptide epoxides
The present invention provides compositions for inhibiting proteases, methods for synthesizing the compositions, and methods of using the disclosed protease inhibitors. Aspects of the invention include aza-peptide epoxide compositions that inhibit proteases, for exa...
06/06/2006
7049285Biocompatible polymers including peptide spacer
The present invention relates to new biocompatible polymer derivatives including peptide spacers of formula (I) and their methods of preparation. The present invention also relates to the conjugates formed by covalent or non-covalent bonding and their methods of pre...
05/23/2006
7045531Composition comprising a metal chelator and a method of treating amyloidosis by administering the metal chelator
The invention relates to the identification of pharmacological agents to be used in the treatment of Alzheimer's disease and related pathological conditions. Methods and compositions for treatment of conditions caused by amyloidosis, Aβ-mediated ROS formation, or b...
05/16/2006
7019046Aqueous suspension agent for water insoluble compounds
This invention relates to an improved aqueous suspension concentrate for water insoluble chemicals comprising a mixture of an anionic suspension agent and a homo- and/or a co-polymer of a heterocyclic vinyl lactam combined in a mole ratio of between about 0.1:1 and ...
03/28/2006
6995283Benzophenones as inhibitors of reverse transcriptase
The present invention is directed to beazophenone compounds useful in the inhibition of HIV reverse transcriptase, particularly its resistant varieties. ...
02/07/2006
RE38915Nonpeptide insulin receptor agonists
Modulation of the activity of the insulin receptor, enhancement of glucose uptake by cells, and other effects significant in the control and management of diabetes are accomplished using compounds of the formula wherein ...
12/06/2005
6960571Methods and compositions for administration of iron for the treatment of restless leg syndrome
A method of treating Restless Leg Syndrome, includes administering to a subject an iron complex having an iron release rate greater than IDI. The iron release rate is determined at a concentration of at least 2,000 μg/dl. ...
11/01/2005
6838482Fungicidal composition
The present invention provides a fungicidal composition characterized by containing as active ingredients (a) a compound represented by the formula I: (wherein Ar is a substituted or unsubstituted phenyl group, ...
01/04/2005
6815557Tryptase inhibitors
Compounds of formula (I), in which M, A1, A2, K1 and K2 have the meanings as indicated in the description are novel active tryptase inhibitors. ...
11/09/2004
6815464Carbamate compounds for use in the treatment of pain
This invention is directed to a method for the treatment of pain comprising administering to a subject in need thereof a therapeutically effective amount of a compound selected from the group consisting of Formula (I) and Formula (II):
11/09/2004
6790853Contraception method using competitive progesterone antagonists and novel compounds useful therein
Competitive progesterone antagonists, including two novel steroids, viz., 11β,19-[4-(cyanophenyl)-o-phenylene]-17β-hydroxy-17α-(3-hydroxyprop-1(Z)-enyl)-4-androsten-3-one and 11β,19-[4-(3-pyridinyl)-o-phenylene]-17β-hydroxy-17α-(3-hydroxyprop-1(Z)-enyl)-4-andr...
09/14/2004
6649591Polydithicarbamate-containing non-targeting marcomolecules and the use thereof for therapeutic and diagnostic applications
In accordance with the present invention, there is provided a new class of drugs for therapeutic treatment of such indications as cerebral stroke and other ischemia/reperfusion injury. Thus, in accordance with the present invention, dithiocarbamates are l...
11/18/2003
6608074Contraception method using competitive progesterone antagonists and novel compounds useful therein
Competitive progesterone antagonists, including two novel steroids, viz., 11ଲ,19-[4-(cyanophenyl)-o-phenylene]-17ଲ-hydroxy-17଱-(3-hy droxyprop-1(Z)-enyl)-4-androsten-3-one and 11ଲ,19-[4-(3-pyridinyl)-o-phenylene]-17ଲ-hydroxy-1...
08/19/2003
6599935Felbamate derived compounds
The present invention relates to novel felbamate derivatives and their use to treat neurological diseases such as epilepsy and to treat tissue damage resulting form ischemic events. The felbamate derivatives are modified to prevent the formation of metabo...
07/29/2003
6589985Carbamate compounds for use in preventing or treating movement disorders
This invention is directed to a method for preventing or treating movement disorders comprising administering to a subject in need thereof a therapeutically effective amount of a compound selected from the group consisting of Formula (I) and Formula (II):...
07/08/2003
6586466Carbohydrazide-protease inhibitors
The present invention provides compounds which inhibit proteases, including cathepsin K, pharmaceutical compositions of such compounds, and methods for treating diseases of excessive bone loss or cartilage or matrix degradation, including osteoporosis; gi...
07/01/2003
6548540Method of treating cancer using dithiocarbamate derivatives
Dithiocarbamate, particularly tetraethylthiuram disulfide, and thiocarbamate anions strongly inhibit the growth of cancer cells of a variety of cell types. Such inhibitory effect is enhanced by heavy metal ions such as copper ions, cytokines and cerulopla...
04/15/2003
6545027Methods of modulating NF-kB transcription factor
A method of modulating NF-kB transcription factor comprising administering to a human in need thereof an effective amount of a compound having the formula ##STR1## wherein R1 and R3 are independently hydrogen, ##STR2## wherein ...
04/08/2003
6541513Carbamate compounds for use in preventing or treating psychotic disorders
This invention is directed to a method for preventing or treating psychotic disorders comprising administering to a subject in need thereof a therapeutically effective amount of a compound selected from the group consisting of Formula (I) and Formula (II)...
04/01/2003
6538024Felbamate derived compounds
The present invention relates to novel felbamate derivatives and their use to treat neurological diseases such as epilepsy and to treat tissue damage resulting form ischemic events. The felbamate derivatives are modified to prevent the formation of metabo...
03/25/2003
6515019Methods of providing symptomatic and prophylactic treatment for medical and neurological conditions
Methods are disclosed for prophylactically and chronically preventing symptomatic depression, neuronal cell injury and cell death in systemic and neurological conditions, populations with cerebrovascular risk factors, and invasive vascular procedures, emp...
02/04/2003
6436421Pesticide compositions
The present invention relates to pesticide compositions. In particular, the present invention relates to pesticide compositions comprising a pesticide and a redispersible polymer and to a method for controlling agricultural pests by applying to the pest o...
08/20/2002
6416789Synergistic combination of fungicides to protect wood and wood-based products from fungal decay, mold and mildew damage
A wood treatment material having a synergistic combination of fungicides including boron-containing compounds, organo-iodine compounds and amine-oxides is provided. This combination is shown to be especially effective in providing resistance to decay, mol...
07/09/2002
6331542Protease inhibitors
The present invention provides compounds which inhibit proteases, including cathepsin K, pharmaceutical compositions of such compounds, and methods for treating diseases of excessive bone loss or cartilage or matrix degradation, including osteoporosis; gi...
12/18/2001
6319949Pesticidal sprays
A method for preventing fungal diseases in crops which comprises the steps of: (a) applying to a crop an aqueous or a non-aqueous spray composition which includes a pesticide and a spray adjuvant including a solvent and an emulsifier, wherein the solvent ...
11/20/2001
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