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Patent No. 6681419

Forehead support apparatus 

A forehead support apparatus for resting a standing users forehead against a wall above a bathroom commode or urinal or beneath a showerhead.

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Class 514/443 - Polycyclo ring system having the hetero ring as one of the cyclos


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the five-membered sulfur containing
No. of patents: 915
Last issue date: 05/08/2012


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NumberTitleIssue Date
RE43372C16 unsaturated FP-selective prostaglandins analogs
Compounds having the general structure: which are useful for the treatment of a variety of diseases and conditions, such as bone disorders. ...
05/08/2012
8153683Methods of treatment using a prodrug of an excitatory amino acid
This invention relates to synthetic excitatory amino acid prodrugs and processes for their preparation. The invention further relates to methods of using, and pharmaceutical compositions comprising, the compounds for the treatment of neurological disorders and psych...
04/10/2012
8153682Sulfonamides as TRPM8 modulators
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula I as follows: wherein A, B, G, Y, R1...
04/10/2012
8148422Sulfonamides as TRPM8 modulators
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula (I) and Formula (II) as follows: wherein Y, R
04/03/2012
8143307Benzothiophen-2-carbonylguanidine derivatives, preparation thereof, and pharmaceutical composition containing the same
The present invention is related to benzothiophen-2-carbonylguanidine derivatives, a preparation method thereof, and pharmaceutical compositions containing the same. The derivatives have potent inhibitory effect on the sodium/hydrogen exchanger NHE-I, improve the fu...
03/27/2012
8129425Small organic molecule regulators of cell proliferation
The present invention makes available methods and reagents for modulating proliferation or differentiation in a cell or tissue comprising contacting the cell with a hedgehog agonist, such as the compounds depicted in FIGS. 32 and 33. In certain embodim...
03/06/2012
8101651Compounds with activity at estrogen receptors
Disclosed herein are compounds of Formula I as disclosed herein, methods of modulating the activity of an estrogen receptor and methods of treating a disorder associated with estrogen receptors. ...
01/24/2012
8063099Trans-3-aza-bicyclo[3.1.0]hexane derivatives
The invention relates to novel trans-3-aza-bicyclo[3.1.0]hexane derivatives of formula (I), wherein A, B, n and R1 are as described in the description, and to the use of such compounds, or of pharmaceutically acceptable salts of such compounds, as medicam...
11/22/2011
8003684Crystal form and pharmaceutical compositions of (+)-R-zileuton
Crystalline forms of (+)-R-zileuton, which may be used in pharmaceutical applications, are disclosed. Particular single crystalline forms of (+)-R-zileuton are characterized by a variety of properties and physical measurements. As well, methods of producing crystall...
08/23/2011
7999001Antiviral compounds and methods of using thereof
Disclosed herein are compounds which exhibit antiviral activity against a plurality of viruses belonging to different families such as Bornaviridae, Filoviridae, Paramyxoviridae, Rhabdoviridae, Arenaviridae, Bunyaviridae, Orthomyxoviridae, and Poxviridae. Thus, meth...
08/16/2011
7985768Compounds as cannabinoid receptor ligands
The present invention relates to thiophene containing compounds of formula (I) wherein R1, R2, R3, and n are as defined in the specification, pharmaceutical compositions comprising such comp...
07/26/2011
7981924Thiophene derivatives
The invention relates to novel thiophene derivatives, their preparation and their use as pharmaceutically active compounds. Said compounds particularly act as immunosuppressive agents. ...
07/19/2011
7973074π-conjugated mono-, oligo- and polymeric compounds, and photovoltaic cells comprising them
Monomeric, oligomeric or polymeric compound corresponding to the following formula (I): in which: A represents an optionally substituted polycyclic group, the said polycyclic group ...
07/05/2011
7964632Methods of treatment using a prodrug of an excitatory amino acid
This invention relates to synthetic excitatory amino acid prodrugs and processes for their preparation. The invention further relates to methods of using, and pharmaceutical compositions comprising, the compounds for the treatment of neurological disorders and psych...
06/21/2011
7935725Aryl-substituted bridged or fused diamines as modulators of leukotriene Ahydrolase
Aryl-substituted bridged or fused diamine compounds, pharmaceutical compositions containing them, and methods of using the compounds and the pharmaceutical compositions for leukotriene A4 hydrolase (LTA4H or LTA4H) modulation and for the treatm...
05/03/2011
7935724Thiophene and benzothiophene hydroxamic acid derivatives
The present invention relates to a novel class of hydroxamic acid derivatives having a benzothiophene or thiophene backbone. The hydroxamic acid compounds can be used to treat cancer. The hydroxamic acid compounds can also inhibit historic deacetylase and are suitab...
05/03/2011
RE42327Medicinal compositions improving brain function and method for improving brain function
An alkyl ether derivative represented by the formula: wherein R1, R2, R3, R4, m and n are as defined in the specification, or salts thereof exhibits synergistically improved anti-...
05/03/2011
7888387Electro-optic chromophore having an edot structure, and related methods and apparatuses
In various embodiments, chromophores are described that include novel election acceptors, novel electron donors, and/or novel conjugated bridges that are useful in nonlinear optical applications. In some embodiments, the present invention provides chromophore archit...
02/15/2011
7868038Compounds as cannabinoid receptor ligands
The present invention relates to thiophene containing compounds of formula (I) wherein m, n, p, q, r, s, R1, R2, and R3 are as defined in the description. Included also are pharmaceutical co...
01/11/2011
7855226Treatment of inflammatory bowel disease
Disclosed herein is a method comprising administering a compound to a mammal suffering from an inflammatory bowel disease for the treatment of said disease, said compound having a structure according to Formula I wherein X,...
12/21/2010
7846964Thiophene derivatives as spingosine-1-phosphate-1 receptor agonists
The invention relates to novel thiophene derivatives, their preparation and their use as pharmaceutically active compounds. Said compounds particularly act as immunosuppressive agents. ...
12/07/2010
7834053Medicinal compositions improving brain function and method for improving brain function
An alkyl ether derivative represented by the formula: wherein R1, R2, R3, R4, m and n are as defined in the specification, or salts thereof exhibits synergistically improved anti-...
11/16/2010
7750040Thiophene derivatives
The invention relates to novel thiophene derivatives, their preparation and their use as pharmaceutically active compounds. Said compounds particularly act as immunosuppressive agents. ...
07/06/2010
7737176Substituted arylhexadienoic acids and esters thereof which can be used for the treatment and prevention of diabetes, dyslipidaemia and atherosclerosis, pharmaceutical compositions comprising them and processes for the preparation of them
The invention relates to compounds of the formula I: and to the pharmaceutically acceptable salts thereof, to processes for the preparation of them and to pharmaceutical compositions comprising them, which are useful especi...
06/15/2010
7732483DNA-PK inhibitors
A compound of formula I: and isomers, salts, solvates, chemically protected forms, and prodrugs thereof, wherein: R1 and R2 are independently selected from hydrogen, an optionally substituted C1-7...
06/08/2010
7723378Hydrogenated benzo (C) thiophene derivatives as immunomodulators
The invention relates to novel thiophene derivatives, their preparation and their use as pharmaceutically active compounds particularly as immunosuppressant agents. ...
05/25/2010
7674822PTP1b inhibitors
This invention relates to modulating (e.g., inhibiting) protein tyrosine phosphatase 1B (PTP1B). ...
03/09/2010
7671082Prodrugs of excitatory amino acids
This invention relates to synthetic excitatory amino acid prodrugs and processes for their preparation. The invention further relates to methods of using, and pharmaceutical compositions comprising, the compounds for the treatment of neurological disorders and psych...
03/02/2010
7671081Multifunctional cationic photoinitiators, their preparation and use
Compounds of formula (I): wherein the substituents are as defined herein. ...
03/02/2010
765206310-hydroxy-11-dihydroprostaglandin analogs as selective EP4 agonists
A compound comprising or a pharmaceutically acceptable salt or a prodrug thereof, wherein the dashed line represents the presence or absence of a double bond; J is C═O or CHOH; ...
01/26/2010
7645791Salicylic anilides
Novel salicylic anilides are chemical uncouplers useful e.g. for the treatment of obesity. ...
01/12/2010
7585888Benzofuran and benzothiophene derivatives useful in the treatment of hyper-proliferative disorders
This invention relates to novel benzofuran and benzothiophene derivatives of the general formula and their use for the treatment of hyper-proliferative disorders. ...
09/08/2009
7582673Bissulfonamide compounds as agonists of GalR1, compositions, and methods of use
Embodiments of the present invention provide bissulfonamide compounds that are agonists of GalR1. The present invention further provides compositions comprising bissulfonamide compounds that are agonists of GalR1, and methods of use of such compounds and composition...
09/01/2009
7576122Ophthalmic compositions for treating ocular hypertension
This invention relates to potent potassium channel blocker compounds of Formula I or a formulation thereof for the treatment of glaucoma and other conditions which leads to elevated intraoccular pressure in the eye of a patient. This invention also relates to the us...
08/18/2009
7473704Cyclohexyl prostaglandin analogs as EP-receptor agonists
The invention relates to the use of novel cyclohexyl analogues of E-type prostaglandins as EP4 agonists, in general, and, in particular as ocular hypotensives. The cyclohexyl analogues used in accordance with the invention are represented by the following...
01/06/2009
7465752Pentenoic acid derivatives, processes for the preparation thereof, pharmaceutical compositions comprising them, and therapeutic applications thereof
Compounds of the formula (I): in which R, R1, R2 and R3 are as defined in the description, to their use for the treatment of dyslipidaemia, atherosclerosis and diabe...
12/16/2008
7449490Pharmaceutically active compounds and methods of use
New fused thiophene compounds are provided and methods of using those compounds for a variety of therapeutic indications. Compounds of the invention are particularly useful for treatment of neuropathic pain. ...
11/11/2008
7442808Antidiabetic bicyclic compounds
Tricyclic compounds containing a cyclopropyl carboxylic acid or carboxylic acid derivative (e.g. amide) fused to a bicyclic ring, including pharmaceutically acceptable salts and prodrugs thereof, are agonists of G-protein coupled receptor 40 (GPR40) and are useful a...
10/28/2008
7439271Reduction of hair growth
Mammalian hair growth is reduced by applying an inhibitor of telomerase to the skin. ...
10/21/2008
74358342-thia-dibenzoazulenes as inhibitors of tumour necrosis factor production and intermediates for the preparation thereof
The present invention relates to compounds of 2-thia-dibenzoazulene class, to their pharmacologically acceptable salts and solvates, to processes and intermediates for the preparation thereof as well as to their antiinflammatory effects, especially to the inhibition...
10/14/2008
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