Class 514/435 - Three or more hetero atoms in the hetero ring

Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the six-membered hetero ring contains
No. of patents: 35
Last issue date: 09/27/2011

Number	Title	Issue Date
8026274	Use of oxandrolone in the treatment of burns and other wounds The subject invention provides a method of treating burn-induced weight loss in a burn patient which comprises administering a therapeutically effective amount of an oxandrolone to the patient. The invention also provides a method of treating a wound in a patient su...	09/27/2011
7348322	Glucocorticoid receptor modulators as antiinflammatory agents The present invention relates to compounds of formula I: wherein A, X, R1, R2 and R3 are as defined herein and pharmaceutically acceptable salts thereof. The invention also relates to method...	03/25/2008
7148360	Perfluoropolyether benzotriazole compounds Perfluoropolyether benzotriazole compounds and compositions containing perfluoropolyether benzotriazole compounds are provided. The perfluoropolyether benzotriazole compounds can be attached to a substrate having a metal or metal oxide-containing surface to provide ...	12/12/2006
7144985	Methods and reagents for diagnosis and treatment of diabetes The invention relates to methods of determining islet cell activity by detecting the level of Archipelin or a fragment thereof and comparing the level to a baseline level or range associated with a known islet cell activity. Such methods are useful in diagnosing and...	12/05/2006
7022739	Substituted 1-aminobutan-3-ol compounds Substituted 1-aminobutane-3-ol compounds, methods for producing them, pharmaceutical compounds containing them, and the use of substituted 1-aminobutane-3-ol compounds for producing pharmaceutical compounds. ...	04/04/2006
6916829	Method for enhancing mutant enzyme activity in gaucher disease Method for enhancing in a mammalian cell the activity of an enzyme associated with Gaucher Disease by administering a competitive inhibitor of glucocerebrosidase in an amount effective to enhance the activity of the enzyme. Preferred compounds for use in the method ...	07/12/2005
6825226	Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias The invention relates to the discovery that specific adamantyl or adamantyl group derivatives containing retinoid-related compounds induce apoptosis of cancer cells and therefore may be used for the treatment of cancer, including advanced cancer. Also, the present i...	11/30/2004
6727258	Allosteric adenosine receptor modulators The present invention relates to compounds of formula (IA): the preparation thereof, pharmaceutical formulations thereof, and their use in medicine as allosteric adenosine receptor modulators for uses including protectio...	04/27/2004
6620782	Substituted 2-aminobenzamide caspase inhibitors and the use thereof The present invention is directed to novel 2-aminobenzamide thereof, represented by the general Formula I: ##STR1## where R1 -R3, X, and A--D are defined herein. The present invention also relates to the discovery that compounds havi...	09/16/2003
6548534	Nonsteroidal gestagens This invention describes the new, nonsteroidal gestagens of general formula I ##STR1## in which A, B, Ar1, R1, R2 and R3 have the meanings that are indicated in more detail in the description. The new compounds ...	04/15/2003
6541506	Antifungal enediynes The invention features enediynes and methods for their production and use. The enediynes of the invention have the formula: ##STR1## wherein R1 is a hydroxyl group or a moiety that can be replaced by a hydroxyl group in a hydrolysis reaction; e...	04/01/2003
6462064	Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias The invention relates to the discovery that specific adamantyl or adamantyl group derivatives containing retinoid-related compounds induce apoptosis of cancer cells and therefore may be used for the treatment of cancer, including advanced cancer. Also, th...	10/08/2002
6221896	Insecticidal and miticidal compositions This invention relates to an insecticidal and miticidal composition which contains as active ingredients chlorfenapyr in combination with one or more compounds selected from the group consisting of benzoepin, nereistoxin-type insecticidal agents and diafe...	04/24/2001
6127415	Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents The present invention relates to specific adamantyl or adamantyl group derivative containing retinoid compounds induce apoptosis of cancer cells. These adamantyl retinoid derivatives are useful for the treatment of many cancers and solid tumors, especiall...	10/03/2000
5869520	Carbamoyloxylabdanes Novel carbamoyloxylabdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure and treating cardiac failure utilizing compounds and compositions thereof are disclosed....	02/09/1999
5827876	Inhibition of bone loss by 3-(4-acrylamidobenzoyl) benzob!-thiophenes This invention relates to 3-(4-acrylamidobenzoyl)benzob! thiophenes, to the process for their preparation, to pharmaceutical compositions and to their use for modifying the balance between bone resorption and bone production in a mammal. The compounds u...	10/27/1998
5646175	Carbamoyloxylabdane compounds Novel carbamoyloxylabdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure and treating cardiac failure utilizing compounds and compositions thereof are disclosed....	07/08/1997
5543427	Carbamoyloxylabdanes Novel carbamoyloxylabdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure and treating cardiac failure utilizing compounds and compositions thereof are disclosed....	08/06/1996
5374650	Carbamoyloxylabdanes Novel carbamoyloxylabdanes, intermediates and processes for the preparation thereof, and methods for reducing intraocular pressure and treating cardiac failure utilizing compounds and compositions thereof are disclosed....	12/20/1994
5356925	N-(mercaptoalkyl)ureas and carbamates Novel N-(mercaptoalkyl)urea or carbamates of the formulae I and II ##STR1## wherein A is a monocyclic or bicyclic arylene or heteroarylene; Q is hydrogen or R9 CO--; Y is --O--,--S-- or --NR8 --; R1 is lower alkyl, cyclolower a...	10/18/1994
5140039	Aminomethyl-thiochroman compounds The present invention includes compounds represented by the formula: ##STR1## wherein X is O or S; R1 and R2 are independently selected from the group consisting of hydrogen, hydroxy, halo, loweralkoxy, thioalkoxy and loweralkyl...	08/18/1992
5045562	1,3,5-trithiane derivatives and pharmaceutical compositions thereof 1,3,5-trithiane derivatives represented by the formula (I) ##STR1## wherein the substituents are defined herein, are disclosed. The trithiane derivatives and their compositions are useful as anti-arteriosclerotic or anti-hyperlipemic agents....	09/03/1991
4942161	Use of beta blockers for the treatment of the progression of infantile axial myopia The invention relates to the use of beta blockers for the treatment of the progression of infantile axial myopia....	07/17/1990
4816475	1,3,5-trithian derivatives and pharmaceutical compositions An anti-arteriosclerotic or anti-hyperlipemic 1,3,5-trithiane derivative according to the formula (I): ##STR1## a pharmaceutical composition containing the same, and a process for producing the same....	03/28/1989
4804677	Esters of aryloxypropanolamine derivatives Novel compounds of the general formula ##STR1## wherein R1 is lower alkyl, lower cycloalkyl, lower alkenyl, lower alkynyl, lower alkyl carboxymethyl, aryl carboxymethyl, aryl, or aralkyl; A is a direct bond, lower alkylene, or lower alkeny...	02/14/1989
4725591	ଲ-lactamase inhibitory composition Compounds having one or two substituents at the 3-position, represented by the general formula ##STR1## wherein R1 is an optionally acylated or protected amino group and X is hydrogen atom or methoxy group, or a pharmaceutically acceptable...	02/16/1988
4692455	Certain acyclic, alicyclic, aromatic or heterocyclic derivatives of 3-benzoylamino-2-oxo- butyl-amino-carbonyl-oxy-3-propanoic acids, esters thereof, pharmaceutical compositions containing same and their enkephalinase inhibiting properties Compounds of the formula ##STR1## wherein Y is oxygen or sulfur are disclosed. These compounds are useful as hypotensive agents due to their angiotensin converting enzyme inhibition activity and depending upon the definition of R1 may also...	09/08/1987
4626529	Oily compositions comprising a dermatological active principle, intended for the treatment of the scalp or skin The present invention discloses a homogeneous oily composition essentially consisting of a dermatological active principle, an oily compound and an oil-soluble surface-active component, the oil-soluble surface-active component comprising an anionic surfac...	12/02/1986
4551472	Unsymmetrical bis-carbamate compounds Unsymmetrical N-substituted bis-carbamoyl sulfide compounds exhibit exceptional broad spectrum pesticidal activity coupled with extremely low mammalian toxicity and phytotoxicity....	11/05/1985
4327110	Pesticidal symmetrical N-substituted bis-carbamoyloximino disulfide compounds Symmetrical N-substituted bis-carbamoyloximino disulfide compounds exhibit outstanding nematocidal, miticidal and insecticidal activity, coupled with substantially reduced mammalian toxicity and phytotoxicity as compared to known pesticidal compounds havi...	04/27/1982
4234580	Carbamate thiosulfenylcarbamoyl fluoride compounds Carbamate thiosulfenylcarbamoyl fluoride compounds are insecticidal and miticidal compounds and are also useful intermediates in the preparation of pesticidally active bis-carbamate disulfide compounds....	11/18/1980
4179514	Ketoalkanesulfenyl and ketoalkanethiosulfenyl carbamates Ketoalkanesulfenyl and ketoalkanethiosulfenyl carbamates exhibit exceptional pesticidal activity....	12/18/1979
4169894	Pesticidal unsymmetrical N-substituted bis-carbamoyloxy disulfide compounds Unsymmetrical N-substituted bis-carbamoyloxy disulfide compounds exhibit outstanding nematocidal, miticidal and insecticidal activity, coupled with substantially reduced mammalian toxicity and phytotoxicity as compared to known pesticidal compounds having...	10/02/1979
4073930	Carbamoyloximes and oximes and insecticidal and miticidal compositions and methods employing them 2-Oximino-1,3,5-trithiane compounds are useful intermediates in the preparation of 1,3,5-trithiane carbamoyloxime compounds which exhibit outstanding pesticidal activity....	02/14/1978
4072750	1,3,5-Trithiane and 1,3,5-oxadithiane carbamoyloxime compounds and insecticidal and miticidal compositions and methods employing them 1,3,5-Trithiane and 1,3,5-oxadithiane carbamoyloximes exhibit outstanding pesticidal activity....	02/07/1978

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Class 514/435 - Three or more hetero atoms in the hetero ring