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Mountable Printable Placard With Headband

A resilient headband in a shape for being mounted on the head of the user. The headband is equipped with a longitudinal slotted member for holding a placard.

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Class 514/365 - 1,3-thiazoles (including hydrogenated)


Subclass of Class 514 - Drug, bio-affecting and body treating compositions
Definition: Subject matter wherein the five-membered hetero ring is
No. of patents: 1866
Last issue date: 05/22/2012


1                      
NumberTitleIssue Date
8183270Insecticidal -substituted (2-substituted-1,3-thiazol)alkyl sulfoximines
N-Substituted (2-substituted-1,3-thiazol)alkyl sulfoximines are effective at controlling insects. ...
05/22/2012
8178566Crystal form of epothilone B and use in pharmaceutical compositions
The invention relates to new crystal forms of epothilone B. ...
05/15/2012
81484112-hetarylthiazole-4-carboxamide derivatives, their preparation and use as pharmaceuticals
The present invention relates to 2-hetarylthiazole-4-carboxamide derivatives of the formula (I), the use thereof as medicament for the treatment of various disorders, and processes for the preparation thereof ...
04/03/2012
8114897Pesticidal composition and method for controlling a pest
A pesticidal composition containing 4-methoxymethyl-2,3,5,6-tetrafluorobenzyl 3-(2-cyano-1-propenyl)-2,2-dimethylcyclopropanecarboxylate and 1-(2-chloro-1,3-thiazolyl)methyl-3-methyl-2-nitroguanidine has a high pesticidal activity. ...
02/14/2012
8110590Synthesis of epothilones, intermediates thereto and analogues thereof
The present invention provides compounds of formula (I): as described generally and in classes and subclasses herein. The present invention additionally provides pharmaceutical compositions comprisi...
02/07/2012
8106078Human protein tyrosine phosphatase inhibitors and methods of use
The present disclosure relates to compounds effective as human protein tyrosine phosphatase beta (HPTP-β) inhibitors thereby regulating angiogenesis. The present disclosure further relates to compositions comprising said human protein tyrosine phosphatase beta (HPT...
01/31/2012
8088804N-hydroxyamide derivatives possessing antibacterial activity
Described herein are N-hydroxyamide antibacterial compounds, methods for making the compounds, pharmaceutical compositions containing the compounds and methods of treating bacterial infections utilizing the compounds and pharmaceutical compositions compound of Formu...
01/03/2012
8071633Pharmaceutical composition for treating
This invention provide to a pharmaceutical composition for treating spinocerebellar ataxia (or atrophy, degeneration) or multiple system atrophy, or for improving ataxia or equilibrium disturbance comprising a compound of the formula (I):
12/06/2011
8067449Modulators of pharmacokinetic properties of therapeutics
The present application provides for a compound of Formula I, or a pharmaceutically acceptable salt, solvate, and/or ester thereof, compositions containing such compounds, therapeutic methods that include the administration of such compounds, and therapeutic methods...
11/29/2011
8048900Use of 15-lipoxygenase inhibitors for treating obesity
The invention concerns the treatment of obesity, in particular abdominal visceral obesity. More specifically, the invention concerns the use of selective 15-lipoxygenase (LO) inhibitors for preparing medicines useful in the treatment of obesity, or at least abdomina...
11/01/2011
8039495Biphenyl carboxylic acids and bioisosteres as glycogen synthase activators
Provided herein are compounds of the formula (I): as well as pharmaceutically acceptable salts thereof, wherein the substituents are as those disclosed in the specification. These compounds, and the pharmaceutical compositi...
10/18/2011
8026263Methods for inhibiting neoproliferative changes in blood vessel walls
Methods, compositions and devices for inhibiting neoproliferative changes in blood vessel walls or other anatomical structures. One or more compounds of Formula I or I-A set forth herein are administered systemically and/or locally to human or veterinary patients to...
09/27/2011
8008330Combinations comprising epothilones and pharmaceutical uses thereof
The invention relates to a combination which comprises (a) a bisphosphonate, a platinum compound or a vasculostatic compound and (b) an epothilone derivative of formula I wherein A represents O or NRN, wherein R
08/30/2011
8008329Method of treating or preventing osteoporosis comprising administering to a patient in need thereof an effective amount of pharmacuetical composition comprising benzamidine derivative or it's salt, and bisphosphonate
The present invention provides a method of treating or preventing osteoporosis comprising administering to a patient in need thereof an effective amount of pharmaceutical composition comprising benzamidine derivative or its salt, and bisphosphonate for the purpose o...
08/30/2011
7994202Bicyclic nitrogen-containing heterocyclic compounds
A nitrogen-containing bicyclic heterocyclic compound represented by the following formula (1) is provided. When the compound or a salt thereof is administered to a human being or an animal, the compound has a strong antagonistic action against EP1 receptors, and is ...
08/09/2011
7989480Aryl amino acid derivatives as inhibitors for treating inflammation
The present invention relates to a chemical genus of 3-(triaryl)-2-aminopropanol derivative inhibitors of LTA4H (leukotriene A4 hydrolase) useful for the treatment and prevention of inflammatory diseases and disorders. The compounds have general formula III: ...
08/02/2011
7981911Pharmaceutical formulations
Improved pharmaceutical compositions are provided comprising one or more solubilized HIV protease inhibiting compounds having improved solubility properties in a medium and/or long chain fatty acid, or mixtures thereof, a pharmaceutically acceptable alcohol, and wat...
07/19/2011
7977363Biphenyl-thiazolo-carboxamides
Novel biphenyl thiazole carboxamides of Formula (I) where R1, R2, R3, R4, R5 and n have the meanings specified in the description, several method...
07/12/2011
7968575Nitric oxide donors and uses thereof
Disclosed are novel NO-donating compounds, designed such that when NO is released from the compound a residue which is a naturally occurring metabolite is formed, and thus a development of tolerance to the compounds upon repetitive administration is prevented or dec...
06/28/2011
7964622Indole acetic acid derivatives and their use as pharmaceutical agents
This invention is directed to indole acetic acid derivatives and their use in pharmaceutical compositions for the treatment of diseases such as diabetes, obesity, hyperlipidemia, and atherosclerotic disease. The invention is also directed to intermediates useful in ...
06/21/2011
7956075Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
The invention relates to thiazole, oxazole, imidazole, isoxazole and isoxazoline derivatives of general formula (I) wherein Het is thiazole, oxazole, imidazole, isoxazole or isoxazoline, n is an integer from 0 to 6, A is no...
06/07/2011
7943646Benzamidine derivative, process for the preparation thereof and pharmaceutical composition comprising same
The present invention relates to a novel benzamidine derivative, a process for the preparation thereof, and a pharmaceutical composition comprising the same. The benzamidine derivative of the present invention effectively inhibits osteoclast differentiation at an ex...
05/17/2011
7939553Modulators of pharmacokinetic properties of therapeutics
The present application provides for a compound of Formula I, or a pharmaceutically acceptable salt, solvate, and/or ester thereof, compositions containing such compounds, therapeutic methods that include the administration...
05/10/2011
7902236Antagonists of the vanilloid receptor subtype 1 (VR1) and use thereof
The present invention is directed to compounds of formula (I) wherein variables W, X, Y, D, A, n, R1, R2 and R9 are as defined in the description. ...
03/08/2011
78976262-substituted thiazole-4-carboxamide derivatives, their preparation and use as pharmaceuticals
The present invention relates to 2-substituted thiazole-4-carboxamide derivatives of the formula (I), the use thereof as medicament for the treatment of various disorders, and processes for the preparation thereof ...
03/01/2011
7893097Methods and compositions for increasing solubility of azole drug compounds that are poorly soluble in water
The combination of any two of a polyol, a polyol ether, and a low carbon organic alcohol provides a synergistic effect on the solubility of azole compounds, such as metronidazole, in aqueous fluid. ...
02/22/2011
7879886Iron binding agents
Composition, article of manufacture for and method of treating malaria in a human having an infestation of Plasmodium protozoans are described. The method comprises administering a therapeutically-effective amount of a compound of formula (I) or (IV), i.e. su...
02/01/2011
7875638Synthesis of epothilones, intermediates thereto, analogues and uses thereof
The present invention provides compounds of formula (I): as described generally and in classes and subclasses herein. The present invention additionally provides pharmaceutical compositions comprisi...
01/25/2011
7863303Insecticidal -substituted (2-substituted-1,3-thiazol)alkyl sulfoximines
N-Substituted (2-substituted-1,3-thiazol)alkyl sulfoximines are effective at controlling insects. ...
01/04/2011
7863304Analogs of glycyl-prolyl-glutamate
Embodiments of this invention include novel analogs of Glycyl-Prolyl-Glutamate (GPE) and compositions containing such analogs of GPE. Of these, certain analogs have modified proline residues. Other embodiments of this invention include uses of analogs of GPE to prot...
01/04/2011
RE41990Synthesis of epothilones, intermediates thereto, analogues and uses thereof
The present invention provides convergent processes for preparing epothilone A and B, desoxyepothilones A and B, and analogues thereof. Also provided are analogues related to epothilone A and B and intermediates useful for preparing same. The present invention furth...
12/07/2010
7846952Epothilones C, D, E, and F, preparation and compositions
The present invention relates to epothilones C, D, E, and F, their preparation and their use for the production of therapeutic compositions and compositions for plant protection. ...
12/07/2010
7846951Thiazoles and oxazoles useful as modulators of ATP-binding cassette transporters
The present invention relates to modulators of ATP-Binding Cassette (“ABC”) transporters or fragments thereof, including Cystic Fibrosis Transmembrane Regulator (“CFTR”), compositions thereof, and methods therewith. The present invention also relates to meth...
12/07/2010
7825141Epothilone derivatives
Epothilone derivatives of Formula (I) and their use as a pharmaceutical. ...
11/02/2010
7825142Heterocyclic compounds, compositions comprising them and methods of their use
Heterocyclic compounds, compositions comprising them, and methods of their use for the treatment, prevention and management of inflammatory and autoimmune diseases and disorders are disclosed. Particular compounds are of formula I:
11/02/2010
RE41911Epothilone derivatives
The present invention relates to epothilone derivatives, having the following formula in which the variables G, W, Q, X, Y, B1, B2, Z1, Z2, and R1-R7 are as define...
11/02/2010
RE41895Epothilone derivatives
The present invention relates to epothilone derivatives, having the following formula in which the variables G, W, Q, X, Y, B1, B2, Z1, Z2, and R1-R7 are as define...
10/26/2010
7812041Heterocyclic NF-κB inhibitors
The present invention relates to compounds of the general formula (I) and salts and physiologically functional derivatives thereof, wherein R1 is independently hydrogen; alkyl, cycloalkyl, hydroxyalk...
10/12/2010
78038232-amino-4,5-trisubstituted thiazolyl derivatives
This invention concerns the use of a compound of formula (I′) a N-oxide, a pharmaceutically acceptable addition salt, a quaternary amine and a stereochemically isomeric form thereof, wherein Z is halo; C1-6alky...
09/28/2010
7799813Salts of substituted 5-membered azacycle and use thereof in the treatment of diseases related to protein aging
The present invention relates to 5-membered azacycle compounds of formula (I), pharmaceutically acceptable salts thereof and hydrates thereof, wherein the groups are as defined in the specification. The present invention further relates to pharmaceutical composition...
09/21/2010
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