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Class 564/98 - Substituent Q is alkyl


Subclass of Class 564 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the sulfonic acid residue consists of
No. of patents: 166
Last issue date: 02/14/2012


1          
NumberTitleIssue Date
8115030Process for the preparation of sulfomate-carboxylate derivatives
Disclosed is a process for the preparation of Compound (III), salt or solvate thereof by reacting Compound (I), salt or solvate thereof with Compound (II) in a toluene solvent in the presence of an additive such as water or an alcohol. Also disclosed is a process fo...
02/14/2012
7453010Phenylcyclohexylpropanolamine derivatives, preparation and therapeutic application thereof
The invention relates to compounds of general formula (I): where R1 represents H or a (C1-C4)alkyl, —CO(C1-C4)alkyl, (C1-C4
11/18/2008
7411002Polycationic sulfonamides and use thereof
Certain lipophilic polycationic sulfonamides are provided and are useful for treating various diseases or conditions and particularly sepsis. ...
08/12/2008
7365196Sulphonamido-substituted bridged bicycloalkyl derivatives
A class of compounds is disclosed, comprising sulphonamido-substituted bridged bicycloalkyl structures. The compounds are inhibitors of gamma-secretase, and hence are useful in the treatment of and/or prevention of Alzheimer's disease. ...
04/29/2008
7232817α- and β-amino acid hydroxyethlamino sulfonyl urea derivatives useful as retroviral protease inhibitors
α- and β-amino acid hydroxyethylamino sulfonyl urea derivative compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. ...
06/19/2007
7220914Zwitterionic compounds and photovoltaic cells containing same
Zwitterionic compounds, photovoltaic cell charge carrier layers containing such compounds, photovoltaic cells including such charge carrier layers, and related methods are disclosed. ...
05/22/2007
7169952Process to prepare sulfonamides
A process for the preparation of a sulfonamide of formula (II), comprising reacting at elevated temperature an aniline of formula (I), with a sulfonating agent A of the formula R1—SO2-Z in the presence of a catalytic amount of either: (i) an ...
01/30/2007
6984757Process for preparing 2-amino-4-(4-fluorphenyl)-6-alkylpyrimidine-5-carboxylate
A process for the preparation of a 4-(4-flourophenyl)-6-alkyl-2-N-alkansulfonyl-N-alkylamino)pyrimidine-5-carboxylic acid ester of formula (Ib), in which R1, R2, R3 and R4 are identical or different and are each a C1-...
01/10/2006
6963010Hydrophobic polyamine analogs and methods for their use
The disclosed invention provides new polyamine analogs and derivatives containing a hydrophobic region and a polyamine region as well as methods and compositions for their use. ...
11/08/2005
6958416Valproyltaurinamide derivatives as anticonvulsant amd CNS active agents
The invention relates to derivatives of valproyltaurinamide of formula (I) in which R1 and R2 are independently hydrogen, a C1-C6-alkyl group, an arylalkyl group or an aryl group. The derivatives are especially useful for ...
10/25/2005
6911595Charge transfer material, and photoelectric conversion device and photoelectric cell using same, and pyridine compound
A charge transfer material comprising a basic compound having negative charge and represented by the following general formula (I): (A1-L)n1-A2·M  (I), wherein A1 represents a group having negativ...
06/28/2005
6908947Sulfonamide-substituted fused 7-membered ring compounds, their use as a medicament, and pharmaceutical preparations comprising them
The present invention relates to compounds of formula I, in which X1, X2, X3, X4, Y1, Y2, Y3, Y4, R(3), R(4) and R(5) have the meanings mentioned in the specification, their preparation and their use, in particular in ...
06/21/2005
6900353Cyclopentyl sulfonamide derivatives
The present invention provides compounds of formula (I): useful for potentiating glutamate receptor function in a mammal and therefore, useful for treating a wide variety of conditions, such as psychiatric and neurological disorders. ...
05/31/2005
6743929Sulfonylalkanoylamino hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
Sulfonamide-containing hydroxyethylamine compounds are effecive as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. ...
06/01/2004
6706755Cyclopentane heptan(ene) acyl sulfonamide, 2-alkyl or 2-arylalkyl, or 2-heteroarylalkenyl derivatives as therapeutic agents
The present invention provides a method of treating ocular hypertension or glaucoma which comprises administering to an animal having ocular hypertension or glaucoma therapeutically effective amount of a compound represented by the general formula I;
03/16/2004
6620858Colorants containing copolymerizable vinyl groups and sulfonamide linkages
Disclosed are thermally-stable, colored, photopolymerizable compounds containing a vinyl group which are capable of being copolymerized with reactive vinyl monomers to produce colored compositions such as polyacrylates, polymethacrylates, polystyrene, etc...
09/16/2003
6596863Medical composition containing nitroetheneamine Derivative or salt there of as active constituent
Process for producing a nitroetheneamine derivative ##STR1## or its stereoisomer, its tautomer or a salt thereof comprising reacting a compound of the formula ##STR2## with a compound of the formula R6 --CH2 NO2 to obtain ...
07/22/2003
6583318Method for synthesis of ଱-sulfonamido amide, carboxylic acid and hydroxamic acid derivatives
A method of synthesizing ଱-sulfonamido amide, carboxylic acid or hydroxamic acid derivatives comprising providing a set of polymer-bound reactant(s) (sulfonamide, aldehyde or ketone, isocyanide or acid) to react with three sets of the other three re...
06/24/2003
6562782Oligocycloalkanoid compounds and methods of use
The present invention related to an oligocycloalkanoid compound comprising formula (I) ##STR1## wherein m, n, and o are independently an integer from 0 to 2; A1 through A10 are independently a direct link, alkylene, alkylene-O--, ...
05/13/2003
6559137Sulphonamide derivatives as prodrugs of aspartyl protease inhibitors
The present invention relates to prodrugs of a class of sulfonamides which are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of prodrugs of HIV aspartyl protease inhibitors characterized by favorable aqueous solu...
05/06/2003
6451792Medical composition containing nitroetheneamine derivative or salt thereof as active constituent
A medical composition containing, as an active constituent, a nitroetheneamine derivative represented by the formula (I): ##STR1## wherein the substituents are as defined in the disclosure, its stereoisomers, its tautomers or a salt thereof....
09/17/2002
6410749Process for the preparation of optically active amino alcohols
Process for preparing optically active ଲ-amino alcohols represented by a general formula (2): Ra--C*H(OH)--C*H(Rb)--Rc wherein Ra and Rc are each independently hydrogen, optionally substituted alkyl, optionally substituted cycloalkyl, Rb is one memb...
06/25/2002
6387954Alkenyl sulphonamide derivatives
The present invention provides certain alkenyl sulphonamide derivatives useful for potentiating glutamate receptor function in a mammal and therefore, useful for treating a wide variety of conditions, such as psychiatric and neurological disorders....
05/14/2002
6319428Perfluorinated amide salts and their uses as ionic conducting materials
The invention concerns ionic compounds in which the anionic load has been delocalized. A compound disclosed by the invention is comprised of an amide or one of its salts, including an anionic portion combined with at least one cationic portion M+m
11/20/2001
6284795Sulfonamide compounds and methods of treating atherosclerosis and restenosis
The present invention provides compounds having the Formula I ##STR1## The present invention also provides methods of treating or preventing atherosclerosis, coronary heart disease, and restenosis using the compounds of Formula I, and pharmaceutical compo...
09/04/2001
6271262Metalloproteinase inhibitors
A compound of formula (I) ##STR1## useful as metalloproteinase inhibitors....
08/07/2001
6200967Anticoagulant agents
This invention relates to a compound of the Formula I X--C(O)--Y--G--R I (wherein X, Y, G and R have the values defined in the description), or a pharmaceutically acceptable salt thereof, processes and intermediates for the preparation of such a compound or s...
03/13/2001
6159989Antagonists of gonadotropin releasing hormone
There are disclosed compounds of formula (I) ##STR1## and pharmaceutically acceptable salts thereof which are useful as antagonists of GnRH and as such may be useful for the treatment of a variety of sex-hormone related and other conditions in both m...
12/12/2000
6054613Process for the production of sulphonamides
A process for the preparation of a sulfonamide of formula: RSO2 NR1 R2 wherein R represents C1 -C10 alkyl; and R1 and R2 independently represent hydrogen, C1 -C10 alk...
04/25/2000
6022872଱- and ଲ-amino acid hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors
଱- and ଲ-amino acid hydroxyethylamino sulfonyl urea derivative compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease....
02/08/2000
6015822Sulfonamide-substituted fused 5-membered ring compounds, their use as a medicament, and pharmaceutical preparations comprising them
Compounds of the formula I ##STR1## having the meanings of the substituents indicated in the claims are outstandingly active substances for the production of medicaments for the prophylaxis and for the therapy of cardiovascular disorders, in particul...
01/18/2000
5968916Fluoroalkenyl compounds and their use as pest control agents
Fluorinated alkene compounds useful for and methods of controlling nematodes, insects, and acarids that prey on agricultural crops. Polar compounds are particularly useful for systemic control of pests....
10/19/1999
5965588Sulfonylalkanoylamino hydroxyethylamimo sulfonamides useful as retroviral protease inhibitors
Sulfonamide-containing hydroxyethylamine compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease....
10/12/1999
5856353Sulfonamide inhibitors of aspartyl protease
The present invention relates to a novel class of sulfonamides which are aspartyl protease inhibitors. In one embodiment, this invention relates to a novel class of HIV aspartyl protease inhibitors characterized by specific structural and physicochemical ...
01/05/1999
5830917L-N6 -(1-iminoethyl) lysine derivatives useful as nitric oxide synthase inhibitors
There is disclosed a novel amino alcohol amine derivatives of L-N6 -(1-iminoethyl)lysine, pharmaceutical compositions containing these novel compounds, and to their use in therapy, in particular their use as nitric oxide synthase inhibitors....
11/03/1998
5789618Synthetic method for a halogen-containing condensation product
A method for synthesizing a halogen-containing condensation product, the method comprising the step of: reacting a compound represented by Formula (I) with a compound represented by Formula (II) or (III) in the presence of a halogenating agent whereby deh...
08/04/1998
5739085O-(oximino)ethylcyclohexenone oxime ethers and their use as herbicides
O-(Oximino)ethylcyclohexenone oxime ethers I ##STR1## (R1 and R2 =C1 -C6 -alkyl; R3 =unsubstituted or substituted phenyl, C1 -C4 -alkyl, C3 -C4 -alkenyl or ...
04/14/1998
5716980Alcohol or aldehyde derivatives and their use
The present invention provides a cathepsin L inhibitor containing a compound of the formula: ##STR1## wherein R1 is a hydrogen atom or an arylalkyl, heterocyclic-alkyl or lower alkyl group which may be substituted; R2 and R...
02/10/1998
5705691Chemical process
A process for the preparation of an N-(alkylsulphonyl)amide, the process comprising reacting a primary amide with a sulphonyl halide in the presence of a base which is sufficiently strong to cause at least partial deprotonation of the amide....
01/06/1998
5684195Method of preparing sulfmonamides from sulfones
A one-pot synthesis of sulfonamides from sulfones has been developed. Conversion of sulfones to the corresponding sulfinic acid salts is followed by oxidative-amination to give the sulfonamides....
11/04/1997
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