Class 564/56 - Aralkyl bonded directly to urea nitrogen

Subclass of Class 564 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein an aralkyl group is bonded directly to
No. of patents: 153
Last issue date: 06/14/2011

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Number	Title	Issue Date
7960584	Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same This present invention relates to novel compounds, isomer thereof or pharmaceutically acceptable salts thereof as vanilloid receptor (Vanilloid Receptor 1; VR1; TRPV1) antagonist; and a pharmaceutical composition containing the same. The present invention provides a...	06/14/2011
7351738	Substituted ureas and carbamates The invention provides compounds of formula I: useful in treating Alzheimer's disease and other similar diseases. These compounds include inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer...	04/01/2008
7326746	Curable electron donor compositions Electron donor compounds, suitable for use as adhesives or as components in adhesives, contain a carbon to carbon double bond attached to an aromatic ring and conjugated with the unsaturation in the aromatic ring. ...	02/05/2008
6908957	Curable electron donor compounds Electron donor compounds, suitable for use as adhesives or as components in adhesives, contain a carbon to carbon double bond attached to an aromatic ring and conjugated with the unsaturation in the aromatic ring. ...	06/21/2005
6900213	Bisaryl derivatives having FSH modulatory activity The invention relates to bisaryl derivatives of the formula I, wherein (R,R) is selected from (H,H), O, (H,CH3), (H,OH) and (H,CN); Ar is substituted phenyl and A is a group of formula II, III, IV ...	05/31/2005
6872851	Substituted cyclic compounds, preparation method and pharmaceutical compositions containing them The invention concerns compounds of formula (I): R—A—R′ wherein: A is as defined in the description; R represent, a group (V), wherein R′a and R″a are as defined in the description, or R forms with A a cyclic structure as defined in t...	03/29/2005
6841701	Inhibitors for the blood-clotting factor Xa The invention relates to derivatives of amidino-benzylamine, especially derivatives of 4-amidino-benzylamine, with two bonded amino acids. These derivatives represent a novel group of highly active and very selective F Xa-inhibitors for treating cardiovascular disea...	01/11/2005
6777561	Compounds Compounds of general formula I are disclosed and claimed in the present application, as well as their pharmaceutically acceptable salts, pharmaceutical compositions comprising the novel compounds and their use in therapy...	08/17/2004
6730784	Urea derivatives useful as synthetic intermediates Objects of the present invention are to create compounds having urea structure as basic structure and having a sulfur atom and an amide bond in side chains and to find pharmacological effects thereof, particularly TNF-α production inhibitory effects. The pre...	05/04/2004
6723875	Process to prepare alkyl-ureas from O,S-dimethyl dithiocarbonate The present invention relates to the preparation of alkyl-ureas, starting from O,S-dimethyl dithiocarbonate, which provides the following steps: A) causing the O,S-dimethyl dithiocarbonate to react with a primary amine of general formula R1NH2...	04/20/2004
6683200	N-substituted-N'-substituted urea derivatives and pharmaceutical compositions containing the derivatives N-Substituted-N'-substituted urea derivatives represented by the following formula, analogs thereof or pharmaceutically acceptable salts thereof are herein provided. These compounds show a TNF-଱ production inhibitory activity. ##STR1##...	01/27/2004
6635650	Substituted dimeric compounds The invention relates to compounds of formula (I): wherein: A represents NR1 C(Q)R2, C(Q)NR2 R3 or NR1 C(Q)NR2 R3, B represents NR1 C(Q)R2, C(Q)NR2...	10/21/2003
6620961	Biarylalkylenecarbamic acid derivatives and bacteriocides for agricultural and horticultural use Biarylalkylenecarbamic acid derivative represented by general formula (I): ##STR1## [wherein Q is a phenyl group which may be substituted or the like, X is a halogen atom, a (C1 -C6) alkyl group or the like, n is 0 or an integer of f...	09/16/2003
6528543	Urea derivatives Glucokinase activating compounds of the formula ##STR1## wherein R1 and R2 are independently hydrogen, halo, amino, nitro, cyano, sulfonamido, lower alkyl, perfluoro-lower alkyl, lower alkyl thio, perfluoro-lower alkyl thio, lower al...	03/04/2003
6423870	Tricyclic compounds, preparation method and pharmaceutical compositions containing same The invention concerns compounds of formula (I) in which: A forms a tricyclic system of formula A1, A2, A3 or A4 ; R1 represents a hydrogen atom, an alkyl, hydroxy, alkoxy or oxo group; (R2...	07/23/2002
6329529	Nitrogen-based halogenating agents and process for preparing halogen-containing compounds Disclosed are a fluorinating agent represented by the general formula (1): ##STR1## wherein R1 to R4 are a substituted or unsubstituted, saturated or unsaturated alkyl group or a substituted or unsubstituted aryl group, and can be th...	12/11/2001
6319930	Substituted dimeric compounds The invention relates to compounds of formula (I): A--G1 --Cy--G2 --Cy--G3 --B (I) wherein: A represents NR1 C(Q)R2, C(Q)NR2 R3 or NR1 C(Q)NR2 R3, B repre...	11/20/2001
6313071	Phenylacetylene derivatives and agricultural/horticultural fungicides A phenylacetylene derivative represented by the formula [I]: ##STR1## {wherein X is a halogen atom, a C1 -C6 alkyl group, a C2 -C6 alkoxy group, a C2 -C6 haloalkyl group, etc., n is 0 or an...	11/06/2001
6310074	Substituted dimeric compounds The invention relates to compound of formula (I): A--G1 --Cy--G2 --Cy'--G3 --B (I) wherein: A represents a grouping NR1 C(Q)R2, C(Q)NR2 R3 or NR1 C(Q)NR2 R3	10/30/2001
6235789	Benzocycloalkene compounds, their production and use A compound of the formula ##STR1## wherein R1 and R2 are H, a hydrocarbon group or a heterocyclic group, or R1 and R2 are combinedly a spiro ring; R3 is a hydrocarbon group, a substituted amino group,...	05/22/2001
6184410	Carbodiimides based on 1,3-bis(1-methyl-1-isocyanatoethyl)benzene Carbodiimides based on 1,3-bis(1-methyl-1-isocyanatoethyl)benzene contain from 12 to 40% by weight of ethylene oxide units [--CH2 --CH2 --O--], based on the weight of the carbodiimides....	02/06/2001
6152968	Water-soluble Quinacridones The use of water-soluble quinacridones of the formula I ##STR1## where M.sym. is a lithium, sodium, potassium or ammonium cation, R1, R2, R3 and R4 independently are hydrogen, C1 -C8	11/28/2000
6140531	Method of preparing N-1-alkenyl carbonylamino compounds Describes a method of producing N-1-alkenyl carbonylamino compounds represented by the following general formula I, ##STR1## wherein R1 is the residue of an active hydrogen functional material, n is a number from 1 to a number equal to the...	10/31/2000
6140368	Naphthols useful in antiviral methods The present invention relates to a novel class of compounds that are potent inhibitors of HIV reverse transcriptase and HIV integrase. In addition to being multienzyme inhibitors, the inventive compounds of the present invention are remarkable in at least...	10/31/2000
6127414	NPY antagonists There is provided pharmaceutically useful compounds of formula I, ##STR1## wherein Ar1, R1, R2, R3, R4, R5 and R6 have meanings given in the description, which are useful as anta...	10/03/2000
6114390	Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them NPY-antagonistic compounds of the formula ##STR1## Exemplary are: (A) (R)-N-[[4-(Aminocarbonylaminomethyl)phenyl]methyl]-N.sup.2 -bis(4-hydroxyphenyl)acetyl]-argininamide-trifluoracetate; (B) (R)-N-[[4-(Aminocarbonylaminomethyl)phenyl]methyl]-N.sup.2...	09/05/2000
6080874	Synthesis and isolation of N-(aryl or heteroaryl)-alkyl-N-hydroxyurea The present invention provides a simple, 1-step process for preparing a N-(aryl or heteroaryl)-hydroxyurea comprising reacting the corresponding alcohol, ester or ether with hydroxyurea and acid. This reaction is particularly useful for preparing a benzo[...	06/27/2000
6022899	Substituted benzyloxy-carbonylguanidines, a process for their preparation, their use as a medicament or diagnostic, and a medicament containing them There are described compounds of the formula I ##STR1## in which the substituents R(1) to R(7) and X have the meanings shown in the claims, and their pharmaceutically tolerable salts. These are effective inhibitors of the cellular sodium proton antip...	02/08/2000
5962530	Amino acid derivatives, medicaments containing said compounds and methods of producing them The invention relates to new amino acid derivatives of general formula ##STR1## wherein R, U, V, Y, n, m and R1 to R3 are defined as in claim 1, their tautomers, diastereomers, enantiomers, mixtures thereof and salts thereof, pa...	10/05/1999
5932595	Matrix metalloprotease inhibitors The present invention relates to compounds of Formula I: ##STR1## that are matrix metalloprotease inhibitors, pharmaceutical compositions containing them, methods for their use and methods of preparing these compounds....	08/03/1999
5922771	Benzocycloalkene compounds, their production and use A compound of the formula ##STR1## wherein R1 and R2 independently represent H or an optionally substituted hydrocarbon group; R3 represents an optionally substituted hydrocarbon group; R4 represents H or a...	07/13/1999
5892100	Method for producing N-acyl carbamate The present invention provides a method for producing N-acyl carbamate in high yield. The method of the present invention comprises the step of reacting an unsaturated acid halide with a carbamate in the presence of a hindered amine. Another method of the...	04/06/1999
5849732	Phenol compound having antioxidative activity and the process for preparing the same Disclosed are a phenol compound represented by the formula (1): ##STR1## wherein R0 represents H, alkyl or alkyloxy; R1 represents alkyl; R2 represents alkyl or alkyloxy; OR3 represents OH; R4 re...	12/15/1998
5811456	Monoamine oxidase B inhibitors, processes for their preparation and use thereof Novel monoamine oxidase B inhibitors of formula (I), wherein R1 .dbd.H, an optionally substituted benzyloxy or phenylethoxy group; p=0-3; R3 .dbd.H, a CN, OH, CCH group, a C1 -C3 alkoxy-carbonyl group, or a C	09/22/1998
5807875	Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them Amino acid derivatives, suitable for the treatment of obesity. The following compound is exemplary of the class: (R,S)-N2 -(diphenylacetyl)-N-(4-hydroxyphenyl)methyl!-N5 -(1H-imidazol-2-yl)-ornithinamide....	09/15/1998
5780512	Alkylated (hetero) cyclic compounds The invention relates to a compounds selected from these of formula (I): ##STR1## in which: R1, R2, R3 and A are as defined in the description, and a medicinal product containing the same useful for treating a melaton...	07/14/1998
5760071	Aryl(alkyl)propylamides The invention relates to a compound selected from those of formula (I): ##STR1## in which A, R1, R'1, R2, R3 and n are as defined in the description, and medicinal product containing the same useful for tre...	06/02/1998
5714633	Process for the preparation of arylalkynyl-N-hydroxyurea derivatives having lipoxygenase inhibitory activity The present invention provides a process for the preparation of a compound of formula ##STR1## wherein R is a straight or branched alkyl group of from one to twelve carbon atoms; M represents hydrogen or a pharmaceutically acceptable cation; and...	02/03/1998
5712312	Tricyclic amides The invention relates to a compound selected from these of formula (I): ##STR1## in which R7, R8, Y, n and A are as defined in the description, and medicinal product containing the same useful for treating a disorder of the mela...	01/27/1998
5703076	Retroviral protease inhibitors Urea-containing hydroxyethylamine compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease....	12/30/1997

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Class 564/56 - Aralkyl bonded directly to urea nitrogen