Class 564/352 - The aryl ring or ring system is polycyclo

Subclass of Class 564 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the ring system is polycyclo.
No. of patents: 40
Last issue date: 07/25/2006

Number	Title	Issue Date
7081465	Alpha-substituted naphthyloxy omega-substituted alky/aryl amino-substituted alkane derivatives as agent for treatment or prophylaxis of diabetes and related metabolic disorders This invention relates to novel {overscore (ω)}-substituted-naphthyloxy-amino alkanes, their preparation and use as antihyperglycemic agents and for the treatment and prevention of cardiovascular disorders (CVS) such as lipid lowering effects. ...	07/25/2006
6610705	Process for the preparation of diaryl naphthyl methanes The invention relates to novel diaryl naphthyl methane compounds having general formula I as shown herein below, and said compounds useful in the treatment of esterogen related disease or syndrome, ##STR1## Pharmaceutical compositions comprising said nove...	08/26/2003
6545053	Tricyclic compounds and drug compositions containing same Compounds having a ଲ-3 adrenaline receptor agonist and are useful as drugs for the treatment and prevention of diabetes, obesity, hyperlipemia, etc., represented by a general formula (I) and salts thereof, and a process for producing these, and thei...	04/08/2003
6437137	Naphthyl compounds, intermediates, processes, compositions, and methods The invention is a process for preparing a compound of formula Ia ##STR1## comprising reducing the compound of formula IIId ##STR2## wherein R3 is 1-piperidinyl, 1-pyrrolidinyl, dimethylamino, diethylamino or 1-hexamethyleneimino, R1a	08/20/2002
6057371	Sigma receptor ligands and the use thereof The invention relates to methods for the treatment of central nervous system disorders, gastrointestinal disorders, drug abuse, angina, migraine, hypertension and depression by administering a pharmaceutical composition comprising an effective amount of c...	05/02/2000
6004959	Alkyloxyamino substituted fluorenones and their use as protein kinase-C inhibitors The present invention describes certain alkyloxyamino-substituted fluorenones which inhibit protein kinase C, as well as pharmaceutical compositions including these compounds and methods of using these compounds to control protein kinase C activity in mam...	12/21/1999
5736568	2-(aminoalkoxy) phenylalkylamines with antiinflammatory activity Compounds of the formula I ##STR1## including pharmaceutically acceptable salts thereof are disclosed in which R1, R2, R3, and R4 independently represent hydrogen, hydroxy, halo, halogenated alkyl, halogena...	04/07/1998
5698733	Use of 9-deoxy prostaglandin derivatives to treat glaucoma Disclosed are 9-deoxyprostaglandins which are useful in the treatment of glaucoma and ocular hypertension. Some of these 9-deoxyprostaglandins are novel. Also disclosed are ophthalmic, pharmaceutical compositions comprising such prostaglandins....	12/16/1997
5650476	Process for production of polycarbodiimide resin powder A process for producing a polycarbodiimide resin powder, which includes reacting an organic diisocyanate in the presence of a carbodiimidization catalyst in a solvent to produce a polycarbodiimide resin and obtaining the resin in a powder form, where the ...	07/22/1997
5420294	Cycloalkylaminoalkoxyindoles This invention provides a method of selectively antagonizing the 5-HT1A receptor in mammals by administering aryloxypropanolamines. Aryloxypropanolamines are also claimed....	05/30/1995
5358971	Substituted 2-aminotetralins Optically active or racemic compounds are provided having the formula ##STR1## where R2, R3 and R4 are selected from the group consisting of H and OA with the provision that at least one of R2, R3 and...	10/25/1994
5310756	Aryloxyphenylpropylamines and their calcium overload blocking compositions and methods of use Novel aryloxyphenylpropylamines having the formula ##STR1## wherein X is H, cyano, halogen, halogenoalkyl, C1-6 -alkoxy, C1- -alkyl, C1-5 -alkanoyl, C3-5 -alkylene, aryloxy- or aralkoxy, and R is 3,4-methyl...	05/10/1994
5274003	Substituted 2-aminotetralins Optically active or racemic compounds are provided having the formula ##STR1## where R2, R3 and R4 are each selected from the group consisting of H and OH with the provision that at least one of R2, R3...	12/28/1993
5272144	Aryloxy-, arylthio-, heteroaryloxy-, heteroarylthio-alkenylene derivatives of amines and pharmaceutical use Aryloxy- and heteroaryloxy-alkylene derivatives of amines of formula ##STR1## wherein each of A and B is a group of formula (i) to (iii): ##STR2## wherein Y is --O--, --S-- or --NR-- in which R is hydrogen or C1 -C6 alkyl;...	12/21/1993
5216178	Process of reducing olefins Novel aminoalkylthiodibenzoxepins, physiologically tolerable acid addition salts thereof, a method of preparing same, pharmaceutical and veterinary preparations including same and methods of treating by administering same are disclosed. These compounds ar...	06/01/1993
5192765	Certain amines which are muscarinic receptor antagonists Amines of the following formula: ##STR1## where the variables are defined in the specification are useful in the treatment of diseases associated with altered motility and/or tone of smooth muscle....	03/09/1993
5145870	Aryloxyphenylpropylamines their preparation and use Novel aryloxyphenylpropylamines having the formula ##STR1## wherein X is H, cyano, halogen, halogenoalkyl, C1-6 -alkoxy, C1-6 -alkyl, C1-5 -alkanoyl, C3-5 -alkylene, aryloxy or aralkoxy, and R is 3,4-methyl...	09/08/1992
5135947	1-phenyl-3-naphthalenyloxypropanamines and their use as selective serotonin reuptake inhibitors The present invention provides 1-phenyl-3-naphthalenyloxypropanamines which are selective inhibitors of serotonin uptake....	08/04/1992
4994616	Anilide herbicides A novel herbicide of formula I ##STR1## wherein R1 represents a halogen atom or an alkyl, haloalkoxy, haloalkyl or alkoxycarbonyl group; R2 represents a hydrogen or halogen atom; each of R3 to R6 independently r...	02/19/1991
4968679	8-substituted 2-aminotetralins New 8-substituted 2-aminotetralins can be prepared from the corresponding aminotetralins or tetralones. They can be used in medicaments....	11/06/1990
4956388	3-aryloxy-3-substituted propanamines The present invention provides 3-aryloxy-3-substituted propanamines capable of inhibiting the uptake of serotonin and norepinephrine....	09/11/1990
4853408	4-phenylpropyl-indoles having antiarythmic activity Novel 4-phenylpropyl-indoles of the formula ##STR1## wherein R and R1 are individually selected from the group consisting of hydrogen, linear alkyl of 1 to 5 carbon atoms, branched alkyl of 3 to 5 carbon atoms, cycloalkyl of 3 to 7 carbon ...	08/01/1989
4831051	Aromatic derivatives comprising an aminoalkoxy chain, the salts thereof, the process for preparing these derivatives and salts and the application thereof in therapeutics New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar represents a group of structure: ##STR3## ...	05/16/1989
4792570	3- and 4-biphenyloxyaminoalkanes and related compounds as anti-inflammatory and analgetic agents Compounds useful for treating inflammation, swelling and associated pain, represented by the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein: a is an integer of 0-3; b is an integer of 0-2; n is an integer o...	12/20/1988
4792551	9-anthryloxyaminoalkanes and related compounds as anti-inflammatory and analgetic agents Compounds useful for treating inflammation, pain and swelling, represented by the formula: ##STR1## and the pharmaceutically acceptable acid addition salts thereof, wherein: Y and Z are each independently halo, alkyl or alkoxy; l and m are each indep...	12/20/1988
4732896	Aromatic derivatives comprising an aminoalkoxy chain, the salts thereof, the process for preparing these derivatives and salts and the application thereof in therapeutics New aromatic derivatives having an activity antagonistic to calcium and corresponding to formula: ##STR1## in which: A represents a chain having any one of the following structures: ##STR2## Ar represents a group of structure: ##STR3## ...	03/22/1988
4661297	Basic ethers of 7-oxo-7H-benzo(c) fluorene and a process for their production Basic ethers of 7-oxo-7H-benzo(c) fluorene have been shown to evidence a pronounced antineoplastic and immunosuppressive effect in mammals suffering from leukemia. The technique for preparing the described ethers and the addition salts thereof with pharma...	04/28/1987
4605673	7H-dibenzo(a,c,)cyclohepten-5-one-(7) derivatives The invention is concerned with 7H-dibenzo(a,c)-cyclohepten-5-one-(7) derivatives of general formula I ##STR1## wherein R1 and R2 can be the same or different, a hydrogen atom, an alkyl radical containing 1 to 3 carbon atoms, or...	08/12/1986
4508732	Basic ethers useful as antidepressant agents Basic ethers of the formula ##STR1## wherein Z is CH3 -NR2 -CH2 CH2 -CHR1 --, (1-R2 -3-piperidyl)-CHR3 --, (1-R2 -2-piperidyl)-CH2 -CHR3 -- ...	04/02/1985
4376123	Hexahydroazepinyloxy-chromones useful as antidepressants Basic ethers of the formula ##STR1## wherein Z is CH3 --NR2 --CH2 CH2 --CHR1 --, (1-R2 -3-piperidyl)-CHR3 --, (1-R2 -2-piperidyl)-CH2 --CHR3...	03/08/1983
4327214	Substituted alkylammonium salts, the manufacture thereof, the use thereof for regulating plant growth, and agents therefor Substituted alkylammonium salts of the formula ##STR1## where R1, R2 and R3 are hydrogen, C1-4 -alkyl, fluorine, chlorine or bromine, X is oxygen or sulfur, n denotes one of the integers 2, 3 and 4, A denot...	04/27/1982
4313005	Inhibiting amidine formation during hydrogenation of organo nitriles This invention relates to a process for reducing amidine formation during reduction of organonitriles. The process comprises including a boron compound in the reaction medium in sufficient amount to complex the amidine compound as it is formed....	01/26/1982
4231942	Styryl compounds There are described new styryl compounds of the formula ##STR1## in which X is .dbd.CH2, --O--, --S-- or the grouping .dbd.NR3 wherein R3 is hydrogen or an alkyl group having 1 to 4 carbon atoms, Z is the --O-- or --S-- at...	11/04/1980
4194009	Aryloxyphenylpropylamines for obtaining a psychotropic effect 3-Aryloxy-3-phenylpropylamines and acid additions salts thereof, useful as psychotropic agents, particularly as anti-depressants....	03/18/1980
4169897	2,7-Bis-basic ethers of 9-phenanthrol and 9-loweralkoxy phenanthrol Novel bis-basic ethers of 9-substituted phenanthrene and related 10-oxa and 10-aza derivatives, their method of preparation and their use as pharmaceutical agents for the prevention and inhibition of viral infections are disclosed....	10/02/1979
4140779	Aryloxy propyldiamines Disclosed herein are compounds of the formula ##STR1## in which Ar is l-naphthyl; R1 and R2 are either the same or different selected from the group consisting of hydrogen or lower alkyl, or R1 and R2 toget...	02/20/1979
4119666	2-Decarboxy-2-amino-methyl-9-deoxy-9-methylene-PGF-type compounds This invention comprises certain analogs PGE or 11-deoxy-PGE compounds in which the carbonyl at C-9 is replaced by methylene. Also provided in this invention, are novel chemical processes and novel chemical intermediates useful in the preparation of the a...	10/10/1978
4067903	Manufacture of arylamines Arylamines are manufactured by reacting alcohols with amines in the presence of phosphorus-III compounds. The arylamines I manufactured by the process of the invention are intermediates for the manufacture of crop protection agents, optical brighteners, e...	01/10/1978
4059702	3,8-Bis-basic ethers of 6H-dibenzo[b,d]pyran-6-one Bis-basic ethers of 9-sustituted phenanthrene and related 10-oxa and 10-aza derivatives, their method of preparation and their use as pharmaceutical agents for the prevention and inhibition of viral infections are disclosed....	11/22/1977
4051166	Araliphatic diisocyanates Novel araliphatic diisocyanates having the formula are disclosed wherein X is oxygen or a single bond and Ar is an arylene radical. The araliphatic diisocyanates are prepared from well known and readily obtainable starting materials. When X represents a single...	09/27/1977

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Class 564/352 - The aryl ring or ring system is polycyclo