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Patent No. 5678617

Method and apparatus for making a drink hop along a bar or counter

A method for generating a drink which appears to hop from a remote spot on the bar or counter and take one or more leaps, before landing in a patron's glass.

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Class 564/345 - Halogen bonded directly to the aryl ring or ring system


Subclass of Class 564 - Organic compounds -- part of the class 532-570 series
Definition: Compounds wherein the aryl ring or ring system contains
No. of patents: 69
Last issue date: 06/30/2009


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NumberTitleIssue Date
7553992Modified release formulations of a bupropion salt
The present invention relates to pharmaceutical compositions, formulations and medicaments comprising a bupropion salt, in particular, modified-release tablets comprising an effective amount of bupropion hydrobromide, and the use of the bupropion salt to prepare a m...
06/30/2009
7091382Synthesis of N-methyl-N-phenylaminoacrolein
A process is disclosed for manufacturing N-methyl-N-phenylaminoacrolein of formula (I) which comprises reacting N-methylformanilide and an alkyl vinyl ether of formula (III)
08/15/2006
6765022Cyclohexylamine derivatives as subtype selective nmda receptor antagonists
Described are cyclobexylamine derivatives of Formula I, Formula II, or Formula III and their pharmaceutically acceptable salts thereof: The compounds are antagonists of NMDA receptor channel complexes useful for treating...
07/20/2004
66535083-amino-2-benzyl-1-phenylpropane derivatives
Substituted 3-amino-2-benzyl-1-phenlypropane derivatives, methods for preparing them, pharmaceutical compositions containing them, and methods of using them to treat various medical conditions....
11/25/2003
6482987Pharmaceutical composition containing bupropion hydrochloride and a stabilizer
Novel, stable formulations of bupropion hydrochloride are provided which will maintain at least 80% of initial bupropion hydrochloride potency after one year. Methods of inhibiting degradation of bupropion hydrochloride and methods of preparing stable for...
11/19/2002
6462237Cyclodextrin stabilized pharmaceutical compositions of bupropion hydrochloride
An inclusion complex of bupropion hydrochloride with beta cyclodextrin that stabilizes the bupropion hydrochloride against degradation. A method of preparing an inclusion complex of bupropion hydrochloride with beta cyclodextrin that stabilizes the buprop...
10/08/2002
6350767Compounds with growth hormone releasing properties
The present invention relates to compounds, compositions containing them, and their use for treating medical disorders resulting from a deficiency in growth hormone....
02/26/2002
6235791Use of amines to produce drugs for preventing tumor cell proliferation
The present invention relates to the use of compounds capable of displacing tritiated cis-N-cyclohexyl-N-ethyl [3-(3-chloro-4-cyclohexylphenyl)-allyl]amine from its receptors for the preparation of pharmaceutical compositions intended to combat cell ...
05/22/2001
6087346Sigma receptor ligands and the use thereof
The invention relates to methods for the treatment of central nervous system disorders, neurological disorders, gastrointestinal disorders, drug abuse, angina, migraine, hypertension and depression by administering a pharmaceutical composition comprising ...
07/11/2000
6057371Sigma receptor ligands and the use thereof
The invention relates to methods for the treatment of central nervous system disorders, gastrointestinal disorders, drug abuse, angina, migraine, hypertension and depression by administering a pharmaceutical composition comprising an effective amount of c...
05/02/2000
5977178Compounds with growth hormone releasing properties
Compounds of peptide mimetic nature having the general formula I ##STR1## wherein a and b are independently 1 or 2, R1 and R2 are independently H or C1-6 alkyl, G and J are independently, inter alia, aromats, and D an...
11/02/1999
5789448Benzoylethylene derivative
Disclosed is a benzoylethylene derivative represented by the following formula (I) or a salt thereof. ##STR1## R1 to R5 : a hydrogen atom, --OR9 (R9 : a hydrogen atom, a C1 -C5 alkyl g...
08/04/1998
5780505Substituted N-arylmethylamino derivatives of cyclobutene-3, 4-diones
The compounds of the formula: ##STR1## wherein R1 is straight chain alkyl, branched chain alkyl, cycloalkyl, hydroxyalkyl, fluoroalkyl or polyfluoroalkyl; R7 and R8 are, independently, hydrogen or an acyl substituent ...
07/14/1998
5741821Use of natural products and related synthetic compounds for the treatment of cardiovascular disease
Use of a compound of formula (I), wherein Ar is an aromatic ring system comprising one or more optionally substituted phenyl rings optionally linked to or fused with one or more other optionally substituted phenyl rings or one or more 5 or 6-membered, opt...
04/21/1998
5674909Derivatives of 2-amino-1,2,3,4-tetrahydronaphthalene active on the cardiovascular system
Compounds of formula ##STR1## wherein R, R', R", R1, R2, R3, R4, R5, R6, X, Y, m, n and p have the meanings reported in the description; and their pharmaceutically acceptable salts are desc...
10/07/1997
5561135N,N,N',N'-tetrasubstituted-1,2-ethanediamine derivative compounds
The invention relates to new N,N,N'N'-tetra-substituted-1,2-ethanediamine compounds of the general formula (I): ##STR1## wherein X is a carbonyl (CO), hydroxymethylen (CHOH) or p-fluorophenyl-methylen (p--F--C6 H4 --CH) group an...
10/01/1996
5037980Phenyl imidazo[1,2-a]pyrimidines
A compound of the formula: ##STR1## wherein R1 is ##STR2## where R3, R4 and R5 may be the same or different and are hydrogen, trihalomethyl, halogen or lower alkoxy having from 1 to 3 carbon atom...
08/06/1991
50361071,7-substituted heptyn-2-ones and use
1-Phenyl-7-substituted-hept-5-yn-2-ones substituted with a C1 to C7 alkyl, C3 to C6 cycloalkyl, aryl, heteroaryl or heterocycloalkyl group at the 1-position and an amino, a dialkylamino, a piperidyl, a pyrrolidy...
07/30/1991
4996318Amino-9,10-secosteroids useful for treating head injury, spinal cord trauma or stroke
The amino-9,10-secosteroids ##STR1## of the present invention contain an amino group attached to the terminal carbon atom of the C17 -side chain and are useful as pharmaceutical agents for treating a number of conditions including spinal t...
02/26/1991
4981990Intermediates in the preparation of 4-phenylpyrrole derivatives
The invention relates to a process for the preparation of 4-phenylpyrrole derivatives of the formula I ##STR1## wherein Rn, R1 and R2 are as defined in claim 1, which comprises reacting a phenacylamine of formula II ...
01/01/1991
49803771-(aminophenyl)-2-aminopropanone derivatives
The present invention relates to the preparation of new 1-(aminophenyl)-2-aminopropanone derivatives of the general formula: ##STR1## in which X is NH2, Y is H or a halogen atom, Z is H or a halogen atom, R1 is C1 -C
12/25/1990
4948813Benzylketone phospholipase A2 inhibitors
The invention relates to benzylketone phospholipase A2 inhibitors, pharmaceutical compositions containing them, and methods of treating phospholipase A2 -mediated conditions in mammals by administration of a therapeutically effective...
08/14/1990
49333701-aminophenyl-2-dimethylaminopropanone derivatives, method of preparation and use in therapy
The present invention relates, by way of novel industrial products, to 1-(4-aminophenyl)-2-dimethylaminopropanone derivatives which are selected from: (a) the compounds having the general formula ##STR1## in which R is H or CH3 CO, and (b...
06/12/1990
4906781Method for the preparation of 4'-(substituted)-amino-2-(substituted) amino-3',5'-dichloroacetophenone and salts thereof
A method for the preparation of 4'-(substituted)-amino-2-(substituted)amino-3',5'-dichloroacetophenone and salts thereof. The method involves the chlorination of the corresponding 4'-(substituted)amino-2-(substituted) aminoacetophenone and acid addition ...
03/06/1990
4861854Photosensitive polyimide precursor
A photosensitive polyimide precursor composed of the structural units (A) represented by the following general formula (I) and the structural units (B) represented by the following general formula (II), in which the ratio of the molar quantity of the stru...
08/29/1989
48472564,5-dihydro and 4,5,6,7-tetrahydropyrazolo(1,5-A)-pyrimidines
Novel compounds having the following structural formula: ##STR1## wherein - - - may represent the presence of a double bond between the C6 and C7 position, Ia, or the absence of a double bond between the C6 and C...
07/11/1989
4835315Fluorophenacyl-amine derivatives and application thereof in therapeutics
The present invention relates to new compounds belonging to the family of fluorophenacyl-amine derivates of formula: ##STR1## [wherein A is CO or CHOH and R is CH(CH3)2 or C(CH3)3 ] and selected from the gr...
05/30/1989
48164891-(aminophenyl)-2-aminoethanone derivatives
The present invention relates to the preparation of new derivatives selected from the group consisting of: (i) 1-(aminophenyl)-2-(alkylamino)ethanones of the formula: ##STR1## in which R is CH(CH3)2 or C(CH3)3 ...
03/28/1989
4803225Dihydroxy-phenethylamino compounds useful as pharmaceuticals
There are provided compounds of formula I, ##STR1## and pharmaceutically acceptable derivatives thereof. There are also described the use of the compounds of formula I as pharmaceuticals, methods for making the compounds and pharmaceutical, e.g. card...
02/07/1989
4762829Polyprenyl compound, process for the production thereof and drug containing the same
A novel polyprenyl compound such as a polyprenyl carboxylic acid amide is disclosed. It has antithrombic and antiplatelet aggregation activity....
08/09/1988
4749792Diamino ketones and alcohols as analgesic agents
Analgesic activity is exhibited by compounds having the formula ##STR1## and pharmaceutically acceptable salts thereof wherein R1, R2 and R4 are each independently hydrogen, alkyl, carboxyalkyl, halosubstituted alkyl,...
06/07/1988
4742058Polyprenyl compound, process for the production thereof and drug containing the same
A novel polyprenyl compound such as a polyprenyl carboxylic acid amide is disclosed. It has antithrombic and antiplatelet aggregation activity....
05/03/1988
4728659Aminomethyl derivatives and preparation process thereof as well as platelet aggregation inhibitors containing same
Disclosed herein are aminomethyl derivatives each of which is of the following general formula (I): ##STR1## wherein A represents a group --C.tbd.C-- or --CH.dbd.CH--, Y represents a group ##STR2## (in which R3 being a lower alky...
03/01/1988
4723039Phenylacetaldehydes substituted by basic groups, their preparation and drugs containing these compounds
Phenylacetaldehydes which are substituted by basic groups, of the formula ##STR1## where R1 to R8, m and n have the meanings stated in the description, and their preparation are described. The substances are useful for the treat...
02/02/1988
4720586Substituted 3,4-dihydroxy-phenylethylamino compounds
There are provided compounds of formula I, ##STR1## in which R1 represents OH, R2 and R3, which may be the same or different, each independently represent hydrogen, fluorine, chlorine, bromine, alkyl C1 to 6, nitro, n...
01/19/1988
4670535Photosensitive polyimide precursor and process for producing the same
The photosensitive polyimide precursor of the invention has a recurring unit represented by the following general formula [I]: ##STR1## (R1 represents a tetravalent aromatic hydrocarbon residue; R2 and R3 each represe...
06/02/1987
4467094Precursors to ethylenediamine derivatives
New derivatives of 1,2-ethylenediamine and salts thereof endowed with vascular antispasmodic and antiallergic activity; processes for preparing them, some new intermediates useful in their preparation and pharmaceutical compositions containing them....
08/21/1984
4438138Reduction of cholesterol with meta-chloro ଱-t-butylaminopropiophenone
A method of treatment for reducing cholesterol in humans by the administration of the compound of the formula I ##STR1## or a pharmaceutically acceptable acid addition salt thereof in a non-toxic, effective therapeutic amount (calculated as base) to ...
03/20/1984
4400380Antiviral 1-aryl-5-amino-1-penten-3-ones
Compounds of the formula ##STR1## wherein R is H, halo, C1-4 alkyl, C1-4 alkoxy, 3,4-methylenedioxy, CF3, NO2, NH2, N(C1-4 alkyl)2, CN, OH, --S(C1-4 alkyl) or --S...
08/23/1983
4326077N-Haloacetylphenylamino carbonyl cyclic intermediates
Novel N-haloacetylphenylamino carbonyl oximes represented by the formula ##STR1## wherein Ar is phenyl or substituted phenyl; R1 is halomethyl; R2 and R3 are each independently hydrogen, alkyl, phenyl, benzyl, substit...
04/20/1982
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